4MA3
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![BU of 4ma3 by Molmil](/molmil-images/mine/4ma3) | Crystal structure of anti-hinge rabbit antibody C2095 | 分子名称: | ACETATE ION, C2095 heavy chain, C2095 light chain, ... | 著者 | Malia, T, Teplyakov, A, Gilliland, G.L. | 登録日 | 2013-08-15 | 公開日 | 2014-03-26 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Structure and specificity of an antibody targeting a proteolytically cleaved IgG hinge. Proteins, 82, 2014
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4LPX
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![BU of 4lpx by Molmil](/molmil-images/mine/4lpx) | |
4M6M
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![BU of 4m6m by Molmil](/molmil-images/mine/4m6m) | Crystal structure of anti-IL-23 antibody CNTO1959 at pH 9.5 | 分子名称: | CNTO1959 heavy chain, CNTO1959 light chain, DI(HYDROXYETHYL)ETHER, ... | 著者 | Teplyakov, A, Obmolova, G, Gilliland, G.L. | 登録日 | 2013-08-09 | 公開日 | 2014-03-26 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Antibody modeling assessment II. Structures and models. Proteins, 82, 2014
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4KQ3
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![BU of 4kq3 by Molmil](/molmil-images/mine/4kq3) | Crystal structure of Anti-IL-17A antibody CNTO3186 | 分子名称: | 1,2-ETHANEDIOL, 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, CNTO3186 heavy chain, ... | 著者 | Teplyakov, A, Obmolova, G, Malia, T, Gilliland, G.L. | 登録日 | 2013-05-14 | 公開日 | 2014-03-26 | 最終更新日 | 2019-12-25 | 実験手法 | X-RAY DIFFRACTION (1.92 Å) | 主引用文献 | Structural evidence for a constrained conformation of short CDR-L3 in antibodies. Proteins, 82, 2014
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4KMT
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![BU of 4kmt by Molmil](/molmil-images/mine/4kmt) | Crystal structure of human germline antibody 5-51/O12 | 分子名称: | 2-[N-CYCLOHEXYLAMINO]ETHANE SULFONIC ACID, GLYCEROL, SULFATE ION, ... | 著者 | Teplyakov, A, Obmolova, G, Malia, T, Gilliland, G.L. | 登録日 | 2013-05-08 | 公開日 | 2014-03-26 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | Antibody modeling assessment II. Structures and models. Proteins, 82, 2014
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4KQ4
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![BU of 4kq4 by Molmil](/molmil-images/mine/4kq4) | Crystal structure of Anti-IL-17A antibody CNTO7357 | 分子名称: | CNTO7357 heavy chain, CNTO7357 light chain, NICKEL (II) ION | 著者 | Teplyakov, A, Obmolova, G, Malia, T, Gilliland, G.L. | 登録日 | 2013-05-14 | 公開日 | 2014-03-26 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (2.45 Å) | 主引用文献 | Antibody modeling assessment II. Structures and models. Proteins, 82, 2014
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4LPU
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![BU of 4lpu by Molmil](/molmil-images/mine/4lpu) | |
4LPT
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![BU of 4lpt by Molmil](/molmil-images/mine/4lpt) | |
4MAU
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![BU of 4mau by Molmil](/molmil-images/mine/4mau) | Crystal structure of anti-ST2L antibody C2244 | 分子名称: | C2244 heavy chain, C2244 light chain, FORMIC ACID, ... | 著者 | Teplyakov, A, Obmolova, G, Malia, T, Gilliland, G.L. | 登録日 | 2013-08-16 | 公開日 | 2014-03-26 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Antibody modeling assessment II. Structures and models. Proteins, 82, 2014
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4M6O
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![BU of 4m6o by Molmil](/molmil-images/mine/4m6o) | Crystal structure of anti-NGF antibody CNTO7309 | 分子名称: | 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, CNTO7309 heavy chain, CNTO7309 light chain, ... | 著者 | Teplyakov, A, Obmolova, G, Malia, T, Gilliland, G.L. | 登録日 | 2013-08-09 | 公開日 | 2014-03-26 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (2.8 Å) | 主引用文献 | Antibody modeling assessment II. Structures and models. Proteins, 82, 2014
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6J1M
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![BU of 6j1m by Molmil](/molmil-images/mine/6j1m) | |
6J1N
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![BU of 6j1n by Molmil](/molmil-images/mine/6j1n) | Anisodus acutangulus type III polyketide sythase AaPKS2 in complex with 4-carboxy-3-oxobutanoyl-CoA | 分子名称: | (3R,5R,9R)-1-[(2R,3S,4R,5R)-5-(6-amino-9H-purin-9-yl)-4-hydroxy-3-(phosphonooxy)tetrahydrofuran-2-yl]-3,5,9-trihydroxy-8,8-dimethyl-10,14,19,21-tetraoxo-2,4,6-trioxa-18-thia-11,15-diaza-3,5-diphosphatricosan-23-oic acid 3,5-dioxide (non-preferred name), A. acutangulus PKS2 | 著者 | Fang, C.L, Zhang, Y. | 登録日 | 2018-12-28 | 公開日 | 2019-09-11 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (2.532 Å) | 主引用文献 | Tropane alkaloids biosynthesis involves an unusual type III polyketide synthase and non-enzymatic condensation. Nat Commun, 10, 2019
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6JRX
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![BU of 6jrx by Molmil](/molmil-images/mine/6jrx) | EGFR T790M/C797S in complex with compound 6i | 分子名称: | Epidermal growth factor receptor, N-{trans-4-[3-(2-chlorophenyl)-7-{[3-methyl-4-(4-methylpiperazin-1-yl)phenyl]amino}-2-oxo-3,4-dihydropyrimido[4,5-d]pyrimidin-1(2H)-yl]cyclohexyl}propanamide | 著者 | Zhu, S.J, Yun, C.H. | 登録日 | 2019-04-06 | 公開日 | 2020-04-15 | 最終更新日 | 2024-03-27 | 実験手法 | X-RAY DIFFRACTION (2.201 Å) | 主引用文献 | Design, Synthesis, and Structure-Activity Relationships of 1,2,3-Triazole Benzenesulfonamides as New Selective Leucine-Zipper and Sterile-alpha Motif Kinase (ZAK) Inhibitors. J.Med.Chem., 63, 2020
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6JUU
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![BU of 6juu by Molmil](/molmil-images/mine/6juu) | Crystal structure of ZAK in complex with compound 6r | 分子名称: | Mitogen-activated protein kinase kinase kinase MLT, ~{N}-[2,4-bis(fluoranyl)-3-[4-(3-methoxy-1~{H}-pyrazolo[3,4-b]pyridin-5-yl)-1,2,3-triazol-1-yl]phenyl]naphthalene-1-sulfonamide | 著者 | Kong, L.L, Yun, C.H. | 登録日 | 2019-04-15 | 公開日 | 2020-04-22 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (1.903 Å) | 主引用文献 | Design, Synthesis, and Structure-Activity Relationships of 1,2,3-Triazole Benzenesulfonamides as New Selective Leucine-Zipper and Sterile-alpha Motif Kinase (ZAK) Inhibitors. J.Med.Chem., 63, 2020
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6JUT
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![BU of 6jut by Molmil](/molmil-images/mine/6jut) | Crystal structure of ZAK in complex with compound 6k | 分子名称: | Mitogen-activated protein kinase kinase kinase MLT, ~{N}-[2,4-bis(fluoranyl)-3-[4-(3-methoxy-1~{H}-pyrazolo[3,4-b]pyridin-5-yl)-1,2,3-triazol-1-yl]phenyl]-3-bromanyl-benzenesulfonamide | 著者 | Kong, L.L, Yun, C.H. | 登録日 | 2019-04-15 | 公開日 | 2019-07-24 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | Design, Synthesis, and Structure-Activity Relationships of 1,2,3-Triazole Benzenesulfonamides as New Selective Leucine-Zipper and Sterile-alpha Motif Kinase (ZAK) Inhibitors. J.Med.Chem., 63, 2020
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6AL4
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![BU of 6al4 by Molmil](/molmil-images/mine/6al4) | |
7FBJ
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![BU of 7fbj by Molmil](/molmil-images/mine/7fbj) | Crystal structure of SARS-CoV-2 receptor binding domain in complex with neutralizing nanobody 17F6 | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, New antigen receptor variable domain, ... | 著者 | Zhu, J, Xu, T, Feng, B, Liu, J. | 登録日 | 2021-07-11 | 公開日 | 2022-07-13 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (2.85 Å) | 主引用文献 | A Class of Shark-Derived Single-Domain Antibodies can Broadly Neutralize SARS-Related Coronaviruses and the Structural Basis of Neutralization and Omicron Escape. Small Methods, 6, 2022
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7FBK
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![BU of 7fbk by Molmil](/molmil-images/mine/7fbk) | Crystal structure of SARS-CoV-2 receptor binding domain N501Y mutant in complex with neutralizing nanobody 20G6 | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-[alpha-L-fucopyranose-(1-6)]2-acetamido-2-deoxy-beta-D-glucopyranose, New antigen receptor variable domain, Spike protein S1 | 著者 | Zhu, J, Xu, T, Feng, B, Liu, J. | 登録日 | 2021-07-11 | 公開日 | 2022-07-13 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | A Class of Shark-Derived Single-Domain Antibodies can Broadly Neutralize SARS-Related Coronaviruses and the Structural Basis of Neutralization and Omicron Escape. Small Methods, 6, 2022
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7CA8
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![BU of 7ca8 by Molmil](/molmil-images/mine/7ca8) | The crystal structure of COVID-19 main protease in complex with an inhibitor Shikonin | 分子名称: | 2-[(1R)-4-methyl-1-oxidanyl-pent-3-enyl]-5,8-bis(oxidanyl)naphthalene-1,4-dione, 3C-like proteinase | 著者 | Zhou, X.L, Zhong, F.L, Lin, C, Li, J, Zhang, J. | 登録日 | 2020-06-08 | 公開日 | 2021-04-07 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (2.45 Å) | 主引用文献 | Crystal structure of SARS-CoV-2 main protease in complex with the natural product inhibitor shikonin illuminates a unique binding mode. Sci Bull (Beijing), 66, 2021
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6AL5
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![BU of 6al5 by Molmil](/molmil-images/mine/6al5) | COMPLEX BETWEEN CD19 (N138Q MUTANT) AND B43 FAB | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, B-lymphocyte antigen CD19, B43 HEAVY CHAIN, ... | 著者 | Teplyakov, A, Obmolova, G, Gilliland, G.L. | 登録日 | 2017-08-07 | 公開日 | 2018-03-28 | 最終更新日 | 2023-10-04 | 実験手法 | X-RAY DIFFRACTION (3 Å) | 主引用文献 | Crystal structure of B-cell co-receptor CD19 in complex with antibody B43 reveals an unexpected fold. Proteins, 86, 2018
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7E6M
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![BU of 7e6m by Molmil](/molmil-images/mine/7e6m) | Crystal structure of Human coronavirus NL63 3C-like protease | 分子名称: | 3C-like proteinase | 著者 | Gao, H.X, Zhang, Y.T, Zhong, F.L, Zhou, X.L, Li, J, Zhang, J. | 登録日 | 2021-02-22 | 公開日 | 2021-10-06 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (1.83445024 Å) | 主引用文献 | Crystal structures of human coronavirus NL63 main protease at different pH values Acta Crystallogr.,Sect.F, 77, 2021
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7E6L
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![BU of 7e6l by Molmil](/molmil-images/mine/7e6l) | Crystal structure of HCoV-NL63 3C-like protease,pH5.0 | 分子名称: | 3C-like proteinase | 著者 | Gao, H.X, Zhang, Y.T, Zhou, X.L, Zhong, F.L, Li, J, Zhang, J. | 登録日 | 2021-02-22 | 公開日 | 2021-10-06 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (1.78037143 Å) | 主引用文献 | Crystal structures of human coronavirus NL63 main protease at different pH values Acta Crystallogr.,Sect.F, 77, 2021
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7E6R
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![BU of 7e6r by Molmil](/molmil-images/mine/7e6r) | Crystal structure of HCoV-NL63 3C-like protease,pH5.6 | 分子名称: | 3C-like proteinase | 著者 | Gao, H.X, Zhang, Y.T, Zhong, F.L, Zhou, X.L, Li, J, Zhang, J. | 登録日 | 2021-02-23 | 公開日 | 2021-10-06 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Crystal structures of human coronavirus NL63 main protease at different pH values Acta Crystallogr.,Sect.F, 77, 2021
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7E6N
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![BU of 7e6n by Molmil](/molmil-images/mine/7e6n) | Crystal structure of HCoV-NL63 3C-like protease,pH5.2 | 分子名称: | 3C-like proteinase | 著者 | Gao, H.X, Zhang, Y.T, Zhou, X.L, Zhong, F.L, Li, J, Zhang, J. | 登録日 | 2021-02-22 | 公開日 | 2021-10-06 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (1.8413 Å) | 主引用文献 | Crystal structures of human coronavirus NL63 main protease at different pH values Acta Crystallogr.,Sect.F, 77, 2021
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7VQ2
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![BU of 7vq2 by Molmil](/molmil-images/mine/7vq2) | Structure of Apo-hsTRPM2 channel TM domain | 分子名称: | Transient receptor potential cation channel subfamily M member 2 | 著者 | Yu, X.F, Xie, Y, Zhang, X.K, Ma, C, Guo, J.T, Yang, F, Yang, W. | 登録日 | 2021-10-18 | 公開日 | 2021-12-22 | 実験手法 | ELECTRON MICROSCOPY (3.68 Å) | 主引用文献 | Structural and functional basis of the selectivity filter as a gate in human TRPM2 channel. Cell Rep, 37, 2021
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