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2SBL
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BU of 2sbl by Molmil
THE THREE-DIMENSIONAL STRUCTURE OF AN ARACHIDONIC ACID 15-LIPOXYGENASE
分子名称: FE (III) ION, LIPOXYGENASE-1
著者Amzel, L.M, Boyington, J.C.
登録日1993-07-22
公開日1995-02-27
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献The three-dimensional structure of an arachidonic acid 15-lipoxygenase.
Science, 260, 1993
1A78
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BU of 1a78 by Molmil
COMPLEX OF TOAD OVARY GALECTIN WITH THIO-DIGALACTOSE
分子名称: 2,3-DIHYDROXY-1,4-DITHIOBUTANE, GALECTIN-1, beta-D-galactopyranose-(1-1)-1-thio-beta-D-galactopyranose
著者Amzel, L.M, Bianchet, M.A, Ahmed, H, Vasta, G.R.
登録日1998-03-20
公開日1998-10-14
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Soluble beta-galactosyl-binding lectin (galectin) from toad ovary: crystallographic studies of two protein-sugar complexes
Proteins, 40, 2000
1GAN
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BU of 1gan by Molmil
COMPLEX OF TOAD OVARY GALECTIN WITH N-ACETYLGALACTOSE
分子名称: GALECTIN-1, beta-D-galactopyranose-(1-4)-2-acetamido-2-deoxy-alpha-D-glucopyranose
著者Amzel, L.M, Bianchet, M.A, Ahmed, H, Vasta, G.R.
登録日1996-11-06
公開日1997-09-04
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (2.23 Å)
主引用文献Soluble beta-galactosyl-binding lectin (galectin) from toad ovary: crystallographic studies of two protein-sugar complexes.
Proteins, 40, 2000
3HHM
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BU of 3hhm by Molmil
Crystal structure of p110alpha H1047R mutant in complex with niSH2 of p85alpha and the drug wortmannin
分子名称: (1S,6BR,9AS,11R,11BR)-9A,11B-DIMETHYL-1-[(METHYLOXY)METHYL]-3,6,9-TRIOXO-1,6,6B,7,8,9,9A,10,11,11B-DECAHYDRO-3H-FURO[4, 3,2-DE]INDENO[4,5-H][2]BENZOPYRAN-11-YL ACETATE, Phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit alpha isoform, ...
著者Amzel, L.M, Vogelstein, B, Gabelli, S.B, Mandelker, D.
登録日2009-05-15
公開日2009-09-29
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献A frequent kinase domain mutation that changes the interaction between PI3K{alpha} and the membrane.
Proc.Natl.Acad.Sci.USA, 106, 2009
3HIZ
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BU of 3hiz by Molmil
Crystal structure of p110alpha H1047R mutant in complex with niSH2 of p85alpha
分子名称: Phosphatidylinositol 3-kinase regulatory subunit alpha, Phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit alpha isoform
著者Amzel, L.M, Vogelstein, B, Gabelli, S.B, Mandelker, D.
登録日2009-05-20
公開日2009-09-29
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (3.3 Å)
主引用文献A frequent kinase domain mutation that changes the interaction between PI3K{alpha} and the membrane.
Proc.Natl.Acad.Sci.USA, 106, 2009
3ID0
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BU of 3id0 by Molmil
Trypanosoma cruzi farnesyl diphosphate synthase homodimer in complex with 3-Fluoro-1-(2-hydroxy-2,2-bisphosphono-ethyl)pyridinium
分子名称: 3-FLUORO-1-(2-HYDROXY-2,2-DIPHOSPHONOETHYL)PYRIDINIUM, Farnesyl pyrophosphate synthase, MAGNESIUM ION, ...
著者Amzel, L.M, Huang, C.H, Gabelli, S.B, Oldfield, E.
登録日2009-07-19
公開日2010-02-09
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (2.81 Å)
主引用文献Binding of nitrogen-containing bisphosphonates (N-BPs) to the Trypanosoma cruzi farnesyl diphosphate synthase homodimer.
Proteins, 78, 2010
3ICZ
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BU of 3icz by Molmil
Trypanosoma cruzi farnesyl diphosphate synthase homodimer in complex with 1-(2,2-Bis-phosphono-ethyl)-3-butyl-pyridinium and isopentenyl pyrophosphate
分子名称: 3-METHYLBUT-3-ENYL TRIHYDROGEN DIPHOSPHATE, 3-[(1E)-but-1-en-1-yl]-1-(2,2-diphosphonoethyl)pyridinium, Farnesyl pyrophosphate synthase, ...
著者Amzel, L.M, Huang, C.H, Gabelli, S.B, Oldfield, E.
登録日2009-07-19
公開日2010-02-09
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (2.15 Å)
主引用文献Binding of nitrogen-containing bisphosphonates (N-BPs) to the Trypanosoma cruzi farnesyl diphosphate synthase homodimer.
Proteins, 78, 2010
3IBA
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BU of 3iba by Molmil
Crystal structure of the complex of Trypanosoma cruzi farnesyl diphosphate synthase with zoledronate, IPP and Mg2+
分子名称: 3-METHYLBUT-3-ENYL TRIHYDROGEN DIPHOSPHATE, Farnesyl pyrophosphate synthase, MAGNESIUM ION, ...
著者Amzel, L.M, Huang, C.H, Gabelli, S.B, Oldfield, E.
登録日2009-07-15
公開日2010-02-09
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Binding of nitrogen-containing bisphosphonates (N-BPs) to the Trypanosoma cruzi farnesyl diphosphate synthase homodimer.
Proteins, 78, 2010
3ICK
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BU of 3ick by Molmil
Trypanosoma cruzi farnesyl diphosphate synthase homodimer in complex with minodronate and isopentenyl disphosphate
分子名称: (1-HYDROXY-2-IMIDAZO[1,2-A]PYRIDIN-3-YLETHANE-1,1-DIYL)BIS(PHOSPHONIC ACID), 3-METHYLBUT-3-ENYL TRIHYDROGEN DIPHOSPHATE, ACETIC ACID, ...
著者Amzel, L.M, Huang, C.H, Gabelli, S.B, Oldfield, E.
登録日2009-07-17
公開日2010-02-09
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Binding of nitrogen-containing bisphosphonates (N-BPs) to the Trypanosoma cruzi farnesyl diphosphate synthase homodimer.
Proteins, 78, 2010
3ICN
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BU of 3icn by Molmil
Trypanosoma cruzi farnesyl diphosphate synthase homodimer in complex with isopentenyl pyrophosphate and 3-Fluoro-1-(2-hydroxy-2,2-bis-phosphono-ethyl)-pyridinium
分子名称: 3-FLUORO-1-(2-HYDROXY-2,2-DIPHOSPHONOETHYL)PYRIDINIUM, 3-METHYLBUT-3-ENYL TRIHYDROGEN DIPHOSPHATE, Farnesyl pyrophosphate synthase, ...
著者Amzel, L.M, Huang, C.H, Gabelli, S.B, Oldfield, E.
登録日2009-07-17
公開日2010-02-09
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Binding of nitrogen-containing bisphosphonates (N-BPs) to the Trypanosoma cruzi farnesyl diphosphate synthase homodimer.
Proteins, 78, 2010
3ICM
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BU of 3icm by Molmil
Trypanosoma cruzi farnesyl diphosphate synthase homodimer in complex with isopentenyl pyrophosphate, Mg2+ and 1-(2-Hydroxy-2,2-bis-phosphono-ethyl)-3-phenyl-pyridinium
分子名称: 1-(2-hydroxy-2,2-diphosphonoethyl)-3-phenylpyridinium, 3-METHYLBUT-3-ENYL TRIHYDROGEN DIPHOSPHATE, Farnesyl pyrophosphate synthase, ...
著者Amzel, L.M, Huang, C.H, Gabelli, S.B, Oldfield, E.
登録日2009-07-17
公開日2010-02-09
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Binding of nitrogen-containing bisphosphonates (N-BPs) to the Trypanosoma cruzi farnesyl diphosphate synthase homodimer.
Proteins, 78, 2010
1PBO
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BU of 1pbo by Molmil
COMPLEX OF BOVINE ODORANT BINDING PROTEIN (OBP) WITH A SELENIUM CONTAINING ODORANT
分子名称: 4-butyl-5-propyl-1,3-selenazol-2-amine, ODORANT BINDING PROTEIN
著者Amzel, L.M, Bianchet, M.A, Monaco, H, Bains, G.
登録日1996-07-15
公開日1997-07-23
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献The three-dimensional structure of bovine odorant binding protein and its mechanism of odor recognition.
Nat.Struct.Biol., 3, 1996
3O6Z
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BU of 3o6z by Molmil
Structure of the D152A E.coli GDP-mannose hydrolase (yffh) in complex with Mg++
分子名称: 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, CHLORIDE ION, DI(HYDROXYETHYL)ETHER, ...
著者Amzel, L.M, Gabelli, S.B, Boto, A.N.
登録日2010-07-29
公開日2011-05-11
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (2.05 Å)
主引用文献Structural studies of the Nudix GDP-mannose hydrolase from E. coli reveals a new motif for mannose recognition.
Proteins, 79, 2011
3O69
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BU of 3o69 by Molmil
Structure of the E100A E.coli GDP-mannose hydrolase (yffh) in complex with Mg++
分子名称: CHLORIDE ION, DI(HYDROXYETHYL)ETHER, GDP-mannose pyrophosphatase nudK, ...
著者Amzel, L.M, Gabelli, S.B, Boto, A.N.
登録日2010-07-28
公開日2011-05-11
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Structural studies of the Nudix GDP-mannose hydrolase from E. coli reveals a new motif for mannose recognition.
Proteins, 79, 2011
3O61
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BU of 3o61 by Molmil
Structure of the E100A E.coli GDP-mannose hydrolase (yffh) in complex with GDP-mannose and Mg++
分子名称: CHLORIDE ION, GDP-mannose pyrophosphatase nudK, GUANOSINE-5'-DIPHOSPHATE-ALPHA-D-MANNOSE, ...
著者Amzel, L.M, Gabelli, S.B, Boto, A.N.
登録日2010-07-28
公開日2011-05-11
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (2.45 Å)
主引用文献Structural studies of the Nudix GDP-mannose hydrolase from E. coli reveals a new motif for mannose recognition.
Proteins, 79, 2011
3O52
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BU of 3o52 by Molmil
Structure of the E.coli GDP-mannose hydrolase (yffh) in complex with tartrate
分子名称: CHLORIDE ION, D(-)-TARTARIC ACID, GDP-mannose pyrophosphatase nudK, ...
著者Amzel, L.M, Gabelli, S.B, Boto, A.N.
登録日2010-07-27
公開日2011-05-11
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Structural studies of the Nudix GDP-mannose hydrolase from E. coli reveals a new motif for mannose recognition.
Proteins, 79, 2011
6MBA
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BU of 6mba by Molmil
Crystal Structure of Human Nav1.4 CTerminal Domain in Complex with apo Calmodulin
分子名称: 1,2-ETHANEDIOL, 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, CARBONATE ION, ...
著者Yoder, J, Gabelli, S.B, Amzel, L.M.
登録日2018-08-29
公開日2019-04-10
最終更新日2023-10-11
実験手法X-RAY DIFFRACTION (1.799 Å)
主引用文献Ca2+-dependent regulation of sodium channels NaV1.4 and NaV1.5 is controlled by the post-IQ motif.
Nat Commun, 10, 2019
6ALA
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BU of 6ala by Molmil
Crystal structure of H108A peptidylglycine alpha-hydroxylating monooxygenase (PHM) in complex with citrate
分子名称: CITRATE ANION, COPPER (II) ION, GLYCEROL, ...
著者Maheshwari, S, Rudzka, K, Gabelli, S.B, Amzel, L.M.
登録日2017-08-07
公開日2018-07-18
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (2.59 Å)
主引用文献Effects of copper occupancy on the conformational landscape of peptidylglycine alpha-hydroxylating monooxygenase.
Commun Biol, 1, 2018
6E0T
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BU of 6e0t by Molmil
C-terminal domain of Fission Yeast OFD1
分子名称: Prolyl 3,4-dihydroxylase ofd1
著者Bianchet, M.A, Amzel, L.M, Espenshade, P.J, Yeh, T.
登録日2018-07-06
公開日2019-09-11
最終更新日2024-03-13
実験手法X-RAY DIFFRACTION (2.02 Å)
主引用文献The hypoxic regulator of sterol synthesis nro1 is a nuclear import adaptor.
Structure, 19, 2011
3U1P
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BU of 3u1p by Molmil
Crystal Structure of M. tuberculosis LD-transpeptidase type 2 with Modified Catalytic Cysteine (C354)
分子名称: DI(HYDROXYETHYL)ETHER, Mycobacteria Tuberculosis LD-transpeptidase type 2
著者Erdemli, S, Bianchet, M.A, Gupta, R, Lamichhane, G, Amzel, L.M.
登録日2011-09-30
公開日2012-12-05
最終更新日2018-04-04
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献Targeting the Cell Wall of Mycobacterium tuberculosis: Structure and Mechanism of L,D-Transpeptidase 2.
Structure, 20, 2012
3TX4
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BU of 3tx4 by Molmil
Crystal Structure of Mutant (C354A) M. tuberculosis LD-transpeptidase type 2
分子名称: Mycobacterium Tuberculosis LD-transpeptidase type 2
著者Erdemli, S, Bianchet, M.A, Gupta, R, Lamichhane, G, Amzel, L.M.
登録日2011-09-22
公開日2012-12-05
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (2.32 Å)
主引用文献Targeting the Cell Wall of Mycobacterium tuberculosis: Structure and Mechanism of L,D-Transpeptidase 2.
Structure, 20, 2012
1MAB
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BU of 1mab by Molmil
RAT LIVER F1-ATPASE
分子名称: ADENOSINE-5'-DIPHOSPHATE, ADENOSINE-5'-TRIPHOSPHATE, MAGNESIUM ION, ...
著者Bianchet, M.A, Amzel, L.M.
登録日1998-08-06
公開日1998-09-30
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献The 2.8-A structure of rat liver F1-ATPase: configuration of a critical intermediate in ATP synthesis/hydrolysis.
Proc.Natl.Acad.Sci.USA, 95, 1998
4TXI
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BU of 4txi by Molmil
Construct of MICAL-1 containing the monooxygenase and calponin homology domains
分子名称: CHLORIDE ION, DI(HYDROXYETHYL)ETHER, FLAVIN-ADENINE DINUCLEOTIDE, ...
著者Alqassim, S.S, Amzel, L.M, Bianchet, M.A.
登録日2014-07-03
公開日2016-01-13
最終更新日2023-12-27
実験手法X-RAY DIFFRACTION (2.309 Å)
主引用文献Modulation of MICAL Monooxygenase Activity by its Calponin Homology Domain: Structural and Mechanistic Insights.
Sci Rep, 6, 2016
4TXK
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BU of 4txk by Molmil
Construct of MICAL-1 containing the monooxygenase and calponin homology domains
分子名称: DI(HYDROXYETHYL)ETHER, FLAVIN-ADENINE DINUCLEOTIDE, Protein-methionine sulfoxide oxidase MICAL1
著者Alqassim, S.S, Amzel, L.M, Bianchet, M.A.
登録日2014-07-03
公開日2015-12-23
最終更新日2023-12-27
実験手法X-RAY DIFFRACTION (2.878 Å)
主引用文献Structural insights into modulation of MICAL activity by its Calponin Homology (CH) domain
To Be Published
3VAE
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BU of 3vae by Molmil
Crystal Structure of M. tuberculosis LD-transpeptidase type 2 with Modified Catalytic Cysteine (C354)
分子名称: DI(HYDROXYETHYL)ETHER, LD-transpeptidase type 2
著者Erdemli, S, Bianchet, M.A, Gupta, R, Lamichhane, G, Amzel, L.M.
登録日2011-12-29
公開日2012-12-12
最終更新日2018-04-04
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献Targeting the Cell Wall of Mycobacterium tuberculosis: Structure and Mechanism of L,D-Transpeptidase 2.
Structure, 20, 2012

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