3P45
| Crystal structure of apo-caspase-6 at physiological pH | 分子名称: | caspase-6 | 著者 | Mueller, I, Lamers, M.B.A.C, Ritchie, A.J, Dominguez, C, Munoz, I, Maillard, M, Kiselyov, A. | 登録日 | 2010-10-06 | 公開日 | 2011-06-15 | 最終更新日 | 2024-02-21 | 実験手法 | X-RAY DIFFRACTION (2.53 Å) | 主引用文献 | Crystal structures of active and inhibitor-bound human Casp6 To be Published
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3P4U
| Crystal structure of active caspase-6 in complex with Ac-VEID-CHO inhibitor | 分子名称: | Ac-VEID-CHO inhibitor, Caspase-6 | 著者 | Mueller, I, Lamers, M.B.A.C, Ritchie, A.J, Dominguez, C, Munoz, I, Maillard, M, Kiselyov, A. | 登録日 | 2010-10-07 | 公開日 | 2011-09-28 | 最終更新日 | 2015-12-02 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Crystal structures of active and inhibitor-bound human Casp6 To be Published
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3QNW
| Caspase-6 in complex with Z-VAD-FMK inhibitor | 分子名称: | Caspase-6, Z-VAD-FMK | 著者 | Mueller, I, Lamers, M, Ritchie, A, Park, H, Dominguez, C, Munoz, I, Maillard, M, Kiselyov, A. | 登録日 | 2011-02-09 | 公開日 | 2011-09-21 | 最終更新日 | 2023-09-13 | 実験手法 | X-RAY DIFFRACTION (2.65 Å) | 主引用文献 | Structure of human caspase-6 in complex with Z-VAD-FMK: New peptide binding mode observed for the non-canonical caspase conformation. Bioorg.Med.Chem.Lett., 21, 2011
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6TPA
| CDK8/CyclinC in complex with drug ETP-50775 | 分子名称: | (2~{R})-butane-1,2-diol, 1-[4-chloranyl-3-(trifluoromethyl)phenyl]-3-(5-oxidanylidene-6-pyridin-4-yl-pyrido[2,3-b][1,5]benzoxazepin-9-yl)urea, Cyclin-C, ... | 著者 | Munoz, I.G, Pastor, J, Martinez, S. | 登録日 | 2019-12-12 | 公開日 | 2020-11-18 | 最終更新日 | 2024-01-24 | 実験手法 | X-RAY DIFFRACTION (2.8 Å) | 主引用文献 | Pyrido[2,3-b][1,5]benzoxazepin-5(6H)-one derivatives as CDK8 inhibitors. Eur.J.Med.Chem., 201, 2020
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