5Z9K

BRD4 Bromodomain 1 with an inhibitor

Summary for 5Z9K

• Entry DOI: 10.2210/pdb5z9k/pdb
• Descriptor: Bromodomain-containing protein 4, 1-ethyl-6-[(2R)-2-(hydroxymethyl)pyrrolidin-1-yl]sulfonyl-benzo[cd]indol-2-one (3 entities in total)
• Functional Keywords: brd4 bromodomain 1, inhibitor, complex, transcription-inhibitor complex, transcription/inhibitor
• Biological source: Homo sapiens (Human)
• Total number of polymer chains: 1
• Total formula weight: 15459.81

Authors

Xiao, S.,Chen, S.,Chen, H. (deposition date: 2018-02-03, release date: 2019-02-06, Last modification date: 2024-03-27)

• Primary citation: Xiao, S.,Chen, S.,Chen, H.; BRD4 Bromodomain 1 with an inhibitor; To Be Published,

Experimental method

X-RAY DIFFRACTION (1.89 Å)