7W0K
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![BU of 7w0k by Molmil](/molmil-images/mine/7w0k) | plant glycosyltransferase | 分子名称: | GLYCEROL, Glycosyltransferase, URIDINE-5'-DIPHOSPHATE | 著者 | Wei, H, Feng, L. | 登録日 | 2021-11-18 | 公開日 | 2022-03-02 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (2.04 Å) | 主引用文献 | Functional and Structural Dissection of a Plant Steroid 3-O-Glycosyltransferase Facilitated the Engineering Enhancement of Sugar Donor Promiscuity Acs Catalysis, 2022
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7W1B
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![BU of 7w1b by Molmil](/molmil-images/mine/7w1b) | Glycosyltransferase | 分子名称: | 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, DIGITOXIGENIN, Glycosyltransferase, ... | 著者 | Wei, H, Feng, L. | 登録日 | 2021-11-19 | 公開日 | 2022-03-02 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (2.15 Å) | 主引用文献 | Functional and Structural Dissection of a Plant Steroid 3-O-Glycosyltransferase Facilitated the Engineering Enhancement of Sugar Donor Promiscuity Acs Catalysis, 2022
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2KIU
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![BU of 2kiu by Molmil](/molmil-images/mine/2kiu) | |
5W0Q
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![BU of 5w0q by Molmil](/molmil-images/mine/5w0q) | CREBBP Bromodomain in complex with Cpd17 (N,2,7-trimethyl-2,3-dihydro-4H-benzo[b][1,4]oxazine-4-carboxamide) | 分子名称: | (2R)-N,2,7-trimethyl-2,3-dihydro-4H-1,4-benzoxazine-4-carboxamide, CREB-binding protein, SULFATE ION | 著者 | Murray, J.M. | 登録日 | 2017-05-31 | 公開日 | 2018-03-07 | 最終更新日 | 2023-10-04 | 実験手法 | X-RAY DIFFRACTION (1.7 Å) | 主引用文献 | GNE-781, A Highly Advanced Potent and Selective Bromodomain Inhibitor of Cyclic Adenosine Monophosphate Response Element Binding Protein, Binding Protein (CBP). J. Med. Chem., 60, 2017
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1VZB
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![BU of 1vzb by Molmil](/molmil-images/mine/1vzb) | |
1VZE
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![BU of 1vze by Molmil](/molmil-images/mine/1vze) | L. CASEI THYMIDYLATE SYNTHASE MUTANT E60Q TERNARY COMPLEX WITH DUMP AND CB3717 | 分子名称: | 10-PROPARGYL-5,8-DIDEAZAFOLIC ACID, 2'-DEOXYURIDINE 5'-MONOPHOSPHATE, THYMIDYLATE SYNTHASE | 著者 | Birdsall, D.L, Finer-Moore, J, Stroud, R.M. | 登録日 | 1996-09-18 | 公開日 | 1997-03-12 | 最終更新日 | 2021-11-03 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | The separate effects of E60Q in Lactobacillus casei thymidylate synthase delineate between mechanisms for formation of intermediates in catalysis. Protein Eng., 11, 1998
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1VZD
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![BU of 1vzd by Molmil](/molmil-images/mine/1vzd) | L. CASEI THYMIDYLATE SYNTHASE MUTANT E60Q TERNARY COMPLEX WITH FDUMP AND CB3717 | 分子名称: | 10-PROPARGYL-5,8-DIDEAZAFOLIC ACID, 5-FLUORO-2'-DEOXYURIDINE-5'-MONOPHOSPHATE, THYMIDYLATE SYNTHASE | 著者 | Birdsall, D.L, Finer-Moore, J, Stroud, R.M. | 登録日 | 1996-09-18 | 公開日 | 1997-03-12 | 最終更新日 | 2024-02-14 | 実験手法 | X-RAY DIFFRACTION (2.5 Å) | 主引用文献 | The separate effects of E60Q in Lactobacillus casei thymidylate synthase delineate between mechanisms for formation of intermediates in catalysis. Protein Eng., 11, 1998
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1VZC
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![BU of 1vzc by Molmil](/molmil-images/mine/1vzc) | |
1VZA
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![BU of 1vza by Molmil](/molmil-images/mine/1vza) | |
4U3F
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![BU of 4u3f by Molmil](/molmil-images/mine/4u3f) | Cytochrome bc1 complex from chicken with designed inhibitor bound | 分子名称: | 1,2-dioleoyl-sn-glycero-3-phosphoethanolamine, 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, CARDIOLIPIN, ... | 著者 | Huang, L.-S, Zhu, X.-L, Yang, G.F, Berry, E.A. | 登録日 | 2014-07-21 | 公開日 | 2015-07-29 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (3.2312 Å) | 主引用文献 | Rational Design of Highly Potent and Slow-Binding Cytochrome bc1 Inhibitor as Fungicide by Computational Substitution Optimization Sci Rep, 5, 2015
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4ONA
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![BU of 4ona by Molmil](/molmil-images/mine/4ona) | |
5VOJ
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![BU of 5voj by Molmil](/molmil-images/mine/5voj) | |
7LRF
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![BU of 7lrf by Molmil](/molmil-images/mine/7lrf) | Netrin-1 in complex with SOS | 分子名称: | 1,2-ETHANEDIOL, 1,3,4,6-tetra-O-sulfo-beta-D-fructofuranose-(2-1)-2,3,4,6-tetra-O-sulfonato-alpha-D-glucopyranose, 2-[N-CYCLOHEXYLAMINO]ETHANE SULFONIC ACID, ... | 著者 | Gupta, M, McDougall, M, Torres, A.M, Stetefeld, J. | 登録日 | 2021-02-16 | 公開日 | 2022-02-23 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (3.21 Å) | 主引用文献 | The dynamic nature of netrin-1 and the structural basis for glycosaminoglycan fragment-induced filament formation. Nat Commun, 14, 2023
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7LER
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![BU of 7ler by Molmil](/molmil-images/mine/7ler) | Netrin-1 filament assembly | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Netrin-1, ... | 著者 | McDougall, M, Gupta, M, Stetefeld, J. | 登録日 | 2021-01-14 | 公開日 | 2022-02-23 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (5.99 Å) | 主引用文献 | The dynamic nature of netrin-1 and the structural basis for glycosaminoglycan fragment-induced filament formation. Nat Commun, 14, 2023
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5KU3
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![BU of 5ku3 by Molmil](/molmil-images/mine/5ku3) | BRD4 bromodomain in complex with Cpd59 ((S)-1-(3-((2-fluoro-4-(1-methyl-1H-pyrazol-4-yl)phenyl)amino)-1-(tetrahydrofuran-3-yl)-6,7-dihydro-1H-pyrazolo[4,3-c]pyridin-5(4H)-yl)ethanone) | 分子名称: | 1,2-ETHANEDIOL, 1-[3-[[2-fluoranyl-4-(1-methylpyrazol-4-yl)phenyl]amino]-1-[(3~{S})-oxolan-3-yl]-6,7-dihydro-4~{H}-pyrazolo[4,3-c]pyridin-5-yl]ethanone, Bromodomain-containing protein 4, ... | 著者 | Murray, J.M, Huang, W. | 登録日 | 2016-07-12 | 公開日 | 2016-11-02 | 最終更新日 | 2024-03-06 | 実験手法 | X-RAY DIFFRACTION (1.14 Å) | 主引用文献 | Discovery of a Potent and Selective in Vivo Probe (GNE-272) for the Bromodomains of CBP/EP300. J. Med. Chem., 59, 2016
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1D2B
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![BU of 1d2b by Molmil](/molmil-images/mine/1d2b) | THE MMP-INHIBITORY, N-TERMINAL DOMAIN OF HUMAN TISSUE INHIBITOR OF METALLOPROTEINASES-1 (N-TIMP-1), SOLUTION NMR, 29 STRUCTURES | 分子名称: | Metalloproteinase inhibitor 1 | 著者 | Wu, B, Arumugam, S, Semenchenko, V, Brew, K, Van Doren, S.R. | 登録日 | 1999-09-22 | 公開日 | 1999-12-22 | 最終更新日 | 2022-03-23 | 実験手法 | SOLUTION NMR | 主引用文献 | NMR structure of tissue inhibitor of metalloproteinases-1 implicates localized induced fit in recognition of matrix metalloproteinases. J.Mol.Biol., 295, 2000
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4TZR
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![BU of 4tzr by Molmil](/molmil-images/mine/4tzr) | Calcium-Dependent Protein Kinase 1 from Toxoplasma gondii (TgCDPK1) in complex with inhibitor UW1561 | 分子名称: | 1-{4-amino-3-[2-(cyclopropyloxy)quinolin-6-yl]-1H-pyrazolo[3,4-d]pyrimidin-1-yl}-2-methylpropan-2-ol, Calmodulin-domain protein kinase 1 | 著者 | Merritt, E.A. | 登録日 | 2014-07-10 | 公開日 | 2014-08-27 | 最終更新日 | 2023-12-27 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Development of an Orally Available and Central Nervous System (CNS) Penetrant Toxoplasma gondii Calcium-Dependent Protein Kinase 1 (TgCDPK1) Inhibitor with Minimal Human Ether-a-go-go-Related Gene (hERG) Activity for the Treatment of Toxoplasmosis. J. Med. Chem., 59, 2016
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8CWV
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![BU of 8cwv by Molmil](/molmil-images/mine/8cwv) | |
8CWU
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![BU of 8cwu by Molmil](/molmil-images/mine/8cwu) | |
7BTN
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![BU of 7btn by Molmil](/molmil-images/mine/7btn) | |
8E0G
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![BU of 8e0g by Molmil](/molmil-images/mine/8e0g) | Re-refined model of active mu-opioid receptor (PDB 5c1m) as an adduct with BU72 | 分子名称: | (2R)-2,3-dihydroxypropyl (9Z)-octadec-9-enoate, (2R,3S,3aR,5aR,6R,11bR,11cS)-3a-methoxy-3,14-dimethyl-2-phenyl-2,3,3a,6,7,11c-hexahydro-1H-6,11b-(epiminoethano)-3,5a-methanonaphtho[2,1-g]indol-10-ol, CHOLESTEROL, ... | 著者 | Munro, T.A. | 登録日 | 2022-08-09 | 公開日 | 2023-10-18 | 最終更新日 | 2023-11-15 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | Reanalysis of a mu opioid receptor crystal structure reveals a covalent adduct with BU72. Bmc Biol., 21, 2023
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3KCU
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![BU of 3kcu by Molmil](/molmil-images/mine/3kcu) | Structure of formate channel | 分子名称: | 2-(6-(2-CYCLOHEXYLETHOXY)-TETRAHYDRO-4,5-DIHYDROXY-2(HYDROXYMETHYL)-2H-PYRAN-3-YLOXY)-TETRAHYDRO-6(HYDROXYMETHYL)-2H-PY RAN-3,4,5-TRIOL, Probable formate transporter 1 | 著者 | Wang, Y, Huang, Y, Wang, J, Yan, N, Shi, Y. | 登録日 | 2009-10-22 | 公開日 | 2009-12-01 | 最終更新日 | 2024-03-20 | 実験手法 | X-RAY DIFFRACTION (2.243 Å) | 主引用文献 | Structure of the formate transporter FocA reveals a pentameric aquaporin-like channel Nature, 462, 2009
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3KCV
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![BU of 3kcv by Molmil](/molmil-images/mine/3kcv) | Structure of formate channel | 分子名称: | Probable formate transporter 1 | 著者 | Wang, Y, Huang, Y, Wang, J, Yan, N, Shi, Y. | 登録日 | 2009-10-22 | 公開日 | 2009-12-01 | 最終更新日 | 2023-11-01 | 実験手法 | X-RAY DIFFRACTION (3.198 Å) | 主引用文献 | Structure of the formate transporter FocA reveals a pentameric aquaporin-like channel Nature, 462, 2009
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4APV
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![BU of 4apv by Molmil](/molmil-images/mine/4apv) | The Klebsiella pneumoniae primosomal PriB protein: identification, crystal structure, and ssDNA binding mode | 分子名称: | PRIMOSOMAL REPLICATION PROTEIN N | 著者 | Lo, Y.H, Huang, Y.H, Hsiao, C.D, Huang, C.Y. | 登録日 | 2012-04-06 | 公開日 | 2012-04-25 | 最終更新日 | 2023-12-20 | 実験手法 | X-RAY DIFFRACTION (2.095 Å) | 主引用文献 | Crystal Structure and DNA-Binding Mode of Klebsiella Pneumoniae Primosomal Prib Protein. Genes Cells, 17, 2012
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4R4B
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![BU of 4r4b by Molmil](/molmil-images/mine/4r4b) | Crystal structure of the anti-hiv-1 antibody 2.2c | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, FAB 2.2C HEAVY CHAIN, FAB 2.2C LIGHT CHAIN, ... | 著者 | McLellan, J.S, Acharya, P, Huang, C.-C, Robinson, J, Kwong, P.D. | 登録日 | 2014-08-19 | 公開日 | 2014-09-10 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (2.199 Å) | 主引用文献 | Structural Definition of an Antibody-Dependent Cellular Cytotoxicity Response Implicated in Reduced Risk for HIV-1 Infection. J.Virol., 88, 2014
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