2AKP
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![BU of 2akp by Molmil](/molmil-images/mine/2akp) | Hsp90 Delta24-N210 mutant | 分子名称: | ATP-dependent molecular chaperone HSP82 | 著者 | Richter, K, Moser, S, Hagn, F, Friedrich, R, Hainzl, O, Heller, M, Schlee, S, Kessler, H, Reinstein, J, Buchner, J. | 登録日 | 2005-08-03 | 公開日 | 2006-01-31 | 最終更新日 | 2023-08-23 | 実験手法 | X-RAY DIFFRACTION (1.94 Å) | 主引用文献 | Intrinsic inhibition of the Hsp90 ATPase activity. J.Biol.Chem., 281, 2006
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4JA9
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![BU of 4ja9 by Molmil](/molmil-images/mine/4ja9) | Rat PP5 apo | 分子名称: | MAGNESIUM ION, Serine/threonine-protein phosphatase 5 | 著者 | Haslbeck, V, Helmuth, M, Alte, F, Popowicz, G, Schmidt, W, Weiwad, M, Fischer, G, Gemmecker, G, Sattler, M, Striggow, F, Groll, M, Richter, K. | 登録日 | 2013-02-18 | 公開日 | 2014-02-19 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Selective activators of protein phosphatase 5 target the auto-inhibitory mechanism. Biosci.Rep., 35, 2015
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4JA7
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![BU of 4ja7 by Molmil](/molmil-images/mine/4ja7) | Rat PP5 co-crystallized with P5SA-2 | 分子名称: | MAGNESIUM ION, Serine/threonine-protein phosphatase 5 | 著者 | Haslbeck, V, Helmuth, M, Alte, F, Popowicz, G, Schmidt, W, Weiwad, M, Fischer, G, Gemmecker, G, Sattler, M, Striggow, F, Groll, M, Richter, K. | 登録日 | 2013-02-18 | 公開日 | 2014-02-19 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Selective activators of protein phosphatase 5 target the auto-inhibitory mechanism. Biosci.Rep., 35, 2015
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3WHW
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![BU of 3whw by Molmil](/molmil-images/mine/3whw) | MTH1 in complex with Ruthenium-based inhibitor | 分子名称: | 7,8-dihydro-8-oxoguanine triphosphatase, SULFATE ION, [4-amino-2-methyl-6-(pyridin-2-yl-kappaN)quinazolin-7-yl-kappaC~7~](carbonyl){1-[(2,6-dimethoxyphenoxy)carbonyl]cyclopenta-2,4-dien-1-yl}ruthenium | 著者 | Streib, M, Kraeling, K, Richter, K, Steuber, H, Meggers, E. | 登録日 | 2013-09-03 | 公開日 | 2014-02-12 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (2.701 Å) | 主引用文献 | An Organometallic Inhibitor for the Human Repair Enzyme 7,8-Dihydro-8-oxoguanosine Triphosphatase. Angew.Chem.Int.Ed.Engl., 53, 2014
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2LLV
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![BU of 2llv by Molmil](/molmil-images/mine/2llv) | Solution structure of the yeast Sti1 DP1 domain | 分子名称: | Heat shock protein STI1 | 著者 | Schmid, A.B, Lagleder, S, Graewert, M.A, Roehl, A, Hagn, F, Wandinger, S.K, Cox, M.B, Demmer, O, Richter, K, Groll, M, Kessler, H, Buchner, J. | 登録日 | 2011-11-17 | 公開日 | 2012-01-25 | 最終更新日 | 2024-05-01 | 実験手法 | SOLUTION NMR | 主引用文献 | The architecture of functional modules in the Hsp90 co-chaperone Sti1/Hop. Embo J., 31, 2012
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2LLW
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![BU of 2llw by Molmil](/molmil-images/mine/2llw) | Solution structure of the yeast Sti1 DP2 domain | 分子名称: | Heat shock protein STI1 | 著者 | Schmid, A.B, Lagleder, S, Graewert, M.A, Roehl, A, Hagn, F, Wandinger, S.K, Cox, M.B, Demmer, O, Richter, K, Groll, M, Kessler, H, Buchner, J. | 登録日 | 2011-11-17 | 公開日 | 2012-01-25 | 最終更新日 | 2024-05-01 | 実験手法 | SOLUTION NMR | 主引用文献 | The architecture of functional modules in the Hsp90 co-chaperone Sti1/Hop. Embo J., 31, 2012
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3UQ3
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![BU of 3uq3 by Molmil](/molmil-images/mine/3uq3) | TPR2AB-domain:pHSP90-complex of yeast Sti1 | 分子名称: | Heat shock protein, Heat shock protein STI1 | 著者 | Schmid, A.B, Lagleder, S, Graewert, M.A, Roehl, A, Hagn, F, Wandinger, S.K, Cox, M.B, Demmer, O, Richter, K, Groll, M, Kessler, H, Buchner, J. | 登録日 | 2011-11-19 | 公開日 | 2012-01-18 | 最終更新日 | 2023-09-13 | 実験手法 | X-RAY DIFFRACTION (2.6 Å) | 主引用文献 | The architecture of functional modules in the Hsp90 co-chaperone Sti1/Hop. Embo J., 31, 2012
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3UPV
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![BU of 3upv by Molmil](/molmil-images/mine/3upv) | TPR2B-domain:pHsp70-complex of yeast Sti1 | 分子名称: | Heat shock protein SSA4, Heat shock protein STI1 | 著者 | Schmid, A.B, Lagleder, S, Graewert, M.A, Roehl, A, Hagn, F, Wandinger, S.K, Cox, M.B, Demmer, O, Richter, K, Groll, M, Kessler, H. | 登録日 | 2011-11-18 | 公開日 | 2012-01-25 | 最終更新日 | 2023-09-13 | 実験手法 | X-RAY DIFFRACTION (1.6 Å) | 主引用文献 | The architecture of functional modules in the Hsp90 co-chaperone Sti1/Hop. Embo J., 31, 2012
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5QU6
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![BU of 5qu6 by Molmil](/molmil-images/mine/5qu6) | |
5QU8
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![BU of 5qu8 by Molmil](/molmil-images/mine/5qu8) | |
5QU3
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![BU of 5qu3 by Molmil](/molmil-images/mine/5qu3) | |
5QUA
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![BU of 5qua by Molmil](/molmil-images/mine/5qua) | |
5QU1
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![BU of 5qu1 by Molmil](/molmil-images/mine/5qu1) | Crystal Structure of the monomeric human Nck SH3.1 domain, triclinic, 1.08A | 分子名称: | Cytoplasmic protein NCK1, SULFATE ION | 著者 | Burger, D, Ruf, A, Benz, J, Schlatter, D, Rudolph, M.G. | 登録日 | 2019-12-13 | 公開日 | 2020-02-12 | 最終更新日 | 2024-04-03 | 実験手法 | X-RAY DIFFRACTION (1.08 Å) | 主引用文献 | Small molecule AX-024 reduces T cell proliferation independently of CD3ε/Nck1 interaction, which is governed by a domain swap in the Nck1-SH3.1 domain. J.Biol.Chem., 295, 2020
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5QU5
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![BU of 5qu5 by Molmil](/molmil-images/mine/5qu5) | Domain Swap in the first SH3 domain of human Nck1 | 分子名称: | Cytoplasmic protein NCK1 | 著者 | Burger, D, Ruf, A, Benz, J, Schlatter, D, Rudolph, M.G. | 登録日 | 2019-12-13 | 公開日 | 2020-02-12 | 最終更新日 | 2024-04-03 | 実験手法 | X-RAY DIFFRACTION (1.11 Å) | 主引用文献 | Small molecule AX-024 reduces T cell proliferation independently of CD3ε/Nck1 interaction, which is governed by a domain swap in the Nck1-SH3.1 domain. J.Biol.Chem., 295, 2020
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5QU2
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![BU of 5qu2 by Molmil](/molmil-images/mine/5qu2) | Crystal Structure of human Nck SH3.1 in complex with peptide PPPVPNPDY | 分子名称: | ACE-PRO-PRO-PRO-VAL-PRO-ASN-PRO-ASP-TYR-NH2, Cytoplasmic protein NCK1, SULFATE ION | 著者 | Rudolph, M.G. | 登録日 | 2019-12-13 | 公開日 | 2020-02-12 | 最終更新日 | 2024-04-03 | 実験手法 | X-RAY DIFFRACTION (1.04 Å) | 主引用文献 | Small molecule AX-024 reduces T cell proliferation independently of CD3ε/Nck1 interaction, which is governed by a domain swap in the Nck1-SH3.1 domain. J.Biol.Chem., 295, 2020
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5QU7
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![BU of 5qu7 by Molmil](/molmil-images/mine/5qu7) | |
5QU4
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![BU of 5qu4 by Molmil](/molmil-images/mine/5qu4) | |
3C7X
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![BU of 3c7x by Molmil](/molmil-images/mine/3c7x) | Hemopexin-like domain of matrix metalloproteinase 14 | 分子名称: | CHLORIDE ION, Matrix metalloproteinase-14, SODIUM ION | 著者 | Tochowicz, A, Itoh, Y, Maskos, K, Bode, W, Goettig, P. | 登録日 | 2008-02-08 | 公開日 | 2009-02-10 | 最終更新日 | 2023-11-01 | 実験手法 | X-RAY DIFFRACTION (1.7 Å) | 主引用文献 | The dimer interface of the membrane type 1 matrix metalloproteinase hemopexin domain: crystal structure and biological functions J.Biol.Chem., 286, 2011
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4UQF
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![BU of 4uqf by Molmil](/molmil-images/mine/4uqf) | CRYSTAL STRUCTURE OF LISTERIA MONOCYTOGENES GTP CYCLOHYDROLASE I | 分子名称: | GTP cyclohydrolase 1 | 著者 | Schuessler, S, Perbandt, M, Fischer, M, Graewert, T. | 登録日 | 2014-06-23 | 公開日 | 2015-07-01 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (2.4 Å) | 主引用文献 | Structure of GTP cyclohydrolase I from Listeria monocytogenes, a potential anti-infective drug target. Acta Crystallogr.,Sect.F, 75, 2019
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6EK4
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![BU of 6ek4 by Molmil](/molmil-images/mine/6ek4) | |
6EL1
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![BU of 6el1 by Molmil](/molmil-images/mine/6el1) | YaxAB pore complex | 分子名称: | YaxA, YaxB | 著者 | Braeuning, B, Bertosin, E, Dietz, H, Groll, M. | 登録日 | 2017-09-27 | 公開日 | 2018-05-16 | 最終更新日 | 2024-05-15 | 実験手法 | ELECTRON MICROSCOPY (6.1 Å) | 主引用文献 | Structure and mechanism of the two-component alpha-helical pore-forming toxin YaxAB. Nat Commun, 9, 2018
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6EK7
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![BU of 6ek7 by Molmil](/molmil-images/mine/6ek7) | YaxA from Yersinia enterocolitica | 分子名称: | (4S)-2-METHYL-2,4-PENTANEDIOL, YaxA | 著者 | Braeuning, B, Groll, M. | 登録日 | 2017-09-25 | 公開日 | 2018-05-16 | 最終更新日 | 2024-05-01 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | Structure and mechanism of the two-component alpha-helical pore-forming toxin YaxAB. Nat Commun, 9, 2018
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5DL1
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![BU of 5dl1 by Molmil](/molmil-images/mine/5dl1) | ClpP from Staphylococcus aureus in complex with AV145 | 分子名称: | 1-(propan-2-yl)-N-{[2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}-1H-pyrazolo[3,4-b]pyridine-5-carboxamide, ATP-dependent Clp protease proteolytic subunit | 著者 | Vielberg, M.-T, Groll, M. | 登録日 | 2015-09-04 | 公開日 | 2015-11-25 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (3 Å) | 主引用文献 | Reversible Inhibitors Arrest ClpP in a Defined Conformational State that Can Be Revoked by ClpX Association. Angew.Chem.Int.Ed.Engl., 54, 2015
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5LIR
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![BU of 5lir by Molmil](/molmil-images/mine/5lir) | |
1NU7
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![BU of 1nu7 by Molmil](/molmil-images/mine/1nu7) | Staphylocoagulase-Thrombin Complex | 分子名称: | IMIDAZOLE, MERCURY (II) ION, N-(sulfanylacetyl)-D-phenylalanyl-N-[(2S,3S)-6-{[amino(iminio)methyl]amino}-1-chloro-2-hydroxyhexan-3-yl]-L-prolinamide, ... | 著者 | Friedrich, R, Bode, W, Fuentes-Prior, P, Panizzi, P, Bock, P.E. | 登録日 | 2003-01-31 | 公開日 | 2003-10-07 | 最終更新日 | 2012-12-12 | 実験手法 | X-RAY DIFFRACTION (2.2 Å) | 主引用文献 | Staphylocoagulase is a prototype for the mechanism of cofactor-induced zymogen activation NATURE, 425, 2003
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