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6WHR
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BU of 6whr by Molmil
GluN1b-GluN2B NMDA receptor in non-active 2 conformation at 4 angstrom resolution
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Glutamate receptor ionotropic, ...
著者Chou, T, Tajima, N, Furukawa, H.
登録日2020-04-08
公開日2020-08-05
実験手法ELECTRON MICROSCOPY (3.99 Å)
主引用文献Structural Basis of Functional Transitions in Mammalian NMDA Receptors.
Cell, 182, 2020
6WI1
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BU of 6wi1 by Molmil
GluN1b-GluN2B NMDA receptor in active conformation stabilized by inter-GluN1b-GluN2B subunit cross-linking
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Ionotropic glutamate receptor , ...
著者Chou, T, Tajima, N, Furukawa, H.
登録日2020-04-08
公開日2020-07-15
最終更新日2020-08-05
実験手法ELECTRON MICROSCOPY (3.62 Å)
主引用文献Structural Basis of Functional Transitions in Mammalian NMDA Receptors.
Cell, 182, 2020
6WHX
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BU of 6whx by Molmil
GluN1b-GluN2B NMDA receptor in complex with GluN2B antagonist SDZ 220-040, class 2
分子名称: (2S)-2-amino-3-[2',4'-dichloro-4-hydroxy-5-(phosphonomethyl)biphenyl-3-yl]propanoic acid, 2-acetamido-2-deoxy-beta-D-glucopyranose, Ionotropic glutamate receptor , ...
著者Chou, T, Tajima, N, Furukawa, H.
登録日2020-04-08
公開日2020-07-15
最終更新日2020-08-05
実験手法ELECTRON MICROSCOPY (4.09 Å)
主引用文献Structural Basis of Functional Transitions in Mammalian NMDA Receptors.
Cell, 182, 2020
6WHU
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BU of 6whu by Molmil
GluN1b-GluN2B NMDA receptor in complex with SDZ 220-040 and L689,560, class 1
分子名称: (2R,4S)-5,7-dichloro-4-[(phenylcarbamoyl)amino]-1,2,3,4-tetrahydroquinoline-2-carboxylic acid, (2S)-2-amino-3-[2',4'-dichloro-4-hydroxy-5-(phosphonomethyl)biphenyl-3-yl]propanoic acid, 2-acetamido-2-deoxy-beta-D-glucopyranose, ...
著者Chou, T, Tajima, N, Furukawa, H.
登録日2020-04-08
公開日2020-08-05
実験手法ELECTRON MICROSCOPY (3.93 Å)
主引用文献Structural Basis of Functional Transitions in Mammalian NMDA Receptors.
Cell, 182, 2020
6WHW
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BU of 6whw by Molmil
GluN1b-GluN2B NMDA receptor in complex with GluN2B antagonist SDZ 220-040, class 1
分子名称: (2S)-2-amino-3-[2',4'-dichloro-4-hydroxy-5-(phosphonomethyl)biphenyl-3-yl]propanoic acid, 2-acetamido-2-deoxy-beta-D-glucopyranose, Ionotropic glutamate receptor , ...
著者Chou, T, Tajima, N, Furukawa, H.
登録日2020-04-08
公開日2020-07-15
最終更新日2020-08-05
実験手法ELECTRON MICROSCOPY (4.09 Å)
主引用文献Structural Basis of Functional Transitions in Mammalian NMDA Receptors.
Cell, 182, 2020
6WHY
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BU of 6why by Molmil
GluN1b-GluN2B NMDA receptor in complex with GluN1 antagonist L689,560, class 1
分子名称: (2R,4S)-5,7-dichloro-4-[(phenylcarbamoyl)amino]-1,2,3,4-tetrahydroquinoline-2-carboxylic acid, 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ...
著者Chou, T, Tajima, N, Furukawa, H.
登録日2020-04-08
公開日2020-07-15
最終更新日2020-08-05
実験手法ELECTRON MICROSCOPY (4.03 Å)
主引用文献Structural Basis of Functional Transitions in Mammalian NMDA Receptors.
Cell, 182, 2020
6WHS
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BU of 6whs by Molmil
GluN1b-GluN2B NMDA receptor in non-active 1 conformation at 3.95 angstrom resolution
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Glutamate receptor ionotropic, ...
著者Chou, T, Tajima, N, Furukawa, H.
登録日2020-04-08
公開日2020-08-05
実験手法ELECTRON MICROSCOPY (4 Å)
主引用文献Structural Basis of Functional Transitions in Mammalian NMDA Receptors.
Cell, 182, 2020
6WHV
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BU of 6whv by Molmil
GluN1b-GluN2B NMDA receptor in complex with SDZ 220-040 and L689,560, class 2
分子名称: (2R,4S)-5,7-dichloro-4-[(phenylcarbamoyl)amino]-1,2,3,4-tetrahydroquinoline-2-carboxylic acid, (2S)-2-amino-3-[2',4'-dichloro-4-hydroxy-5-(phosphonomethyl)biphenyl-3-yl]propanoic acid, 2-acetamido-2-deoxy-beta-D-glucopyranose, ...
著者Chou, T, Tajima, N, Furukawa, H.
登録日2020-04-08
公開日2020-08-05
実験手法ELECTRON MICROSCOPY (4.05 Å)
主引用文献Structural Basis of Functional Transitions in Mammalian NMDA Receptors.
Cell, 182, 2020
6WHT
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BU of 6wht by Molmil
GluN1b-GluN2B NMDA receptor in active conformation at 4.4 angstrom resolution
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Glutamate receptor ionotropic, ...
著者Chou, T, Tajima, N, Furukawa, H.
登録日2020-04-08
公開日2020-08-05
実験手法ELECTRON MICROSCOPY (4.39 Å)
主引用文献Structural Basis of Functional Transitions in Mammalian NMDA Receptors.
Cell, 182, 2020
6WI0
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BU of 6wi0 by Molmil
GluN1b-GluN2B NMDA receptor in complex with GluN1 antagonist L689,560, class 2
分子名称: (2R,4S)-5,7-dichloro-4-[(phenylcarbamoyl)amino]-1,2,3,4-tetrahydroquinoline-2-carboxylic acid, 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ...
著者Chou, T, Tajima, N, Furukawa, H.
登録日2020-04-08
公開日2020-07-15
最終更新日2020-08-05
実験手法ELECTRON MICROSCOPY (4.27 Å)
主引用文献Structural Basis of Functional Transitions in Mammalian NMDA Receptors.
Cell, 182, 2020
6USU
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BU of 6usu by Molmil
Crystal structure of GluN1/GluN2A ligand-binding domain in complex with L689,560 and glutamate
分子名称: (2R,4S)-5,7-dichloro-4-[(phenylcarbamoyl)amino]-1,2,3,4-tetrahydroquinoline-2-carboxylic acid, GLUTAMIC ACID, Glutamate receptor ionotropic, ...
著者Romero-Hernandez, A, Tajima, N, Chou, T, Furukawa, H.
登録日2019-10-28
公開日2020-07-15
最終更新日2023-10-11
実験手法X-RAY DIFFRACTION (2.092 Å)
主引用文献Structural Basis of Functional Transitions in Mammalian NMDA Receptors.
Cell, 182, 2020
6USV
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BU of 6usv by Molmil
Crystal structure of GluN1/GluN2A ligand-binding domain in complex with glycine and SDZ 220-040
分子名称: (2S)-2-amino-3-[2',4'-dichloro-4-hydroxy-5-(phosphonomethyl)biphenyl-3-yl]propanoic acid, GLYCEROL, GLYCINE, ...
著者Romero-Hernandez, A, Tajima, N, Chou, T, Furukawa, h.
登録日2019-10-28
公開日2020-07-15
最終更新日2023-10-11
実験手法X-RAY DIFFRACTION (2.304 Å)
主引用文献Structural Basis of Functional Transitions in Mammalian NMDA Receptors.
Cell, 182, 2020
6DBP
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BU of 6dbp by Molmil
RNA-recognition motif 1 of human MSI2
分子名称: RNA-binding protein Musashi homolog 2
著者Goldgur, Y, Kharas, M.G, Minuesa, G.
登録日2018-05-03
公開日2019-05-08
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (1.603 Å)
主引用文献Small-molecule targeting of MUSASHI RNA-binding activity in acute myeloid leukemia.
Nat Commun, 10, 2019
8P43
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BU of 8p43 by Molmil
Structure of the MHC class Ib molecule Qa-1b in complex with Q001 peptide
分子名称: Beta-2-microglobulin, H-2 class I histocompatibility antigen, Qa-1b, ...
著者Sala, B.M, Achour, A.
登録日2023-05-19
公開日2024-06-12
実験手法X-RAY DIFFRACTION (2.43 Å)
主引用文献MHC-E is a convergent checkpoint ligand for LILRB1 on macrophages and during inflammation for NKG2A on lymphocytes
To Be Published
8ANO
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BU of 8ano by Molmil
Fucosylated mixed-chirality linear peptide FHP8 bound to the fucose binding lectin LecB PA-IIL from Pseudomonas aeruginosa at 1.3 Angstrom resolution.
分子名称: 3,7-anhydro-2,8-dideoxy-L-glycero-D-gluco-octonic acid, CALCIUM ION, Fucose-binding lectin PA-IIL, ...
著者Personne, H, Stocker, A, Reymond, J.-L.
登録日2022-08-05
公開日2023-05-31
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (1.29 Å)
主引用文献To Fold or Not to Fold: Diastereomeric Optimization of an alpha-Helical Antimicrobial Peptide.
J.Med.Chem., 66, 2023
8AOO
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BU of 8aoo by Molmil
Fucosylated mixed-chirality linear peptide FHP31 bound to the fucose binding lectin LecB PA-IIL from Pseudomonas aeruginosa at 1.2 Angstrom resolution.
分子名称: 3,7-anhydro-2,8-dideoxy-L-glycero-D-gluco-octonic acid, CALCIUM ION, Fucose-binding lectin PA-IIL, ...
著者Personne, H, Stocker, A, Reymond, J.-L.
登録日2022-08-08
公開日2023-05-31
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (1.18 Å)
主引用文献To Fold or Not to Fold: Diastereomeric Optimization of an alpha-Helical Antimicrobial Peptide.
J.Med.Chem., 66, 2023
8ANR
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BU of 8anr by Molmil
Fucosylated alternate chirality linear peptide FHP30 bound to the fucose binding lectin LecB PA-IIL from Pseudomonas aeruginosa at 1.6 Angstrom resolution.
分子名称: 3,7-anhydro-2,8-dideoxy-L-glycero-D-gluco-octonic acid, CALCIUM ION, Fucose-binding lectin PA-IIL, ...
著者Personne, H, Stocker, A, Reymond, J.-L.
登録日2022-08-05
公開日2023-05-31
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (1.62 Å)
主引用文献To Fold or Not to Fold: Diastereomeric Optimization of an alpha-Helical Antimicrobial Peptide.
J.Med.Chem., 66, 2023
8AN9
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BU of 8an9 by Molmil
Fucosylated mixed-chirality linear peptide FHP5 bound to the fucose binding lectin LecB PA-IIL from Pseudomonas aeruginosa at 1.3 Angstrom resolution.
分子名称: 3,7-anhydro-2,8-dideoxy-L-glycero-D-gluco-octonic acid, CALCIUM ION, Fucose-binding lectin PA-IIL, ...
著者Personne, H, Stocker, A, Reymond, J.-L.
登録日2022-08-04
公開日2023-05-31
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (1.273 Å)
主引用文献To Fold or Not to Fold: Diastereomeric Optimization of an alpha-Helical Antimicrobial Peptide.
J.Med.Chem., 66, 2023

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件を2024-07-24に公開中

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