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2Z2T

Crystal structure of the complex between gp41 fragment N36 and fusion inhibitor SC34EK

Summary for 2Z2T
Entry DOI10.2210/pdb2z2t/pdb
Descriptorgp41 fragment N36, Fusion inhibitor peptide SC34EK, ACETIC ACID, ... (5 entities in total)
Functional Keywordscoiled-coil, viral protein-inhibitor complex, viral protein/inhibitor
Total number of polymer chains6
Total formula weight26015.82
Authors
Nakamura, S.,Ohkubo, T.,Kobayashi, Y. (deposition date: 2007-05-28, release date: 2008-06-03, Last modification date: 2023-11-15)
Primary citationNishikawa, H.,Nakamura, S.,Kodama, E.,Ito, S.,Kajiwara, K.,Izumi, K.,Sakagami, Y.,Oishi, S.,Ohkubo, T.,Kobayashi, Y.,Fujii, N.,Matsuoka, M.
Intrahelical Salt-bridges in a-Helical Peptide Enhances its Binding to the Target: A New Design for HIV-1 Fusion Inhibitors
To be Published,
Experimental method
X-RAY DIFFRACTION (2.1 Å)
Structure validation

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