4YAA
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![BU of 4yaa by Molmil](/molmil-images/mine/4yaa) | YopH W354Y Yersinia enterocolitica PTPase apo form | 分子名称: | ACETATE ION, SULFATE ION, Tyrosine-protein phosphatase YopH | 著者 | Moise, G.E, Johnson, S.J, Hengge, A.C. | 登録日 | 2015-02-17 | 公開日 | 2015-10-28 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (1.05 Å) | 主引用文献 | Conservative Tryptophan Mutants of the Protein Tyrosine Phosphatase YopH Exhibit Impaired WPD-Loop Function and Crystallize with Divanadate Esters in Their Active Sites. Biochemistry, 54, 2015
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4ZI4
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6DT6
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![BU of 6dt6 by Molmil](/molmil-images/mine/6dt6) | Crystal Structure of the YopH PTP1B Chimera 3 PTPase bound to vanadate | 分子名称: | Targeted effector protein, VANADATE ION | 著者 | Morales, Y, Johnson, S.J, Hengge, A.C. | 登録日 | 2018-06-15 | 公開日 | 2018-08-29 | 最終更新日 | 2023-10-11 | 実験手法 | X-RAY DIFFRACTION (2.101 Å) | 主引用文献 | A YopH PTP1B Chimera Shows the Importance of the WPD-Loop Sequence to the Activity, Structure, and Dynamics of Protein Tyrosine Phosphatases. Biochemistry, 57, 2018
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6DRB
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![BU of 6drb by Molmil](/molmil-images/mine/6drb) | Crystal Structure of the YopH PTP1B WPD loop Chimera 3 PTPase bound to tungstate | 分子名称: | TUNGSTATE(VI)ION, Targeted effector protein | 著者 | Morales, Y, Johnson, S.J, Hengge, A.C. | 登録日 | 2018-06-11 | 公開日 | 2018-08-29 | 最終更新日 | 2023-10-11 | 実験手法 | X-RAY DIFFRACTION (2.745 Å) | 主引用文献 | A YopH PTP1B Chimera Shows the Importance of the WPD-Loop Sequence to the Activity, Structure, and Dynamics of Protein Tyrosine Phosphatases. Biochemistry, 57, 2018
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6DR1
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![BU of 6dr1 by Molmil](/molmil-images/mine/6dr1) | YopH PTP1B Chimera 2 PTPase | 分子名称: | Targeted effector protein | 著者 | Morales, Y, Johnson, S.J, Hengge, A.C. | 登録日 | 2018-06-11 | 公開日 | 2018-08-29 | 最終更新日 | 2023-10-11 | 実験手法 | X-RAY DIFFRACTION (2.5 Å) | 主引用文献 | A YopH PTP1B Chimera Shows the Importance of the WPD-Loop Sequence to the Activity, Structure, and Dynamics of Protein Tyrosine Phosphatases. Biochemistry, 57, 2018
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6DR7
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![BU of 6dr7 by Molmil](/molmil-images/mine/6dr7) | YopH PTP1B WPD loop Chimera 2 PTPase bound to vanadate | 分子名称: | ACETATE ION, Targeted effector protein, VANADATE ION | 著者 | Moise, G, Morales, Y, Johnson, S.J, Hengge, A.C. | 登録日 | 2018-06-11 | 公開日 | 2018-08-29 | 最終更新日 | 2023-10-11 | 実験手法 | X-RAY DIFFRACTION (1.849 Å) | 主引用文献 | A YopH PTP1B Chimera Shows the Importance of the WPD-Loop Sequence to the Activity, Structure, and Dynamics of Protein Tyrosine Phosphatases. Biochemistry, 57, 2018
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3I7Z
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![BU of 3i7z by Molmil](/molmil-images/mine/3i7z) | Protein Tyrosine Phosphatase 1B - Transition state analog for the first catalytic step | 分子名称: | 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, EGFR receptor fragment, GLYCEROL, ... | 著者 | Brandao, T.A.S, Johnson, S.J, Hengge, A.C. | 登録日 | 2009-07-09 | 公開日 | 2010-03-16 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Insights into the reaction of protein-tyrosine phosphatase 1B: crystal structures for transition state analogs of both catalytic steps. J.Biol.Chem., 285, 2010
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3I80
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![BU of 3i80 by Molmil](/molmil-images/mine/3i80) | Protein Tyrosine Phosphatase 1B - Transition state analog for the second catalytic step | 分子名称: | 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, GLYCEROL, Tyrosine-protein phosphatase non-receptor type 1, ... | 著者 | Brandao, T.A.S, Johnson, S.J, Hengge, A.C. | 登録日 | 2009-07-09 | 公開日 | 2010-03-16 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (2.25 Å) | 主引用文献 | Insights into the reaction of protein-tyrosine phosphatase 1B: crystal structures for transition state analogs of both catalytic steps. J.Biol.Chem., 285, 2010
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4H43
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4HAH
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4Z6B
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4ZN5
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![BU of 4zn5 by Molmil](/molmil-images/mine/4zn5) | YopH W354Y Yersinia enterocolitica PTPase bond with Divanadate glycerol ester in the active site | 分子名称: | ACETATE ION, Divanadate Glycerol ester, GLYCEROL, ... | 著者 | Moise, G.E, Johnson, S.J, Hengge, A.C. | 登録日 | 2015-05-04 | 公開日 | 2015-10-28 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (1.12 Å) | 主引用文献 | Conservative Tryptophan Mutants of the Protein Tyrosine Phosphatase YopH Exhibit Impaired WPD-Loop Function and Crystallize with Divanadate Esters in Their Active Sites. Biochemistry, 54, 2015
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7MPD
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![BU of 7mpd by Molmil](/molmil-images/mine/7mpd) | Structure of SsoPTP bound to 2-chloroethylsulfonate | 分子名称: | 2-chloroethane-1-sulfonic acid, 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, SsoPTP | 著者 | Pinkston, J.A, Olsen, K.J, Hengge, A.C, Johnson, S.J. | 登録日 | 2021-05-04 | 公開日 | 2021-09-22 | 最終更新日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (1.05 Å) | 主引用文献 | Significant Loop Motions in the SsoPTP Protein Tyrosine Phosphatase Allow for Dual General Acid Functionality. Biochemistry, 60, 2021
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7MPC
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![BU of 7mpc by Molmil](/molmil-images/mine/7mpc) | Structure of SsoPTP bound to vanadate | 分子名称: | SsoPTP, VANADATE ION | 著者 | Pinkston, J.A, Olsen, K.J, Hengge, A.C, Johnson, S.J. | 登録日 | 2021-05-04 | 公開日 | 2021-09-22 | 最終更新日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (1.75 Å) | 主引用文献 | Significant Loop Motions in the SsoPTP Protein Tyrosine Phosphatase Allow for Dual General Acid Functionality. Biochemistry, 60, 2021
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6DR9
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7S4F
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![BU of 7s4f by Molmil](/molmil-images/mine/7s4f) | Protein Tyrosine Phosphatase 1B - F182Q mutant bound with Hepes | 分子名称: | 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, GLYCEROL, MAGNESIUM ION, ... | 著者 | Brandao, T.A.S, Hengge, A.C, Johnson, S.J. | 登録日 | 2021-09-08 | 公開日 | 2022-09-21 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (1.65 Å) | 主引用文献 | Insights into the importance of WPD-loop sequence for activity and structure in protein tyrosine phosphatases. Chem Sci, 13, 2022
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3QKQ
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![BU of 3qkq by Molmil](/molmil-images/mine/3qkq) | Protein Tyrosine Phosphatase 1B - W179F mutant bound with vanadate | 分子名称: | 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, GLYCEROL, Tyrosine-protein phosphatase non-receptor type 1, ... | 著者 | Brandao, T.A.S, Johnson, S.J, Hengge, A.C. | 登録日 | 2011-02-01 | 公開日 | 2012-08-08 | 最終更新日 | 2023-09-13 | 実験手法 | X-RAY DIFFRACTION (2.2 Å) | 主引用文献 | The molecular details of WPD-loop movement differ in the protein-tyrosine phosphatases YopH and PTP1B. Arch.Biochem.Biophys., 525, 2012
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3QKP
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![BU of 3qkp by Molmil](/molmil-images/mine/3qkp) | Protein Tyrosine Phosphatase 1B - Apo W179F mutant with open WPD-loop | 分子名称: | 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, GLYCEROL, Tyrosine-protein phosphatase non-receptor type 1 | 著者 | Brandao, T.A.S, Johnson, S.J, Hengge, A.C. | 登録日 | 2011-02-01 | 公開日 | 2012-08-08 | 最終更新日 | 2023-09-13 | 実験手法 | X-RAY DIFFRACTION (2.05 Å) | 主引用文献 | The molecular details of WPD-loop movement differ in the protein-tyrosine phosphatases YopH and PTP1B. Arch.Biochem.Biophys., 525, 2012
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7L0C
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![BU of 7l0c by Molmil](/molmil-images/mine/7l0c) | Ligand-free PTP1B T177G | 分子名称: | Tyrosine-protein phosphatase non-receptor type 1 | 著者 | Shen, R.D, Hengge, A.C, Johnson, S.J. | 登録日 | 2020-12-11 | 公開日 | 2021-05-12 | 最終更新日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | Single Residue on the WPD-Loop Affects the pH Dependency of Catalysis in Protein Tyrosine Phosphatases. Jacs Au, 1, 2021
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7L0M
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![BU of 7l0m by Molmil](/molmil-images/mine/7l0m) | Vanadate-bound YopH G352T | 分子名称: | Protein-tyrosine-phosphatase, VANADATE ION | 著者 | Shen, R.D, Hengge, A.C, Johnson, S.J. | 登録日 | 2020-12-11 | 公開日 | 2021-05-12 | 最終更新日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Single Residue on the WPD-Loop Affects the pH Dependency of Catalysis in Protein Tyrosine Phosphatases. Jacs Au, 1, 2021
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7L0I
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![BU of 7l0i by Molmil](/molmil-images/mine/7l0i) | Ligand-free YopH G352T | 分子名称: | 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, Protein-tyrosine-phosphatase | 著者 | Shen, R.D, Hengge, A.C, Johnson, S.J. | 登録日 | 2020-12-11 | 公開日 | 2021-05-12 | 最終更新日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (2.02 Å) | 主引用文献 | Single Residue on the WPD-Loop Affects the pH Dependency of Catalysis in Protein Tyrosine Phosphatases. Jacs Au, 1, 2021
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7L0H
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![BU of 7l0h by Molmil](/molmil-images/mine/7l0h) | Vanadate-bound PTP1B T177G | 分子名称: | Tyrosine-protein phosphatase non-receptor type 1, VANADATE ION | 著者 | Shen, R.D, Hengge, A.C, Johnson, S.J. | 登録日 | 2020-12-11 | 公開日 | 2021-05-12 | 最終更新日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | Single Residue on the WPD-Loop Affects the pH Dependency of Catalysis in Protein Tyrosine Phosphatases. Jacs Au, 1, 2021
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3F9A
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![BU of 3f9a by Molmil](/molmil-images/mine/3f9a) | W354F Yersinia enterocolitica PTPase complexed with tungstate | 分子名称: | TUNGSTATE(VI)ION, Tyrosine-protein phosphatase yopH | 著者 | Brandao, T.A.S, Robinson, H, Johnson, S.J, Hengge, A.C. | 登録日 | 2008-11-13 | 公開日 | 2009-01-20 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (1.69 Å) | 主引用文献 | Impaired acid catalysis by mutation of a protein loop hinge residue in a YopH mutant revealed by crystal structures. J.Am.Chem.Soc., 131, 2009
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3F9B
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![BU of 3f9b by Molmil](/molmil-images/mine/3f9b) | W354F Yersinia enterocolitica PTPase complexed with divanadate | 分子名称: | Divanadate ion, GLYCEROL, Tyrosine-protein phosphatase yopH, ... | 著者 | Brandao, T.A.S, Robinson, H, Johnson, S.J, Hengge, A.C. | 登録日 | 2008-11-13 | 公開日 | 2009-01-20 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (1.42 Å) | 主引用文献 | Impaired acid catalysis by mutation of a protein loop hinge residue in a YopH mutant revealed by crystal structures. J.Am.Chem.Soc., 131, 2009
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3D03
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![BU of 3d03 by Molmil](/molmil-images/mine/3d03) | 1.9A structure of Glycerophoshphodiesterase (GpdQ) from Enterobacter aerogenes | 分子名称: | COBALT (II) ION, Phosphohydrolase | 著者 | Hadler, K.S, Tanifum, E, Yip, S.H.-C, Miti, N, Guddat, L.W, Jackson, C.J, Gahan, L.R, Carr, P.D, Nguyen, K, Ollis, D.L, Hengge, A.C, Larrabee, J.A, Schenk, G. | 登録日 | 2008-04-30 | 公開日 | 2008-10-14 | 最終更新日 | 2023-08-30 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Substrate-promoted formation of a catalytically competent binuclear center and regulation of reactivity in a glycerophosphodiesterase from Enterobacter aerogenes. J.Am.Chem.Soc., 130, 2008
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