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8VP4
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BU of 8vp4 by Molmil
Crystal Structure of JF1cpCasp2 with Peptide Inhibitor AcVDVAD-CHO
分子名称: AcVDVAD-CHO, JF1cpCasp2
著者Fuller, J.L, Shi, K, Walters, M.A, Finzel, B.C.
登録日2024-01-16
公開日2025-04-09
最終更新日2025-04-30
実験手法X-RAY DIFFRACTION (1.51 Å)
主引用文献Reengineering of Circularly Permuted Caspase-2 to Enhance Enzyme Stability and Enable Crystallographic Studies.
Acs Chem.Biol., 20, 2025
9C2Y
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BU of 9c2y by Molmil
Crystal Structure of JF1cpCasp2 in complex with MUR-65
分子名称: JF1cpCasp2, MUR-65
著者Fuller, J.L, Finzel, B.C, Shi, K.
登録日2024-05-31
公開日2025-04-09
最終更新日2025-04-30
実験手法X-RAY DIFFRACTION (1.96 Å)
主引用文献Reengineering of Circularly Permuted Caspase-2 to Enhance Enzyme Stability and Enable Crystallographic Studies.
Acs Chem.Biol., 20, 2025
7SEO
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BU of 7seo by Molmil
Crystal Structure of Caspase-3 with Peptide Inhibitor Ac-VDV(DAB)D-CHO
分子名称: ACE-VAL-ASP-VAL-DAB-ASP, Caspase-3 subunit p12, Caspase-3 subunit p17
著者Fuller, J.L, Finzel, B.C.
登録日2021-09-30
公開日2022-01-05
最終更新日2024-10-30
実験手法X-RAY DIFFRACTION (3.25 Å)
主引用文献Structure-Based Design and Biological Evaluation of Novel Caspase-2 Inhibitors Based on the Peptide AcVDVAD-CHO and the Caspase-2-Mediated Tau Cleavage Sequence YKPVD314.
Acs Pharmacol Transl Sci, 5, 2022
7USQ
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BU of 7usq by Molmil
Crystal Structure of Caspase-3 with Peptide Inhibitor AcDVPD-CHO
分子名称: Caspase-3 subunit p12, Caspase-3 subunit p17, Peptide Inhibitor AcDVPD-CHO
著者Fuller, J.L, Finzel, B.C.
登録日2022-04-25
公開日2022-06-01
最終更新日2024-10-23
実験手法X-RAY DIFFRACTION (2.71 Å)
主引用文献Characterization of caspase-2 inhibitors based on specific sites of caspase-2-mediated proteolysis.
Arch Pharm, 355, 2022
7USO
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BU of 7uso by Molmil
Crystal Structure of Caspase-3 with Peptide Inhibitor AcITVKD-CHO
分子名称: Caspase-3 subunit p12, Caspase-3 subunit p17, Peptide Inhibitor AcITVKD-CHO
著者Fuller, J.L, Finzel, B.C.
登録日2022-04-25
公開日2022-06-01
最終更新日2024-11-06
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Characterization of caspase-2 inhibitors based on specific sites of caspase-2-mediated proteolysis.
Arch Pharm, 355, 2022
7USP
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BU of 7usp by Molmil
Crystal Structure of Caspase-3 with Peptide Inhibitor AcITV(Orn)D-CHO
分子名称: Caspase-3 subunit p12, Caspase-3 subunit p17, Peptide Inhibitor AcITV(Orn)D-CHO
著者Fuller, J.L, Finzel, B.C.
登録日2022-04-25
公開日2022-06-01
最終更新日2023-10-18
実験手法X-RAY DIFFRACTION (2.85 Å)
主引用文献Characterization of caspase-2 inhibitors based on specific sites of caspase-2-mediated proteolysis.
Arch Pharm, 355, 2022

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件を2025-07-09に公開中

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