3G80
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![BU of 3g80 by Molmil](/molmil-images/mine/3g80) | |
3U7T
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![BU of 3u7t by Molmil](/molmil-images/mine/3u7t) | |
4FC1
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![BU of 4fc1 by Molmil](/molmil-images/mine/4fc1) | |
2BCE
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![BU of 2bce by Molmil](/molmil-images/mine/2bce) | CHOLESTEROL ESTERASE FROM BOS TAURUS | 分子名称: | CHOLESTEROL ESTERASE | 著者 | Chen, J.C.-H, Miercke, L.J.W, Krucinski, J, Starr, J.R, Saenz, G, Wang, X, Spilburg, C.A, Lange, L.G, Ellsworth, J.L, Stroud, R.M. | 登録日 | 1998-01-28 | 公開日 | 1999-02-02 | 最終更新日 | 2023-08-09 | 実験手法 | X-RAY DIFFRACTION (1.6 Å) | 主引用文献 | Structure of bovine pancreatic cholesterol esterase at 1.6 A: novel structural features involved in lipase activation. Biochemistry, 37, 1998
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1EXQ
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![BU of 1exq by Molmil](/molmil-images/mine/1exq) | CRYSTAL STRUCTURE OF THE HIV-1 INTEGRASE CATALYTIC CORE DOMAIN | 分子名称: | CADMIUM ION, CHLORIDE ION, POL POLYPROTEIN, ... | 著者 | Chen, J.C.-H, Krucinski, J, Miercke, L.J.W, Finer-Moore, J.S, Tang, A.H, Leavitt, A.D, Stroud, R.M. | 登録日 | 2000-05-03 | 公開日 | 2000-11-03 | 最終更新日 | 2024-02-07 | 実験手法 | X-RAY DIFFRACTION (1.6 Å) | 主引用文献 | Crystal structure of the HIV-1 integrase catalytic core and C-terminal domains: a model for viral DNA binding. Proc.Natl.Acad.Sci.USA, 97, 2000
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1EX4
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![BU of 1ex4 by Molmil](/molmil-images/mine/1ex4) | HIV-1 INTEGRASE CATALYTIC CORE AND C-TERMINAL DOMAIN | 分子名称: | 3-[(3-CHOLAMIDOPROPYL)DIMETHYLAMMONIO]-1-PROPANESULFONATE, INTEGRASE | 著者 | Chen, J.C.-H, Krucinski, J, Miercke, L.J.W, Finer-Moore, J.S, Tang, A.H, Leavitt, A.D, Stroud, R.M. | 登録日 | 2000-04-28 | 公開日 | 2000-06-07 | 最終更新日 | 2024-02-07 | 実験手法 | X-RAY DIFFRACTION (2.8 Å) | 主引用文献 | Crystal structure of the HIV-1 integrase catalytic core and C-terminal domains: a model for viral DNA binding. Proc.Natl.Acad.Sci.USA, 97, 2000
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3KGG
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![BU of 3kgg by Molmil](/molmil-images/mine/3kgg) | X-ray structure of perdeuterated diisopropyl fluorophosphatase (DFPase): Perdeuteration of proteins for neutron diffraction | 分子名称: | CALCIUM ION, Diisopropyl-fluorophosphatase | 著者 | Blum, M.-M, Tomanicek, S.J, John, H, Hanson, B.L, terjans, H.R, Schoenborn, B.P, Langan, P, Chen, J.C.-H. | 登録日 | 2009-10-29 | 公開日 | 2010-04-07 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | X-ray structure of perdeuterated diisopropyl fluorophosphatase (DFPase): perdeuteration of proteins for neutron diffraction. Acta Crystallogr.,Sect.F, 66, 2010
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3LI5
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![BU of 3li5 by Molmil](/molmil-images/mine/3li5) | Diisopropyl fluorophosphatase (DFPase), E21Q,N120D,N175D,D229N mutant | 分子名称: | 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, CALCIUM ION, Diisopropyl-fluorophosphatase | 著者 | Chen, J.C.-H. | 登録日 | 2010-01-24 | 公開日 | 2010-04-07 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (1.36 Å) | 主引用文献 | Structural characterization of the catalytic calcium-binding site in diisopropyl fluorophosphatase (DFPase)-Comparison with related beta-propeller enzymes. Chem.Biol.Interact, 187, 2010
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1OSF
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![BU of 1osf by Molmil](/molmil-images/mine/1osf) | Human Hsp90 in complex with 17-desmethoxy-17-N,N-Dimethylaminoethylamino-Geldanamycin | 分子名称: | (4S)-2-METHYL-2,4-PENTANEDIOL, 17-DESMETHOXY-17-N,N-DIMETHYLAMINOETHYLAMINO-GELDANAMYCIN, ACETIC ACID, ... | 著者 | Jez, J.M, Chen, J.C.-H, Rastelli, G, Stroud, R.M, Santi, D.V. | 登録日 | 2003-03-19 | 公開日 | 2003-05-27 | 最終更新日 | 2024-02-14 | 実験手法 | X-RAY DIFFRACTION (1.75 Å) | 主引用文献 | Crystal Structure and Molecular Modeling of 17-DMAG in Complex with Human Hsp90 Chem.Biol., 10, 2003
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3BYC
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![BU of 3byc by Molmil](/molmil-images/mine/3byc) | Joint neutron and X-ray structure of diisopropyl fluorophosphatase. Deuterium occupancies are 1-Q, where Q is occupancy of H | 分子名称: | CALCIUM ION, Diisopropyl-fluorophosphatase | 著者 | Blum, M.-M, Mustyakimov, M, Ruterjans, H, Schoenborn, B.P, Langan, P, Chen, J.C.-H. | 登録日 | 2008-01-15 | 公開日 | 2009-01-27 | 最終更新日 | 2024-02-21 | 実験手法 | NEUTRON DIFFRACTION (2.2 Å), X-RAY DIFFRACTION | 主引用文献 | Rapid determination of hydrogen positions and protonation states of diisopropyl fluorophosphatase by joint neutron and X-ray diffraction refinement. Proc.Natl.Acad.Sci.Usa, 106, 2009
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5VG0
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![BU of 5vg0 by Molmil](/molmil-images/mine/5vg0) | |
3HLI
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![BU of 3hli by Molmil](/molmil-images/mine/3hli) | |
3HLH
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![BU of 3hlh by Molmil](/molmil-images/mine/3hlh) | |
5VG1
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![BU of 5vg1 by Molmil](/molmil-images/mine/5vg1) | |
1KEZ
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![BU of 1kez by Molmil](/molmil-images/mine/1kez) | Crystal Structure of the Macrocycle-forming Thioesterase Domain of Erythromycin Polyketide Synthase (DEBS TE) | 分子名称: | ERYTHRONOLIDE SYNTHASE | 著者 | Tsai, S.-C, Miercke, L.J.W, Krucinski, J, Gokhale, R, Chen, J.C.-H, Foster, P.G, Cane, D.E, Khosla, C, Stroud, R.M. | 登録日 | 2001-11-19 | 公開日 | 2002-01-09 | 最終更新日 | 2024-02-07 | 実験手法 | X-RAY DIFFRACTION (2.8 Å) | 主引用文献 | Crystal structure of the macrocycle-forming thioesterase domain of the erythromycin polyketide synthase: versatility from a unique substrate channel. Proc.Natl.Acad.Sci.USA, 98, 2001
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2GVV
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![BU of 2gvv by Molmil](/molmil-images/mine/2gvv) | |
2GVU
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![BU of 2gvu by Molmil](/molmil-images/mine/2gvu) | |
2GVW
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![BU of 2gvw by Molmil](/molmil-images/mine/2gvw) | |
3LI4
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![BU of 3li4 by Molmil](/molmil-images/mine/3li4) | Diisopropyl fluorophosphatase (DFPase), N120D,N175D,D229N mutant | 分子名称: | CALCIUM ION, Diisopropyl-fluorophosphatase | 著者 | Chen, J.C.-H. | 登録日 | 2010-01-24 | 公開日 | 2010-04-07 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (1.35 Å) | 主引用文献 | Structural characterization of the catalytic calcium-binding site in diisopropyl fluorophosphatase (DFPase)-Comparison with related beta-propeller enzymes. Chem.Biol.Interact, 187, 2010
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3LI3
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![BU of 3li3 by Molmil](/molmil-images/mine/3li3) | Diisopropyl fluorophosphatase (DFPase), D121E mutant | 分子名称: | CALCIUM ION, Diisopropyl-fluorophosphatase | 著者 | Chen, J.C.-H. | 登録日 | 2010-01-24 | 公開日 | 2010-04-07 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (1.66 Å) | 主引用文献 | Structural characterization of the catalytic calcium-binding site in diisopropyl fluorophosphatase (DFPase)-Comparison with related beta-propeller enzymes. Chem.Biol.Interact, 187, 2010
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6LN1
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![BU of 6ln1 by Molmil](/molmil-images/mine/6ln1) | A natural inhibitor of DYRK1A for treatment of diabetes mellitus | 分子名称: | 1,3,5,8-tetrakis(oxidanyl)xanthen-9-one, Dual specificity tyrosine-phosphorylation-regulated kinase 1A | 著者 | Li, H, Chen, L.X, Zheng, M.Z, Zhang, Q.Z, Zhang, C.L, Wu, C.R, Yang, K.Y, Song, Z.R, Wang, Q.Q, Li, C, Zhou, Y.R, Chen, J.C. | 登録日 | 2019-12-28 | 公開日 | 2021-10-06 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (2.699 Å) | 主引用文献 | A natural DYRK1A inhibitor as a potential stimulator for beta-cell proliferation in diabetes. Clin Transl Med, 11, 2021
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2NUB
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![BU of 2nub by Molmil](/molmil-images/mine/2nub) | Structure of Aquifex aeolicus Argonuate | 分子名称: | Argonaute | 著者 | Rashid, U.J, Paterok, D, Koglin, A, Gohlke, H, Piehler, J, Chen, J.C.-H. | 登録日 | 2006-11-09 | 公開日 | 2007-02-06 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (3.2 Å) | 主引用文献 | Structure of Aquifex aeolicus argonaute highlights conformational flexibility of the PAZ domain as a potential regulator of RNA-induced silencing complex function. J.Biol.Chem., 282, 2007
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5VLM
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![BU of 5vlm by Molmil](/molmil-images/mine/5vlm) | Crystal structure of EilR in complex with crystal violet | 分子名称: | CRYSTAL VIOLET, Regulatory protein TetR | 著者 | Pereira, J.H, Ruegg, T.L, Chen, J, Novichkov, P, DeGiovani, A, Tomaleri, G.P, Singer, S, Simmons, B, Thelen, M, Adams, P.D. | 登録日 | 2017-04-25 | 公開日 | 2018-06-27 | 最終更新日 | 2024-03-13 | 実験手法 | X-RAY DIFFRACTION (3.403 Å) | 主引用文献 | Jungle Express is a versatile repressor system for tight transcriptional control. Nat Commun, 9, 2018
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5VL9
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![BU of 5vl9 by Molmil](/molmil-images/mine/5vl9) | Crystal structure of EilR in complex with eilO DNA element | 分子名称: | DNA (5'-D(*GP*AP*AP*AP*GP*TP*TP*GP*GP*AP*CP*AP*TP*A)-3'), DNA (5'-D(*TP*AP*TP*GP*TP*CP*CP*AP*AP*CP*TP*TP*TP*C)-3'), HEXANE-1,6-DIOL, ... | 著者 | Pereira, J.H, Ruegg, T.L, Chen, J, Novichkov, P, DeGiovani, A, Tomaleri, G.P, Singer, S, Simmons, B, Thelen, M, Adams, P.D. | 登録日 | 2017-04-25 | 公開日 | 2018-06-27 | 最終更新日 | 2022-03-16 | 実験手法 | X-RAY DIFFRACTION (2.16 Å) | 主引用文献 | Jungle Express is a versatile repressor system for tight transcriptional control. Nat Commun, 9, 2018
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5VLG
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![BU of 5vlg by Molmil](/molmil-images/mine/5vlg) | Crystal structure of EilR in complex with malachite green | 分子名称: | MALACHITE GREEN, Regulatory protein TetR | 著者 | Pereira, J.H, Ruegg, T.L, Chen, J, Novichkov, P, DeGiovani, A, Tomaleri, G.P, Singer, S, Simmons, B, Thelen, M, Adams, P.D. | 登録日 | 2017-04-25 | 公開日 | 2018-06-27 | 最終更新日 | 2024-03-13 | 実験手法 | X-RAY DIFFRACTION (2.932 Å) | 主引用文献 | Jungle Express is a versatile repressor system for tight transcriptional control. Nat Commun, 9, 2018
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