3AZ1
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 3az1 by Molmil](/molmil-images/mine/3az1) | Crystal Structure Analysis of Vitamin D receptor | 分子名称: | Vitamin D3 receptor, {4-[3-(4-{[(2R)-2-hydroxy-3,3-dimethylbutyl]oxy}-3-methylphenyl)pentan-3-yl]-2-methylphenoxy}acetic acid | 著者 | Itoh, S, Iijima, S. | 登録日 | 2011-05-20 | 公開日 | 2011-11-02 | 最終更新日 | 2024-03-13 | 実験手法 | X-RAY DIFFRACTION (1.5 Å) | 主引用文献 | Novel nonsecosteroidal vitamin D(3) carboxylic acid analogs for osteoporosis, and SAR analysis. Bioorg.Med.Chem., 19, 2011
|
|
3AZ2
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 3az2 by Molmil](/molmil-images/mine/3az2) | Crystal Structure Analysis of Vitamin D receptor | 分子名称: | 5-{4-[3-(4-{[(2R)-2-hydroxy-3,3-dimethylbutyl]oxy}-3-methylphenyl)pentan-3-yl]-2-methylphenoxy}pentanoic acid, Vitamin D3 receptor | 著者 | Itoh, S, Iijima, S. | 登録日 | 2011-05-20 | 公開日 | 2011-11-02 | 最終更新日 | 2024-03-13 | 実験手法 | X-RAY DIFFRACTION (1.69 Å) | 主引用文献 | Novel nonsecosteroidal vitamin D(3) carboxylic acid analogs for osteoporosis, and SAR analysis. Bioorg.Med.Chem., 19, 2011
|
|
3AZ3
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 3az3 by Molmil](/molmil-images/mine/3az3) | Crystal Structure Analysis of Vitamin D receptor | 分子名称: | (4S)-4-hydroxy-5-[4-(3-{4-[(3S)-3-hydroxy-4,4-dimethylpentyl]-3-methylphenyl}pentan-3-yl)-2-methylphenoxy]pentanoic acid, Vitamin D3 receptor | 著者 | Itoh, S, Iijima, S. | 登録日 | 2011-05-20 | 公開日 | 2011-11-02 | 最終更新日 | 2024-03-13 | 実験手法 | X-RAY DIFFRACTION (1.36 Å) | 主引用文献 | Novel nonsecosteroidal vitamin D(3) carboxylic acid analogs for osteoporosis, and SAR analysis. Bioorg.Med.Chem., 19, 2011
|
|
3A2B
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 3a2b by Molmil](/molmil-images/mine/3a2b) | |
3A4P
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 3a4p by Molmil](/molmil-images/mine/3a4p) | human c-MET kinase domain complexed with 6-benzyloxyquinoline inhibitor | 分子名称: | (2E)-3-{6-[(1R)-1-(2,6-dichloro-3-fluorophenyl)ethoxy]quinolin-3-yl}-N-methylprop-2-enamide, CHLORIDE ION, Hepatocyte growth factor receptor, ... | 著者 | Fukami, T.A, Kadono, S, Yamamuro, M, Matsuura, T. | 登録日 | 2009-07-13 | 公開日 | 2010-02-16 | 最終更新日 | 2023-11-01 | 実験手法 | X-RAY DIFFRACTION (2.54 Å) | 主引用文献 | Discovery of 6-benzyloxyquinolines as c-Met selective kinase inhibitors Bioorg.Med.Chem.Lett., 20, 2010
|
|
6OAP
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 6oap by Molmil](/molmil-images/mine/6oap) | Crystal structure of a dual sensor histidine kinase in the green-light absorbing Pg state | 分子名称: | Dual sensor histidine kinase, MAGNESIUM ION, PHYCOCYANOBILIN | 著者 | Heewhan, S, Zhong, R, Xiaoli, Z, Sepalika, B, Xiaojing, Y. | 登録日 | 2019-03-18 | 公開日 | 2019-09-18 | 最終更新日 | 2023-10-11 | 実験手法 | X-RAY DIFFRACTION (1.97 Å) | 主引用文献 | Structural basis of molecular logic OR in a dual-sensor histidine kinase. Proc.Natl.Acad.Sci.USA, 116, 2019
|
|
6OAQ
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 6oaq by Molmil](/molmil-images/mine/6oaq) | Crystal structure of a dual sensor histidine kinase in BeF3- bound state | 分子名称: | BERYLLIUM TRIFLUORIDE ION, Dual sensor histidine kinase, MAGNESIUM ION, ... | 著者 | Heewhan, S, Zhong, R, Xiaoli, Z, Sepalika, B, Xiaojing, Y. | 登録日 | 2019-03-18 | 公開日 | 2019-09-18 | 最終更新日 | 2023-10-11 | 実験手法 | X-RAY DIFFRACTION (2.54 Å) | 主引用文献 | Structural basis of molecular logic OR in a dual-sensor histidine kinase. Proc.Natl.Acad.Sci.USA, 116, 2019
|
|
6OB8
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 6ob8 by Molmil](/molmil-images/mine/6ob8) | Crystal structure of a dual sensor histidine kinase in green light illuminated state | 分子名称: | Dual sensor histidine kinase, MAGNESIUM ION, PHYCOCYANOBILIN | 著者 | Heewhan, S, Zhong, R, Xiaoli, Z, Sepalika, B, Xiaojing, Y. | 登録日 | 2019-03-19 | 公開日 | 2019-09-18 | 最終更新日 | 2023-10-11 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Structural basis of molecular logic OR in a dual-sensor histidine kinase. Proc.Natl.Acad.Sci.USA, 116, 2019
|
|
8JF5
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 8jf5 by Molmil](/molmil-images/mine/8jf5) | Crystal structure of Lysine Specific Demethylase 1 (LSD1) with TAS1440 | 分子名称: | 4-[5-[(3~{R})-3-azanylpyrrolidin-1-yl]carbonyl-2-[2-fluoranyl-4-(2-methyl-2-oxidanyl-propyl)phenyl]phenyl]-2-fluoranyl-benzenecarbonitrile, FLAVIN-ADENINE DINUCLEOTIDE, GLYCEROL, ... | 著者 | Fukushima, H, Machida, T, Yamashita, S, Suzuki, T. | 登録日 | 2023-05-17 | 公開日 | 2024-05-22 | 実験手法 | X-RAY DIFFRACTION (3.2 Å) | 主引用文献 | TAS1440, a histone H3 competitive LSD1 inhibitor, activates both TGF-beta and notch signaling pathways via INSM1 dissociation in neuroendocrine small cell lung cancer To Be Published
|
|
6J5L
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 6j5l by Molmil](/molmil-images/mine/6j5l) | |
1CMN
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 1cmn by Molmil](/molmil-images/mine/1cmn) | |
2RVM
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 2rvm by Molmil](/molmil-images/mine/2rvm) | |
1CMJ
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 1cmj by Molmil](/molmil-images/mine/1cmj) | |
1CL6
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 1cl6 by Molmil](/molmil-images/mine/1cl6) | |
2RVN
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 2rvn by Molmil](/molmil-images/mine/2rvn) | |
2RVL
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 2rvl by Molmil](/molmil-images/mine/2rvl) | |
2Z2T
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 2z2t by Molmil](/molmil-images/mine/2z2t) | |
6JRQ
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 6jrq by Molmil](/molmil-images/mine/6jrq) | Crystal structure of adenylosuccinate synthetase, PurA, from Thermus thermophilus | 分子名称: | 1,2-ETHANEDIOL, Adenylosuccinate synthetase, INOSINIC ACID | 著者 | Sampei, G, Kawai, G, RIKEN Structural Genomics/Proteomics Initiative (RSGI) | 登録日 | 2019-04-05 | 公開日 | 2020-04-08 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | Crystal structure of adenylosuccinate synthetase, PurA, from Thermus thermophilus HB8 To Be Published
|
|
2Z5E
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 2z5e by Molmil](/molmil-images/mine/2z5e) | Crystal Structure of Proteasome Assembling Chaperone 3 | 分子名称: | Proteasome Assembling Chaperone 3 | 著者 | Okamoto, K, Kurimoto, E, Sakata, E, Suzuki, A, Yamane, T, Hirano, Y, Murata, S, Tanaka, K, Kato, K. | 登録日 | 2007-07-06 | 公開日 | 2008-02-19 | 最終更新日 | 2024-03-13 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Crystal structure of a chaperone complex that contributes to the assembly of yeast 20S proteasomes Nat.Struct.Mol.Biol., 15, 2008
|
|
3W0C
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 3w0c by Molmil](/molmil-images/mine/3w0c) | Crystal Structure Analysis of Vitamin D receptor | 分子名称: | (4S)-4-hydroxy-5-[2-methyl-4-(3-{3-methyl-4-[(1E)-4,4,4-trifluoro-3-hydroxy-3-(trifluoromethyl)but-1-en-1-yl]phenyl}pentan-3-yl)phenoxy]pentanoic acid, Vitamin D3 receptor | 著者 | Itoh, S, Iijima, S. | 登録日 | 2012-10-29 | 公開日 | 2013-11-13 | 最終更新日 | 2024-03-20 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | structure analysis of vitamin D receptor To be Published
|
|
3W0A
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 3w0a by Molmil](/molmil-images/mine/3w0a) | Crystal Structure Analysis of Vitamin D receptor | 分子名称: | (4S)-4-hydroxy-5-[2-methyl-4-(3-{3-methyl-4-[4,4,4-trifluoro-3-hydroxy-3-(trifluoromethyl)but-1-yn-1-yl]phenyl}pentan-3-yl)phenoxy]pentanoic acid, Vitamin D3 receptor | 著者 | Itoh, S, Iijima, S. | 登録日 | 2012-10-25 | 公開日 | 2013-11-13 | 最終更新日 | 2024-03-20 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | structure analysis of vitamin D3 receptor To be Published
|
|
2O3Z
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 2o3z by Molmil](/molmil-images/mine/2o3z) | X-ray crystal structure of LpxC complexed with 3-heptyloxybenzoate | 分子名称: | 3-(heptyloxy)benzoic acid, CHLORIDE ION, SULFATE ION, ... | 著者 | Gennadios, H.A, Whittington, D.A, Christianson, D.W. | 登録日 | 2006-12-02 | 公開日 | 2007-02-27 | 最終更新日 | 2023-08-30 | 実験手法 | X-RAY DIFFRACTION (2.25 Å) | 主引用文献 | Amphipathic benzoic acid derivatives: synthesis and binding in the hydrophobic tunnel of the zinc deacetylase LpxC. Bioorg.Med.Chem., 15, 2007
|
|
3UNC
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 3unc by Molmil](/molmil-images/mine/3unc) | Crystal Structure of Bovine Milk Xanthine Dehydrogenase to 1.65A Resolution | 分子名称: | 2-HYDROXYBENZOIC ACID, CALCIUM ION, CARBONATE ION, ... | 著者 | Eger, B.T, Okamoto, K, Nishino, T, Pai, E.F. | 登録日 | 2011-11-15 | 公開日 | 2012-05-09 | 最終更新日 | 2023-09-13 | 実験手法 | X-RAY DIFFRACTION (1.65 Å) | 主引用文献 | Protein conformational gating of enzymatic activity in xanthine oxidoreductase. J.Am.Chem.Soc., 134, 2012
|
|
3VYV
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 3vyv by Molmil](/molmil-images/mine/3vyv) | Crystal structure of subtilisin NAT at 1.36 | 分子名称: | CALCIUM ION, GLYCEROL, Subtilisin NAT | 著者 | Ushijima, H, Fuchita, N, Kajiwara, T, Motoshima, H, Ueno, G, Watanabe, K. | 登録日 | 2012-10-03 | 公開日 | 2013-10-09 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (1.36 Å) | 主引用文献 | Crystal structure of subtilisin NAT at 1.36 TO BE PUBLISHED
|
|
3UNI
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 3uni by Molmil](/molmil-images/mine/3uni) | Crystal Structure of Bovine Milk Xanthine Dehydrogenase with NADH Bound | 分子名称: | 1,4-DIHYDRONICOTINAMIDE ADENINE DINUCLEOTIDE, 2-HYDROXYBENZOIC ACID, CALCIUM ION, ... | 著者 | Eger, B.T, Okamoto, K, Nishino, T, Pai, E.F. | 登録日 | 2011-11-15 | 公開日 | 2012-05-09 | 最終更新日 | 2023-09-13 | 実験手法 | X-RAY DIFFRACTION (2.2 Å) | 主引用文献 | Protein conformational gating of enzymatic activity in xanthine oxidoreductase. J.Am.Chem.Soc., 134, 2012
|
|