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4A6W
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BU of 4a6w by Molmil
X-ray structures of oxazole hydroxamate EcMetAp-Mn complexes
分子名称: 5-(2-chlorophenyl)-N-hydroxy-1,3-oxazole-2-carboxamide, MANGANESE (II) ION, METHIONINE AMINOPEPTIDASE
著者Huguet, F, Melet, A, AlvesdeSousa, R, Lieutaud, A, Chevalier, J, Deschamps, P, Tomas, A, Leulliot, N, Pages, J.M, Artaud, I.
登録日2011-11-09
公開日2012-06-13
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (1.46 Å)
主引用文献Hydroxamic Acids as Potent Inhibitors of Fe(II) and Mn(II) E. Coli Methionine Aminopeptidase: Biological Activities and X-Ray Structures of Oxazole Hydroxamate-Ecmetap-Mn Complexes.
Chemmedchem, 7, 2012
4A6V
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BU of 4a6v by Molmil
X-ray structures of oxazole hydroxamate EcMetAp-Mn complexes
分子名称: CARBONATE ION, MANGANESE (II) ION, METHIONINE AMINOPEPTIDASE, ...
著者Huguet, F, Melet, A, AlvesdeSousa, R, Lieutaud, A, Chevalier, J, Deschamps, P, Tomas, A, Leulliot, N, Pages, J.M, Artaud, I.
登録日2011-11-09
公開日2012-06-13
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (1.46 Å)
主引用文献Hydroxamic Acids as Potent Inhibitors of Fe(II) and Mn(II) E. Coli Methionine Aminopeptidase: Biological Activities and X-Ray Structures of Oxazole Hydroxamate-Ecmetap-Mn Complexes.
Chemmedchem, 7, 2012
1A87
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BU of 1a87 by Molmil
COLICIN N
分子名称: COLICIN N
著者Vetter, I.R, Parker, M.W, Tucker, A.D, Lakey, J.H, Pattus, F, Tsernoglou, D.
登録日1998-04-03
公開日1999-04-06
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (3.1 Å)
主引用文献Crystal structure of a colicin N fragment suggests a model for toxicity.
Structure, 6, 1998
5LDT
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BU of 5ldt by Molmil
Crystal Structures of MOMP from Campylobacter jejuni
分子名称: (HYDROXYETHYLOXY)TRI(ETHYLOXY)OCTANE, CALCIUM ION, MOMP porin
著者Ferrara, L.G.M, Wallat, G.D, Moynie, L, Naismith, J.H.
登録日2016-06-27
公開日2016-10-26
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (2.88 Å)
主引用文献MOMP from Campylobacter jejuni Is a Trimer of 18-Stranded beta-Barrel Monomers with a Ca(2+) Ion Bound at the Constriction Zone.
J.Mol.Biol., 428, 2016
5LDV
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BU of 5ldv by Molmil
Crystal Structures of MOMP from Campylobacter jejuni
分子名称: CALCIUM ION, MOMP porin, N-OCTANE, ...
著者Wallat, G.D, Ferrara, L.M.G, Moynie, L, Naismith, J.H.
登録日2016-06-28
公開日2016-10-26
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献MOMP from Campylobacter jejuni Is a Trimer of 18-Stranded beta-Barrel Monomers with a Ca(2+) Ion Bound at the Constriction Zone.
J.Mol.Biol., 428, 2016
5N9I
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BU of 5n9i by Molmil
STRUCTURE OF 206-GVVTSE-211, THE STERIC ZIPPER THAT SUPPORTS THE SELF-ASSOCIATION OF P. STUARTII OMP-PST1 INTO DIMERS OF TRIMERS
分子名称: Porin 1
著者Colletier, J.P, Nasrallah, C.
登録日2017-02-24
公開日2018-02-21
最終更新日2024-05-01
実験手法X-RAY DIFFRACTION (1.91 Å)
主引用文献Porin self-association enables cell-to-cell contact in
Proc. Natl. Acad. Sci. U.S.A., 115, 2018
5N9H
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BU of 5n9h by Molmil
STRUCTURE OF 283-LGNY-286, THE STERIC ZIPPER THAT SUPPORTS THE SELF-ASSOCIATION OF P. STUARTII OMP-PST2 INTO DIMERS OF TRIMERS
分子名称: Porin, SULFATE ION
著者Nasrallah, C, Colletier, J.P.
登録日2017-02-24
公開日2018-02-21
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (0.997 Å)
主引用文献Porin self-association enables cell-to-cell contact in
Proc. Natl. Acad. Sci. U.S.A., 115, 2018
4D65
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BU of 4d65 by Molmil
Structure of porin Omp-Pst2 from P. stuartii; the asymmetric unit contains a dimer of trimers.
分子名称: 3-HYDROXY-TETRADECANOIC ACID, LAURYL DIMETHYLAMINE-N-OXIDE, MYRISTIC ACID, ...
著者Nasrallah, C, Colletier, J.P.
登録日2014-11-08
公開日2016-03-09
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Porin self-association enables cell-to-cell contact inProvidencia stuartiifloating communities.
Proc. Natl. Acad. Sci. U.S.A., 115, 2018
4D64
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BU of 4d64 by Molmil
Structure of porin Omp-Pst1 from P. stuartii; the crystallographic symmetry generates a dimer of trimers.
分子名称: CALCIUM ION, PORIN 1
著者Nasrallah, C, Colletier, J.P.
登録日2014-11-08
公開日2016-03-09
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (3.2 Å)
主引用文献Porin self-association enables cell-to-cell contact inProvidencia stuartiifloating communities.
Proc. Natl. Acad. Sci. U.S.A., 115, 2018
6ENE
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BU of 6ene by Molmil
OmpF orthologue from Enterobacter cloacae (OmpE35)
分子名称: (HYDROXYETHYLOXY)TRI(ETHYLOXY)OCTANE, Outer membrane protein (Porin), SULFATE ION, ...
著者van den Berg, B, Abellon-Ruiz, J, Basle, A.
登録日2017-10-04
公開日2018-10-31
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Getting Drugs into Gram-Negative Bacteria: Rational Rules for Permeation through General Porins.
Acs Infect Dis., 4, 2018
5NXU
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BU of 5nxu by Molmil
Complex structure with maltose of Providencia stuartii Omp-Pst1 porin
分子名称: CALCIUM ION, LAURYL DIMETHYLAMINE-N-OXIDE, Porin 1, ...
著者Colletier, J.P, Nasrallah, C.
登録日2017-05-10
公開日2018-02-21
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (3 Å)
主引用文献Porin self-association enables cell-to-cell contact in
Proc. Natl. Acad. Sci. U.S.A., 115, 2018
5NXN
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BU of 5nxn by Molmil
Structure of a L5-deletion mutant of Providencia stuartii Omp-Pst1
分子名称: CALCIUM ION, Porin 1
著者El Khatib, M, Colletier, J.P.
登録日2017-05-10
公開日2018-02-21
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (3.12 Å)
主引用文献Porin self-association enables cell-to-cell contact in
Proc. Natl. Acad. Sci. U.S.A., 115, 2018
5NXR
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BU of 5nxr by Molmil
Trimeric structure of Omp-Pst1, the major porin from Providencia stuartii
分子名称: CALCIUM ION, CHLORIDE ION, LAURYL DIMETHYLAMINE-N-OXIDE, ...
著者Colletier, J.P, Nasrallah, C.
登録日2017-05-10
公開日2018-02-21
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (2.7 Å)
主引用文献Porin self-association enables cell-to-cell contact in
Proc. Natl. Acad. Sci. U.S.A., 115, 2018
5JF2
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BU of 5jf2 by Molmil
Crystal structure of type 2 PDF from Streptococcus agalactiae in complex with inhibitor AT002
分子名称: (3R)-3-{3-[(4-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}-N-hydroxyheptanamide, ACETATE ION, IMIDAZOLE, ...
著者Fieulaine, S, Giglione, C, Meinnel, T, Hamiche, K.
登録日2016-04-19
公開日2016-11-30
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献A unique peptide deformylase platform to rationally design and challenge novel active compounds.
Sci Rep, 6, 2016
5JF1
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BU of 5jf1 by Molmil
Crystal structure of type 2 PDF from Streptococcus agalactiae in complex with actinonin
分子名称: ACETATE ION, ACTINONIN, Peptide deformylase, ...
著者Fieulaine, S, Giglione, C, Meinnel, T.
登録日2016-04-19
公開日2016-11-30
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献A unique peptide deformylase platform to rationally design and challenge novel active compounds.
Sci Rep, 6, 2016
5JF5
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BU of 5jf5 by Molmil
Crystal structure of type 2 PDF from Streptococcus agalactiae in complex with inhibitor AT020
分子名称: (3R)-3-{3-[(2H-1,3-benzodioxol-5-yl)methyl]-1,2,4-oxadiazol-5-yl}-4-cyclopentyl-N-hydroxybutanamide, ACETATE ION, IMIDAZOLE, ...
著者Fieulaine, S, Giglione, C, Meinnel, T.
登録日2016-04-19
公開日2016-11-30
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献A unique peptide deformylase platform to rationally design and challenge novel active compounds.
Sci Rep, 6, 2016
5JEZ
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BU of 5jez by Molmil
Crystal structure of type 2 PDF from Streptococcus agalactiae in complex with tripeptide Met-Ala-Ser
分子名称: ACETATE ION, Met-Ala-Ser, Peptide deformylase, ...
著者Fieulaine, S, Giglione, C, Meinnel, T.
登録日2016-04-19
公開日2016-11-30
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献A unique peptide deformylase platform to rationally design and challenge novel active compounds.
Sci Rep, 6, 2016
5JF7
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BU of 5jf7 by Molmil
Crystal structure of type 2 PDF from Streptococcus agalactiae in complex with inhibitor SMP289
分子名称: 2-(3-benzyl-5-bromo-1H-indol-1-yl)-N-hydroxyacetamide, ACETATE ION, IMIDAZOLE, ...
著者Fieulaine, S, Giglione, C, Meinnel, T, Hamiche, K.
登録日2016-04-19
公開日2016-11-30
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献A unique peptide deformylase platform to rationally design and challenge novel active compounds.
Sci Rep, 6, 2016
5JF0
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BU of 5jf0 by Molmil
Crystal structure of type 2 PDF from Streptococcus agalactiae in complex with tripeptide Met-Ala-Arg
分子名称: ACETATE ION, MET-ALA-ARG, NICKEL (II) ION, ...
著者Fieulaine, S, Giglione, C, Meinnel, T.
登録日2016-04-19
公開日2016-11-30
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (1.6 Å)
主引用文献A unique peptide deformylase platform to rationally design and challenge novel active compounds.
Sci Rep, 6, 2016
5JEX
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BU of 5jex by Molmil
Crystal structure of type 2 PDF from Streptococcus agalactiae, crystallized in imidazole buffer
分子名称: IMIDAZOLE, Peptide deformylase, ZINC ION
著者Fieulaine, S, Giglione, C, Meinnel, T.
登録日2016-04-19
公開日2016-11-30
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献A unique peptide deformylase platform to rationally design and challenge novel active compounds.
Sci Rep, 6, 2016
5JF3
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BU of 5jf3 by Molmil
Crystal structure of type 2 PDF from Streptococcus agalactiae in complex with inhibitor AT018
分子名称: ACETATE ION, IMIDAZOLE, Peptide deformylase, ...
著者Fieulaine, S, Giglione, C, Meinnel, T.
登録日2016-04-19
公開日2016-11-30
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (1.6 Å)
主引用文献A unique peptide deformylase platform to rationally design and challenge novel active compounds.
Sci Rep, 6, 2016
5JEY
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BU of 5jey by Molmil
Crystal structure of type 2 PDF from Streptococcus agalactiae, crystallized in cacodylate buffer
分子名称: NICKEL (II) ION, Peptide deformylase
著者Fieulaine, S, Giglione, C, Meinnel, T.
登録日2016-04-19
公開日2016-11-30
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献A unique peptide deformylase platform to rationally design and challenge novel active compounds.
Sci Rep, 6, 2016
5JF6
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BU of 5jf6 by Molmil
Crystal structure of type 2 PDF from Streptococcus agalactiae in complex with inhibitor 6b (AB47)
分子名称: 2-(5-bromo-1H-indol-3-yl)-N-hydroxyacetamide, ACETATE ION, Peptide deformylase, ...
著者Fieulaine, S, Giglione, C, Meinnel, T, Hamiche, K.
登録日2016-04-19
公開日2016-11-30
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献A unique peptide deformylase platform to rationally design and challenge novel active compounds.
Sci Rep, 6, 2016
5JF8
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BU of 5jf8 by Molmil
Crystal structure of type 2 PDF from Streptococcus agalactiae in complex with inhibitor RAS358 (21)
分子名称: ACETATE ION, IMIDAZOLE, Peptide deformylase, ...
著者Fieulaine, S, Giglione, C, Meinnel, T.
登録日2016-04-19
公開日2016-11-30
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献A unique peptide deformylase platform to rationally design and challenge novel active compounds.
Sci Rep, 6, 2016
5JF4
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BU of 5jf4 by Molmil
Crystal structure of type 2 PDF from Streptococcus agalactiae in complex with inhibitor AT019
分子名称: (3R)-3-{3-[(1-benzofuran-3-yl)methyl]-1,2,4-oxadiazol-5-yl}-4-cyclopentyl-N-hydroxybutanamide, ACETATE ION, IMIDAZOLE, ...
著者Fieulaine, S, Giglione, C, Meinnel, T.
登録日2016-04-19
公開日2016-11-30
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献A unique peptide deformylase platform to rationally design and challenge novel active compounds.
Sci Rep, 6, 2016

 

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