5NOB
| Crystal structure of human tankyrase 2 in complex with OD336 | 分子名称: | 1-[3-[4-(2-chlorophenyl)-5-pyrimidin-4-yl-1,2,4-triazol-3-yl]cyclobutyl]-2-oxidanylidene-3~{H}-benzimidazole-5-carbonitrile, Tankyrase-2, ZINC ION | 著者 | Ignatev, A, Lehtio, L. | 登録日 | 2017-04-11 | 公開日 | 2017-11-29 | 最終更新日 | 2024-01-17 | 実験手法 | X-RAY DIFFRACTION (1.85 Å) | 主引用文献 | Discovery of a Novel Series of Tankyrase Inhibitors by a Hybridization Approach. J. Med. Chem., 60, 2017
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3CPI
| Crystal structure of yeast Rab-GDI | 分子名称: | Rab GDP-dissociation inhibitor | 著者 | Kravchenko, S, Ignatev, A, Goody, R.S, Rak, A, Pylypenko, O. | 登録日 | 2008-03-31 | 公開日 | 2008-05-06 | 最終更新日 | 2023-11-01 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | A structural model of the GDP dissociation inhibitor rab membrane extraction mechanism. J.Biol.Chem., 283, 2008
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3CPJ
| Crystal structure of Ypt31 in complex with yeast Rab-GDI | 分子名称: | CHLORIDE ION, GTP-binding protein YPT31/YPT8, GUANOSINE-5'-DIPHOSPHATE, ... | 著者 | Kravchenko, S, Ignatev, A, Goody, R.S, Rak, A, Pylypenko, O. | 登録日 | 2008-03-31 | 公開日 | 2008-05-06 | 最終更新日 | 2023-11-01 | 実験手法 | X-RAY DIFFRACTION (2.35 Å) | 主引用文献 | A structural model of the GDP dissociation inhibitor rab membrane extraction mechanism. J.Biol.Chem., 283, 2008
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3CPH
| Crystal structure of Sec4 in complex with Rab-GDI | 分子名称: | GUANOSINE-5'-DIPHOSPHATE, MAGNESIUM ION, Rab GDP-dissociation inhibitor, ... | 著者 | Kravchenko, S, Ignatev, A, Goody, R.S, Rak, A, Pylypenko, O. | 登録日 | 2008-03-31 | 公開日 | 2008-05-06 | 最終更新日 | 2023-11-01 | 実験手法 | X-RAY DIFFRACTION (2.9 Å) | 主引用文献 | A structural model of the GDP dissociation inhibitor rab membrane extraction mechanism. J.Biol.Chem., 283, 2008
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5AEH
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4CBU
| Crystal structure of Plasmodium falciparum actin I | 分子名称: | ADENOSINE-5'-TRIPHOSPHATE, Actin-1, CALCIUM ION, ... | 著者 | Vahokoski, J, Bhargav, S.P, Desfosses, A, Andreadaki, M, Kumpula, E.P, Ignatev, A, Munico Martinez, S, Lepper, S, Frischknecht, F, Siden-Kiamos, I, Sachse, C, Kursula, I. | 登録日 | 2013-10-16 | 公開日 | 2014-04-30 | 最終更新日 | 2024-05-08 | 実験手法 | X-RAY DIFFRACTION (1.3 Å) | 主引用文献 | Structural Differences Explain Diverse Functions of Plasmodium Actins. Plos Pathog., 10, 2014
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4CBX
| Crystal structure of Plasmodium berghei actin II | 分子名称: | ACTIN-2, ADENOSINE-5'-TRIPHOSPHATE, CALCIUM ION, ... | 著者 | Vahokoski, J, Bhargav, S.P, Desfosses, A, Andreadaki, M, Kumpula, E.P, Ignatev, A, Munico Martinez, S, Lepper, S, Frischknecht, F, Siden-Kiamos, I, Sachse, C, Kursula, I. | 登録日 | 2013-10-17 | 公開日 | 2014-04-30 | 最終更新日 | 2023-12-20 | 実験手法 | X-RAY DIFFRACTION (2.2 Å) | 主引用文献 | Structural Differences Explain Diverse Functions of Plasmodium Actins. Plos Pathog., 10, 2014
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4CBW
| Crystal structure of Plasmodium berghei actin I with D-loop from muscle actin | 分子名称: | 1,4-DIETHYLENE DIOXIDE, ACTIN, ALPHA SKELETAL MUSCLE, ... | 著者 | Vahokoski, J, Bhargav, S.P, Desfosses, A, Andreadaki, M, Kumpula, E.P, Ignatev, A, Munico Martinez, S, Lepper, S, Frischknecht, F, Siden-Kiamos, I, Sachse, C, Kursula, I. | 登録日 | 2013-10-17 | 公開日 | 2014-04-30 | 最終更新日 | 2023-12-20 | 実験手法 | X-RAY DIFFRACTION (2.501 Å) | 主引用文献 | Structural Differences Explain Diverse Functions of Plasmodium Actins. Plos Pathog., 10, 2014
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5ADS
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5NSP
| Crystal structure of TNKS2 in complex with OD334 | 分子名称: | 1-[4-[4-(2-chlorophenyl)-5-pyrimidin-4-yl-1,2,4-triazol-3-yl]phenyl]-2-oxidanylidene-3~{H}-benzimidazole-5-carbonitrile, BICARBONATE ION, GLYCEROL, ... | 著者 | Nkizinkiko, Y, Haikarainen, T, Lehtio, L. | 登録日 | 2017-04-26 | 公開日 | 2017-11-29 | 最終更新日 | 2024-01-17 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Discovery of a Novel Series of Tankyrase Inhibitors by a Hybridization Approach. J. Med. Chem., 60, 2017
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5ADQ
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5ADR
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5ADT
| Crystal structure of human tankyrase 2 in complex with OD73 | 分子名称: | BICARBONATE ION, N-[3-chloranyl-4-[[4-(4-methoxyphenyl)oxan-4-yl]methylcarbamoyl]phenyl]-2-methyl-1,3-oxazole-5-carboxamide, SULFATE ION, ... | 著者 | Haikarainen, T, Lehtio, L. | 登録日 | 2015-08-24 | 公開日 | 2016-01-13 | 最終更新日 | 2024-05-08 | 実験手法 | X-RAY DIFFRACTION (2.15 Å) | 主引用文献 | Development and Structural Analysis of Adenosine Site Binding Tankyrase Inhibitors. Bioorg.Med.Chem.Lett., 26, 2016
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