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4EYM
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BU of 4eym by Molmil
MAPK13 complex with inhibitor
分子名称: 2-(morpholin-4-yl)-N-[4-(pyridin-4-yloxy)phenyl]pyridine-4-carboxamide, Mitogen-activated protein kinase 13
著者Miller, C.A, Brett, T.J.
登録日2012-05-01
公開日2012-12-19
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (2.353 Å)
主引用文献IL-13-induced airway mucus production is attenuated by MAPK13 inhibition.
J.Clin.Invest., 122, 2012
4EYJ
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BU of 4eyj by Molmil
MAPK13 Complex with inhibitor
分子名称: 1-(3-tert-butyl-1-methyl-1H-pyrazol-5-yl)-3-[4-(pyridin-4-yloxy)phenyl]urea, Mitogen-activated protein kinase 13
著者Miller, C.A, Brett, T.J.
登録日2012-05-01
公開日2012-12-19
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (2.102 Å)
主引用文献IL-13-induced airway mucus production is attenuated by MAPK13 inhibition.
J.Clin.Invest., 122, 2012
4YNO
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BU of 4yno by Molmil
Crystal structure of MAPK13 at INACTIVE FORM
分子名称: Mitogen-activated protein kinase 13
著者Miller, C.A, Brett, T.J.
登録日2015-03-10
公開日2015-04-08
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献IL-13-induced airway mucus production is attenuated by MAPK13 inhibition.
J.Clin.Invest., 122, 2012
5EKO
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BU of 5eko by Molmil
Crystal structure of MAPK13 complex with inhibitor
分子名称: 3-(4-methyl-1H-imidazol-1-yl)-N-[4-(pyridin-4-yloxy)phenyl]benzamide, Mitogen-activated protein kinase 13
著者Brett, T.J, Miller, C.A, Yurtsever, Z.
登録日2015-11-03
公開日2016-07-06
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献First comprehensive structural and biophysical analysis of MAPK13 inhibitors targeting DFG-in and DFG-out binding modes.
Biochim.Biophys.Acta, 1860, 2016
5EKN
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BU of 5ekn by Molmil
Crystal structure of MAPK13 complex with inhibitor
分子名称: 1-(3-tert-butyl-1-methyl-1H-pyrazol-5-yl)-3-[4-(pyridin-4-ylsulfanyl)phenyl]urea, Mitogen-activated protein kinase 13
著者Brett, T.J, Miller, C.A, Yurtsever, Z.
登録日2015-11-03
公開日2016-07-06
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (2.594 Å)
主引用文献First comprehensive structural and biophysical analysis of MAPK13 inhibitors targeting DFG-in and DFG-out binding modes.
Biochim.Biophys.Acta, 1860, 2016

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件を2024-07-03に公開中

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