2ZYN
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![BU of 2zyn by Molmil](/molmil-images/mine/2zyn) | Crystal structure of cyclo/maltodextrin-binding protein complexed with beta-cyclodextrin | 分子名称: | Cycloheptakis-(1-4)-(alpha-D-glucopyranose), Solute-binding protein | 著者 | Matsumoto, M, Yamada, M, Kurakata, Y, Yoshida, H, Kamitori, S, Nishikawa, A, Tonozuka, T. | 登録日 | 2009-01-27 | 公開日 | 2009-03-31 | 最終更新日 | 2023-11-01 | 実験手法 | X-RAY DIFFRACTION (1.7 Å) | 主引用文献 | Crystal structures of open and closed forms of cyclo/maltodextrin-binding protein Febs J., 276, 2009
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3ALJ
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![BU of 3alj by Molmil](/molmil-images/mine/3alj) | Crystal structure of 2-methyl-3-hydroxypyridine-5-carboxylic acid oxygenase, reduced form | 分子名称: | 2-methyl-3-hydroxypyridine-5-carboxylic acid oxygenase, BETA-MERCAPTOETHANOL, FLAVIN-ADENINE DINUCLEOTIDE, ... | 著者 | Kobayashi, J, Yoshida, H, Yoshikane, Y, Kamitori, S, Yagi, T. | 登録日 | 2010-08-04 | 公開日 | 2011-08-10 | 最終更新日 | 2023-11-01 | 実験手法 | X-RAY DIFFRACTION (1.48 Å) | 主引用文献 | Crystal structure of 2-methyl-3-hydroxypyridine-5-carboxylic acid oxygenase To be Published
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3A9T
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![BU of 3a9t by Molmil](/molmil-images/mine/3a9t) | X-ray Structure of Bacillus pallidus D-Arabinose Isomerase Complex with L-Fucitol | 分子名称: | D-arabinose isomerase, FUCITOL, MANGANESE (II) ION | 著者 | Takeda, K, Yoshida, H, Izumori, K, Kamitori, S. | 登録日 | 2009-11-05 | 公開日 | 2010-04-07 | 最終更新日 | 2023-11-01 | 実験手法 | X-RAY DIFFRACTION (2.61 Å) | 主引用文献 | X-ray structures of Bacillus pallidusd-arabinose isomerase and its complex with l-fucitol. Biochim.Biophys.Acta, 1804, 2010
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2ZNL
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![BU of 2znl by Molmil](/molmil-images/mine/2znl) | Crystal structure of PA-PB1 complex form influenza virus RNA polymerase | 分子名称: | Polymerase acidic protein, RNA-directed RNA polymerase catalytic subunit | 著者 | Obayashi, E, Yoshida, H, Kawai, F, Shibayama, N, Kawaguchi, A, Nagata, K, Tame, J.R.H, Park, S.-Y. | 登録日 | 2008-04-28 | 公開日 | 2008-09-02 | 最終更新日 | 2024-03-13 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | The structural basis for an essential subunit interaction in influenza virus RNA polymerase Nature, 454, 2008
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3ALM
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![BU of 3alm by Molmil](/molmil-images/mine/3alm) | Crystal structure of 2-methyl-3-hydroxypyridine-5-carboxylic acid oxygenase, mutant C294A | 分子名称: | 2-methyl-3-hydroxypyridine-5-carboxylic acid oxygenase, FLAVIN-ADENINE DINUCLEOTIDE, GLYCEROL | 著者 | Kobayashi, J, Yoshida, H, Yoshikane, Y, Kamitori, S, Yagi, T. | 登録日 | 2010-08-04 | 公開日 | 2011-08-10 | 最終更新日 | 2023-11-01 | 実験手法 | X-RAY DIFFRACTION (1.77 Å) | 主引用文献 | Crystal structure of 2-methyl-3-hydroxypyridine-5-carboxylic acid oxygenase To be Published
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3D3I
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![BU of 3d3i by Molmil](/molmil-images/mine/3d3i) | Crystal structural of Escherichia coli K12 YgjK, a glucosidase belonging to glycoside hydrolase family 63 | 分子名称: | CALCIUM ION, GLYCEROL, Uncharacterized protein ygjK | 著者 | Kurakata, Y, Uechi, A, Yoshida, H, Kamitori, S, Sakano, Y, Nishikawa, A, Tonozuka, T. | 登録日 | 2008-05-12 | 公開日 | 2008-06-03 | 最終更新日 | 2011-07-13 | 実験手法 | X-RAY DIFFRACTION (1.78 Å) | 主引用文献 | Structural insights into the substrate specificity and function of Escherichia coli K12 YgjK, a glucosidase belonging to the glycoside hydrolase family 63. J.Mol.Biol., 381, 2008
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3A9R
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![BU of 3a9r by Molmil](/molmil-images/mine/3a9r) | X-ray Structures of Bacillus pallidus D-Arabinose IsomeraseComplex with (4R)-2-METHYLPENTANE-2,4-DIOL | 分子名称: | (4R)-2-METHYLPENTANE-2,4-DIOL, D-arabinose isomerase, MANGANESE (II) ION | 著者 | Takeda, K, Yoshida, H, Izumori, K, Kamitori, S. | 登録日 | 2009-11-05 | 公開日 | 2010-04-07 | 最終更新日 | 2023-11-01 | 実験手法 | X-RAY DIFFRACTION (1.77 Å) | 主引用文献 | X-ray structures of Bacillus pallidusd-arabinose isomerase and its complex with l-fucitol. Biochim.Biophys.Acta, 1804, 2010
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3A9S
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![BU of 3a9s by Molmil](/molmil-images/mine/3a9s) | X-ray Structure of Bacillus pallidus D-Arabinose Isomerase Complex with Glycerol | 分子名称: | D-arabinose isomerase, GLYCEROL, MANGANESE (II) ION | 著者 | Takeda, K, Yoshida, H, Izumori, K, Kamitori, S. | 登録日 | 2009-11-05 | 公開日 | 2010-04-07 | 最終更新日 | 2023-11-01 | 実験手法 | X-RAY DIFFRACTION (1.6 Å) | 主引用文献 | X-ray structures of Bacillus pallidusd-arabinose isomerase and its complex with l-fucitol. Biochim.Biophys.Acta, 1804, 2010
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3ALL
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![BU of 3all by Molmil](/molmil-images/mine/3all) | Crystal structure of 2-methyl-3-hydroxypyridine-5-carboxylic acid oxygenase, mutant Y270A | 分子名称: | 2-methyl-3-hydroxypyridine-5-carboxylic acid oxygenase, BETA-MERCAPTOETHANOL, FLAVIN-ADENINE DINUCLEOTIDE, ... | 著者 | Kobayashi, J, Yoshida, H, Yoshikane, Y, Kamitori, S, Yagi, T. | 登録日 | 2010-08-04 | 公開日 | 2011-08-10 | 最終更新日 | 2023-11-01 | 実験手法 | X-RAY DIFFRACTION (1.78 Å) | 主引用文献 | Crystal structure of 2-methyl-3-hydroxypyridine-5-carboxylic acid oxygenase To be published
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2ECE
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![BU of 2ece by Molmil](/molmil-images/mine/2ece) | |
2D2O
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![BU of 2d2o by Molmil](/molmil-images/mine/2d2o) | Structure of a complex of Thermoactinomyces vulgaris R-47 alpha-amylase 2 with maltohexaose demonstrates the important role of aromatic residues at the reducing end of the substrate binding cleft | 分子名称: | CALCIUM ION, Neopullulanase 2, alpha-D-glucopyranose-(1-4)-alpha-D-glucopyranose-(1-4)-alpha-D-glucopyranose-(1-4)-alpha-D-glucopyranose-(1-4)-alpha-D-glucopyranose-(1-4)-alpha-D-glucopyranose | 著者 | Ohtaki, A, Mizuno, M, Yoshida, H, Tonozuka, T, Sakano, Y, Kamitori, S. | 登録日 | 2005-09-13 | 公開日 | 2006-08-29 | 最終更新日 | 2024-05-29 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | Structure of a complex of Thermoactinomyces vulgaris R-47 alpha-amylase 2 with maltohexaose demonstrates the important role of aromatic residues at the reducing end of the substrate binding cleft Carbohydr.Res., 341, 2006
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2D0F
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![BU of 2d0f by Molmil](/molmil-images/mine/2d0f) | Crystal Structure of Thermoactinomyces vulgaris R-47 Alpha-Amylase 1 (TVAI) Mutant D356N complexed with P2, a pullulan model oligosaccharide | 分子名称: | (4S)-2-METHYL-2,4-PENTANEDIOL, CALCIUM ION, alpha-D-glucopyranose-(1-4)-alpha-D-glucopyranose-(1-4)-alpha-D-glucopyranose-(1-6)-alpha-D-glucopyranose-(1-4)-beta-D-glucopyranose, ... | 著者 | Abe, A, Yoshida, H, Tonozuka, T, Sakano, Y, Kamitori, S. | 登録日 | 2005-08-02 | 公開日 | 2006-07-11 | 最終更新日 | 2024-05-29 | 実験手法 | X-RAY DIFFRACTION (2.08 Å) | 主引用文献 | Complexes of Thermoactinomyces vulgaris R-47 alpha-amylase 1 and pullulan model oligossacharides provide new insight into the mechanism for recognizing substrates with alpha-(1,6) glycosidic linkages Febs J., 272, 2005
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2D0H
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![BU of 2d0h by Molmil](/molmil-images/mine/2d0h) | Crystal Structure of Thermoactinomyces vulgaris R-47 Alpha-Amylase 1 (TVAI) Mutant D356N/E396Q complexed with P2, a pullulan model oligosaccharide | 分子名称: | (4S)-2-METHYL-2,4-PENTANEDIOL, CALCIUM ION, alpha-D-glucopyranose-(1-6)-alpha-D-glucopyranose-(1-4)-alpha-D-glucopyranose-(1-4)-alpha-D-glucopyranose-(1-6)-alpha-D-glucopyranose-(1-4)-alpha-D-glucopyranose, ... | 著者 | Abe, A, Yoshida, H, Tonozuka, T, Sakano, Y, Kamitori, S. | 登録日 | 2005-08-02 | 公開日 | 2006-07-11 | 最終更新日 | 2024-05-29 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | Complexes of Thermoactinomyces vulgaris R-47 alpha-amylase 1 and pullulan model oligossacharides provide new insight into the mechanism for recognizing substrates with alpha-(1,6) glycosidic linkages Febs J., 272, 2005
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2D0G
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![BU of 2d0g by Molmil](/molmil-images/mine/2d0g) | Crystal Structure of Thermoactinomyces vulgaris R-47 Alpha-Amylase 1 (TVAI) Mutant D356N/E396Q complexed with P5, a pullulan model oligosaccharide | 分子名称: | (4S)-2-METHYL-2,4-PENTANEDIOL, CALCIUM ION, alpha-D-glucopyranose, ... | 著者 | Abe, A, Yoshida, H, Tonozuka, T, Sakano, Y, Kamitori, S. | 登録日 | 2005-08-02 | 公開日 | 2006-07-11 | 最終更新日 | 2024-05-29 | 実験手法 | X-RAY DIFFRACTION (2.6 Å) | 主引用文献 | Complexes of Thermoactinomyces vulgaris R-47 alpha-amylase 1 and pullulan model oligossacharides provide new insight into the mechanism for recognizing substrates with alpha-(1,6) glycosidic linkages Febs J., 272, 2005
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2RQL
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![BU of 2rql by Molmil](/molmil-images/mine/2rql) | |
7BV9
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![BU of 7bv9 by Molmil](/molmil-images/mine/7bv9) | The NMR structure of the BEN domain from human NAC1 | 分子名称: | Nucleus accumbens-associated protein 1 | 著者 | Nagata, T, Kobayashi, N, Nakayama, N, Obayashi, E, Urano, T. | 登録日 | 2020-04-09 | 公開日 | 2021-02-17 | 最終更新日 | 2024-05-15 | 実験手法 | SOLUTION NMR | 主引用文献 | Nucleus Accumbens-Associated Protein 1 Binds DNA Directly through the BEN Domain in a Sequence-Specific Manner. Biomedicines, 8, 2020
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2RVH
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![BU of 2rvh by Molmil](/molmil-images/mine/2rvh) | NMR structure of eIF1 | 分子名称: | Eukaryotic translation initiation factor eIF-1 | 著者 | Nagata, T, Obayashi, E, Asano, K. | 登録日 | 2015-10-16 | 公開日 | 2016-10-26 | 最終更新日 | 2024-05-15 | 実験手法 | SOLUTION NMR | 主引用文献 | Molecular Landscape of the Ribosome Pre-initiation Complex during mRNA Scanning: Structural Role for eIF3c and Its Control by eIF5 Cell Rep, 18, 2017
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6KRO
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![BU of 6kro by Molmil](/molmil-images/mine/6kro) | Tankyrase-2 in complex with RK-582 | 分子名称: | 6-[(2S,6R)-2,6-dimethylmorpholin-4-yl]-4-fluoranyl-1-methyl-1'-(8-methyl-4-oxidanylidene-3,5,6,7-tetrahydropyrido[2,3-d]pyrimidin-2-yl)spiro[indole-3,4'-piperidine]-2-one, GLYCEROL, PHOSPHATE ION, ... | 著者 | Niwa, H, Shirai, F, Sato, S, Tsumura, T, Okue, M, Shirouzu, M, Seimiya, H, Umehara, T. | 登録日 | 2019-08-22 | 公開日 | 2020-04-01 | 最終更新日 | 2024-03-27 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Design and Discovery of an Orally Efficacious Spiroindolinone-Based Tankyrase Inhibitor for the Treatment of Colon Cancer. J.Med.Chem., 63, 2020
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5ZQQ
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![BU of 5zqq by Molmil](/molmil-images/mine/5zqq) | Tankyrase-2 in complex with compound 52 | 分子名称: | 1-methyl-1'-(4-oxo-3,4,5,6,7,8-hexahydroquinazolin-2-yl)spiro[indole-3,4'-piperidin]-2(1H)-one, GLYCEROL, PHOSPHATE ION, ... | 著者 | Niwa, H, Shirai, F, Sato, S, Yoshimoto, N, Tsumura, T, Okue, M, Shirouzu, M, Seimiya, H, Umehara, T. | 登録日 | 2018-04-19 | 公開日 | 2019-04-03 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (2.29 Å) | 主引用文献 | Discovery of Novel Spiroindoline Derivatives as Selective Tankyrase Inhibitors. J. Med. Chem., 62, 2019
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5ZQO
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![BU of 5zqo by Molmil](/molmil-images/mine/5zqo) | Tankyrase-2 in complex with compound 1a | 分子名称: | 2-[4-(2-methoxyphenyl)piperazin-1-yl]-5,6,7,8-tetrahydroquinazolin-4(3H)-one, GLYCEROL, SULFATE ION, ... | 著者 | Niwa, H, Shirai, F, Sato, S, Yoshimoto, N, Tsumura, T, Okue, M, Shirouzu, M, Seimiya, H, Umehara, T. | 登録日 | 2018-04-19 | 公開日 | 2019-04-03 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (2.06 Å) | 主引用文献 | Discovery of Novel Spiroindoline Derivatives as Selective Tankyrase Inhibitors. J. Med. Chem., 62, 2019
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5ZQP
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![BU of 5zqp by Molmil](/molmil-images/mine/5zqp) | Tankyrase-2 in complex with compound 12 | 分子名称: | 1'-(4-oxo-3,4,5,6,7,8-hexahydroquinazolin-2-yl)-2H-spiro[1-benzofuran-3,4'-piperidin]-2-one, GLYCEROL, PHOSPHATE ION, ... | 著者 | Niwa, H, Shirai, F, Sato, S, Yoshimoto, N, Tsumura, T, Okue, M, Shirouzu, M, Seimiya, H, Umehara, T. | 登録日 | 2018-04-19 | 公開日 | 2019-04-03 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (1.99 Å) | 主引用文献 | Discovery of Novel Spiroindoline Derivatives as Selective Tankyrase Inhibitors. J. Med. Chem., 62, 2019
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5ZQR
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![BU of 5zqr by Molmil](/molmil-images/mine/5zqr) | Tankyrase-2 in complex with compound 40c | 分子名称: | 2-[4,6-difluoro-1-(2-hydroxyethyl)-1,2-dihydro-1'H-spiro[indole-3,4'-piperidin]-1'-yl]-5,6,7,8-tetrahydroquinazolin-4(3H)-one, GLYCEROL, PHOSPHATE ION, ... | 著者 | Niwa, H, Shirai, F, Sato, S, Yoshimoto, N, Tsumura, T, Okue, M, Shirouzu, M, Seimiya, H, Umehara, T. | 登録日 | 2018-04-19 | 公開日 | 2019-04-03 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (1.75 Å) | 主引用文献 | Discovery of Novel Spiroindoline Derivatives as Selective Tankyrase Inhibitors. J. Med. Chem., 62, 2019
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6A84
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![BU of 6a84 by Molmil](/molmil-images/mine/6a84) | Tankyrase-2 in complex with compound 15d | 分子名称: | 2-(4-chloro-1,2-dihydro-1'H-spiro[indole-3,4'-piperidin]-1'-yl)-5,6,7,8-tetrahydroquinazolin-4(3H)-one, GLYCEROL, PHOSPHATE ION, ... | 著者 | Niwa, H, Shirai, F, Sato, S, Yoshimoto, N, Tsumura, T, Okue, M, Shirouzu, M, Seimiya, H, Umehara, T. | 登録日 | 2018-07-06 | 公開日 | 2019-04-03 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (1.98 Å) | 主引用文献 | Discovery of Novel Spiroindoline Derivatives as Selective Tankyrase Inhibitors. J. Med. Chem., 62, 2019
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6L6B
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![BU of 6l6b by Molmil](/molmil-images/mine/6l6b) | X-ray structure of human galectin-10 in complex with L-fucose | 分子名称: | Galectin-10, beta-L-fucopyranose | 著者 | Kamitori, S. | 登録日 | 2019-10-28 | 公開日 | 2020-03-04 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (1.802 Å) | 主引用文献 | Structures of human galectin-10/monosaccharide complexes demonstrate potential of monosaccharides as effectors in forming Charcot-Leyden crystals. Biochem.Biophys.Res.Commun., 2020
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6L6C
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![BU of 6l6c by Molmil](/molmil-images/mine/6l6c) | |