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2VHX
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BU of 2vhx by Molmil
Crystal structure of the ternary complex of L-alanine dehydrogenase from Mycobacterium tuberculosis with NAD+ and pyruvate
分子名称: ALANINE DEHYDROGENASE, MAGNESIUM ION, NICOTINAMIDE-ADENINE-DINUCLEOTIDE, ...
著者Agren, D, Schneider, G.
登録日2007-11-26
公開日2008-03-11
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Three-Dimensional Structures of Apo- and Holo-L-Alanine Dehydrogenase from Mycobacterium Tuberculosis Reveal Conformational Changes Upon Coenzyme Binding.
J.Mol.Biol., 377, 2008
5M35
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BU of 5m35 by Molmil
The molecular tweezer CLR01 stabilizes a disordered protein-protein interface
分子名称: 14-3-3 protein zeta/delta, BENZOIC ACID, GLYCEROL, ...
著者Bier, D, Ottmann, C.
登録日2016-10-14
公開日2017-11-15
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (2.38 Å)
主引用文献The Molecular Tweezer CLR01 Stabilizes a Disordered Protein-Protein Interface.
J. Am. Chem. Soc., 139, 2017
5M39
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BU of 5m39 by Molmil
Crystal structure of BRD4 BROMODOMAIN 1 IN COMPLEX WITH LIGAND 1
分子名称: 6-(3,4-dimethoxyphenyl)-3-methyl-[1,2,4]triazolo[4,3-b]pyridazine, Bromodomain-containing protein 4
著者Kessler, D, Mayer, M, Engelhardt, H, Wolkerstorfer, B, Geist, L.
登録日2016-10-14
公開日2017-09-27
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (1.38 Å)
主引用文献Direct NMR Probing of Hydration Shells of Protein Ligand Interfaces and Its Application to Drug Design.
J. Med. Chem., 60, 2017
1M72
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BU of 1m72 by Molmil
Crystal Structure of Caspase-1 from Spodoptera frugiperda
分子名称: 1,2-ETHANEDIOL, Ace-Asp-Glu-Val-Asp-chloromethylketone, Caspase-1
著者Forsyth, C.M, Lemongello, D, Friesen, P.D, Fisher, A.J.
登録日2002-07-18
公開日2004-01-20
最終更新日2013-02-27
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Crystal structure of an invertebrate caspase.
J.Biol.Chem., 279, 2004
2V9F
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BU of 2v9f by Molmil
L-RHAMNULOSE-1-PHOSPHATE ALDOLASE FROM ESCHERICHIA COLI (MUTANT E192A- K248W-A273S)
分子名称: ACETATE ION, RHAMNULOSE-1-PHOSPHATE ALDOLASE, ZINC ION
著者Grueninger, D, Schulz, G.E.
登録日2007-08-23
公開日2008-01-15
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Designed Protein-Protein Association.
Science, 319, 2008
1MBM
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BU of 1mbm by Molmil
NSP4 proteinase from Equine Arteritis Virus
分子名称: chymotrypsin-like serine protease
著者Barrette-Ng, I.H, Ng, K.K.-S, Mark, B.L, van Aken, D, Cherney, M.M, Garen, C, Kolodenko, Y, Gorbalenya, A.E, Snijder, E.J, James, M.N.G.
登録日2002-08-03
公開日2002-10-23
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Structure of Arterivirus nsp4: the smallest chymotrypsin-like proteinase with an alpha/beta C-terminal extension and alternate conformations of the oxyanion hole
J.Biol.Chem., 277, 2002
1MC7
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BU of 1mc7 by Molmil
Solution Structure of mDvl1 PDZ domain
分子名称: Segment polarity protein dishevelled homolog DVL-1
著者Wong, H.-C, Bourdelas, A, Shao, Y, Wu, D, Shi, D.L, Zheng, J.
登録日2002-08-05
公開日2003-09-23
最終更新日2024-05-22
実験手法SOLUTION NMR
主引用文献Direct binding of the PDZ domain of Dishevelled to a conserved internal sequence in the C-terminal region of Frizzled
Mol.Cell, 12, 2003
2UY6
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BU of 2uy6 by Molmil
Crystal structure of the P pilus rod subunit PapA
分子名称: PAP FIMBRIAL MAJOR PILIN PROTEIN, PERIPLASMID CHAPERONE PAPD PROTEIN
著者Verger, D, Bullitt, E, Hultgren, S.J, Waksman, G.
登録日2007-04-02
公開日2007-05-29
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Crystal Structure of the P Pilus Rod Subunit Papa.
Plos Pathog., 3, 2007
5MG7
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BU of 5mg7 by Molmil
New Insights into the Role of DNA Shape on Its Recognition by p53 Proteins (complex p53DBD-p53R2)
分子名称: Cellular tumor antigen p53, DNA, ZINC ION
著者Rozenberg, H, Braeuning, B, Golovenko, D, Shakked, Z.
登録日2016-11-21
公開日2018-06-13
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (1.45 Å)
主引用文献New Insights into the Role of DNA Shape on Its Recognition by p53 Proteins.
Structure, 26, 2018
5MGF
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BU of 5mgf by Molmil
Crystal Structure of BAZ2B bromodomain in complex with 4-propionyl-pyrrole derivative 2
分子名称: Bromodomain adjacent to zinc finger domain protein 2B, methyl 4-propanoyl-1~{H}-pyrrole-2-carboxylate
著者Lolli, G, Spiliotopoulos, D, Caflisch, A.
登録日2016-11-21
公開日2017-04-12
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Discovery of BAZ2A bromodomain ligands.
Eur J Med Chem, 139, 2017
5MGI
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BU of 5mgi by Molmil
Crystal structure of KPC-2 carbapenemase in complex with a phenyl boronic inhibitor.
分子名称: (~{E})-3-[2-(dihydroxyboranyl)phenyl]prop-2-enoic acid, Carbapenem-hydrolyzing beta-lactamase KPC
著者Vicario, M, Celenza, G, Bellio, P, Perilli, M.G, Tondi, D, Cendron, L.
登録日2016-11-21
公開日2018-03-14
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (1.5 Å)
主引用文献Phenylboronic Acid Derivatives as Validated Leads Active in Clinical Strains Overexpressing KPC-2: A Step against Bacterial Resistance.
Chemmedchem, 13, 2018
2VKG
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BU of 2vkg by Molmil
COMPLEXES OF DODECIN WITH FLAVIN AND FLAVIN-LIKE LIGANDS
分子名称: CHLORIDE ION, DODECIN, MAGNESIUM ION, ...
著者Grininger, M, Noell, G, Trawoeger, S, Sinner, E, Oesterhelt, D.
登録日2007-12-19
公開日2008-09-30
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Electrochemical Switching of the Flavoprotein Dodecin at Gold Surfaces Modified by Flavin-DNA Hybrid Linkers
Biointerphases, 3, 2008
1ML4
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BU of 1ml4 by Molmil
The PALA-liganded Aspartate transcarbamoylase catalytic subunit from Pyrococcus abyssi
分子名称: Aspartate Transcarbamoylase, N-(PHOSPHONACETYL)-L-ASPARTIC ACID
著者Van Boxstael, S, Cunin, R, Maes, D.
登録日2002-08-30
公開日2003-02-25
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Aspartate Transcarbamylase from the Hyperthermophilic Archaeon Pyrococcus abyssi: Thermostability and 1.8A Resolution Crystal Structure of the Catalytic Subunit Complexed With the Bisubstrate Analogue N-Phosphonacetyl-L-aspartate.
J.Mol.Biol., 326, 2003
5MEV
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BU of 5mev by Molmil
MCL1 FAB COMPLEX IN COMPLEX WITH COMPOUND 21
分子名称: (5~{R},13~{S},17~{S})-5-[(3,4-dichlorophenyl)methyl]-8-methyl-13-[(4-methylsulfonylphenyl)methyl]-1,4,8,12,16-pentazatricyclo[15.8.1.0^{20,25}]hexacosa-20,22,24-triene-3,7,15,26-tetrone, Fab Heavy Chain, Fab Light Chain, ...
著者Hargreaves, D.
登録日2016-11-16
公開日2017-01-18
最終更新日2017-03-08
実験手法X-RAY DIFFRACTION (2.94 Å)
主引用文献Structure Based Design of Non-Natural Peptidic Macrocyclic Mcl-1 Inhibitors
Acs Med.Chem.Lett., 8, 2017
5MGM
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BU of 5mgm by Molmil
Crystal Structure of BAZ2A bromodomain in complex with acetophenone derivative 4
分子名称: 1-(3-pyrimidin-2-yloxyphenyl)ethanone, Bromodomain adjacent to zinc finger domain protein 2A
著者Lolli, G, Spiliotopoulos, D, Caflisch, A.
登録日2016-11-21
公開日2017-04-12
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献Discovery of BAZ2A bromodomain ligands.
Eur J Med Chem, 139, 2017
2WSN
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BU of 2wsn by Molmil
Structure of Enhanced Cyan Fluorescent Protein at physiological pH
分子名称: GREEN FLUORESCENT PROTEIN
著者Lelimousin, M, Noirclerc-Savoye, M, Lazareno-Saez, C, Paetzold, B, Le Vot, S, Chazal, R, Macheboeuf, P, Field, M.J, Bourgeois, D, Royant, A.
登録日2009-09-08
公開日2009-09-29
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (1.37 Å)
主引用文献Intrinsic Dynamics in Ecfp and Cerulean Control Fluorescence Quantum Yield.
Biochemistry, 48, 2009
1MN4
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BU of 1mn4 by Molmil
Structure of Ndt80 (Residues 59-340) DNA-binding domain core
分子名称: NDT80 PROTEIN
著者Lamoureux, J.S, Stuart, D, Tsang, R, Wu, C, Glover, J.N.M.
登録日2002-09-04
公開日2002-11-06
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Structure of the sporulation-specific transcription factor Ndt80 bound to DNA
Embo J., 21, 2002
1MOF
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BU of 1mof by Molmil
COAT PROTEIN
分子名称: CHLORIDE ION, MOLONEY MURINE LEUKEMIA VIRUS P15
著者Fass, D, Harrison, S.C, Kim, P.S.
登録日1996-04-02
公開日1996-10-14
最終更新日2022-12-21
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Retrovirus envelope domain at 1.7 angstrom resolution.
Nat.Struct.Biol., 3, 1996
5MMJ
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BU of 5mmj by Molmil
Structure of the small subunit of the chloroplast ribosome
分子名称: 16S ribosomal RNA, 30S ribosomal protein 2, chloroplastic, ...
著者Bieri, P, Leibundgut, M, Saurer, M, Boehringer, D, Ban, N.
登録日2016-12-10
公開日2017-01-11
最終更新日2024-05-15
実験手法ELECTRON MICROSCOPY (3.6 Å)
主引用文献The complete structure of the chloroplast 70S ribosome in complex with translation factor pY.
EMBO J., 36, 2017
1MOZ
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BU of 1moz by Molmil
ADP-ribosylation factor-like 1 (ARL1) from Saccharomyces cerevisiae
分子名称: ADP-ribosylation factor-like protein 1, GUANOSINE-5'-DIPHOSPHATE
著者Amor, J.C, Horton, J.R, Zhu, X, Wang, Y, Sullards, C, Ringe, D, Cheng, X, Kahn, R.A.
登録日2002-09-10
公開日2002-10-09
最終更新日2017-10-11
実験手法X-RAY DIFFRACTION (3.17 Å)
主引用文献Structures of Yeast ARF2 and ARL1: DISTINCT ROLES FOR THE N TERMINUS IN THE STRUCTURE AND FUNCTION OF ARF FAMILY GTPases
J.Biol.Chem., 276, 2001
1MIO
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BU of 1mio by Molmil
X-RAY CRYSTAL STRUCTURE OF THE NITROGENASE MOLYBDENUM-IRON PROTEIN FROM CLOSTRIDIUM PASTEURIANUM AT 3.0 ANGSTROMS RESOLUTION
分子名称: 3-HYDROXY-3-CARBOXY-ADIPIC ACID, CALCIUM ION, FE-MO-S CLUSTER, ...
著者Kim, J, Woo, D, Rees, D.C.
登録日1993-03-24
公開日1993-10-31
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (3 Å)
主引用文献X-ray crystal structure of the nitrogenase molybdenum-iron protein from Clostridium pasteurianum at 3.0-A resolution.
Biochemistry, 32, 1993
1MPV
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BU of 1mpv by Molmil
Structure of bhpBR3, the BAFF-binding loop of BR3 embedded in a beta-hairpin peptide
分子名称: BLyS Receptor 3
著者Kayagaki, N, Yan, M, Seshasayee, D, Wang, H, Lee, W, French, D.M, Grewal, I.S, Cochran, A.G, Gordon, N.C, Yin, J, Starovasnik, M.A, Dixit, V.M.
登録日2002-09-12
公開日2002-10-30
最終更新日2022-02-23
実験手法SOLUTION NMR
主引用文献BAFF/BLyS receptor 3 binds the B cell survival factor BAFF ligand through a discrete surface loop and promotes processing of NF-kappaB2.
Immunity, 17, 2002
2X96
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BU of 2x96 by Molmil
Crystal structure of AnCE-RXPA380 complex
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, ANGIOTENSIN CONVERTING ENZYME, ...
著者Akif, M, Georgiadis, D, Mahajan, A, Dive, V, Sturrock, E.D, Isaac, R.E, Acharya, K.R.
登録日2010-03-14
公開日2010-06-02
最終更新日2020-07-29
実験手法X-RAY DIFFRACTION (1.85 Å)
主引用文献High Resolution Crystal Structures of Drosophila Melanogaster Angiotensin Converting Enzyme in Complex with Novel Inhibitors and Anti- Hypertensive Drugs.
J.Mol.Biol., 400, 2010
5MSG
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BU of 5msg by Molmil
Influenza B polymerase bound to vRNA promoter and capped RNA primer
分子名称: PHOSPHATE ION, Polymerase acidic protein, Polymerase basic protein 2, ...
著者Cusack, S, Guilligay, D.
登録日2017-01-04
公開日2017-02-08
最終更新日2024-03-06
実験手法X-RAY DIFFRACTION (3.8 Å)
主引用文献An in vitro fluorescence based study of initiation of RNA synthesis by influenza B polymerase.
Nucleic Acids Res., 45, 2017
5MQN
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Glycoside hydrolase BT_0986
分子名称: CALCIUM ION, Glycosyl hydrolases family 2, sugar binding domain
著者Basle, A, Ndeh, D, Rogowski, A, Cartmell, A, Luis, A.S, Venditto, I, Labourel, A, Gilbert, H.J.
登録日2016-12-20
公開日2017-03-22
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Complex pectin metabolism by gut bacteria reveals novel catalytic functions.
Nature, 544, 2017

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