2MT4
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4NJC
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2VY9
| Molecular architecture of the stressosome, a signal integration and transduction hub | 分子名称: | ANTI-SIGMA-FACTOR ANTAGONIST | 著者 | Marles-Wright, J, Grant, T, Delumeau, O, van Duinen, G, Firbank, S.J, Lewis, P.J, Murray, J.W, Newman, J.A, Quin, M.B, Race, P.R, Rohou, A, Tichelaar, W, van Heel, M, Lewis, R.J. | 登録日 | 2008-07-21 | 公開日 | 2008-10-14 | 最終更新日 | 2024-10-16 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Molecular Architecture of the "Stressosome," a Signal Integration and Transduction Hub Science, 322, 2008
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1S9G
| CRYSTAL STRUCTURE OF HIV-1 REVERSE TRANSCRIPTASE (RT) IN COMPLEX WITH JANSSEN-R120394. | 分子名称: | 4-[4-AMINO-6-(5-CHLORO-1H-INDOL-4-YLMETHYL)-[1,3,5]TRIAZIN-2-YLAMINO]-BENZONITRILE, POL polyprotein [Contains: Reverse transcriptase] | 著者 | Das, K, Clark Jr, A.D, Ludovici, D.W, Kukla, M.J, Decorte, B, Lewi, P.J, Hughes, S.H, Janssen, P.A, Arnold, E. | 登録日 | 2004-02-04 | 公開日 | 2004-05-11 | 最終更新日 | 2024-02-14 | 実験手法 | X-RAY DIFFRACTION (2.8 Å) | 主引用文献 | Roles of Conformational and Positional Adaptability in Structure-Based Design of TMC125-R165335 (Etravirine) and Related Non-nucleoside Reverse Transcriptase Inhibitors That Are Highly Potent and Effective against Wild-Type and Drug-Resistant HIV-1 Variants. J.Med.Chem., 47, 2004
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1S9E
| CRYSTAL STRUCTURE OF HIV-1 REVERSE TRANSCRIPTASE (RT) IN COMPLEX WITH JANSSEN-R129385 | 分子名称: | 4-[4-AMINO-6-(2,6-DICHLORO-PHENOXY)-[1,3,5]TRIAZIN-2-YLAMINO]-BENZONITRILE, POL polyprotein [Contains: Reverse transcriptase], POL polyprotein [Contains:Reverse transcriptase] | 著者 | Das, K, Clark Jr, A.D, Ludovici, D.W, Kukla, M.J, Decorte, B, Lewi, P.J, Hughes, S.H, Janssen, P.A, Arnold, E. | 登録日 | 2004-02-04 | 公開日 | 2004-05-11 | 最終更新日 | 2024-02-14 | 実験手法 | X-RAY DIFFRACTION (2.6 Å) | 主引用文献 | Roles of Conformational and Positional Adaptability in Structure-Based Design of TMC125-R165335 (Etravirine) and Related Non-nucleoside Reverse Transcriptase Inhibitors That Are Highly Potent and Effective against Wild-Type and Drug-Resistant HIV-1 Variants. J.Med.Chem., 47, 2004
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4OVG
| E. coli sliding clamp in complex with (R)-9-(2-amino-2-oxoethyl)-6-chloro-2,3,4,9-tetrahydro-1H-carbazole-2-carboxylic acid | 分子名称: | (2R)-9-(2-amino-2-oxoethyl)-6-chloro-2,3,4,9-tetrahydro-1H-carbazole-2-carboxylic acid, 1,2-ETHANEDIOL, CALCIUM ION, ... | 著者 | Yin, Z, Oakley, A.J. | 登録日 | 2014-02-21 | 公開日 | 2014-03-05 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Bacterial Sliding Clamp Inhibitors that Mimic the Sequential Binding Mechanism of Endogenous Linear Motifs. J.Med.Chem., 58, 2015
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2LY7
| B-flap domain of RNA polymerase (B. subtilis) | 分子名称: | DNA-directed RNA polymerase subunit beta | 著者 | Mobli, M. | 登録日 | 2012-09-12 | 公開日 | 2014-03-12 | 最終更新日 | 2024-05-15 | 実験手法 | SOLUTION NMR | 主引用文献 | RNA polymerase-induced remodelling of NusA produces a pause enhancement complex. Nucleic Acids Res., 43, 2015
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4U6N
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6WVJ
| Cryo-EM structure of Bacillus subtilis RNA Polymerase elongation complex | 分子名称: | DNA (5'-D(*TP*GP*TP*CP*GP*GP*GP*CP*GP*TP*CP*CP*GP*CP*GP*CP*GP*CP*C)-3'), DNA (5'-D(P*AP*CP*GP*CP*CP*CP*GP*AP*CP*A)-3'), DNA-directed RNA polymerase subunit alpha, ... | 著者 | Newing, T, Tolun, G, Oakley, A.J. | 登録日 | 2020-05-06 | 公開日 | 2020-11-18 | 最終更新日 | 2024-05-29 | 実験手法 | ELECTRON MICROSCOPY (3.36 Å) | 主引用文献 | Molecular basis for RNA polymerase-dependent transcription complex recycling by the helicase-like motor protein HelD. Nat Commun, 11, 2020
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6WVK
| Cryo-EM structure of Bacillus subtilis RNA Polymerase in complex with HelD | 分子名称: | DNA helicase IV, DNA-directed RNA polymerase subunit alpha, DNA-directed RNA polymerase subunit beta, ... | 著者 | Newing, T, Tolun, G, Oakley, A.J. | 登録日 | 2020-05-06 | 公開日 | 2020-11-18 | 最終更新日 | 2024-05-29 | 実験手法 | ELECTRON MICROSCOPY (3.36 Å) | 主引用文献 | Molecular basis for RNA polymerase-dependent transcription complex recycling by the helicase-like motor protein HelD. Nat Commun, 11, 2020
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7SSG
| Mfd DNA complex | 分子名称: | DNA (5'-D(P*TP*GP*GP*CP*GP*GP*CP*GP*AP*GP*GP*C)-3'), DNA (5'-D(P*TP*TP*GP*CP*CP*TP*CP*GP*CP*TP*GP*CP*CP*A)-3'), Transcription-repair-coupling factor | 著者 | Oakley, A.J, Xu, Z.-Q. | 登録日 | 2021-11-11 | 公開日 | 2022-05-25 | 最終更新日 | 2024-06-05 | 実験手法 | ELECTRON MICROSCOPY (5.2 Å) | 主引用文献 | Mechanism of transcription modulation by the transcription-repair coupling factor. Nucleic Acids Res., 50, 2022
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8GJ3
| E. coli clamp loader on primed template DNA | 分子名称: | ADENOSINE-5'-DIPHOSPHATE, DNA polymerase III subunit delta, DNA polymerase III subunit delta', ... | 著者 | Oakley, A.J, Xu, Z.-Q, Dixon, N.E. | 登録日 | 2023-03-14 | 公開日 | 2024-03-27 | 最終更新日 | 2024-10-16 | 実験手法 | ELECTRON MICROSCOPY (2.8 Å) | 主引用文献 | Structural characterisation of the complete cycle of sliding clamp loading in Escherichia coli. Nat Commun, 15, 2024
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8GJ1
| E. coli clamp loader with open clamp on primed template DNA (form 2) | 分子名称: | ADENOSINE-5'-DIPHOSPHATE, Beta sliding clamp, DNA polymerase III subunit delta, ... | 著者 | Oakley, A.J, Xu, Z.-Q, Dixon, N.E. | 登録日 | 2023-03-14 | 公開日 | 2024-03-27 | 最終更新日 | 2024-10-16 | 実験手法 | ELECTRON MICROSCOPY (3 Å) | 主引用文献 | Structural characterisation of the complete cycle of sliding clamp loading in Escherichia coli. Nat Commun, 15, 2024
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8GIZ
| E. coli clamp loader with open clamp | 分子名称: | Beta sliding clamp, DNA polymerase III subunit delta, DNA polymerase III subunit delta', ... | 著者 | Oakley, A.J, Xu, Z.-Q, Dixon, N.E. | 登録日 | 2023-03-14 | 公開日 | 2024-03-27 | 最終更新日 | 2024-10-16 | 実験手法 | ELECTRON MICROSCOPY (2.7 Å) | 主引用文献 | Structural characterisation of the complete cycle of sliding clamp loading in Escherichia coli. Nat Commun, 15, 2024
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8GIY
| E. coli clamp loader with closed clamp | 分子名称: | Beta sliding clamp, DNA polymerase III subunit delta, DNA polymerase III subunit delta', ... | 著者 | Oakley, A.J, Xu, Z.-Q, Dixon, N.E. | 登録日 | 2023-03-14 | 公開日 | 2024-03-27 | 最終更新日 | 2024-10-16 | 実験手法 | ELECTRON MICROSCOPY (3.7 Å) | 主引用文献 | Structural characterisation of the complete cycle of sliding clamp loading in Escherichia coli. Nat Commun, 15, 2024
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8GJ2
| E. coli clamp loader with closed clamp on primed template DNA | 分子名称: | ADENOSINE-5'-DIPHOSPHATE, Beta sliding clamp, DNA polymerase III subunit delta, ... | 著者 | Oakley, A.J, Xu, Z.-Q, Dixon, N.E. | 登録日 | 2023-03-14 | 公開日 | 2024-03-27 | 最終更新日 | 2024-10-16 | 実験手法 | ELECTRON MICROSCOPY (2.6 Å) | 主引用文献 | Structural characterisation of the complete cycle of sliding clamp loading in Escherichia coli. Nat Commun, 15, 2024
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8GJ0
| E. coli clamp loader with open clamp on primed template DNA (form 1) | 分子名称: | ADENOSINE-5'-DIPHOSPHATE, Beta sliding clamp, DNA polymerase III subunit delta, ... | 著者 | Oakley, A.J, Xu, Z.-Q, Dixon, N.E. | 登録日 | 2023-03-14 | 公開日 | 2024-03-27 | 最終更新日 | 2024-10-16 | 実験手法 | ELECTRON MICROSCOPY (2.9 Å) | 主引用文献 | Structural characterisation of the complete cycle of sliding clamp loading in Escherichia coli. Nat Commun, 15, 2024
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4OVF
| E. coli sliding clamp in complex with (R)-6-chloro-2,3,4,9-tetrahydro-1H-carbazole-2-carboxylic acid | 分子名称: | (2R)-6-chloro-2,3,4,9-tetrahydro-1H-carbazole-2-carboxylic acid, CALCIUM ION, CHLORIDE ION, ... | 著者 | Yin, Z, Oakley, A.J. | 登録日 | 2014-02-21 | 公開日 | 2014-03-05 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (2.05 Å) | 主引用文献 | Bacterial Sliding Clamp Inhibitors that Mimic the Sequential Binding Mechanism of Endogenous Linear Motifs. J.Med.Chem., 58, 2015
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4OVH
| E. coli sliding clamp in complex with (R)-6-bromo-9-(2-(carboxymethylamino)-2-oxoethyl)-2,3,4,9-tetrahydro-1H-carbazole-2-carboxylic acid | 分子名称: | (2R)-6-bromo-9-{2-[(carboxymethyl)amino]-2-oxoethyl}-2,3,4,9-tetrahydro-1H-carbazole-2-carboxylic acid, CALCIUM ION, CHLORIDE ION, ... | 著者 | Yin, Z, Oakley, A.J. | 登録日 | 2014-02-21 | 公開日 | 2014-03-05 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (2.25 Å) | 主引用文献 | Bacterial Sliding Clamp Inhibitors that Mimic the Sequential Binding Mechanism of Endogenous Linear Motifs. J.Med.Chem., 58, 2015
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5DCF
| C-terminal domain of XerD recombinase in complex with gamma domain of FtsK | 分子名称: | Tyrosine recombinase XerD,DNA translocase FtsK | 著者 | Keller, A.N, Xin, Y, Lowe, J, Grainge, I. | 登録日 | 2015-08-24 | 公開日 | 2016-09-07 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Activation of Xer-recombination at dif: structural basis of the FtsK gamma-XerD interaction. Sci Rep, 6, 2016
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4PNW
| E. coli sliding clamp in complex with (R)-6-bromo-9-(2-((S)-1-carboxy-2-phenylethylamino)-2-oxoethyl)-2,3,4,9-tetrahydro-1H-carbazole-2-carboxylic acid | 分子名称: | (2R)-6-bromo-9-(2-{[(1S)-1-carboxy-2-phenylethyl]amino}-2-oxoethyl)-2,3,4,9-tetrahydro-1H-carbazole-2-carboxylic acid, CALCIUM ION, CHLORIDE ION, ... | 著者 | Yin, Z, Oakley, A.J. | 登録日 | 2014-02-21 | 公開日 | 2014-03-05 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Bacterial Sliding Clamp Inhibitors that Mimic the Sequential Binding Mechanism of Endogenous Linear Motifs. J.Med.Chem., 58, 2015
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4PNU
| E. coli sliding clamp in complex with (R)-6-bromo-9-(2-((R)-1-carboxy-2-phenylethylamino)-2-oxoethyl)-2,3,4,9-tetrahydro-1H-carbazole-2-carboxylic acid | 分子名称: | (2R)-6-bromo-9-(2-{[(1R)-1-carboxy-2-phenylethyl]amino}-2-oxoethyl)-2,3,4,9-tetrahydro-1H-carbazole-2-carboxylic acid, CALCIUM ION, CHLORIDE ION, ... | 著者 | Yin, Z, Oakley, A.J. | 登録日 | 2014-02-21 | 公開日 | 2014-03-05 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Bacterial Sliding Clamp Inhibitors that Mimic the Sequential Binding Mechanism of Endogenous Linear Motifs. J.Med.Chem., 58, 2015
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4PNV
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3BGR
| Crystal structure of K103N/Y181C mutant HIV-1 reverse transcriptase (RT) in complex with TMC278 (Rilpivirine), a non-nucleoside RT inhibitor | 分子名称: | 1,2-ETHANEDIOL, 4-{[4-({4-[(E)-2-cyanoethenyl]-2,6-dimethylphenyl}amino)pyrimidin-2-yl]amino}benzonitrile, Reverse transcriptase/ribonuclease H, ... | 著者 | Das, K, Bauman, J.D, Clark Jr, A.D, Shatkin, A.J, Arnold, E. | 登録日 | 2007-11-27 | 公開日 | 2008-02-12 | 最終更新日 | 2023-11-01 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | High-resolution structures of HIV-1 reverse transcriptase/TMC278 complexes: Strategic flexibility explains potency against resistance mutations. Proc.Natl.Acad.Sci.Usa, 105, 2008
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2ZD1
| Crystal Structure of HIV-1 Reverse Transcriptase (RT) in Complex with TMC278 (Rilpivirine), A Non-nucleoside RT Inhibitor | 分子名称: | 1,2-ETHANEDIOL, 4-{[4-({4-[(E)-2-cyanoethenyl]-2,6-dimethylphenyl}amino)pyrimidin-2-yl]amino}benzonitrile, Reverse transcriptase/ribonuclease H, ... | 著者 | Das, K, Bauman, J.D, Clark Jr, A.D, Shatkin, A.J, Arnold, E. | 登録日 | 2007-11-16 | 公開日 | 2008-02-12 | 最終更新日 | 2023-11-01 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | High-resolution structures of HIV-1 reverse transcriptase/TMC278 complexes: Strategic flexibility explains potency against resistance mutations. Proc.Natl.Acad.Sci.Usa, 105, 2008
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