6SZL
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![BU of 6szl by Molmil](/molmil-images/mine/6szl) | Crystal structure of YTHDC1 with fragment 7 (DHU_DC1_021) | 分子名称: | 6-phenyl-1~{H}-pyrimidine-2,4-dione, SULFATE ION, YTH domain-containing protein 1 | 著者 | Bedi, R.K, Huang, D, Sledz, P, Caflisch, A. | 登録日 | 2019-10-02 | 公開日 | 2020-03-04 | 最終更新日 | 2024-01-24 | 実験手法 | X-RAY DIFFRACTION (1.45 Å) | 主引用文献 | Selectively Disrupting m6A-Dependent Protein-RNA Interactions with Fragments. Acs Chem.Biol., 15, 2020
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6T09
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![BU of 6t09 by Molmil](/molmil-images/mine/6t09) | Crystal structure of YTHDC1 with fragment 24 (PSI_DC1_003) | 分子名称: | SULFATE ION, YTHDC1, ~{N}-pyridin-3-ylethanamide | 著者 | Bedi, R.K, Huang, D, Sledz, P, Caflisch, A. | 登録日 | 2019-10-02 | 公開日 | 2020-03-04 | 最終更新日 | 2024-01-24 | 実験手法 | X-RAY DIFFRACTION (1.75 Å) | 主引用文献 | Selectively Disrupting m6A-Dependent Protein-RNA Interactions with Fragments. Acs Chem.Biol., 15, 2020
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8XYZ
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![BU of 8xyz by Molmil](/molmil-images/mine/8xyz) | The structure of fox ACE2 and PT RBD complex | 分子名称: | Angiotensin-converting enzyme, Signal peptide, Spike protein S1, ... | 著者 | sun, J.Q. | 登録日 | 2024-01-20 | 公開日 | 2024-07-03 | 最終更新日 | 2024-07-24 | 実験手法 | ELECTRON MICROSCOPY (2.96 Å) | 主引用文献 | The binding and structural basis of fox ACE2 to RBDs from different sarbecoviruses. Virol Sin, 2024
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7VLN
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![BU of 7vln by Molmil](/molmil-images/mine/7vln) | NSD2-PWWP1 domain bound with an imidazol-5-yl benzonitrile compound | 分子名称: | 4-[5-[4-(aminomethyl)-2,6-dimethoxy-phenyl]-3-methyl-imidazol-4-yl]benzenecarbonitrile, Histone-lysine N-methyltransferase NSD2 | 著者 | Cao, D.Y, Li, Y.L, Li, J, Xiong, B. | 登録日 | 2021-10-05 | 公開日 | 2022-07-06 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (3.09 Å) | 主引用文献 | Structure-Based Discovery of a Series of NSD2-PWWP1 Inhibitors. J.Med.Chem., 65, 2022
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6CCG
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![BU of 6ccg by Molmil](/molmil-images/mine/6ccg) | Crystal structure MBD3 MBD domain in complex with methylated CpG DNA | 分子名称: | DNA, Methyl-CpG-binding domain protein 3, UNKNOWN ATOM OR ION | 著者 | Liu, K, Tempel, W, Bountra, C, Arrowsmith, C.H, Edwards, A.M, Min, J, Structural Genomics Consortium (SGC) | 登録日 | 2018-02-07 | 公開日 | 2018-05-09 | 最終更新日 | 2024-03-13 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Structural analyses reveal that MBD3 is a methylated CG binder. Febs J., 286, 2019
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5Y4O
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![BU of 5y4o by Molmil](/molmil-images/mine/5y4o) | Cryo-EM structure of MscS channel, YnaI | 分子名称: | Low conductance mechanosensitive channel YnaI | 著者 | Zhang, Y, Yu, J. | 登録日 | 2017-08-04 | 公開日 | 2019-03-20 | 実験手法 | ELECTRON MICROSCOPY (3.8 Å) | 主引用文献 | A binding-block ion selective mechanism revealed by a Na/K selective channel. Protein Cell, 9, 2018
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6CKM
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6CKL
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![BU of 6ckl by Molmil](/molmil-images/mine/6ckl) | N. meningitidis CMP-sialic acid synthetase in the presence of CMP and Neu5Ac2en | 分子名称: | 2-DEOXY-2,3-DEHYDRO-N-ACETYL-NEURAMINIC ACID, CHLORIDE ION, CITRATE ANION, ... | 著者 | Matthews, M.M, Fisher, A.J, Chen, X. | 登録日 | 2018-02-28 | 公開日 | 2019-03-06 | 最終更新日 | 2023-10-04 | 実験手法 | X-RAY DIFFRACTION (2.684 Å) | 主引用文献 | Catalytic Cycle ofNeisseria meningitidisCMP-Sialic Acid Synthetase Illustrated by High-Resolution Protein Crystallography. Biochemistry, 2019
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5V0L
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![BU of 5v0l by Molmil](/molmil-images/mine/5v0l) | Crystal structure of the AHR-ARNT heterodimer in complex with the DRE | 分子名称: | Aryl hydrocarbon receptor, Aryl hydrocarbon receptor nuclear translocator, CITRIC ACID, ... | 著者 | Seok, S.-H, Lee, W, Jiang, L, Bradfield, C.A, Xing, Y. | 登録日 | 2017-02-28 | 公開日 | 2017-04-19 | 最終更新日 | 2023-10-04 | 実験手法 | X-RAY DIFFRACTION (4 Å) | 主引用文献 | Structural hierarchy controlling dimerization and target DNA recognition in the AHR transcriptional complex. Proc. Natl. Acad. Sci. U.S.A., 114, 2017
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5H3W
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8JOP
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![BU of 8jop by Molmil](/molmil-images/mine/8jop) | Crystal structure of the SARS-CoV-2 main protease in complex with 11a | 分子名称: | 3C-like proteinase nsp5, methyl (6~{R})-5-ethanoyl-7-oxidanylidene-6-[4-(trifluoromethyl)phenyl]-8,9,10,11-tetrahydro-6~{H}-benzo[b][1,4]benzodiazepine-2-carboxylate | 著者 | Zeng, R, Liu, Y.Z, Wang, F.L, Yang, S.Y, Lei, J. | 登録日 | 2023-06-08 | 公開日 | 2023-08-16 | 実験手法 | X-RAY DIFFRACTION (2.7 Å) | 主引用文献 | Discovery of benzodiazepine derivatives as a new class of covalent inhibitors of SARS-CoV-2 main protease. Bioorg.Med.Chem.Lett., 92, 2023
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1RAO
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1LPO
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![BU of 1lpo by Molmil](/molmil-images/mine/1lpo) | |
1LPP
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![BU of 1lpp by Molmil](/molmil-images/mine/1lpp) | |
1SCJ
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![BU of 1scj by Molmil](/molmil-images/mine/1scj) | |
5OFP
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![BU of 5ofp by Molmil](/molmil-images/mine/5ofp) | |
6EQB
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![BU of 6eqb by Molmil](/molmil-images/mine/6eqb) | HLA class I histocompatibility antigen | 分子名称: | 1,2-ETHANEDIOL, 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, ALA-ALA-GLY-ILE-GLY-ILE-LEU-THR-VAL, ... | 著者 | Rizkallah, P.J, Cole, D.K. | 登録日 | 2017-10-12 | 公開日 | 2018-10-10 | 最終更新日 | 2024-01-17 | 実験手法 | X-RAY DIFFRACTION (2.81 Å) | 主引用文献 | TCR-induced alteration of primary MHC peptide anchor residue. Eur.J.Immunol., 49, 2019
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6EAY
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![BU of 6eay by Molmil](/molmil-images/mine/6eay) | |
6CEV
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![BU of 6cev by Molmil](/molmil-images/mine/6cev) | MBD3 MBD in complex with methylated, non-palindromic CpG DNA: alternative interpretation of crystallographic data | 分子名称: | DNA (5'-D(*GP*CP*CP*AP*AP*(5CM)P*GP*CP*TP*GP*GP*C)-3'), DNA (5'-D(*GP*CP*CP*AP*GP*(5CM)P*GP*TP*TP*GP*GP*C)-3'), Methyl-CpG-binding domain protein 3, ... | 著者 | Liu, K, Tempel, W, Wernimont, A.K, Bountra, C, Arrowsmith, C.H, Edwards, A.M, Min, J, Structural Genomics Consortium (SGC) | 登録日 | 2018-02-12 | 公開日 | 2018-05-09 | 最終更新日 | 2023-10-04 | 実験手法 | X-RAY DIFFRACTION (2.005 Å) | 主引用文献 | Structural analyses reveal that MBD3 is a methylated CG binder. Febs J., 286, 2019
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5H6I
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![BU of 5h6i by Molmil](/molmil-images/mine/5h6i) | Crystal Structure of GBS CAMP Factor | 分子名称: | CHLORIDE ION, Protein B, SULFATE ION | 著者 | Jin, T.C, Brefo-Mensah, E.K. | 登録日 | 2016-11-13 | 公開日 | 2017-11-22 | 最終更新日 | 2024-03-20 | 実験手法 | X-RAY DIFFRACTION (2.45 Å) | 主引用文献 | Crystal structure of theStreptococcus agalactiaeCAMP factor provides insights into its membrane-permeabilizing activity. J.Biol.Chem., 293, 2018
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6CEU
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![BU of 6ceu by Molmil](/molmil-images/mine/6ceu) | MBD3 MBD in complex with methylated, non-palindromic CpG DNA: alternative interpretation of crystallographic data | 分子名称: | DNA (5'-D(*GP*CP*CP*AP*AP*(5CM)P*GP*CP*TP*GP*GP*C)-3'), DNA (5'-D(*GP*CP*CP*AP*GP*(5CM)P*GP*TP*TP*GP*GP*C)-3'), Methyl-CpG-binding domain protein 3, ... | 著者 | Liu, K, Tempel, W, Wernimont, A.K, Bountra, C, Arrowsmith, C.H, Edwards, A.M, Min, J, Structural Genomics Consortium (SGC) | 登録日 | 2018-02-12 | 公開日 | 2018-05-09 | 最終更新日 | 2023-10-04 | 実験手法 | X-RAY DIFFRACTION (2.005 Å) | 主引用文献 | Structural analyses reveal that MBD3 is a methylated CG binder. Febs J., 286, 2019
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6CKK
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7XCZ
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7XDK
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![BU of 7xdk by Molmil](/molmil-images/mine/7xdk) | Cryo-EM structure of SARS-CoV-2 Delta Spike protein in complex with BA7054 and BA7125 fab | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, BA7054 fab, ... | 著者 | Liu, Z, Lui, S, Gao, Y. | 登録日 | 2022-03-27 | 公開日 | 2023-03-01 | 実験手法 | ELECTRON MICROSCOPY (3.2 Å) | 主引用文献 | Biparatopic antibody BA7208/7125 effectively neutralizes SARS-CoV-2 variants including Omicron BA.1-BA.5. Cell Discov, 9, 2023
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7XDA
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![BU of 7xda by Molmil](/molmil-images/mine/7xda) | |