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6EXW
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BU of 6exw by Molmil
Crystal structure of cIAP1-BIR3 in complex with a covalently bound SM
分子名称: (3~{S},6~{S},7~{R},9~{a}~{S})-6-[[(2~{S})-2-(methylamino)propanoyl]amino]-5-oxidanylidene-~{N}-(phenylmethyl)-7-[(propanoylamino)methyl]-3,6,7,8,9,9~{a}-hexahydropyrrolo[1,2-a]azepine-3-carboxamide, Baculoviral IAP repeat-containing protein 2, ZINC ION
著者Corti, A, Cossu, F, Milani, M, Mastrangelo, E.
登録日2017-11-10
公開日2018-08-08
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Structure-based design and molecular profiling of Smac-mimetics selective for cellular IAPs.
FEBS J., 285, 2018
6EY2
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BU of 6ey2 by Molmil
Crystal structure of XIAP-BIR3 in complex with a cIAP1-selective SM
分子名称: (3~{S},6~{S},7~{S},9~{a}~{S})-~{N}-[(4-~{tert}-butylphenyl)methyl]-7-(hydroxymethyl)-6-[[(2~{S})-2-(methylamino)butanoyl]amino]-5-oxidanylidene-1,2,3,6,7,8,9,9~{a}-octahydropyrrolo[1,2-a]azepine-3-carboxamide, E3 ubiquitin-protein ligase XIAP, ZINC ION
著者Cossu, F, Corti, A, Milani, M, Mastrangelo, E.
登録日2017-11-10
公開日2018-08-08
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (2.7 Å)
主引用文献Structure-based design and molecular profiling of Smac-mimetics selective for cellular IAPs.
FEBS J., 285, 2018
6R2X
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BU of 6r2x by Molmil
NMR structure of Chromogranin A (F39-D63)
分子名称: Chromogranin-A
著者Nardelli, F, Quilici, G, Ghitti, M, Curnis, F, Gori, A, Berardi, A, Corti, A, Musco, G.
登録日2019-03-19
公開日2019-12-04
最終更新日2024-06-19
実験手法SOLUTION NMR
主引用文献A stapled chromogranin A-derived peptide is a potent dual ligand for integrins alpha v beta 6 and alpha v beta 8.
Chem.Commun.(Camb.), 55, 2019
1RAV
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BU of 1rav by Molmil
RECOMBINANT AVIDIN
分子名称: AVIDIN
著者Rosano, C, Arosio, P, Bolognesi, M.
登録日1998-03-27
公開日1998-07-15
最終更新日2023-08-09
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Biochemical characterization and crystal structure of a recombinant hen avidin and its acidic mutant expressed in Escherichia coli.
Eur.J.Biochem., 256, 1998
4MTZ
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BU of 4mtz by Molmil
Structure of XIAP-BIR1 in complex with NF023
分子名称: 8-({3-[({3-[(4,6,8-trisulfonaphthalen-1-yl)carbamoyl]phenyl}carbamoyl)amino]benzoyl}amino)naphthalene-1,3,5-trisulfonic acid, E3 ubiquitin-protein ligase XIAP, SULFATE ION, ...
著者Cossu, F, Milani, M, Grassi, S, Mastrangelo, E, Bolognesi, M.
登録日2013-09-20
公開日2014-09-24
最終更新日2023-09-20
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Protein-protein interactions in nfkb pathway: novel tools to promote apoptosis in cancer therapy
To be Published
4OXC
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BU of 4oxc by Molmil
Crystal structure of XIAP BIR1 domain
分子名称: E3 ubiquitin-protein ligase XIAP, ZINC ION
著者Milani, M, Cossu, F, Mastrangelo, E.
登録日2014-02-05
公開日2015-02-11
最終更新日2023-12-27
実験手法X-RAY DIFFRACTION (2.9 Å)
主引用文献NF023 binding to XIAP-BIR1: Searching drugs for regulation of the NF-kappa B pathway.
Proteins, 83, 2015
2CAM
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BU of 2cam by Molmil
AVIDIN MUTANT (K3E,K9E,R26D,R124L)
分子名称: AVIDIN
著者Rosano, C, Arosio, P, Bolognesi, M.
登録日1998-03-27
公開日1998-07-15
最終更新日2023-08-09
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Biochemical characterization and crystal structure of a recombinant hen avidin and its acidic mutant expressed in Escherichia coli.
Eur.J.Biochem., 256, 1998
8AKP
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BU of 8akp by Molmil
Crystal structure of the catalytic domain of G7048 from Penicillium sumatraense
分子名称: 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, alpha-D-mannopyranose-(1-3)-[alpha-D-mannopyranose-(1-6)]alpha-D-mannopyranose-(1-6)-[alpha-D-mannopyranose-(1-3)]beta-D-mannopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, catalytic domain of G7048
著者Troilo, F, Scafati, V, Giovannoni, M, Mattei, B, Benedetti, M, Angelucci, F, Di Matteo, A.
登録日2022-07-30
公開日2022-12-28
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Characterization of two 1,3-beta-glucan-modifying enzymes from Penicillium sumatraense reveals new insights into 1,3-beta-glucan metabolism of fungal saprotrophs.
Biotechnol Biofuels Bioprod, 15, 2022

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件を2024-07-31に公開中

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