5INB
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![BU of 5inb by Molmil](/molmil-images/mine/5inb) | RepoMan-PP1g (protein phosphatase 1, gamma isoform) holoenzyme complex | 分子名称: | Cell division cycle-associated protein 2, GLYCEROL, MALONATE ION, ... | 著者 | Kumar, G.S, Peti, W, Page, R. | 登録日 | 2016-03-07 | 公開日 | 2016-10-05 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (1.3 Å) | 主引用文献 | The Ki-67 and RepoMan mitotic phosphatases assemble via an identical, yet novel mechanism. Elife, 5, 2016
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5IOH
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![BU of 5ioh by Molmil](/molmil-images/mine/5ioh) | RepoMan-PP1a (protein phosphatase 1, alpha isoform) holoenzyme complex | 分子名称: | Cell division cycle-associated protein 2, Serine/threonine-protein phosphatase PP1-alpha catalytic subunit | 著者 | Kumar, G.S, Peti, W, Page, R. | 登録日 | 2016-03-08 | 公開日 | 2016-10-05 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (2.566 Å) | 主引用文献 | The Ki-67 and RepoMan mitotic phosphatases assemble via an identical, yet novel mechanism. Elife, 5, 2016
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5J28
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![BU of 5j28 by Molmil](/molmil-images/mine/5j28) | Ki67-PP1g (protein phosphatase 1, gamma isoform) holoenzyme complex | 分子名称: | Antigen KI-67, MALONATE ION, SODIUM ION, ... | 著者 | Kumar, G.S, Peti, W, Page, R. | 登録日 | 2016-03-29 | 公開日 | 2016-10-05 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | The Ki-67 and RepoMan mitotic phosphatases assemble via an identical, yet novel mechanism. Elife, 5, 2016
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2KTC
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![BU of 2ktc by Molmil](/molmil-images/mine/2ktc) | Solution Structure of a Novel hKv1.1 inhibiting scorpion toxin from Mesibuthus tamulus | 分子名称: | Potassium channel toxin alpha-KTx 9.4 | 著者 | Kumar, G.S, Upadhyay, S, Mathew, M.K, Sarma, S.P. | 登録日 | 2010-01-26 | 公開日 | 2011-02-02 | 最終更新日 | 2019-12-25 | 実験手法 | SOLUTION NMR | 主引用文献 | Solution structure of BTK-2, a novel hK(v)1.1 inhibiting scorpion toxin, from the eastern Indian scorpion Mesobuthus tamulus. Biochim.Biophys.Acta, 1814, 2011
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6DNO
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![BU of 6dno by Molmil](/molmil-images/mine/6dno) | Crystal structure of Protein Phosphatase 1 (PP1) bound to the muscle glycogen-targeting subunit (Gm) | 分子名称: | Microcystin-LR, Protein phosphatase 1 regulatory subunit 3A, Serine/threonine-protein phosphatase PP1-alpha catalytic subunit | 著者 | Choy, M.S, Kumar, G.S, Peti, W, Page, R. | 登録日 | 2018-06-07 | 公開日 | 2019-01-23 | 最終更新日 | 2023-11-15 | 実験手法 | X-RAY DIFFRACTION (1.45 Å) | 主引用文献 | Identification of the substrate recruitment mechanism of the muscle glycogen protein phosphatase 1 holoenzyme. Sci Adv, 4, 2018
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4HTM
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![BU of 4htm by Molmil](/molmil-images/mine/4htm) | Mechanism of CREB Recognition and Coactivation by the CREB Regulated Transcriptional Coactivator CRTC2 | 分子名称: | CREB-regulated transcription coactivator 2, ZINC ION | 著者 | Luo, Q, Viste, K, Urday-Zaa, J.C, Kumar, G.S, Tsai, W.-W, Talai, A, Mayo, K, Montminy, M, Radhakrishnan, I. | 登録日 | 2012-11-01 | 公開日 | 2012-12-05 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Protein kinase N1, a cell inhibitor of Akt kinase, has a central role in quality control of germinal center formation Proc.Natl.Acad.Sci.USA, 2012
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1YZ2
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![BU of 1yz2 by Molmil](/molmil-images/mine/1yz2) | Solution structure of Am2766 | 分子名称: | Delta-conotoxin Am 2766 | 著者 | Sarma, S.P, Kumar, G.S, Sudarslal, S, Iengar, P, Sikdar, S.K, Krishnan, K.S, Balaram, P. | 登録日 | 2005-02-26 | 公開日 | 2006-02-07 | 最終更新日 | 2019-11-06 | 実験手法 | SOLUTION NMR | 主引用文献 | Solution Structure of delta-Am2766: A Highly Hydrophobic delta-Conotoxin from Conus amadis That Inhibits Inactivation of Neuronal Voltage-Gated Sodium Channels CHEM.BIODIVERS., 2, 2005
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2M61
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![BU of 2m61 by Molmil](/molmil-images/mine/2m61) | NMR and Mass Spectrometric Studies of M-2 Branch Mini-M Conotoxins from Indian Cone Snails | 分子名称: | Conotoxin Ar1446 | 著者 | Sarma, S.P, Rajesh, R.P, Kumar, G.S, Sudarslal, S, Sabareesh, V, Gowd, K.H, Gupta, K, Krishnan, K.S, Balaram, P. | 登録日 | 2013-03-18 | 公開日 | 2014-04-16 | 実験手法 | SOLUTION NMR | 主引用文献 | NMR and Mass Spectrometric Studies of M-2 Branch Mini-M Conotoxins from Indian Cone Snails To be Published
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2L9S
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![BU of 2l9s by Molmil](/molmil-images/mine/2l9s) | Solution structure of Pf1 SID1-mSin3A PAH2 Complex | 分子名称: | PHD finger protein 12, Paired amphipathic helix protein Sin3a | 著者 | Senthil Kumar, G, Xie, T, Zhang, Y, Radhakrishnan, I. | 登録日 | 2011-02-23 | 公開日 | 2011-05-11 | 最終更新日 | 2024-05-15 | 実験手法 | SOLUTION NMR | 主引用文献 | Solution Structure of the mSin3A PAH2-Pf1 SID1 Complex: A Mad1/Mxd1-Like Interaction Disrupted by MRG15 in the Rpd3S/Sin3S Complex. J.Mol.Biol., 408, 2011
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6S15
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![BU of 6s15 by Molmil](/molmil-images/mine/6s15) | Pyridine derivative of the natural alkaloid Berberine as Human Telomeric G-quadruplex Binder | 分子名称: | Berberine, DNA TAGGGTTAGGGT, POTASSIUM ION | 著者 | Ferraroni, M, Bazzicalupi, C, Gratteri, P, Papi, F. | 登録日 | 2019-06-18 | 公開日 | 2020-06-03 | 最終更新日 | 2024-01-24 | 実験手法 | X-RAY DIFFRACTION (1.7 Å) | 主引用文献 | Pyridine Derivative of the Natural Alkaloid Berberine as Human Telomeric G4-DNA Binder: A Solution and Solid-State Study. Acs Med.Chem.Lett., 11, 2020
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6ZQS
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![BU of 6zqs by Molmil](/molmil-images/mine/6zqs) | Crystal structure of double-phosphorylated p38alpha with ATF2(83-102) | 分子名称: | 2-[(2,4-difluorophenyl)amino]-7-{[(2R)-2,3-dihydroxypropyl]oxy}-10,11-dihydro-5H-dibenzo[a,d][7]annulen-5-one, Cyclic AMP-dependent transcription factor ATF-2, Mitogen-activated protein kinase 14 | 著者 | Kirsch, K, Sok, P, Poti, A.L, Remenyi, A. | 登録日 | 2020-07-10 | 公開日 | 2020-11-18 | 最終更新日 | 2024-01-31 | 実験手法 | X-RAY DIFFRACTION (1.95 Å) | 主引用文献 | Co-regulation of the transcription controlling ATF2 phosphoswitch by JNK and p38. Nat Commun, 11, 2020
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6ZR5
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![BU of 6zr5 by Molmil](/molmil-images/mine/6zr5) | Crystal structure of JNK1 in complex with ATF2(19-58) | 分子名称: | Cyclic AMP-dependent transcription factor ATF-2, MAGNESIUM ION, Mitogen-activated protein kinase 8, ... | 著者 | Kirsch, K, Zeke, A, Remenyi, A. | 登録日 | 2020-07-10 | 公開日 | 2020-11-18 | 最終更新日 | 2024-01-31 | 実験手法 | X-RAY DIFFRACTION (2.699 Å) | 主引用文献 | Co-regulation of the transcription controlling ATF2 phosphoswitch by JNK and p38. Nat Commun, 11, 2020
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6TCA
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![BU of 6tca by Molmil](/molmil-images/mine/6tca) | Phosphorylated p38 and MAPKAPK2 complex with inhibitor | 分子名称: | MAP kinase-activated protein kinase 2, Mitogen-activated protein kinase 14, N-[5-(dimethylsulfamoyl)-2-methylphenyl]-1-phenyl-5-propyl-1H-pyrazole-4-carboxamide | 著者 | Sok, P, Remenyi, A. | 登録日 | 2019-11-05 | 公開日 | 2020-07-22 | 最終更新日 | 2024-01-24 | 実験手法 | X-RAY DIFFRACTION (3.7 Å) | 主引用文献 | MAP Kinase-Mediated Activation of RSK1 and MK2 Substrate Kinases. Structure, 28, 2020
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1JO1
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![BU of 1jo1 by Molmil](/molmil-images/mine/1jo1) | N7-Guanine Adduct of 2,7-diaminomitosene with DNA | 分子名称: | 5'-D(*GP*TP*GP*(DAJ)GP*TP*AP*TP*AP*CP*CP*AP*C)-3', DECARBAMOYL-2,7-DIAMINOMITOSENE | 著者 | Subramaniam, G, Paz, M.M, Kumar, G.S, Das, A, Palom, Y, Clement, C.C, Patel, D.J, Tomasz, M. | 登録日 | 2001-07-26 | 公開日 | 2001-09-12 | 最終更新日 | 2024-05-22 | 実験手法 | SOLUTION NMR | 主引用文献 | Solution structure of a guanine-N7-linked complex of the mitomycin C metabolite 2,7-diaminomitosene and DNA. Basis of sequence selectivity. Biochemistry, 40, 2001
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6GHM
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![BU of 6ghm by Molmil](/molmil-images/mine/6ghm) | Structure of PP1 alpha phosphatase bound to ASPP2 | 分子名称: | 1,2-ETHANEDIOL, 2-[N-CYCLOHEXYLAMINO]ETHANE SULFONIC ACID, Apoptosis-stimulating of p53 protein 2, ... | 著者 | Mouilleron, S, Bertran, T.M, Tapon, N, Zhou, Y. | 登録日 | 2018-05-08 | 公開日 | 2019-02-27 | 最終更新日 | 2024-01-17 | 実験手法 | X-RAY DIFFRACTION (2.15 Å) | 主引用文献 | ASPP proteins discriminate between PP1 catalytic subunits through their SH3 domain and the PP1 C-tail. Nat Commun, 10, 2019
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7T0Y
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![BU of 7t0y by Molmil](/molmil-images/mine/7t0y) | The Ribosomal RNA Processing 1B Protein Phosphatase-1 Holoenzyme | 分子名称: | 1,2-ETHANEDIOL, BROMIDE ION, FLUORIDE ION, ... | 著者 | Srivastava, G, Page, R, Peti, W. | 登録日 | 2021-11-30 | 公開日 | 2022-12-07 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | The ribosomal RNA processing 1B:protein phosphatase 1 holoenzyme reveals non-canonical PP1 interaction motifs. Cell Rep, 41, 2022
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4MOV
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![BU of 4mov by Molmil](/molmil-images/mine/4mov) | 1.45 A Resolution Crystal Structure of Protein Phosphatase 1 | 分子名称: | CHLORIDE ION, MANGANESE (II) ION, PHOSPHATE ION, ... | 著者 | Choy, M.S, Peti, W, Page, R. | 登録日 | 2013-09-12 | 公開日 | 2014-03-26 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (1.4503 Å) | 主引用文献 | Understanding the antagonism of retinoblastoma protein dephosphorylation by PNUTS provides insights into the PP1 regulatory code. Proc.Natl.Acad.Sci.USA, 111, 2014
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4MP0
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![BU of 4mp0 by Molmil](/molmil-images/mine/4mp0) | Structure of a second nuclear PP1 Holoenzyme, crystal form 2 | 分子名称: | GLYCEROL, MANGANESE (II) ION, PHOSPHATE ION, ... | 著者 | Choy, M.S, Hieke, M, Peti, W, Page, R. | 登録日 | 2013-09-12 | 公開日 | 2014-03-26 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (2.1003 Å) | 主引用文献 | Understanding the antagonism of retinoblastoma protein dephosphorylation by PNUTS provides insights into the PP1 regulatory code. Proc.Natl.Acad.Sci.USA, 111, 2014
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4MOY
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![BU of 4moy by Molmil](/molmil-images/mine/4moy) | Structure of a second nuclear PP1 Holoenzyme, crystal form 1 | 分子名称: | CHLORIDE ION, GLYCEROL, MANGANESE (II) ION, ... | 著者 | Choy, M.S, Hieke, M, Peti, W, Page, R. | 登録日 | 2013-09-12 | 公開日 | 2014-03-26 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (2.1953 Å) | 主引用文献 | Understanding the antagonism of retinoblastoma protein dephosphorylation by PNUTS provides insights into the PP1 regulatory code. Proc.Natl.Acad.Sci.USA, 111, 2014
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2LKM
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![BU of 2lkm by Molmil](/molmil-images/mine/2lkm) | |
8F3H
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![BU of 8f3h by Molmil](/molmil-images/mine/8f3h) | Crystal structure of Penicillin Binding Protein 5 (PBP5) S466 insertion variant apo form from Enterococcus faecium | 分子名称: | Penicillin binding protein 5, SULFATE ION | 著者 | D'Andrea, E.D, Choy, M.S, Schoenle, M.V, Page, R, Peti, W. | 登録日 | 2022-11-10 | 公開日 | 2023-07-05 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (2.6 Å) | 主引用文献 | The Molecular Basis for Resistance of E. faecium PBP5 to beta-lactam Antibiotics Nat Commun, 2023
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8F3L
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![BU of 8f3l by Molmil](/molmil-images/mine/8f3l) | Crystal structure of Penicillin Binding Protein 5 (PBP5) T485A variant penicillin bound form from Enterococcus faecium | 分子名称: | OPEN FORM - PENICILLIN G, Penicillin binding protein 5, SULFATE ION | 著者 | D'Andrea, E.D, Choy, M.S, Schoenle, M.V, Page, R, Peti, W. | 登録日 | 2022-11-10 | 公開日 | 2023-07-05 | 最終更新日 | 2024-03-13 | 実験手法 | X-RAY DIFFRACTION (3.4 Å) | 主引用文献 | The Molecular Basis for Resistance of E. faecium PBP5 to beta-lactam Antibiotics Nat Commun, 2023
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8F3O
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![BU of 8f3o by Molmil](/molmil-images/mine/8f3o) | Crystal structure of Penicillin Binding Protein 5 (PBP5) R464A variant apo form from Enterococcus faecium | 分子名称: | Penicillin binding protein 5, SULFATE ION | 著者 | D'Andrea, E.D, Choy, M.S, Schoenle, M.V, Peti, W, Page, R. | 登録日 | 2022-11-10 | 公開日 | 2023-07-05 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (3 Å) | 主引用文献 | The Molecular Basis for Resistance of E. faecium PBP5 to beta-lactam Antibiotics Nat Commun, 2023
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8F3S
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![BU of 8f3s by Molmil](/molmil-images/mine/8f3s) | Crystal structure of Penicillin Binding Protein 5 (PBP5) T485M T499I variant penicillin bound form from Enterococcus faecium | 分子名称: | OPEN FORM - PENICILLIN G, Penicillin binding protein 5, SULFATE ION | 著者 | D'Andrea, E.D, Choy, M.S, Schoenle, M.V, Page, R, Peti, W. | 登録日 | 2022-11-10 | 公開日 | 2023-07-05 | 最終更新日 | 2024-03-13 | 実験手法 | X-RAY DIFFRACTION (3.5 Å) | 主引用文献 | The Molecular Basis for Resistance of E. faecium PBP5 to beta-lactam Antibiotics Nat Commun, 2023
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8F3T
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![BU of 8f3t by Molmil](/molmil-images/mine/8f3t) | Crystal structure of Penicillin Binding Protein 5 (PBP5) T485M T499I V629E variant apo form from Enterococcus faecium | 分子名称: | Penicillin binding protein 5, SODIUM ION, SULFATE ION | 著者 | D'Andrea, E.D, Choy, M.S, Schoenle, M.V, Page, R, Peti, W. | 登録日 | 2022-11-10 | 公開日 | 2023-07-05 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (2.56 Å) | 主引用文献 | The Molecular Basis for Resistance of E. faecium PBP5 to beta-lactam Antibiotics Nat Commun, 2023
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