5YY9
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![BU of 5yy9 by Molmil](/molmil-images/mine/5yy9) | Crystal structure of Tandem Tudor Domain of human UHRF1 in complex with LIG1-K126me3 | 分子名称: | E3 ubiquitin-protein ligase UHRF1, Ligase 1 | 著者 | Kori, S, Defossez, P.A, Arita, K. | 登録日 | 2017-12-08 | 公開日 | 2018-12-12 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (2.653 Å) | 主引用文献 | Structure of the UHRF1 Tandem Tudor Domain Bound to a Methylated Non-histone Protein, LIG1, Reveals Rules for Binding and Regulation. Structure, 27, 2019
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5YYA
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![BU of 5yya by Molmil](/molmil-images/mine/5yya) | Crystal structure of Tandem Tudor Domain of human UHRF1 | 分子名称: | 1,2-ETHANEDIOL, E3 ubiquitin-protein ligase UHRF1, SULFATE ION | 著者 | Kori, S, Defossez, P.A, Arita, K. | 登録日 | 2017-12-08 | 公開日 | 2018-12-12 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (1.7 Å) | 主引用文献 | Structure of the UHRF1 Tandem Tudor Domain Bound to a Methylated Non-histone Protein, LIG1, Reveals Rules for Binding and Regulation. Structure, 27, 2019
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7FB7
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![BU of 7fb7 by Molmil](/molmil-images/mine/7fb7) | Crystal structure of human UHRF1 TTD in complex with 5-amino-2,4-dimethylpyridine | 分子名称: | (4S)-2-METHYL-2,4-PENTANEDIOL, 5-amino-2,4-dimethylpyridine, DIMETHYL SULFOXIDE, ... | 著者 | Kori, S, Arita, K, Yoshimi, S. | 登録日 | 2021-07-08 | 公開日 | 2022-01-05 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (1.45 Å) | 主引用文献 | Structure-based screening combined with computational and biochemical analyses identified the inhibitor targeting the binding of DNA Ligase 1 to UHRF1. Bioorg.Med.Chem., 52, 2021
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7XI9
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![BU of 7xi9 by Molmil](/molmil-images/mine/7xi9) | Cryo-EM structure of human DNMT1 (aa:351-1616) in complex with ubiquitinated H3 and hemimethylated DNA analog (CXXC-ordered form) | 分子名称: | DNA (5'-D(*AP*CP*TP*TP*AP*(5CM)P*GP*GP*AP*AP*GP*G)-3'), DNA (5'-D(*CP*CP*TP*TP*CP*(C55)P*GP*TP*AP*AP*GP*T)-3'), DNA (cytosine-5)-methyltransferase 1, ... | 著者 | Onoda, H, Kikuchi, A, Kori, S, Yoshimi, S, Yamagata, A, Arita, K. | 登録日 | 2022-04-12 | 公開日 | 2022-11-30 | 最終更新日 | 2022-12-07 | 実験手法 | ELECTRON MICROSCOPY (2.52 Å) | 主引用文献 | Structural basis for activation of DNMT1. Nat Commun, 13, 2022
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7XIB
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![BU of 7xib by Molmil](/molmil-images/mine/7xib) | Cryo-EM structure of human DNMT1 (aa:351-1616) in complex with ubiquitinated H3 and hemimethylated DNA analog (CXXC-disordered form) | 分子名称: | DNA (5'-D(*AP*CP*TP*TP*AP*(5CM)P*GP*GP*AP*AP*GP*G)-3'), DNA (5'-D(*CP*CP*TP*TP*CP*(C55)P*GP*TP*AP*AP*GP*T)-3'), DNA (cytosine-5)-methyltransferase 1, ... | 著者 | Onoda, H, Kikuchi, A, Kori, S, Yoshimi, S, Yamagata, A, Arita, K. | 登録日 | 2022-04-12 | 公開日 | 2022-11-30 | 最終更新日 | 2022-12-07 | 実験手法 | ELECTRON MICROSCOPY (2.23 Å) | 主引用文献 | Structural basis for activation of DNMT1. Nat Commun, 13, 2022
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