Search by PDB author

A modular route to novel potent and selective inhibitors of rhomboid intramembrane proteases
分子名称:	CHLORIDE ION, Rhomboid protease GlpG, inhibitor, ...
著者	Ticha, A, Stanchev, S, Vinothkumar, K.R, Mikles, D.C, Pachl, P, Svehlova, K, Nguyen, M.T.N, Verhelst, S.H.L, Johnson, D, Bachovchin, D, Lepsik, M, Majer, P, Strisovsky, K.
登録日	2017-01-09
公開日	2017-11-15
最終更新日	2024-01-17
実験手法	X-RAY DIFFRACTION (1.79 Å)
主引用文献	General and Modular Strategy for Designing Potent, Selective, and Pharmacologically Compliant Inhibitors of Rhomboid Proteases. Cell Chem Biol, 24, 2017

Structure of E.coli GlpG in complex with peptide derived inhibitor Ac-VRHA-cmk
分子名称:	ACE-VAL-ARG-HIS-ALA-0QE, Rhomboid protease GlpG
著者	Vinothkumar, K.R.
登録日	2017-01-06
公開日	2017-11-15
最終更新日	2024-11-06
実験手法	X-RAY DIFFRACTION (2.05 Å)
主引用文献	General and Modular Strategy for Designing Potent, Selective, and Pharmacologically Compliant Inhibitors of Rhomboid Proteases. Cell Chem Biol, 24, 2017

Structure of E.coli GlpG in complex with peptide derived inhibitor Ac-RVRHA-phenylethyl-ketoamide
分子名称:	ACE-ARG-VAL-ARG-HIS-ALA-V9C, Rhomboid protease GlpG, nonyl beta-D-glucopyranoside
著者	Vinothkumar, K.R.
登録日	2017-01-06
公開日	2017-11-15
最終更新日	2024-01-17
実験手法	X-RAY DIFFRACTION (2.16 Å)
主引用文献	General and Modular Strategy for Designing Potent, Selective, and Pharmacologically Compliant Inhibitors of Rhomboid Proteases. Cell Chem Biol, 24, 2017

Structure of E.coli GlpG in complex with peptide derived inhibitor Ac-RVRHA-cmk
分子名称:	ACE-ARG-VAL-ARG-HIS-ALA-0QE, CHLORIDE ION, Rhomboid protease GlpG, ...
著者	Vinothkumar, K.R.
登録日	2017-01-06
公開日	2017-11-15
最終更新日	2024-10-09
実験手法	X-RAY DIFFRACTION (1.95 Å)
主引用文献	General and Modular Strategy for Designing Potent, Selective, and Pharmacologically Compliant Inhibitors of Rhomboid Proteases. Cell Chem Biol, 24, 2017