7QPR
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7QR9
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![BU of 7qr9 by Molmil](/molmil-images/mine/7qr9) | Crystal structure of CK1 delta in complex with PK-09-82 | 分子名称: | 1,2-ETHANEDIOL, 4-[5-(4-fluorophenyl)-3-(pyridin-4-ylmethyl)imidazol-4-yl]-1~{H}-pyrrolo[2,3-b]pyridine, Casein kinase I isoform delta, ... | 著者 | Chaikuad, A, Khirsariya, P, Paruch, K, Knapp, S, Structural Genomics Consortium (SGC) | 登録日 | 2022-01-10 | 公開日 | 2023-01-18 | 最終更新日 | 2024-02-07 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Discovery of Potent and Exquisitely Selective Inhibitors of Kinase CK1 with Tunable Isoform Selectivity. Angew.Chem.Int.Ed.Engl., 62, 2023
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7QRM
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![BU of 7qrm by Molmil](/molmil-images/mine/7qrm) | Cryo-EM structure of catalytically active Spinacia oleracea cytochrome b6f in complex with endogenous plastoquinones at 2.7 A resolution | 分子名称: | (1S)-2-{[{[(2R)-2,3-DIHYDROXYPROPYL]OXY}(HYDROXY)PHOSPHORYL]OXY}-1-[(PALMITOYLOXY)METHYL]ETHYL STEARATE, 1,2-DI-O-ACYL-3-O-[6-DEOXY-6-SULFO-ALPHA-D-GLUCOPYRANOSYL]-SN-GLYCEROL, 2,3-DIMETHYL-5-(3,7,11,15,19,23,27,31,35-NONAMETHYL-2,6,10,14,18,22,26,30,34-HEXATRIACONTANONAENYL-2,5-CYCLOHEXADIENE-1,4-DIONE-2,3-DIMETHYL-5-SOLANESYL-1,4-BENZOQUINONE, ... | 著者 | Sarewicz, M, Szwalec, M, Indyka, P, Rawski, M, Pintscher, S, Pietras, R, Mielecki, B, Jaciuk, M, Glatt, S, Osyczka, A. | 登録日 | 2022-01-11 | 公開日 | 2023-01-25 | 実験手法 | ELECTRON MICROSCOPY (2.7 Å) | 主引用文献 | High-resolution cryo-EM structures of plant cytochrome b 6 f at work. Sci Adv, 9, 2023
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7QRB
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![BU of 7qrb by Molmil](/molmil-images/mine/7qrb) | Crystal structure of CK1 delta in complex with PK-09-129 | 分子名称: | 3-(dimethylamino)-~{N}-[4-[4-(4-fluorophenyl)-5-(1~{H}-pyrrolo[2,3-b]pyridin-4-yl)imidazol-1-yl]cyclohexyl]propane-1-sulfonamide, Casein kinase I isoform delta, SULFATE ION | 著者 | Chaikuad, A, Khirsariya, P, Paruch, K, Knapp, S, Structural Genomics Consortium (SGC) | 登録日 | 2022-01-10 | 公開日 | 2023-01-18 | 最終更新日 | 2024-02-07 | 実験手法 | X-RAY DIFFRACTION (2.6 Å) | 主引用文献 | Discovery of Potent and Exquisitely Selective Inhibitors of Kinase CK1 with Tunable Isoform Selectivity. Angew.Chem.Int.Ed.Engl., 62, 2023
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7QUI
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![BU of 7qui by Molmil](/molmil-images/mine/7qui) | Crystal structure of the N-terminal domain of Siglec-8 in complex with sulfonamide sialoside analogue | 分子名称: | (2~{S},4~{S},5~{R},6~{R})-5-acetamido-2-[(2~{S},3~{R},4~{S},5~{S},6~{R})-2-[(2~{R},3~{S},4~{R},5~{R},6~{R})-5-acetamido-2-(hydroxymethyl)-4,6-bis(oxidanyl)oxan-3-yl]oxy-3,5-bis(oxidanyl)-6-(sulfooxymethyl)oxan-4-yl]oxy-6-[(1~{R},2~{R})-3-(naphthalen-2-ylsulfonylamino)-1,2-bis(oxidanyl)propyl]-4-oxidanyl-oxane-2-carboxylic acid, Sialic acid-binding Ig-like lectin 8 | 著者 | Lenza, M.P, Oyenarte, I, Atxabal, U, Nycholat, C, Franconetti, A, Quintana, J.I, Delgado, S, Unione, L, Paulson, J, Jimenez-Barbero, J, Ereno-Orbea, J. | 登録日 | 2022-01-18 | 公開日 | 2023-01-18 | 最終更新日 | 2024-02-07 | 実験手法 | X-RAY DIFFRACTION (3.352 Å) | 主引用文献 | Structures of the Inhibitory Receptor Siglec-8 in Complex with a High-Affinity Sialoside Analogue and a Therapeutic Antibody. Jacs Au, 3, 2023
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7QU6
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![BU of 7qu6 by Molmil](/molmil-images/mine/7qu6) | Crystal structure of the N-terminal domain of Siglec-8 | 分子名称: | Sialic acid-binding Ig-like lectin 8 | 著者 | Lenza, M.P, Atxabal, U, Nycholat, C.M, Oyenarte, I, Paulson, J.C, Franconetti, A, Quintana, J.I, Unione, L, Delgado, S, Jimenez-Barbero, J, Ereno-Orbea, J. | 登録日 | 2022-01-17 | 公開日 | 2023-01-18 | 最終更新日 | 2024-02-07 | 実験手法 | X-RAY DIFFRACTION (2.34 Å) | 主引用文献 | Structures of the Inhibitory Receptor Siglec-8 in Complex with a High-Affinity Sialoside Analogue and a Therapeutic Antibody. Jacs Au, 3, 2023
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7QSE
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7QWH
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![BU of 7qwh by Molmil](/molmil-images/mine/7qwh) | X-ray structure of the adduct formed upon reaction of a vanadium hydroxyquinoline complex with RNase A | 分子名称: | 2,2-bis($l^{1}-oxidanyl)-3-oxa-1$l^{4}-aza-2$l^{4}-vanadatricyclo[6.3.1.0^{4,12}]dodeca-1(12),4,6,8,10-pentaene, Ribonuclease pancreatic | 著者 | Merlino, A, Ferraro, G. | 登録日 | 2022-01-25 | 公開日 | 2023-02-01 | 最終更新日 | 2024-02-07 | 実験手法 | X-RAY DIFFRACTION (1.573 Å) | 主引用文献 | Interaction of VIVO-8-hydroxyquinoline species with RNase A: the effect of metal ligands in the protein adduct stabilization Inorg Chem Front, 2023
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8E10
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![BU of 8e10 by Molmil](/molmil-images/mine/8e10) | Structure of mouse polymerase beta | 分子名称: | DNA polymerase beta, MALONIC ACID | 著者 | Thompson, M.K, Sharma, N, Prakash, A. | 登録日 | 2022-08-09 | 公開日 | 2023-02-01 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (1.65 Å) | 主引用文献 | Pol beta /XRCC1 heterodimerization dictates DNA damage recognition and basal Pol beta protein levels without interfering with mouse viability or fertility. DNA Repair (Amst), 123, 2023
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8E11
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7QV0
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![BU of 7qv0 by Molmil](/molmil-images/mine/7qv0) | Covalent complex between Scalindua brodae amxFabZ and amxACP | 分子名称: | Acyl carrier protein, Beta-hydroxyacyl-(Acyl-carrier-protein) dehydratase, S-[2-[3-[[(2R)-3,3-dimethyl-2-oxidanyl-4-phosphonooxy-butanoyl]amino]propanoylamino]ethyl] (Z)-hex-2-enethioate | 著者 | Barends, T, Dietl, A. | 登録日 | 2022-01-19 | 公開日 | 2023-02-01 | 最終更新日 | 2024-02-07 | 実験手法 | X-RAY DIFFRACTION (2.49 Å) | 主引用文献 | Structures of an unusual 3-hydroxyacyl dehydratase (FabZ) from a ladderane-producing organism with an unexpected substrate preference. J.Biol.Chem., 299, 2023
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7QWJ
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7QXV
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![BU of 7qxv by Molmil](/molmil-images/mine/7qxv) | Crystal Structure of Haem-Binding Protein HemS Mutant F104A F199A, from Yersinia enterocolitica | 分子名称: | DI(HYDROXYETHYL)ETHER, Hemin transport protein | 著者 | Barker, P.D, Keith, A, Brear, P, Wales, D. | 登録日 | 2022-01-27 | 公開日 | 2023-02-08 | 最終更新日 | 2024-02-07 | 実験手法 | X-RAY DIFFRACTION (1.67 Å) | 主引用文献 | Crystal Structure of Haem-Binding Protein HemS Mutant F104A F199A, from Yersinia enterocolitica To Be Published
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8G5N
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![BU of 8g5n by Molmil](/molmil-images/mine/8g5n) | Cryo-EM structure of the Guide loop Engagement Complex (VI) of Human Mitochondrial DNA Polymerase Gamma | 分子名称: | DNA polymerase subunit gamma-1, DNA polymerase subunit gamma-2, mitochondrial, ... | 著者 | Nayak, A.R, Buchel, G, Herbine, K.H, Sarfallah, A, Sokolova, V.O, Zamudio-Ochoa, A, Temiakov, D. | 登録日 | 2023-02-13 | 公開日 | 2024-01-10 | 実験手法 | ELECTRON MICROSCOPY (2.73 Å) | 主引用文献 | Structural basis for DNA proofreading. Nat Commun, 14, 2023
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4U4I
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![BU of 4u4i by Molmil](/molmil-images/mine/4u4i) | Megavirus chilensis superoxide dismutase | 分子名称: | Cu/Zn superoxide dismutase | 著者 | Lartigue, A, Claverie, J.-M, Burlat, B, Coutard, B, Abergel, C. | 登録日 | 2014-07-23 | 公開日 | 2014-11-05 | 最終更新日 | 2014-12-24 | 実験手法 | X-RAY DIFFRACTION (2.2 Å) | 主引用文献 | The megavirus chilensis cu,zn-superoxide dismutase: the first viral structure of a typical cellular copper chaperone-independent hyperstable dimeric enzyme. J.Virol., 89, 2015
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8G5K
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![BU of 8g5k by Molmil](/molmil-images/mine/8g5k) | Cryo-EM structure of the Wedge Alignment Complex (VIII) of Human Mitochondrial DNA Polymerase Gamma | 分子名称: | DNA polymerase subunit gamma-1, DNA polymerase subunit gamma-2, mitochondrial, ... | 著者 | Nayak, A.R, Buchel, G, Herbine, K.H, Sarfallah, A, Sokolova, V.O, Zamudio-Ochoa, A, Temiakov, D. | 登録日 | 2023-02-13 | 公開日 | 2024-01-10 | 実験手法 | ELECTRON MICROSCOPY (2.9 Å) | 主引用文献 | Structural basis for DNA proofreading. Nat Commun, 14, 2023
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8G5M
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![BU of 8g5m by Molmil](/molmil-images/mine/8g5m) | Cryo-EM structure of the Mismatch Locking Complex (III) of Human Mitochondrial DNA Polymerase Gamma | 分子名称: | DNA polymerase subunit gamma-1, DNA polymerase subunit gamma-2, mitochondrial, ... | 著者 | Nayak, A.R, Buchel, G, Herbine, K.H, Sarfallah, A, Sokolova, V.O, Zamudio-Ochoa, A, Temiakov, D. | 登録日 | 2023-02-13 | 公開日 | 2024-01-10 | 実験手法 | ELECTRON MICROSCOPY (2.58 Å) | 主引用文献 | Structural basis for DNA proofreading. Nat Commun, 14, 2023
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8G5I
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![BU of 8g5i by Molmil](/molmil-images/mine/8g5i) | Cryo-EM structure of the Mismatch Sensing Complex (I) of Human Mitochondrial DNA Polymerase Gamma | 分子名称: | DNA polymerase subunit gamma-1, DNA polymerase subunit gamma-2, mitochondrial, ... | 著者 | Nayak, A.R, Buchel, G, Herbine, K.H, Sarfallah, A, Sokolova, V.O, Zamudio-Ochoa, A, Temiakov, D. | 登録日 | 2023-02-13 | 公開日 | 2024-01-10 | 実験手法 | ELECTRON MICROSCOPY (2.75 Å) | 主引用文献 | Structural basis for DNA proofreading. Nat Commun, 14, 2023
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8G5P
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![BU of 8g5p by Molmil](/molmil-images/mine/8g5p) | Cryo-EM structure of the Guide loop Engagement Complex (V) of Human Mitochondrial DNA Polymerase Gamma | 分子名称: | DNA polymerase subunit gamma-1, DNA polymerase subunit gamma-2, mitochondrial, ... | 著者 | Nayak, A.R, Buchel, G, Herbine, K.H, Sarfallah, A, Sokolova, V.O, Zamudio-Ochoa, A, Temiakov, D. | 登録日 | 2023-02-13 | 公開日 | 2024-01-10 | 実験手法 | ELECTRON MICROSCOPY (2.78 Å) | 主引用文献 | Structural basis for DNA proofreading. Nat Commun, 14, 2023
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8G5J
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![BU of 8g5j by Molmil](/molmil-images/mine/8g5j) | Cryo-EM structure of the Mismatch Uncoupling Complex (II) of Human Mitochondrial DNA Polymerase Gamma | 分子名称: | DNA polymerase subunit gamma-1, DNA polymerase subunit gamma-2, mitochondrial, ... | 著者 | Nayak, A.R, Buchel, G, Herbine, K.H, Sarfallah, A, Sokolova, V.O, Zamudio-Ochoa, A, Temiakov, D. | 登録日 | 2023-02-13 | 公開日 | 2024-01-10 | 実験手法 | ELECTRON MICROSCOPY (2.63 Å) | 主引用文献 | Structural basis for DNA proofreading. Nat Commun, 14, 2023
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8G5L
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![BU of 8g5l by Molmil](/molmil-images/mine/8g5l) | Cryo-EM structure of the Primer Separation Complex (IX) of Human Mitochondrial DNA Polymerase Gamma | 分子名称: | DNA polymerase subunit gamma-1, DNA polymerase subunit gamma-2, mitochondrial, ... | 著者 | Nayak, A.R, Buchel, G, Herbine, K.H, Sarfallah, A, Sokolova, V.O, Zamudio-Ochoa, A, Temiakov, D. | 登録日 | 2023-02-13 | 公開日 | 2024-01-10 | 実験手法 | ELECTRON MICROSCOPY (3 Å) | 主引用文献 | Structural basis for DNA proofreading. Nat Commun, 14, 2023
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8G5O
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![BU of 8g5o by Molmil](/molmil-images/mine/8g5o) | Cryo-EM structure of the Guide loop Engagement Complex (IV) of Human Mitochondrial DNA Polymerase Gamma | 分子名称: | DNA polymerase subunit gamma-1, DNA polymerase subunit gamma-2, mitochondrial, ... | 著者 | Nayak, A.R, Buchel, G, Herbine, K.H, Sarfallah, A, Sokolova, V.O, Zamudio-Ochoa, A, Temiakov, D. | 登録日 | 2023-02-13 | 公開日 | 2024-01-10 | 実験手法 | ELECTRON MICROSCOPY (2.61 Å) | 主引用文献 | Structural basis for DNA proofreading. Nat Commun, 14, 2023
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7QRI
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![BU of 7qri by Molmil](/molmil-images/mine/7qri) | Regulatory domain dimer of tryptophan hydroxylase 2 in complex with L-Phe | 分子名称: | PHENYLALANINE, Tryptophan 5-hydroxylase 2 | 著者 | Vedel, I.M, Prestel, A, Harris, P, Peters, G.H.J, Kragelund, B.B. | 登録日 | 2022-01-11 | 公開日 | 2023-05-03 | 最終更新日 | 2024-06-19 | 実験手法 | SOLUTION NMR | 主引用文献 | Structural characterization of human tryptophan hydroxylase 2 reveals that L-Phe is superior to L-Trp as the regulatory domain ligand. Structure, 31, 2023
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8E7F
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![BU of 8e7f by Molmil](/molmil-images/mine/8e7f) | Crystal structure of the autotransporter Ssp from Serratia marcescens. | 分子名称: | CALCIUM ION, DI(HYDROXYETHYL)ETHER, Extracellular serine protease, ... | 著者 | Hor, L, Pilapitiya, A, Panjikar, S, Paxman, J.J, Heras, B. | 登録日 | 2022-08-23 | 公開日 | 2023-03-08 | 最終更新日 | 2023-03-15 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Crystal structure of a subtilisin-like autotransporter passenger domain reveals insights into its cytotoxic function. Nat Commun, 14, 2023
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7QF8
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![BU of 7qf8 by Molmil](/molmil-images/mine/7qf8) | Crystal structure of a bacterial pyranose 2-oxidase from Pseudoarthrobacter siccitolerans | 分子名称: | 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, FLAVIN-ADENINE DINUCLEOTIDE, GMC oxidoreductase family protein, ... | 著者 | Borges, P.T, Frazao, T, Taborda, A, Frazao, C, Martins, L.O. | 登録日 | 2021-12-04 | 公開日 | 2023-06-14 | 最終更新日 | 2024-02-07 | 実験手法 | X-RAY DIFFRACTION (2.009 Å) | 主引用文献 | Mechanistic insights into glycoside 3-oxidases involved in C-glycoside metabolism in soil microorganisms. Nat Commun, 14, 2023
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