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5VOE
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BU of 5voe by Molmil
DesGla-XaS195A Bound to Aptamer 11F7t
分子名称: Aptamer 11F7t (36-MER), CALCIUM ION, Coagulation factor X, ...
著者Gunaratne, R, Kumar, S, Frederiksen, J.W, Stayrook, S, Lohrmann, J.L, Perry, K, Chabata, C.V, Thalji, N.K, Ho, M.D, Arepally, G, Camire, R.M, Krishnaswamy, S.K, Sullenger, B.A.
登録日2017-05-02
公開日2018-06-20
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Combination of aptamer and drug for reversible anticoagulation in cardiopulmonary bypass.
Nat. Biotechnol., 36, 2018
3DD2
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BU of 3dd2 by Molmil
Crystal structure of an RNA aptamer bound to human thrombin
分子名称: ACETIC ACID, D-phenylalanyl-N-[(2S,3S)-6-{[amino(iminio)methyl]amino}-1-chloro-2-hydroxyhexan-3-yl]-L-prolinamide, DI(HYDROXYETHYL)ETHER, ...
著者Long, S.B, Sullenger, B.A.
登録日2008-06-04
公開日2008-11-11
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Crystal structure of an RNA aptamer bound to thrombin.
Rna, 14, 2008
8TQS
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BU of 8tqs by Molmil
Complex of human thrombin (S195A) bound to a bivalent inhibitor comprised of DNA Aptamer HD22 conjugated to Dabigatran with a linker.
分子名称: 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, 2-acetamido-2-deoxy-beta-D-glucopyranose, DNA (30-MER), ...
著者Krishnaswamy, S, Kumar, S.
登録日2023-08-08
公開日2024-05-01
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (2.207 Å)
主引用文献Aptameric hirudins as selective and reversible EXosite-ACTive site (EXACT) inhibitors.
Nat Commun, 15, 2024
5VOF
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BU of 5vof by Molmil
DesGla-XaS195A Bound to Aptamer 11F7t and Rivaroxaban
分子名称: 5-chloro-N-({(5S)-2-oxo-3-[4-(3-oxomorpholin-4-yl)phenyl]-1,3-oxazolidin-5-yl}methyl)thiophene-2-carboxamide, CALCIUM ION, Coagulation factor X, ...
著者Krishnaswamy, S, Kumar, S.
登録日2017-05-02
公開日2018-06-13
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (2.25 Å)
主引用文献Combination of aptamer and drug for reversible anticoagulation in cardiopulmonary bypass.
Nat. Biotechnol., 36, 2018
8EPC
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BU of 8epc by Molmil
Crystal structure of human coagulation factor IXa (S195A), apo-form
分子名称: CALCIUM ION, Coagulation factor IXa heavy chain, Coagulation factor IXa light chain
著者Kolyadko, V.N, Krishnaswamy, S.
登録日2022-10-05
公開日2024-07-03
実験手法X-RAY DIFFRACTION (2.51 Å)
主引用文献Allosteric Control of Coagulation Factor IXa via Its Exosite II Regulates Blood Clotting
Proc.Natl.Acad.Sci.USA, 2024
8EPH
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BU of 8eph by Molmil
Crystal structure of human coagulation factor IXa (S195A), apo-form, DES-GLA
分子名称: CALCIUM ION, Coagulation factor IXa heavy chain, Coagulation factor IXa light chain, ...
著者Kolyadko, V.N, Krishnaswamy, S.
登録日2022-10-05
公開日2024-07-03
実験手法X-RAY DIFFRACTION (1.88 Å)
主引用文献Allosteric Control of Coagulation Factor IXa via Its Exosite II Regulates Blood Clotting
Proc.Natl.Acad.Sci.USA, 2024
8EPK
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BU of 8epk by Molmil
Complex of anticoagulant RNA aptamer and human coagulation factor IXa (S195A)
分子名称: CALCIUM ION, Coagulation factor IXa heavy chain, Coagulation factor IXa light chain, ...
著者Kolyadko, V.N, Krishnaswamy, S.
登録日2022-10-05
公開日2024-07-03
実験手法X-RAY DIFFRACTION (2.65 Å)
主引用文献Allosteric Control of Coagulation Factor IXa via Its Exosite II Regulates Blood Clotting
Proc.Natl.Acad.Sci.USA, 2024

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件を2024-07-17に公開中

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