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6FT8
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BU of 6ft8 by Molmil
Crystal structure of CLK1 in complex with inhibitor 8g
分子名称: 1,2-ETHANEDIOL, 3-(3-hydroxyphenyl)-1~{H}-pyrrolo[3,4-g]indol-8-one, CHLORIDE ION, ...
著者Chaikuad, A, Walter, A, von Delft, F, Bountra, C, Arrowsmith, C.H, Edwards, A.M, Kunick, C, Knapp, S, Structural Genomics Consortium (SGC)
登録日2018-02-20
公開日2018-05-16
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (1.45 Å)
主引用文献Molecular structures of cdc2-like kinases in complex with a new inhibitor chemotype.
PLoS ONE, 13, 2018
6FT7
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BU of 6ft7 by Molmil
Crystal structure of CLK3 in complex with compound 8a
分子名称: 1,2-ETHANEDIOL, 3-phenyl-1~{H}-pyrrolo[3,4-g]indol-8-one, Dual specificity protein kinase CLK3, ...
著者Chaikuad, A, Walter, A, von Delft, F, Bountra, C, Arrowsmith, C.H, Edwards, A.M, Kunick, C, Knapp, S, Structural Genomics Consortium (SGC)
登録日2018-02-20
公開日2018-05-16
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (2.02 Å)
主引用文献Molecular structures of cdc2-like kinases in complex with a new inhibitor chemotype.
PLoS ONE, 13, 2018
6FT9
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BU of 6ft9 by Molmil
Crystal structure of CLK1 in complex with inhibitor 16
分子名称: 2-bromanyl-3-phenyl-1~{H}-pyrrolo[3,4-g]indol-8-one, BROMIDE ION, Dual specificity protein kinase CLK1, ...
著者Chaikuad, A, Walter, A, von Delft, F, Bountra, C, Arrowsmith, C.H, Edwards, A.M, Kunick, C, Knapp, S, Structural Genomics Consortium (SGC)
登録日2018-02-20
公開日2018-05-16
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (1.87 Å)
主引用文献Molecular structures of cdc2-like kinases in complex with a new inhibitor chemotype.
PLoS ONE, 13, 2018
3DCV
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BU of 3dcv by Molmil
Crystal structure of human Pim1 kinase complexed with 4-(4-hydroxy-3-methyl-phenyl)-6-phenylpyrimidin-2(1H)-one
分子名称: 4-(4-hydroxy-3-methylphenyl)-6-phenylpyrimidin-2(5H)-one, Proto-oncogene serine/threonine-protein kinase Pim-1
著者Bellamacina, C.R, Shafer, C.M, Lindvall, M, Gesner, T.G, Yabannavar, A, Weiping, J, Song, L, Walter, A.
登録日2008-06-04
公開日2008-08-19
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (2.7 Å)
主引用文献4-(1H-indazol-5-yl)-6-phenylpyrimidin-2(1H)-one analogs as potent CDC7 inhibitors.
Bioorg.Med.Chem.Lett., 18, 2008
4XHV
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BU of 4xhv by Molmil
Crystal structure of Drosophila Spinophilin-PDZ and a C-terminal peptide of Neurexin
分子名称: 1,2-ETHANEDIOL, CHLORIDE ION, LP20995p, ...
著者Driller, J.H, Muhammad, K.G.H, Reddy, S, Rey, U, Boehme, M.A, Hollmann, C, Ramesh, N, Depner, H, Luetzkendorf, J, Matkovic, T, Bergeron, D, Quentin, C, Schmoranzer, J, Goettfert, F, Holt, M, Wahl, M.C, Hell, S.W, Walter, A, Sigrist, S.J, Loll, B.
登録日2015-01-06
公開日2015-07-01
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (1.23 Å)
主引用文献Presynaptic spinophilin tunes neurexin signalling to control active zone architecture and function.
Nat Commun, 6, 2015
8RDX
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BU of 8rdx by Molmil
PGGtase I in complex with probe BAY-6092
分子名称: (5~{R})-5-(2-methoxyphenyl)-9-[(2~{R})-3,3,3-tris(fluoranyl)-2-methoxy-2-phenyl-propanoyl]-3,9-diazaspiro[5.5]undecan-2-one, CHLORIDE ION, DIPHOSPHATE, ...
著者Steuber, H.
登録日2023-12-08
公開日2024-02-14
最終更新日2024-04-10
実験手法X-RAY DIFFRACTION (3.67 Å)
主引用文献Discovery of YAP1/TAZ pathway inhibitors through phenotypic screening with potent anti-tumor activity via blockade of Rho-GTPase signaling.
Cell Chem Biol, 2024
8P20
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BU of 8p20 by Molmil
TarM(Se)_G117R-UDP-4RboP-glucose
分子名称: BETA-MERCAPTOETHANOL, CHLORIDE ION, GLYCEROL, ...
著者Guo, Y, Stehle, T.
登録日2023-05-14
公開日2023-12-06
実験手法X-RAY DIFFRACTION (2.848 Å)
主引用文献Invasive Staphylococcus epidermidis uses a unique processive wall teichoic acid glycosyltransferase to evade immune recognition.
Sci Adv, 9, 2023
8P1X
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BU of 8p1x by Molmil
TarM(Se)_G117R-UDP-glucose
分子名称: 1,2-ETHANEDIOL, CHLORIDE ION, PHOSPHATE ION, ...
著者Guo, Y, Stehle, T.
登録日2023-05-13
公開日2023-12-06
実験手法X-RAY DIFFRACTION (2.03 Å)
主引用文献Invasive Staphylococcus epidermidis uses a unique processive wall teichoic acid glycosyltransferase to evade immune recognition.
Sci Adv, 9, 2023
8P60
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BU of 8p60 by Molmil
Spraguea lophii ribosome dimer
分子名称: 40S Ribosomal protein S19, 40S ribosomal protein S0, 40S ribosomal protein S1, ...
著者Gil Diez, P, McLaren, M, Isupov, M.N, Daum, B, Conners, R, Williams, B.
登録日2023-05-24
公開日2023-06-21
最終更新日2023-12-20
実験手法ELECTRON MICROSCOPY (14.3 Å)
主引用文献CryoEM reveals that ribosomes in microsporidian spores are locked in a dimeric hibernating state.
Nat Microbiol, 8, 2023
8P5D
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BU of 8p5d by Molmil
Spraguea lophii ribosome in the closed conformation by cryo sub tomogram averaging
分子名称: 40S Ribosomal protein S19, 40S ribosomal protein S0, 40S ribosomal protein S10, ...
著者Gil Diez, P, McLaren, M, Isupov, M.N, Daum, B, Conners, R, Williams, B.
登録日2023-05-23
公開日2023-06-21
最終更新日2023-12-20
実験手法ELECTRON MICROSCOPY (10.8 Å)
主引用文献CryoEM reveals that ribosomes in microsporidian spores are locked in a dimeric hibernating state.
Nat Microbiol, 8, 2023
7QD7
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BU of 7qd7 by Molmil
TarM(Se)_G117R
分子名称: CHLORIDE ION, GLYCEROL, PENTAETHYLENE GLYCOL, ...
著者Guo, Y, Stehle, T.
登録日2021-11-26
公開日2023-05-10
最終更新日2023-12-06
実験手法X-RAY DIFFRACTION (2.06 Å)
主引用文献Invasive Staphylococcus epidermidis uses a unique processive wall teichoic acid glycosyltransferase to evade immune recognition.
Sci Adv, 9, 2023
7QNT
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BU of 7qnt by Molmil
TarM(Se) native
分子名称: 1,2-ETHANEDIOL, BETA-MERCAPTOETHANOL, CHLORIDE ION, ...
著者Guo, Y, Stehle, T.
登録日2021-12-22
公開日2023-05-10
最終更新日2023-12-06
実験手法X-RAY DIFFRACTION (3.21 Å)
主引用文献Invasive Staphylococcus epidermidis uses a unique processive wall teichoic acid glycosyltransferase to evade immune recognition.
Sci Adv, 9, 2023
7QH9
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BU of 7qh9 by Molmil
TarM(Se)_G117R-4RboP
分子名称: 1,2-ETHANEDIOL, CHLORIDE ION, TarM(Se)_G117R-4RboP, ...
著者Guo, Y, Stehle, T.
登録日2021-12-10
公開日2023-05-10
最終更新日2023-12-06
実験手法X-RAY DIFFRACTION (2.689 Å)
主引用文献Invasive Staphylococcus epidermidis uses a unique processive wall teichoic acid glycosyltransferase to evade immune recognition.
Sci Adv, 9, 2023
7QCA
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BU of 7qca by Molmil
Spraguea lophii ribosome
分子名称: 40S Ribosomal protein S19, 40S ribosomal protein S0, 40S ribosomal protein S10, ...
著者Gil Diez, P, McLaren, M, Isupov, M.N, Daum, B, Conners, R, Williams, B.
登録日2021-11-22
公開日2022-11-30
最終更新日2023-12-20
実験手法ELECTRON MICROSCOPY (2.79 Å)
主引用文献CryoEM reveals that ribosomes in microsporidian spores are locked in a dimeric hibernating state
Nat Microbiol, 2023
4CQF
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BU of 4cqf by Molmil
Crystal structure of Schistosoma mansoni HDAC8 complexed with a mercaptoacetamide inhibitor
分子名称: 6-(2-Mercaptoacetylamino)-N-phenylhexanamide, DIMETHYLFORMAMIDE, GLYCEROL, ...
著者Marek, M, Romier, C.
登録日2014-02-14
公開日2014-04-02
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Molecular Basis for the Anti-Parasitic Activity of a Mercaptoacetamide Derivative that Inhibits Histone Deacetylase 8 (Hdac8) from the Human Pathogen Schistosoma Mansoni
J.Mol.Biol., 426, 2014

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件を2024-06-12に公開中

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