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6TC2
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BU of 6tc2 by Molmil
Monoclinic human insulin in complex with p-coumaric acid
分子名称: 4'-HYDROXYCINNAMIC ACID, Insulin, PHOSPHATE ION, ...
著者Triandafillidis, D.-P, Parthenios, N, Spiliopoulou, M, Valmas, A, Kosinas, C, Gozzo, F, Reinle-Schmitt, M, Beckers, D, Degen, T, Pop, M, Fitch, A, Wollenhaupt, J, Weiss, M.S, Karavassili, F, Margiolaki, I.
登録日2019-11-04
公開日2020-11-11
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (1.36 Å)
主引用文献Insulin polymorphism induced by two polyphenols: new crystal forms and advances in macromolecular powder diffraction.
Acta Crystallogr D Struct Biol, 76, 2020
3I5K
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BU of 3i5k by Molmil
Crystal structure of the NS5B polymerase from Hepatitis C Virus (HCV) strain JFH1
分子名称: PHOSPHATE ION, RNA-directed RNA polymerase
著者Simister, P.C, Schmitt, M, Lohmann, V, Bressanelli, S.
登録日2009-07-05
公開日2009-09-22
最終更新日2024-03-20
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Structural and functional analysis of hepatitis C virus strain JFH1 polymerase
J.Virol., 83, 2009
6SBR
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BU of 6sbr by Molmil
The crystal structure of PfA-M1 in complex with 7-amino-1,4-dibromo-5,7,8,9-tetrahydrobenzocyclohepten-6-one
分子名称: 2-[3-(2-HYDROXY-1,1-DIHYDROXYMETHYL-ETHYLAMINO)-PROPYLAMINO]-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, CHLORIDE ION, GLYCEROL, ...
著者Salomon, E, Schmitt, M, Mouray, E, McEwen, A.G, Torchy, M, Poussin-Courmontagne, P, Alavi, S, Tarnus, C, Cavarelli, J, Florent, I, Albrecht, S.
登録日2019-07-22
公開日2020-03-25
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (1.54 Å)
主引用文献Aminobenzosuberone derivatives as PfA-M1 inhibitors: Molecular recognition and antiplasmodial evaluation.
Bioorg.Chem., 98, 2020
6SBQ
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BU of 6sbq by Molmil
The crystal structure of PfA-M1 in complex with 7-amino-4-phenyl-5,7,8,9-tetrahydrobenzocyclohepten-6-one
分子名称: DI(HYDROXYETHYL)ETHER, M1-family alanyl aminopeptidase, MALONATE ION, ...
著者Salomon, E, Schmitt, M, Mouray, E, McEwen, A.G, Torchy, M, Poussin-Courmontagne, P, Alavi, S, Tarnus, C, Cavarelli, J, Florent, I, Albrecht, S.
登録日2019-07-22
公開日2020-03-25
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (1.33 Å)
主引用文献Aminobenzosuberone derivatives as PfA-M1 inhibitors: Molecular recognition and antiplasmodial evaluation.
Bioorg.Chem., 98, 2020
2XWH
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BU of 2xwh by Molmil
HCV-J6 NS5B polymerase structure at 1.8 Angstrom
分子名称: DI(HYDROXYETHYL)ETHER, POLYETHYLENE GLYCOL (N=34), RNA DEPENDENT RNA POLYMERASE
著者Scrima, N, Bressanelli, S.
登録日2010-11-03
公開日2011-01-12
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献A Comprehensive Structure-Function Comparison of Hepatitis C Virus Strains Jfh1 and J6 Polymerases Reveals a Key Residue Stimulating Replication in Cell Culture Across Genotypes.
J.Virol., 85, 2011
2XXD
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BU of 2xxd by Molmil
HCV-JFH1 NS5B polymerase structure at 1.9 angstrom
分子名称: PHOSPHATE ION, RNA-DIRECTED RNA POLYMERASE
著者Caillet-Saguy, C, Bressanelli, S.
登録日2010-11-10
公開日2011-01-12
最終更新日2024-05-01
実験手法X-RAY DIFFRACTION (1.881 Å)
主引用文献A Comprehensive Structure-Function Comparison of Hepatitis C Virus Strains Jfh1 and J6 Polymerases Reveals a Key Residue Stimulating Replication in Cell Culture Across Genotypes.
J.Virol., 85, 2011
2XYM
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BU of 2xym by Molmil
HCV-JFH1 NS5B T385A mutant
分子名称: PHOSPHATE ION, RNA-DIRECTED RNA POLYMERASE
著者Simister, P.C, Caillet-Saguy, C, Bressanelli, S.
登録日2010-11-18
公開日2011-01-12
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (1.774 Å)
主引用文献A Comprehensive Structure-Function Comparison of Hepatitis C Virus Strains Jfh1 and J6 Polymerases Reveals a Key Residue Stimulating Replication in Cell Culture Across Genotypes.
J.Virol., 85, 2011
6VC1
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BU of 6vc1 by Molmil
Octreotide oxalate
分子名称: OXALATE ION, Octreotide
著者Spiliopoulou, M, Karavassili, F, Triandafillidis, D, Valmas, A, Kosinas, C, Fili, S, Barlos, K, Barlos, K.K, Morin, M, Reinle-Schmitt, M, Gozzo, F, Margiolaki, I.
登録日2019-12-20
公開日2020-12-23
最終更新日2021-05-19
実験手法POWDER DIFFRACTION
主引用文献New perspectives in macromolecular powder diffraction using single-photon-counting strip detectors: high-resolution structure of the pharmaceutical peptide octreotide.
Acta Crystallogr.,Sect.A, 77, 2021
6NOV
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BU of 6nov by Molmil
A Fab derived from ixekizumab
分子名称: DODECAETHYLENE GLYCOL, Fab Heavy Chain, Fab Light Chain
著者Durbin, J.D, Clawson, D.K, Lu, F, Tian, Y, Lu, J, Schmitt, M, Atwell, S.
登録日2019-01-16
公開日2019-06-19
最終更新日2019-08-14
実験手法X-RAY DIFFRACTION (2.14 Å)
主引用文献Development of tibulizumab, a tetravalent bispecific antibody targeting BAFF and IL-17A for the treatment of autoimmune disease.
Mabs, 11, 2019

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件を2024-07-24に公開中

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