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7FSO
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BU of 7fso by Molmil
SDCBP PanDDA analysis group deposition -- The PDZ domans of SDCBP in complex with Z198195770
分子名称: 1,2-ETHANEDIOL, D-GLUTAMIC ACID, GLYCINE, ...
著者Bradshaw, W.J, Katis, V.L, Bountra, C, von Delft, F, Brennan, P.E.
登録日2023-01-24
公開日2023-02-15
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献SDCBP PanDDA analysis group deposition
To Be Published
7FSQ
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BU of 7fsq by Molmil
SDCBP PanDDA analysis group deposition -- The PDZ domans of SDCBP in complex with Z1429867185
分子名称: 1,2-ETHANEDIOL, 4-methoxy-1H-indole, ALANINE, ...
著者Bradshaw, W.J, Katis, V.L, Bountra, C, von Delft, F, Brennan, P.E.
登録日2023-01-24
公開日2023-02-15
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (2.07 Å)
主引用文献SDCBP PanDDA analysis group deposition
To Be Published
7FSS
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BU of 7fss by Molmil
SDCBP PanDDA analysis group deposition -- The PDZ domans of SDCBP in complex with Z839706072
分子名称: 1,2-ETHANEDIOL, 2-(4-bromanylpyrazol-1-yl)-~{N}-cyclopropyl-~{N}-methyl-ethanamide, ALANINE, ...
著者Bradshaw, W.J, Katis, V.L, Bountra, C, von Delft, F, Brennan, P.E.
登録日2023-01-24
公開日2023-02-15
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (2.11 Å)
主引用文献SDCBP PanDDA analysis group deposition
To Be Published
7FSZ
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BU of 7fsz by Molmil
SDCBP PanDDA analysis group deposition -- The PDZ domans of SDCBP in complex with Z3006151474
分子名称: (5S)-5-(difluoromethoxy)pyridin-2(5H)-one, 1,2-ETHANEDIOL, D-GLUTAMIC ACID, ...
著者Bradshaw, W.J, Katis, V.L, Bountra, C, von Delft, F, Brennan, P.E.
登録日2023-01-24
公開日2023-02-15
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (2.05 Å)
主引用文献SDCBP PanDDA analysis group deposition
To Be Published
7FT4
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BU of 7ft4 by Molmil
SDCBP PanDDA analysis group deposition -- The PDZ domans of SDCBP in complex with Z48847594
分子名称: 1,2-ETHANEDIOL, ALANINE, D-GLUTAMIC ACID, ...
著者Bradshaw, W.J, Katis, V.L, Bountra, C, von Delft, F, Brennan, P.E.
登録日2023-01-24
公開日2023-02-15
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (2.17 Å)
主引用文献SDCBP PanDDA analysis group deposition
To Be Published
7FT3
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BU of 7ft3 by Molmil
SDCBP PanDDA analysis group deposition -- The PDZ domans of SDCBP in complex with Z291279160
分子名称: 1,2-ETHANEDIOL, 1-[2-(trifluoromethyloxy)phenyl]thiourea, ALANINE, ...
著者Bradshaw, W.J, Katis, V.L, Bountra, C, von Delft, F, Brennan, P.E.
登録日2023-01-24
公開日2023-02-15
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (2.05 Å)
主引用文献SDCBP PanDDA analysis group deposition
To Be Published
5WBV
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BU of 5wbv by Molmil
Crystal Structure of the SET Domain of Human SUV420H1 In Complex With Inhibitor
分子名称: 2-chloro-5-(4-methyl-6-oxo-3-phenylpyrano[2,3-c]pyrazol-1(6H)-yl)benzoic acid, Histone-lysine N-methyltransferase KMT5B, S-ADENOSYLMETHIONINE, ...
著者Halabelian, L, Tempel, W, Brown, P.J, Bountra, C, Edwards, A.M, Arrowsmith, C.H, Structural Genomics Consortium (SGC)
登録日2017-06-29
公開日2017-07-19
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Crystal Structure of the SET Domain of Human SUV420H1 In Complex With Inhibitor
To be published
5W8R
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BU of 5w8r by Molmil
Toxoplasma Gondii CDPK1 in complex with inhibitor 3CIB-PPI
分子名称: 1-tert-butyl-3-[(3-chlorophenyl)methyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine, CALCIUM ION, Calmodulin-domain protein kinase 1
著者El Bakkouri, M, Lovato, D, Loppnau, P, Lin, Y.H, Rutaganaria, F, Lopez, M.S, Shokat, L, Bountra, C, Edwards, A.M, Arrowsmith, C.H, Sibley, D, Hui, R, Walker, J.R, Structural Genomics Consortium (SGC)
登録日2017-06-22
公開日2017-07-19
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Toxoplasma Gondii CDPK1 in complex with inhibitor 3CIB-PPI
To be published
5WBN
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BU of 5wbn by Molmil
Crystal structure of fragment 3-(3-Benzyl-2-oxo-2H-[1,2,4]triazino[2,3-c]quinazolin-6-yl)propanoic acid bound in the ubiquitin binding pocket of the HDAC6 zinc-finger domain
分子名称: 3-(3-benzyl-2-oxo-2H-[1,2,4]triazino[2,3-c]quinazolin-6-yl)propanoic acid, ACETATE ION, CHLORIDE ION, ...
著者Harding, R.J, Walker, J.R, Ferreira de Freitas, R, Ravichandran, M, Santhakumar, V, Schapira, M, Bountra, C, Edwards, A.M, Arrowsmith, C.H.
登録日2017-06-29
公開日2017-08-02
最終更新日2024-03-13
実験手法X-RAY DIFFRACTION (1.64 Å)
主引用文献Crystal structure of fragment 3-(3-Benzyl-2-oxo-2H-[1,2,4]triazino[2,3-c]quinazolin-6-yl)propanoic acid bound in the ubiquitin binding pocket of the HDAC6 zinc-finger domain
To be published
7G84
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BU of 7g84 by Molmil
ARHGEF2 PanDDA analysis group deposition -- ARHGEF2 and RhoA in complex with Z1102357527
分子名称: DIMETHYL SULFOXIDE, FORMIC ACID, N-[(3R)-6-oxopiperidin-3-yl]-1,3-thiazole-4-carboxamide, ...
著者Bradshaw, W.J, Katis, V.L, Bountra, C, von Delft, F, Brennan, P.E.
登録日2023-06-22
公開日2023-07-12
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (1.811 Å)
主引用文献ARHGEF2 PanDDA analysis group deposition
To Be Published
7G86
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BU of 7g86 by Molmil
ARHGEF2 PanDDA analysis group deposition -- ARHGEF2 and RhoA in complex with Z1137725943
分子名称: DIMETHYL SULFOXIDE, FORMIC ACID, N-[(1H-indol-4-yl)methyl]ethanamine, ...
著者Bradshaw, W.J, Katis, V.L, Bountra, C, von Delft, F, Brennan, P.E.
登録日2023-06-22
公開日2023-07-12
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (1.699 Å)
主引用文献ARHGEF2 PanDDA analysis group deposition
To Be Published
7G8H
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BU of 7g8h by Molmil
ARHGEF2 PanDDA analysis group deposition -- ARHGEF2 and RhoA in complex with Z1198180782
分子名称: 5-methoxy-1H-pyrrolo[3,2-b]pyridine, DIMETHYL SULFOXIDE, FORMIC ACID, ...
著者Bradshaw, W.J, Katis, V.L, Bountra, C, von Delft, F, Brennan, P.E.
登録日2023-06-22
公開日2023-07-12
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (1.67 Å)
主引用文献ARHGEF2 PanDDA analysis group deposition
To Be Published
7G8I
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BU of 7g8i by Molmil
ARHGEF2 PanDDA analysis group deposition -- ARHGEF2 and RhoA in complex with Z1198316457
分子名称: 4,4-difluorocyclohexane-1-carboxamide, DIMETHYL SULFOXIDE, FORMIC ACID, ...
著者Bradshaw, W.J, Katis, V.L, Bountra, C, von Delft, F, Brennan, P.E.
登録日2023-06-22
公開日2023-07-12
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (2.468 Å)
主引用文献ARHGEF2 PanDDA analysis group deposition
To Be Published
7G80
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BU of 7g80 by Molmil
ARHGEF2 PanDDA analysis group deposition -- ARHGEF2 and RhoA in complex with Z1041785508
分子名称: 5-(1,3-thiazol-2-yl)-1H-1,2,4-triazole, DIMETHYL SULFOXIDE, FORMIC ACID, ...
著者Bradshaw, W.J, Katis, V.L, Bountra, C, von Delft, F, Brennan, P.E.
登録日2023-06-22
公開日2023-07-12
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (1.671 Å)
主引用文献ARHGEF2 PanDDA analysis group deposition
To Be Published
7G8K
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BU of 7g8k by Molmil
ARHGEF2 PanDDA analysis group deposition -- ARHGEF2 and RhoA in complex with Z1217131798
分子名称: (3M)-3-(2-methyl-1H-imidazol-1-yl)pyridine, DIMETHYL SULFOXIDE, FORMIC ACID, ...
著者Bradshaw, W.J, Katis, V.L, Bountra, C, von Delft, F, Brennan, P.E.
登録日2023-06-22
公開日2023-07-12
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (1.491 Å)
主引用文献ARHGEF2 PanDDA analysis group deposition
To Be Published
7G88
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BU of 7g88 by Molmil
ARHGEF2 PanDDA analysis group deposition -- ARHGEF2 and RhoA in complex with Z1148747945
分子名称: DIMETHYL SULFOXIDE, FORMIC ACID, N-(3-methylpyridin-4-yl)acetamide, ...
著者Bradshaw, W.J, Katis, V.L, Bountra, C, von Delft, F, Brennan, P.E.
登録日2023-06-22
公開日2023-07-12
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (1.869 Å)
主引用文献ARHGEF2 PanDDA analysis group deposition
To Be Published
7G90
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BU of 7g90 by Molmil
ARHGEF2 PanDDA analysis group deposition -- ARHGEF2 and RhoA in complex with Z1509195674
分子名称: 4-[(3S)-piperidin-3-yl]-1H-indole, DIMETHYL SULFOXIDE, FORMIC ACID, ...
著者Bradshaw, W.J, Katis, V.L, Bountra, C, von Delft, F, Brennan, P.E.
登録日2023-06-22
公開日2023-07-12
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (1.911 Å)
主引用文献ARHGEF2 PanDDA analysis group deposition
To Be Published
7G8B
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BU of 7g8b by Molmil
ARHGEF2 PanDDA analysis group deposition -- ARHGEF2 and RhoA in complex with Z100643660
分子名称: DIMETHYL SULFOXIDE, FORMIC ACID, N,1-dimethyl-1H-indole-3-carboxamide, ...
著者Bradshaw, W.J, Katis, V.L, Bountra, C, von Delft, F, Brennan, P.E.
登録日2023-06-22
公開日2023-07-12
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (1.42 Å)
主引用文献ARHGEF2 PanDDA analysis group deposition
To Be Published
7G93
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BU of 7g93 by Molmil
ARHGEF2 PanDDA analysis group deposition -- ARHGEF2 and RhoA in complex with Z1565771450
分子名称: DIMETHYL SULFOXIDE, FORMIC ACID, N-(8-methyl-1,2,3,4-tetrahydroquinolin-5-yl)acetamide, ...
著者Bradshaw, W.J, Katis, V.L, Bountra, C, von Delft, F, Brennan, P.E.
登録日2023-06-22
公開日2023-07-12
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (1.693 Å)
主引用文献ARHGEF2 PanDDA analysis group deposition
To Be Published
7G8E
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BU of 7g8e by Molmil
ARHGEF2 PanDDA analysis group deposition -- ARHGEF2 and RhoA in complex with Z104479710
分子名称: 1-(1H-benzimidazol-2-yl)methanamine, DIMETHYL SULFOXIDE, FORMIC ACID, ...
著者Bradshaw, W.J, Katis, V.L, Bountra, C, von Delft, F, Brennan, P.E.
登録日2023-06-22
公開日2023-07-12
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (1.79 Å)
主引用文献ARHGEF2 PanDDA analysis group deposition
To Be Published
7G8P
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BU of 7g8p by Molmil
ARHGEF2 PanDDA analysis group deposition -- ARHGEF2 and RhoA in complex with Z1269184613
分子名称: 1,3-benzothiazole-6-sulfonamide, DIMETHYL SULFOXIDE, FORMIC ACID, ...
著者Bradshaw, W.J, Katis, V.L, Bountra, C, von Delft, F, Brennan, P.E.
登録日2023-06-22
公開日2023-07-12
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (2.209 Å)
主引用文献ARHGEF2 PanDDA analysis group deposition
To Be Published
7G81
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BU of 7g81 by Molmil
ARHGEF2 PanDDA analysis group deposition -- ARHGEF2 and RhoA in complex with Z104474512
分子名称: 1-(2-ethoxyphenyl)piperazine, DIMETHYL SULFOXIDE, FORMIC ACID, ...
著者Bradshaw, W.J, Katis, V.L, Bountra, C, von Delft, F, Brennan, P.E.
登録日2023-06-22
公開日2023-07-12
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (1.51 Å)
主引用文献ARHGEF2 PanDDA analysis group deposition
To Be Published
7G8S
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BU of 7g8s by Molmil
ARHGEF2 PanDDA analysis group deposition -- ARHGEF2 and RhoA in complex with Z1270393711
分子名称: 5-(methoxymethyl)-1,2-oxazole-3-carboxamide, DIMETHYL SULFOXIDE, FORMIC ACID, ...
著者Bradshaw, W.J, Katis, V.L, Bountra, C, von Delft, F, Brennan, P.E.
登録日2023-06-22
公開日2023-07-12
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (1.6 Å)
主引用文献ARHGEF2 PanDDA analysis group deposition
To Be Published
7G89
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BU of 7g89 by Molmil
ARHGEF2 PanDDA analysis group deposition -- ARHGEF2 and RhoA in complex with Z1192341021
分子名称: 1-(5-amino-2H-isoindol-2-yl)ethan-1-one, DIMETHYL SULFOXIDE, FORMIC ACID, ...
著者Bradshaw, W.J, Katis, V.L, Bountra, C, von Delft, F, Brennan, P.E.
登録日2023-06-22
公開日2023-07-12
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (1.901 Å)
主引用文献ARHGEF2 PanDDA analysis group deposition
To Be Published
7G94
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BU of 7g94 by Molmil
ARHGEF2 PanDDA analysis group deposition -- ARHGEF2 and RhoA in complex with Z1575337975
分子名称: (2P)-5-fluoro-2-(1H-pyrazol-5-yl)pyridine, DIMETHYL SULFOXIDE, FORMIC ACID, ...
著者Bradshaw, W.J, Katis, V.L, Bountra, C, von Delft, F, Brennan, P.E.
登録日2023-06-22
公開日2023-07-12
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (1.47 Å)
主引用文献ARHGEF2 PanDDA analysis group deposition
To Be Published

221716

件を2024-06-26に公開中

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