6KEE
| Crystal structure of BRD4 Bromodomain1 with an inhibitor | 分子名称: | 6-[2-[2,4-bis(fluoranyl)phenoxy]-5-(methylsulfonylmethyl)pyridin-3-yl]-8-methyl-2H-pyrrolo[1,2-a]pyrazin-1-one, Bromodomain-containing protein 4 | 著者 | Xiao, S, Li, Z, Chen, S, Zhou, B, Luo, C. | 登録日 | 2019-07-04 | 公開日 | 2020-07-08 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (2.12154651 Å) | 主引用文献 | Crystal structure of BRD4 Bromodomain1 with an inhibitor To be published
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6KEG
| BRD4 Bromodomain1 with an inhibitor | 分子名称: | 6-[2-[2,4-bis(fluoranyl)phenoxy]-5-(ethylsulfonylmethyl)pyridin-3-yl]-8-methyl-4H-pyrrolo[1,2-a]pyrazin-1-one, Bromodomain-containing protein 4 | 著者 | Xiao, S, Li, Z, Chen, S, Zhou, B, Luo, C. | 登録日 | 2019-07-04 | 公開日 | 2020-07-08 | 最終更新日 | 2024-03-27 | 実験手法 | X-RAY DIFFRACTION (2.232 Å) | 主引用文献 | BRD4 Bromodomain1 with an inhibitor To Be Published
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6KEF
| BRD4 Bromodomain1 with an inhibitor | 分子名称: | Bromodomain-containing protein 4, N-[3-(8-methyl-1-oxidanylidene-2H-pyrrolo[1,2-a]pyrazin-6-yl)-4-phenoxy-phenyl]methanesulfonamide | 著者 | Xiao, S, Li, Z, Chen, S, Zhou, B, Luo, C. | 登録日 | 2019-07-04 | 公開日 | 2020-07-08 | 最終更新日 | 2024-03-27 | 実験手法 | X-RAY DIFFRACTION (2.44467545 Å) | 主引用文献 | BRD4 Bromodomain1 with an inhibitor To Be Published
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6KED
| BRD4 Bromodomain1 with an inhibitor | 分子名称: | 6-[2-[2,4-bis(fluoranyl)phenoxy]-5-(methylsulfonylmethyl)pyridin-3-yl]-8-methyl-2H-pyrrolo[1,2-d][1,2,4]triazin-1-one, Bromodomain-containing protein 4 | 著者 | Xiao, S, Li, Z, Chen, S, Zhou, B, Luo, C. | 登録日 | 2019-07-04 | 公開日 | 2020-07-08 | 最終更新日 | 2024-03-27 | 実験手法 | X-RAY DIFFRACTION (2.548447 Å) | 主引用文献 | BRD4 Bromodomain1 with an inhibitor To Be Published
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5Z90
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5Z8G
| BRD4 Bromodomain 1 with an inhibitor | 分子名称: | 1-ethyl-6-[(3R)-3-oxidanylpiperidin-1-yl]sulfonyl-benzo[cd]indol-2-one, Bromodomain-containing protein 4, DIMETHYL SULFOXIDE | 著者 | Xiao, S, Chen, S, Chen, H. | 登録日 | 2018-01-31 | 公開日 | 2019-02-06 | 最終更新日 | 2024-03-27 | 実験手法 | X-RAY DIFFRACTION (1.701 Å) | 主引用文献 | BRD4 Bromodomain 1 with an inhibitor To Be Published
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5Z8R
| BRD4 Bromodomain 1 with an inhibitor | 分子名称: | 1-ethyl-6-[(3S)-3-oxidanylpiperidin-1-yl]sulfonyl-benzo[cd]indol-2-one, Bromodomain-containing protein 4 | 著者 | Xiao, S, Chen, S, Chen, H. | 登録日 | 2018-02-01 | 公開日 | 2019-02-06 | 最終更新日 | 2024-03-27 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | BRD4 Bromodomain 1 with an inhibitor To Be Published
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5Z9K
| BRD4 Bromodomain 1 with an inhibitor | 分子名称: | 1-ethyl-6-[(2R)-2-(hydroxymethyl)pyrrolidin-1-yl]sulfonyl-benzo[cd]indol-2-one, Bromodomain-containing protein 4 | 著者 | Xiao, S, Chen, S, Chen, H. | 登録日 | 2018-02-03 | 公開日 | 2019-02-06 | 最終更新日 | 2024-03-27 | 実験手法 | X-RAY DIFFRACTION (1.89 Å) | 主引用文献 | BRD4 Bromodomain 1 with an inhibitor To Be Published
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5Z8Z
| BRD4 Bromodomain 1 with an inhibitor | 分子名称: | 6-[(3S)-3-azanylpiperidin-1-yl]sulfonyl-1-ethyl-benzo[cd]indol-2-one, Bromodomain-containing protein 4 | 著者 | Xiao, S, Chen, S, Chen, H. | 登録日 | 2018-02-01 | 公開日 | 2019-02-06 | 最終更新日 | 2024-03-27 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | BRD4 Bromodomain 1 with an inhibitor To Be Published
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2LSW
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2N9D
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2N2N
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2N31
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5T7Q
| TIRAP phosphoinositide-binding motif | 分子名称: | Toll/interleukin-1 receptor domain-containing adapter protein | 著者 | Capelluto, D.G.S, Ellena, J.F, Armstrong, G, Zhao, X, Xiao, S. | 登録日 | 2016-09-05 | 公開日 | 2017-03-08 | 最終更新日 | 2024-05-15 | 実験手法 | SOLUTION NMR | 主引用文献 | Membrane targeting of TIRAP is negatively regulated by phosphorylation in its phosphoinositide-binding motif. Sci Rep, 7, 2017
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5KZF
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6LKX
| The structure of PRRSV helicase | 分子名称: | CITRIC ACID, GLYCEROL, RNA-dependent RNA polymerase, ... | 著者 | Shi, Y.J, Tong, X.H, Peng, G.Q. | 登録日 | 2019-12-20 | 公開日 | 2020-05-27 | 最終更新日 | 2021-06-09 | 実験手法 | X-RAY DIFFRACTION (2.998 Å) | 主引用文献 | Structural Characterization of the Helicase nsp10 Encoded by Porcine Reproductive and Respiratory Syndrome Virus. J.Virol., 94, 2020
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5KWA
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7YRV
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7YRW
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7YRX
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4XFQ
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4WZF
| Crystal structural basis for Rv0315, an immunostimulatory antigen and pseudo beta-1, 3-glucanase of Mycobacterium tuberculosis | 分子名称: | 1,2-ETHANEDIOL, 1,3-beta-glucanase, CALCIUM ION | 著者 | Dong, W.Y, Fu, Z.F, Peng, G.Q. | 登録日 | 2014-11-19 | 公開日 | 2015-12-09 | 最終更新日 | 2024-03-20 | 実験手法 | X-RAY DIFFRACTION (1.699 Å) | 主引用文献 | Crystal structural basis for Rv0315, an immunostimulatory antigen and inactive beta-1,3-glucanase of Mycobacterium tuberculosis. Sci Rep, 5, 2015
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4ZUH
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6LPA
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6LP9
| the protein of cat virus | 分子名称: | nsp1 protein | 著者 | Shen, Z, Peng, G.Q. | 登録日 | 2020-01-09 | 公開日 | 2020-08-12 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (1.803 Å) | 主引用文献 | Structural and Biological Basis of Alphacoronavirus nsp1 Associated with Host Proliferation and Immune Evasion. Viruses, 12, 2020
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