5E1V
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3U37
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4YX6
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4YXT
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4YXV
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4YXF
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5DZ6
| Acyl transferase from Bacillaene PKS | 分子名称: | 1,2-ETHANEDIOL, BROMIDE ION, CHLORIDE ION, ... | 著者 | Till, M, Race, P.R. | 登録日 | 2015-09-25 | 公開日 | 2016-10-05 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (1.44 Å) | 主引用文献 | Architectural hierarchy of trans-acting enoyl reductases from polyunsaturated fatty acid and trans-acyltransferase polyketide synthases To Be Published
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4NOV
| Xsa43E, a GH43 family enzyme from Butyrivibrio proteoclasticus | 分子名称: | 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, CALCIUM ION, Xylosidase/arabinofuranosidase Xsa43E | 著者 | Till, M, Arcus, V.L. | 登録日 | 2013-11-20 | 公開日 | 2014-10-08 | 実験手法 | X-RAY DIFFRACTION (1.33 Å) | 主引用文献 | Structural analysis of the GH43 enzyme Xsa43E from Butyrivibrio proteoclasticus ACTA CRYSTALLOGR.,SECT.F, 70, 2014
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4DEV
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5DZ7
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4YXQ
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5DZA
| Streptococcus agalactiae AgI/II polypeptide BspA C terminal domain (WT) | 分子名称: | 1,2-ETHANEDIOL, BspA, DI(HYDROXYETHYL)ETHER | 著者 | Rego, S, Till, M, Race, P.R. | 登録日 | 2015-09-25 | 公開日 | 2016-06-22 | 最終更新日 | 2024-06-12 | 実験手法 | X-RAY DIFFRACTION (2.19 Å) | 主引用文献 | Structural and Functional Analysis of Cell Wall-anchored Polypeptide Adhesin BspA in Streptococcus agalactiae. J.Biol.Chem., 291, 2016
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5DZ9
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5DZ8
| Streptococcus agalactiae AgI/II polypeptide BspA variable (V) domain | 分子名称: | 1,2-ETHANEDIOL, ACETATE ION, BspA (BspA_V), ... | 著者 | Rego, S, Till, M, Race, P.R. | 登録日 | 2015-09-25 | 公開日 | 2016-06-22 | 最終更新日 | 2016-08-10 | 実験手法 | X-RAY DIFFRACTION (2.41 Å) | 主引用文献 | Structural and Functional Analysis of Cell Wall-anchored Polypeptide Adhesin BspA in Streptococcus agalactiae. J.Biol.Chem., 291, 2016
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4Q1G
| Structure and mechanism of a dehydratase/decarboxylase enzyme couple involved in polyketide beta-branching | 分子名称: | 1,2-ETHANEDIOL, GLYCEROL, Polyketide biosynthesis enoyl-CoA isomerase PksI | 著者 | Nair, A.V, Race, P.R, Till, M. | 登録日 | 2014-04-03 | 公開日 | 2015-05-06 | 最終更新日 | 2024-05-22 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | Structure and mechanism of a dehydratase/decarboxylase enzyme couple involved in polyketide beta-methyl branch incorporation. Sci Rep, 10, 2020
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4Q1H
| Structure and mechanism of a dehydratase/decarboxylase enzyme couple involved in polyketide beta-branching | 分子名称: | 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, GLYCEROL, Polyketide biosynthesis enoyl-CoA isomerase PksI, ... | 著者 | Nair, A.V, Race, P.R, Till, M. | 登録日 | 2014-04-03 | 公開日 | 2015-05-06 | 最終更新日 | 2024-05-22 | 実験手法 | X-RAY DIFFRACTION (1.93 Å) | 主引用文献 | Structure and mechanism of a dehydratase/decarboxylase enzyme couple involved in polyketide beta-methyl branch incorporation. Sci Rep, 10, 2020
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4Q1K
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4Q1J
| Structure and mechanism of a dehydratase/decarboxylase enzyme couple involved in polyketide beta-branching | 分子名称: | 1,2-ETHANEDIOL, Polyketide biosynthesis enoyl-CoA isomerase PksI, SODIUM ION | 著者 | Nair, A.V, Race, P.R, Till, M. | 登録日 | 2014-04-03 | 公開日 | 2015-05-06 | 最終更新日 | 2024-05-22 | 実験手法 | X-RAY DIFFRACTION (2.17 Å) | 主引用文献 | Structure and mechanism of a dehydratase/decarboxylase enzyme couple involved in polyketide beta-methyl branch incorporation. Sci Rep, 10, 2020
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4Q1I
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4F4P
| SYK in COMPLEX WITH LIGAND LASW836 | 分子名称: | N-{6-[3-(piperazin-1-yl)phenyl]pyridin-2-yl}-4-(trifluoromethyl)pyridin-2-amine, SULFATE ION, Tyrosine-protein kinase SYK | 著者 | Lopez, M, Segarra, V, Vidal, B, Wenzkowski, C, Jestel, A, Krapp, S, Blaesse, M, Nagel, S, Schreiner, P. | 登録日 | 2012-05-11 | 公開日 | 2012-12-12 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (2.37 Å) | 主引用文献 | Highly potent aminopyridines as Syk kinase inhibitors. Bioorg.Med.Chem.Lett., 22, 2012
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8P99
| SARS-CoV-2 S-protein:D614G mutant in 1-up conformation | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Spike protein S1,Spike glycoprotein | 著者 | Adhav, A, Forcada-Nadal, A, Marco-Marin, C, Lopez-Redondo, M.L, Llacer, J.L. | 登録日 | 2023-06-05 | 公開日 | 2023-09-27 | 実験手法 | ELECTRON MICROSCOPY (3.4 Å) | 主引用文献 | C-2 Thiophenyl Tryptophan Trimers Inhibit Cellular Entry of SARS-CoV-2 through Interaction with the Viral Spike (S) Protein. J.Med.Chem., 66, 2023
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8P9Y
| SARS-CoV-2 S protein S:D614G mutant in 3-down with binding site of an entry inhibitor | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, SODIUM ION, ... | 著者 | Adhav, A, Forcada-Nadal, A, Marco-Marin, C, Lopez-Redondo, M.L, Llacer, J.L. | 登録日 | 2023-06-06 | 公開日 | 2023-09-27 | 実験手法 | ELECTRON MICROSCOPY (4.3 Å) | 主引用文献 | C-2 Thiophenyl Tryptophan Trimers Inhibit Cellular Entry of SARS-CoV-2 through Interaction with the Viral Spike (S) Protein. J.Med.Chem., 66, 2023
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5L2D
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2WTN
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2WTM
| Est1E from Butyrivibrio proteoclasticus | 分子名称: | EST1E, GLYCEROL, PHOSPHATE ION | 著者 | Goldstone, D.C, Arcus, V.L. | 登録日 | 2009-09-17 | 公開日 | 2010-01-19 | 最終更新日 | 2024-05-08 | 実験手法 | X-RAY DIFFRACTION (1.6 Å) | 主引用文献 | Structural and Functional Characterization of a Promiscuous Feruloyl Esterase (Est1E) from the Rumen Bacterium Butyrivibrio Proteoclasticus. Proteins, 78, 2010
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