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4EUU
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BU of 4euu by Molmil
Structure of BX-795 Complexed with Human TBK1 Kinase Domain Phosphorylated on Ser172
分子名称: GLYCEROL, IODIDE ION, N-(3-{[5-iodo-4-({3-[(thiophen-2-ylcarbonyl)amino]propyl}amino)pyrimidin-2-yl]amino}phenyl)pyrrolidine-1-carboxamide, ...
著者Ma, X, Helgason, E, Phung, Q.T, Quan, C.L, Iyer, R.S, Lee, M.W, Bowman, K.K, Starovasnik, M.A, Dueber, E.C.
登録日2012-04-25
公開日2012-05-23
最終更新日2017-11-15
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Molecular basis of Tank-binding kinase 1 activation by transautophosphorylation.
Proc.Natl.Acad.Sci.USA, 109, 2012
4EUT
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BU of 4eut by Molmil
Structure of BX-795 Complexed with Unphosphorylated Human TBK1 Kinase-ULD Domain
分子名称: IODIDE ION, N-(3-{[5-iodo-4-({3-[(thiophen-2-ylcarbonyl)amino]propyl}amino)pyrimidin-2-yl]amino}phenyl)pyrrolidine-1-carboxamide, SULFATE ION, ...
著者Ma, X, Helgason, E, Phung, Q.T, Quan, C.L, Iyer, R.S, Lee, M.W, Bowman, K.K, Starovasnik, M.A, Dueber, E.C.
登録日2012-04-25
公開日2012-05-23
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献Molecular basis of Tank-binding kinase 1 activation by transautophosphorylation.
Proc.Natl.Acad.Sci.USA, 109, 2012
7JWQ
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BU of 7jwq by Molmil
Fab CJ11 in complex IL-1beta peptide liberated by Caspase cleavage
分子名称: Fab CJ11 Heavy chain, Fab CJ11 Light chain, IL-1beta peptide
著者Payandeh, J, Ho, H.
登録日2020-08-26
公開日2021-03-24
最終更新日2023-10-18
実験手法X-RAY DIFFRACTION (2.001 Å)
主引用文献Discovery of a caspase cleavage motif antibody reveals insights into noncanonical inflammasome function.
Proc.Natl.Acad.Sci.USA, 118, 2021
7JWP
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BU of 7jwp by Molmil
Fab CJ11 in complex IL-18 peptide liberated by Caspase cleavage
分子名称: Fab CJ11 Heavy chain, Fab CJ11 Light chain, IL-18 peptide
著者Payandeh, J, Ho, H.
登録日2020-08-26
公開日2021-03-24
最終更新日2023-10-18
実験手法X-RAY DIFFRACTION (3 Å)
主引用文献Discovery of a caspase cleavage motif antibody reveals insights into noncanonical inflammasome function.
Proc.Natl.Acad.Sci.USA, 118, 2021

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件を2024-07-24に公開中

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