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5AEB
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BU of 5aeb by Molmil
Crystal structure of the class B3 di-zinc metallo-beta-lactamase LRA- 12 from an Alaskan soil metagenome.
分子名称: COBALT (II) ION, LRA-12, SULFATE ION, ...
著者Power, P, Herman, R, Kerff, F, Bouillenne, F, Rodriguez, M.M, Galleni, M, Handelsman, J, Gutkind, G, Charlier, P, Sauvage, E.
登録日2015-08-27
公開日2015-09-16
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Crystal structure and kinetic analysis of the class B3 di-zinc metallo-beta-lactamase LRA-12 from an Alaskan soil metagenome.
PLoS ONE, 12, 2017
8EHH
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BU of 8ehh by Molmil
Crystal structure of the class A extended-spectrum beta-lactamase CTX-M-96 in complex with relebactam at 1.03 Angstrom resolution
分子名称: (2S,5R)-1-formyl-N-(piperidin-4-yl)-5-[(sulfooxy)amino]piperidine-2-carboxamide, Beta-lactamase
著者Power, P, Ghiglione, B, Bonomo, R.A, Rodriguez, M.M, Gutkind, G, Klinke, S.
登録日2022-09-14
公開日2023-09-20
最終更新日2024-03-13
実験手法X-RAY DIFFRACTION (1.03 Å)
主引用文献Biochemical and structural evidences of the activity of relebactam as inhibitor of the extended-spectrum beta-lactamase CTX-M-96.
To be published
3ZNY
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BU of 3zny by Molmil
Crystal structure of the class A extended-spectrum beta-lactamase CTX- M-96, a natural D240G mutant derived from CTX-M-12
分子名称: CTX-M-12A ENZYME
著者Power, P, Herman, R, Bouillenne, F, Ghiglione, B, Rodriguez, M.M, Galleni, M, Gutkind, G, Charlier, P, Sauvage, E.
登録日2013-02-18
公開日2014-01-08
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (1.2 Å)
主引用文献Structural and Kinetic Insights Into the "Ceftazidimase" Behavior of the Extended-Spectrum Beta-Lactamase Ctx-M-96.
Biochemistry, 54, 2015
6BN3
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BU of 6bn3 by Molmil
CTX-M-151 class A extended-spectrum beta-lactamase apo crystal structure at 1.3 Angstrom resolution
分子名称: 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, Beta-lactamase
著者Power, P, Ghiglione, B, Rodriguez, M.M, Gutkind, G, Ishii, Y, Bonomo, R.A, Klinke, S.
登録日2017-11-16
公開日2018-11-21
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (1.278 Å)
主引用文献Structural and Biochemical Characterization of the Novel CTX-M-151 Extended-Spectrum beta-Lactamase and Its Inhibition by Avibactam.
Antimicrob.Agents Chemother., 65, 2021
6BPF
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BU of 6bpf by Molmil
CTX-M-151 class A extended-spectrum beta-lactamase crystal structure in complex with avibactam at 1.32 Angstrom resolution
分子名称: (2S,5R)-1-formyl-5-[(sulfooxy)amino]piperidine-2-carboxamide, Beta-lactamase
著者Power, P, Ghiglione, B, Rodriguez, M.M, Gutkind, G, Ishii, Y, Bonomo, R.A, Klinke, S.
登録日2017-11-23
公開日2018-11-28
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (1.318 Å)
主引用文献Structural and Biochemical Characterization of the Novel CTX-M-151 Extended-Spectrum beta-Lactamase and Its Inhibition by Avibactam.
Antimicrob.Agents Chemother., 65, 2021
3QM6
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BU of 3qm6 by Molmil
Blackfin tuna deoxy-myoglobin, atomic resolution
分子名称: 1,2-ETHANEDIOL, Myoglobin, PROTOPORPHYRIN IX CONTAINING FE
著者de Serrano, V.S, Schreiter, E.R, Rodriguez, M.M.
登録日2011-02-03
公開日2012-02-08
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (0.91 Å)
主引用文献High Resolution Structures of Blackfin Tuna Myoglobin
To be Published
3QM9
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BU of 3qm9 by Molmil
Blackfin tuna azido-myoglobin, atomic resolution
分子名称: 1,2-ETHANEDIOL, AZIDE ION, Myoglobin, ...
著者de Serrano, V.S, Rodriguez, M.M, Schreiter, E.R.
登録日2011-02-03
公開日2012-02-08
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (0.91 Å)
主引用文献High Resolution Structures of Blackfin Tuna Myoglobin
To be Published
3QM7
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BU of 3qm7 by Molmil
Blackfin tuna carbonmonoxy-myoglobin, atomic resolution
分子名称: 1,2-ETHANEDIOL, CARBON MONOXIDE, Myoglobin, ...
著者de Serrano, V.S, Rodriguez, M.M, Schreiter, E.R.
登録日2011-02-03
公開日2012-02-08
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (0.96 Å)
主引用文献High Resolution Structures of Blackfin Tuna Myoglobin
To be Published
3QM5
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BU of 3qm5 by Molmil
Blackfin tuna oxy-myoglobin, atomic resolution
分子名称: 1,2-ETHANEDIOL, Myoglobin, OXYGEN MOLECULE, ...
著者de Serrano, V.S, Rodriguez, M.M, Schreiter, E.R.
登録日2011-02-03
公開日2012-02-08
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (0.91 Å)
主引用文献High Resolution Structures of Blackfin Tuna Myoglobin
To be Published
3QMA
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BU of 3qma by Molmil
Blackfin tuna myoglobin imidazole complex, atomic resolution
分子名称: 1,2-ETHANEDIOL, IMIDAZOLE, Myoglobin, ...
著者de Serrano, V.S, Rodriguez, M.M, Schreiter, E.R.
登録日2011-02-03
公開日2012-02-08
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (0.94 Å)
主引用文献High Resolution Structures of Blackfin Tuna Myoglobin
To be Published
3QM8
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BU of 3qm8 by Molmil
Blackfin tuna cyanomet-myoglobin, atomic resolution
分子名称: 1,2-ETHANEDIOL, CYANIDE ION, Myoglobin, ...
著者de Serrano, V.S, Rodriguez, M.M, Schreiter, E.R.
登録日2011-02-03
公開日2012-02-08
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (0.91 Å)
主引用文献High Resolution Structures of Blackfin Tuna Myoglobin
To be Published
2NX0
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BU of 2nx0 by Molmil
Ferrous nitrosyl blackfin tuna myoglobin
分子名称: Myoglobin, NITRIC OXIDE, PROTOPORPHYRIN IX CONTAINING FE, ...
著者Schreiter, E.R, Rodriguez, M.M, Weichsel, A, Montfort, W.R, Bonaventura, J.
登録日2006-11-16
公開日2007-05-08
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (0.95 Å)
主引用文献S-nitrosylation-induced conformational change in blackfin tuna myoglobin.
J.Biol.Chem., 282, 2007
7UTB
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BU of 7utb by Molmil
KPC-2 CARBAPENEMASE IN COMPLEX WITH THE BORONIC ACID INHIBITOR MB_076
分子名称: Carbapenem-hydrolyzing beta-lactamase KPC, [(1~{R})-1-[2-[(5-azanyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethanoylamino]-2-(4-carboxy-1,2,3-triazol-1-yl)ethyl]-$l^{3}-oxidanyl-bis(oxidanyl)boron
著者van den Akker, F, Alsenani, T.A.
登録日2022-04-26
公開日2022-12-14
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (1.38 Å)
主引用文献Boronic Acid Transition State Inhibitors as Potent Inactivators of KPC and CTX-M beta-Lactamases: Biochemical and Structural Analyses.
Antimicrob.Agents Chemother., 67, 2023
2NRM
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BU of 2nrm by Molmil
S-nitrosylated blackfin tuna myoglobin
分子名称: GLYCEROL, Myoglobin, PROTOPORPHYRIN IX CONTAINING FE
著者Schreiter, E.R, Rodr guez, M.M, Weichsel, A, Montfort, W.R, Bonaventura, J.
登録日2006-11-02
公開日2007-05-08
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (1.09 Å)
主引用文献S-nitrosylation-induced conformational change in blackfin tuna myoglobin.
J.Biol.Chem., 282, 2007
2NRL
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BU of 2nrl by Molmil
Blackfin tuna myoglobin
分子名称: 1,2-ETHANEDIOL, Myoglobin, PROTOPORPHYRIN IX CONTAINING FE
著者Schreiter, E.R, Rodr guez, M.M, Weichsel, A, Montfort, W.R, Bonaventura, J.
登録日2006-11-02
公開日2007-05-08
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (0.91 Å)
主引用文献S-nitrosylation-induced conformational change in blackfin tuna myoglobin.
J.Biol.Chem., 282, 2007
6ZQK
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BU of 6zqk by Molmil
HER2-binding scFv-Fab fusion 841
分子名称: 1,2-ETHANEDIOL, 841 heavy chain, 841 light chain
著者Kast, F, Schwill, M, Stueber, J.C, Pfundstein, S, Nagy-Davidescu, G, Monne Rodriguez, J.M, Seehusen, F, Richter, C.P, Honegger, A, Hartmann, K.P, Weber, T.G, Kroener, F, Ernst, P, Piehler, J, Plueckthun, A.
登録日2020-07-09
公開日2021-06-30
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Engineering an anti-HER2 biparatopic antibody with a multimodal mechanism of action.
Nat Commun, 12, 2021

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件を2024-08-21に公開中

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