6NUG
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![BU of 6nug by Molmil](/molmil-images/mine/6nug) | hGRNA4-28_3s | 分子名称: | Granulin-4 | 著者 | Dastpeyman, M, Bansal, P, Wilson, D, Loukas, A, Smout, M, Daly, N. | 登録日 | 2019-02-01 | 公開日 | 2020-02-05 | 最終更新日 | 2023-06-14 | 実験手法 | SOLUTION NMR | 主引用文献 | hGRN4-28_3s to be published
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6E1L
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![BU of 6e1l by Molmil](/molmil-images/mine/6e1l) | GRN3Ala | 分子名称: | Granulin | 著者 | Dastpeyman, M, Bansal, P, Wilson, D, Sotillo, J, Brindley, P, Loukas, A, Smout, M, Daly, N. | 登録日 | 2018-07-10 | 公開日 | 2019-02-06 | 最終更新日 | 2023-06-14 | 実験手法 | SOLUTION NMR | 主引用文献 | Structural Variants of a Liver Fluke Derived Granulin Peptide Potently Stimulate Wound Healing. J. Med. Chem., 61, 2018
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5UJH
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![BU of 5ujh by Molmil](/molmil-images/mine/5ujh) | ov-GRN12-34 | 分子名称: | Granulin | 著者 | Bansal, P, Smout, M, Wilson, D, Caceres, C.C, Dastpeyman, M, Sotillo, J, Seifert, J, Brindley, P, Loukas, A, Daly, N. | 登録日 | 2017-01-18 | 公開日 | 2018-01-24 | 最終更新日 | 2023-06-14 | 実験手法 | SOLUTION NMR | 主引用文献 | Development of a Potent Wound Healing Agent Based on the Liver Fluke Granulin Structural Fold. J. Med. Chem., 60, 2017
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1KQH
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![BU of 1kqh by Molmil](/molmil-images/mine/1kqh) | NMR Solution Structure of the cis Pro30 Isomer of ACTX-Hi:OB4219 | 分子名称: | ACTX-Hi:OB4219 | 著者 | Rosengren, K.J, Wilson, D, Daly, N.L, Alewood, P.F, Craik, D.J. | 登録日 | 2002-01-05 | 公開日 | 2002-02-06 | 最終更新日 | 2022-02-23 | 実験手法 | SOLUTION NMR | 主引用文献 | Solution structures of the cis- and trans-Pro30 isomers of a novel 38-residue toxin
from the venom of Hadronyche Infensa sp. that contains a cystine-knot motif within
its four disulfide bonds Biochemistry, 41, 2002
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5UJG
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![BU of 5ujg by Molmil](/molmil-images/mine/5ujg) | ovGRN12-35_3s | 分子名称: | Granulin | 著者 | Bansal, P, Smout, M, Wilson, D, Caceres, C.C, Dastpeyman, M, Sotillo, J, Seifert, J, Brindley, P, Loukas, A, Daly, N. | 登録日 | 2017-01-17 | 公開日 | 2018-01-24 | 最終更新日 | 2023-06-14 | 実験手法 | SOLUTION NMR | 主引用文献 | Development of a Potent Wound Healing Agent Based on the Liver Fluke Granulin Structural Fold. J. Med. Chem., 60, 2017
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1KQI
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![BU of 1kqi by Molmil](/molmil-images/mine/1kqi) | NMR Solution Structure of the trans Pro30 Isomer of ACTX-Hi:OB4219 | 分子名称: | ACTX-Hi:OB4219 | 著者 | Rosengren, K.J, Wilson, D, Daly, N.L, Alewood, P.F, Craik, D.J. | 登録日 | 2002-01-06 | 公開日 | 2002-02-06 | 最終更新日 | 2022-02-23 | 実験手法 | SOLUTION NMR | 主引用文献 | Solution structures of the cis- and trans-Pro30 isomers of a novel 38-residue toxin
from the venom of Hadronyche Infensa sp. that contains a cystine-knot motif within
its four disulfide bonds Biochemistry, 41, 2002
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8QUS
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![BU of 8qus by Molmil](/molmil-images/mine/8qus) | |
8QU7
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![BU of 8qu7 by Molmil](/molmil-images/mine/8qu7) | |
1G9P
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![BU of 1g9p by Molmil](/molmil-images/mine/1g9p) | |
1HP3
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![BU of 1hp3 by Molmil](/molmil-images/mine/1hp3) | |
7JIY
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![BU of 7jiy by Molmil](/molmil-images/mine/7jiy) | |
7JIA
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![BU of 7jia by Molmil](/molmil-images/mine/7jia) | |
6PPC
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![BU of 6ppc by Molmil](/molmil-images/mine/6ppc) | |
3BON
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![BU of 3bon by Molmil](/molmil-images/mine/3bon) | |
3BOO
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![BU of 3boo by Molmil](/molmil-images/mine/3boo) | |
3BOK
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![BU of 3bok by Molmil](/molmil-images/mine/3bok) | |
5J4Y
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![BU of 5j4y by Molmil](/molmil-images/mine/5j4y) | |
5J40
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![BU of 5j40 by Molmil](/molmil-images/mine/5j40) | The X-ray structure of JCV Helicase | 分子名称: | 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, Large T antigen, SULFATE ION, ... | 著者 | Ter Haar, E. | 登録日 | 2016-03-31 | 公開日 | 2016-07-20 | 最終更新日 | 2024-03-06 | 実験手法 | X-RAY DIFFRACTION (2.17 Å) | 主引用文献 | Fragment-Based Discovery of Dual JC Virus and BK Virus Helicase Inhibitors. J.Med.Chem., 59, 2016
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5J4V
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![BU of 5j4v by Molmil](/molmil-images/mine/5j4v) | The crystal structure of Inhibitor Bound to JCV Helicase | 分子名称: | 2-(2-phenoxypyridin-3-yl)[1,3]thiazolo[5,4-c]pyridine, 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, Large T antigen, ... | 著者 | Ter Haar, E. | 登録日 | 2016-04-01 | 公開日 | 2016-07-20 | 最終更新日 | 2024-03-06 | 実験手法 | X-RAY DIFFRACTION (2.94 Å) | 主引用文献 | Fragment-Based Discovery of Dual JC Virus and BK Virus Helicase Inhibitors. J.Med.Chem., 59, 2016
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5J47
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![BU of 5j47 by Molmil](/molmil-images/mine/5j47) | The X-ray structure of Inhibitor Bound to JCV Helicase | 分子名称: | 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, 6-(2-phenoxyphenyl)[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole, Large T antigen, ... | 著者 | Ter Haar, E. | 登録日 | 2016-03-31 | 公開日 | 2016-07-20 | 最終更新日 | 2024-03-06 | 実験手法 | X-RAY DIFFRACTION (1.99 Å) | 主引用文献 | Fragment-Based Discovery of Dual JC Virus and BK Virus Helicase Inhibitors. J.Med.Chem., 59, 2016
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8EL2
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![BU of 8el2 by Molmil](/molmil-images/mine/8el2) | SARS-CoV-2 RBD bound to neutralizing antibody Fab ICO-hu23 | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, Fab ICO-hu23 Heavy Chain, Fab ICO-hu23 Light Chain, ... | 著者 | Besaw, J.E, Kuo, A, Morizumi, T, Ernst, O.P. | 登録日 | 2022-09-22 | 公開日 | 2023-07-19 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (2.89 Å) | 主引用文献 | Broadly neutralizing humanized SARS-CoV-2 antibody binds to a conserved epitope on Spike and provides antiviral protection through inhalation-based delivery in non-human primates. Plos Pathog., 19, 2023
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8ELJ
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![BU of 8elj by Molmil](/molmil-images/mine/8elj) | SARS-CoV-2 spike glycoprotein in complex with the ICO-hu23 neutralizing antibody Fab fragment | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ICO-hu23 antibody Fab heavy chain, ... | 著者 | Yee, A.W, Morizumi, T, Kim, K, Kuo, A, Ernst, O.P. | 登録日 | 2022-09-24 | 公開日 | 2023-07-19 | 最終更新日 | 2023-08-16 | 実験手法 | ELECTRON MICROSCOPY (3.6 Å) | 主引用文献 | Broadly neutralizing humanized SARS-CoV-2 antibody binds to a conserved epitope on Spike and provides antiviral protection through inhalation-based delivery in non-human primates. Plos Pathog., 19, 2023
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2NTA
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![BU of 2nta by Molmil](/molmil-images/mine/2nta) | Crystal Structure of PTP1B-inhibitor Complex | 分子名称: | 5-(4-CHLORO-5-PHENYL-3-THIENYL)-1,2,5-THIADIAZOLIDIN-3-ONE 1,1-DIOXIDE, Tyrosine-protein phosphatase non-receptor type 1 | 著者 | Xu, W, Follows, B. | 登録日 | 2006-11-07 | 公開日 | 2007-04-17 | 最終更新日 | 2023-12-27 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | Probing acid replacements of thiophene PTP1B inhibitors. Bioorg.Med.Chem.Lett., 17, 2007
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2NT7
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![BU of 2nt7 by Molmil](/molmil-images/mine/2nt7) | Crystal structure of PTP1B-inhibitor complex | 分子名称: | Tyrosine-protein phosphatase non-receptor type 1, {[5-(3-{[1-(BENZYLSULFONYL)PIPERIDIN-4-YL]AMINO}PHENYL)-4-BROMO-2-(2H-TETRAZOL-5-YL)-3-THIENYL]OXY}ACETIC ACID | 著者 | Xu, W, Follows, B. | 登録日 | 2006-11-07 | 公開日 | 2007-04-17 | 最終更新日 | 2023-12-27 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | Probing acid replacements of thiophene PTP1B inhibitors. Bioorg.Med.Chem.Lett., 17, 2007
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8D73
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![BU of 8d73 by Molmil](/molmil-images/mine/8d73) | Crystal Structure of EGFR LRTM with compound 7 | 分子名称: | (3S,4R)-3-fluoro-1-(4-{[4-(methylamino)-1-(propan-2-yl)pyrido[3,4-d]pyridazin-7-yl]amino}pyrimidin-2-yl)piperidin-4-ol, Epidermal growth factor receptor, GLYCEROL | 著者 | Kim, J.L. | 登録日 | 2022-06-07 | 公開日 | 2022-07-27 | 最終更新日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (2.17 Å) | 主引用文献 | Discovery of BLU-945, a Reversible, Potent, and Wild-Type-Sparing Next-Generation EGFR Mutant Inhibitor for Treatment-Resistant Non-Small-Cell Lung Cancer. J.Med.Chem., 65, 2022
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