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5SUL
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BU of 5sul by Molmil
Inhibited state structure of yGsy2p
分子名称: Glycogen [starch] synthase isoform 2, URIDINE-5'-DIPHOSPHATE, URIDINE-5'-MONOPHOSPHATE
著者Mahalingan, K.K, Hurley, T.D.
登録日2016-08-03
公開日2017-06-14
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (3.3 Å)
主引用文献Redox Switch for the Inhibited State of Yeast Glycogen Synthase Mimics Regulation by Phosphorylation.
Biochemistry, 56, 2017
6VZV
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BU of 6vzv by Molmil
TTLL6 bound to gamma-elongation analog
分子名称: (2~{S})-2-[[[(3~{R})-3-acetamido-4-oxidanyl-4-oxidanylidene-butyl]-phosphonooxy-phosphoryl]methyl]pentanedioic acid, (2~{S})-2-[[[(3~{S})-3-acetamido-4-oxidanyl-4-oxidanylidene-butyl]-oxidanyl-phosphoryl]methyl]pentanedioic acid, ADENOSINE-5'-DIPHOSPHATE, ...
著者Mahalingan, K.K, Keenen, E.K, Strickland, M, Li, Y, Liu, Y, Ball, H.L, Tanner, M.E, Tjandra, N, Roll-Mecak, A.
登録日2020-02-28
公開日2020-08-12
最終更新日2023-10-11
実験手法X-RAY DIFFRACTION (2.33 Å)
主引用文献Structural basis for polyglutamate chain initiation and elongation by TTLL family enzymes.
Nat.Struct.Mol.Biol., 27, 2020
6VZR
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BU of 6vzr by Molmil
Engineered TTLL6 bound to the initiation analog
分子名称: (2~{S})-2-[[[(3~{R})-3-acetamido-4-(ethylamino)-4-oxidanylidene-butyl]-phosphonooxy-phosphoryl]methyl]pentanedioic acid, ADENOSINE-5'-DIPHOSPHATE, GLYCEROL, ...
著者Mahalingan, K.K, Keenen, E.K, Strickland, M, Li, Y, Liu, Y, Ball, H.L, Tanner, M.E, Tjandra, N, Roll-Mecak, A.
登録日2020-02-28
公開日2020-08-12
最終更新日2023-10-11
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献Structural basis for polyglutamate chain initiation and elongation by TTLL family enzymes.
Nat.Struct.Mol.Biol., 27, 2020
5UW1
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BU of 5uw1 by Molmil
Activated state yGsy2p in complex with UDP-galactose
分子名称: 6-O-phosphono-alpha-D-glucopyranose, GALACTOSE-URIDINE-5'-DIPHOSPHATE, Glycogen [starch] synthase isoform 2
著者Mahalingan, K.K, Hurley, T.D.
登録日2017-02-20
公開日2018-02-28
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (3.26 Å)
主引用文献Activated state yGsy2p in complex with UDP-galactose
To Be Published
8T42
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BU of 8t42 by Molmil
Model of TTLL6 MTBH1-2 bound to microtubule
分子名称: GUANOSINE-5'-TRIPHOSPHATE, MAGNESIUM ION, PHOSPHOMETHYLPHOSPHONIC ACID GUANYLATE ESTER, ...
著者Mahalingan, K.K, Grotjahn, D, Li, Y, Lander, G.C, Zehr, E.A, Roll-Mecak, A.
登録日2023-06-08
公開日2024-05-08
実験手法ELECTRON MICROSCOPY (3.6 Å)
主引用文献Structural basis for alpha-tubulin-specific and modification state-dependent glutamylation.
Nat.Chem.Biol., 2024
5VNC
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BU of 5vnc by Molmil
Glycogen synthase in complex with UDP and glucosamine
分子名称: 2-amino-2-deoxy-beta-D-glucopyranose, 6-O-phosphono-alpha-D-glucopyranose, Glycogen [starch] synthase isoform 2, ...
著者Mahalingan, K.K, Hurley, T.D.
登録日2017-04-30
公開日2018-05-02
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (2.98 Å)
主引用文献Glycogen synthase in complex with UDP and glucosamine
To Be Published
8U3Z
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BU of 8u3z by Molmil
Model of TTLL6 bound to microtubule from composite map
分子名称: ADENOSINE-5'-TRIPHOSPHATE, GUANOSINE-5'-TRIPHOSPHATE, MAGNESIUM ION, ...
著者Mahalingan, K.K, Grotjahn, D, Li, Y, Lander, G.C, Zehr, E.A, Roll-Mecak, A.
登録日2023-09-08
公開日2024-05-29
実験手法ELECTRON MICROSCOPY (3.6 Å)
主引用文献Structural basis for alpha-tubulin-specific and modification state-dependent glutamylation.
Nat.Chem.Biol., 2024
5UW0
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BU of 5uw0 by Molmil
Activated state yGsy2p in complex with UDP-2-fluoro-2-deoxy-glucose
分子名称: 6-O-phosphono-alpha-D-glucopyranose, Glycogen [starch] synthase isoform 2, URIDINE-5'-DIPHOSPHATE, ...
著者Mahalingan, K.K, Hurley, T.D.
登録日2017-02-20
公開日2018-02-28
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (2.73 Å)
主引用文献Activated state yGsy2p in complex with UDP-2-fluoro-2-deoxy-glucose
To Be Published
5UX7
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BU of 5ux7 by Molmil
Activated state yeast Glycogen Synthase in complex with UDP-xylose
分子名称: 6-O-phosphono-alpha-D-glucopyranose, Glycogen [starch] synthase isoform 2, URIDINE-5'-DIPHOSPHATE, ...
著者Mahalingan, K.K, Hurley, T.D.
登録日2017-02-22
公開日2018-02-28
最終更新日2024-03-06
実験手法X-RAY DIFFRACTION (2.69 Å)
主引用文献Activated state yeast Glycogen Synthase in complex with UDP-xylose
To Be Published
6VZS
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BU of 6vzs by Molmil
Engineered TTLL6 mutant bound to gamma-elongation analog
分子名称: (2~{S})-2-[[[(3~{R})-3-acetamido-4-oxidanyl-4-oxidanylidene-butyl]-phosphonooxy-phosphoryl]methyl]pentanedioic acid, ADENOSINE-5'-DIPHOSPHATE, GLYCEROL, ...
著者Mahalingan, K.K, Keenen, E.K, Strickland, M, Li, Y, Liu, Y, Ball, H.L, Tanner, M.E, Tjandra, N, Roll-Mecak, A.
登録日2020-02-28
公開日2020-08-12
最終更新日2023-10-11
実験手法X-RAY DIFFRACTION (2.66 Å)
主引用文献Structural basis for polyglutamate chain initiation and elongation by TTLL family enzymes.
Nat.Struct.Mol.Biol., 27, 2020
6VZW
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BU of 6vzw by Molmil
TTLL6 bound to the initiation analog
分子名称: (2~{S})-2-[[[(3~{R})-3-acetamido-4-(ethylamino)-4-oxidanylidene-butyl]-phosphonooxy-phosphoryl]methyl]pentanedioic acid, ADENOSINE-5'-DIPHOSPHATE, GLYCEROL, ...
著者Mahalingan, K.K, Keenen, E.K, Strickland, M, Li, Y, Liu, Y, Ball, H.L, Tanner, T.E, Tjandra, N, Roll-Mecak, A.
登録日2020-02-28
公開日2020-08-12
最終更新日2023-10-11
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Structural basis for polyglutamate chain initiation and elongation by TTLL family enzymes.
Nat.Struct.Mol.Biol., 27, 2020
6VZU
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BU of 6vzu by Molmil
TTLL6 bound to alpha-elongation analog
分子名称: (2~{S})-2-[[[(1~{R})-1-acetamido-4-oxidanyl-4-oxidanylidene-butyl]-oxidanyl-phosphoryl]methyl]pentanedioic acid, (2~{S})-2-[[[(1~{R})-1-acetamido-4-oxidanyl-4-oxidanylidene-butyl]-phosphonooxy-phosphoryl]methyl]pentanedioic acid, ADENOSINE-5'-DIPHOSPHATE, ...
著者Mahalingan, K.K, Keenen, E.K, Strickland, M, Li, Y, Liu, Y, Ball, H.B, Tanner, M.E, Tjandra, N, Roll-Mecak, A.
登録日2020-02-28
公開日2020-08-12
最終更新日2023-10-11
実験手法X-RAY DIFFRACTION (1.98 Å)
主引用文献Structural basis for polyglutamate chain initiation and elongation by TTLL family enzymes.
Nat.Struct.Mol.Biol., 27, 2020
6VZQ
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BU of 6vzq by Molmil
Engineered TTLL6 mutant bound to alpha-elongation analog
分子名称: (2~{S})-2-[[[(1~{R})-1-acetamido-4-oxidanyl-4-oxidanylidene-butyl]-phosphonooxy-phosphoryl]methyl]pentanedioic acid, (2~{S})-2-[[[(1~{S})-1-acetamidoethyl]-phosphonooxy-phosphoryl]methyl]pentanedioic acid, ADENOSINE-5'-DIPHOSPHATE, ...
著者Mahalingan, K.K, Keenen, E.K, Strickland, E.K, Li, Y, Liu, Y, Ball, H.L, Tanner, M.E, Tjandra, N, Roll-Mecak, A.
登録日2020-02-28
公開日2020-08-12
最終更新日2023-10-11
実験手法X-RAY DIFFRACTION (3.08 Å)
主引用文献Structural basis for polyglutamate chain initiation and elongation by TTLL family enzymes.
Nat.Struct.Mol.Biol., 27, 2020
6VZT
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BU of 6vzt by Molmil
TTLL6 bound to ATP
分子名称: ADENOSINE-5'-TRIPHOSPHATE, GLYCEROL, MAGNESIUM ION, ...
著者Mahalingan, K.K, Keenen, E.K, Strickland, M, Li, Y, Liu, Y, Ball, H.L, Tanner, M.E, Tjandra, N, Roll-Mecak, A.
登録日2020-02-28
公開日2020-08-12
最終更新日2023-10-11
実験手法X-RAY DIFFRACTION (2.18 Å)
主引用文献Structural basis for polyglutamate chain initiation and elongation by TTLL family enzymes.
Nat.Struct.Mol.Biol., 27, 2020
5SUK
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BU of 5suk by Molmil
G6P bound activated state of yeast glycogen synthase 2
分子名称: 6-O-phosphono-alpha-D-glucopyranose, Glycogen [starch] synthase isoform 2
著者Baskaran, S, Mahalingan, K.K, Hurley, T.D.
登録日2016-08-03
公開日2017-06-14
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (2.88 Å)
主引用文献Redox Switch for the Inhibited State of Yeast Glycogen Synthase Mimics Regulation by Phosphorylation.
Biochemistry, 56, 2017
5UW4
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BU of 5uw4 by Molmil
Activated yeast Glycogen Synthase in complex with UDP glucosamine
分子名称: 2-amino-2-deoxy-beta-D-glucopyranose, 6-O-phosphono-alpha-D-glucopyranose, Glycogen [starch] synthase isoform 2, ...
著者Mahalingan, K.K, Hurley, T.D.
登録日2017-02-20
公開日2018-02-28
最終更新日2022-03-23
実験手法X-RAY DIFFRACTION (2.98 Å)
主引用文献Activated state yeast Glycogen Synthase in complex with UDP glucosamine
To Be Published
6U77
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BU of 6u77 by Molmil
yGsy2p in complex with small molecule
分子名称: 2-methoxy-4-(1-{2-[(2S)-1-methylpyrrolidin-2-yl]ethyl}-4-phenyl-1H-imidazol-5-yl)phenol, 6-O-phosphono-alpha-D-glucopyranose, Glycogen [starch] synthase isoform 2
著者Tang, B, Hurley, T.D.
登録日2019-08-31
公開日2020-03-18
最終更新日2023-10-11
実験手法X-RAY DIFFRACTION (2.85 Å)
主引用文献Discovery and Development of Small-Molecule Inhibitors of Glycogen Synthase.
J.Med.Chem., 63, 2020

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件を2024-06-26に公開中

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