8P1P
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![BU of 8p1p by Molmil](/molmil-images/mine/8p1p) | USP28 in complex with AZ1 | 分子名称: | 2-[[5-bromanyl-2-[[4-fluoranyl-3-(trifluoromethyl)phenyl]methoxy]phenyl]methylamino]ethanol, CHLORIDE ION, DIMETHYL SULFOXIDE, ... | 著者 | Sauer, F, Karal-Nair, R, Kisker, C. | 登録日 | 2023-05-12 | 公開日 | 2024-05-22 | 実験手法 | X-RAY DIFFRACTION (2.76 Å) | 主引用文献 | USP28 in complex with AZ1 To Be Published
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6ZVA
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![BU of 6zva by Molmil](/molmil-images/mine/6zva) | |
8P14
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![BU of 8p14 by Molmil](/molmil-images/mine/8p14) | |
8P1Q
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![BU of 8p1q by Molmil](/molmil-images/mine/8p1q) | USP28 in complex with FT206 | 分子名称: | 3-azanyl-N-[(2S)-6-[(1S,5R)-3,8-diazabicyclo[3.2.1]octan-3-yl]-1,2,3,4-tetrahydronaphthalen-2-yl]-6-methyl-thieno[2,3-b]pyridine-2-carboxamide, DIMETHYL SULFOXIDE, Ubiquitin carboxyl-terminal hydrolase 28 | 著者 | Sauer, F, Karal Nair, R, Kisker, C. | 登録日 | 2023-05-12 | 公開日 | 2024-05-22 | 実験手法 | X-RAY DIFFRACTION (2.79 Å) | 主引用文献 | USP28 in complex with FT206 To Be Published
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8P19
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![BU of 8p19 by Molmil](/molmil-images/mine/8p19) | |
3KNB
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![BU of 3knb by Molmil](/molmil-images/mine/3knb) | |
3Q5O
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![BU of 3q5o by Molmil](/molmil-images/mine/3q5o) | |
3QP3
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![BU of 3qp3 by Molmil](/molmil-images/mine/3qp3) | |
3PUC
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![BU of 3puc by Molmil](/molmil-images/mine/3puc) | |
6TUN
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![BU of 6tun by Molmil](/molmil-images/mine/6tun) | Helicase domain complex | 分子名称: | CDK-activating kinase assembly factor MAT1, CHLORIDE ION, General transcription and DNA repair factor IIH helicase subunit XPD | 著者 | Sauer, F, Kisker, C. | 登録日 | 2020-01-07 | 公開日 | 2020-11-11 | 最終更新日 | 2024-05-15 | 実験手法 | X-RAY DIFFRACTION (2.07 Å) | 主引用文献 | In TFIIH the Arch domain of XPD is mechanistically essential for transcription and DNA repair. Nat Commun, 11, 2020
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4F14
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![BU of 4f14 by Molmil](/molmil-images/mine/4f14) | |
6H4I
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![BU of 6h4i by Molmil](/molmil-images/mine/6h4i) | Usp28 catalytic domain apo | 分子名称: | SULFATE ION, Ubiquitin carboxyl-terminal hydrolase 28 | 著者 | Klemm, T.A, Sauer, F, Kisker, C. | 登録日 | 2018-07-21 | 公開日 | 2019-03-27 | 最終更新日 | 2019-05-15 | 実験手法 | X-RAY DIFFRACTION (3.22 Å) | 主引用文献 | Differential Oligomerization of the Deubiquitinases USP25 and USP28 Regulates Their Activities. Mol.Cell, 74, 2019
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6H4H
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![BU of 6h4h by Molmil](/molmil-images/mine/6h4h) | Usp28 catalytic domain variant E593D in complex with UbPA | 分子名称: | Polyubiquitin-B, SULFATE ION, Ubiquitin carboxyl-terminal hydrolase 28, ... | 著者 | Klemm, T.A, Sauer, F, Kisker, C. | 登録日 | 2018-07-21 | 公開日 | 2019-03-27 | 最終更新日 | 2019-05-15 | 実験手法 | X-RAY DIFFRACTION (3.5 Å) | 主引用文献 | Differential Oligomerization of the Deubiquitinases USP25 and USP28 Regulates Their Activities. Mol.Cell, 74, 2019
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6H4K
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6H4L
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![BU of 6h4l by Molmil](/molmil-images/mine/6h4l) | Structure of Titin M4 trigonal form | 分子名称: | CHLORIDE ION, Titin, ZINC ION | 著者 | Sauer, F, Wilmanns, M. | 登録日 | 2018-07-21 | 公開日 | 2019-08-07 | 最終更新日 | 2020-02-19 | 実験手法 | X-RAY DIFFRACTION (1.6 Å) | 主引用文献 | Structural diversity in the atomic resolution 3D fingerprint of the titin M-band segment. Plos One, 14, 2019
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6H4J
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![BU of 6h4j by Molmil](/molmil-images/mine/6h4j) | Usp25 catalytic domain | 分子名称: | CHLORIDE ION, Ubiquitin carboxyl-terminal hydrolase 25 | 著者 | Klemm, T.A, Sauer, F, Kisker, C. | 登録日 | 2018-07-21 | 公開日 | 2019-03-27 | 最終更新日 | 2024-01-17 | 実験手法 | X-RAY DIFFRACTION (3.07 Å) | 主引用文献 | Differential Oligomerization of the Deubiquitinases USP25 and USP28 Regulates Their Activities. Mol.Cell, 74, 2019
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5B5Q
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![BU of 5b5q by Molmil](/molmil-images/mine/5b5q) | |
5LST
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![BU of 5lst by Molmil](/molmil-images/mine/5lst) | |
8REV
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![BU of 8rev by Molmil](/molmil-images/mine/8rev) | |
6FDU
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![BU of 6fdu by Molmil](/molmil-images/mine/6fdu) | Structure of Chlamydia trachomatis effector protein Cdu1 bound to Compound 3 | 分子名称: | (2~{S},3~{S})-2-[[(2~{S})-2-[3,5-bis(chloranyl)phenyl]-2-(dimethylamino)ethanoyl]amino]-~{N}-[[2-(iminomethyl)pyrimidin-4-yl]methyl]-3-methyl-pentanamide, CHLORIDE ION, Deubiquitinase and deneddylase Dub1 | 著者 | Ramirez, Y, Kisker, C, Altmann, E. | 登録日 | 2017-12-26 | 公開日 | 2018-08-15 | 最終更新日 | 2024-01-17 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Structural Basis of Substrate Recognition and Covalent Inhibition of Cdu1 from Chlamydia trachomatis. ChemMedChem, 13, 2018
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6FDQ
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6FDK
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6HCI
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![BU of 6hci by Molmil](/molmil-images/mine/6hci) | |