8AUR
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8AW4
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7Q1E
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![BU of 7q1e by Molmil](/molmil-images/mine/7q1e) | CPAP:TUBULIN:IIH5 ALPHAREP COMPLEX | 分子名称: | Centromere protein J, GLYCEROL, GUANOSINE-5'-TRIPHOSPHATE, ... | 著者 | Campanacci, V, Gigant, b. | 登録日 | 2021-10-19 | 公開日 | 2022-04-13 | 最終更新日 | 2024-01-31 | 実験手法 | X-RAY DIFFRACTION (2.7 Å) | 主引用文献 | Structural convergence for tubulin binding of CPAP and vinca domain microtubule inhibitors. Proc.Natl.Acad.Sci.USA, 119, 2022
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7Q1F
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![BU of 7q1f by Molmil](/molmil-images/mine/7q1f) | CPAP:TUBULIN:IE5 ALPHAREP COMPLEX | 分子名称: | 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, CITRATE ANION, Centromere protein J, ... | 著者 | Campanacci, V, Gigant, b. | 登録日 | 2021-10-19 | 公開日 | 2022-04-20 | 最終更新日 | 2024-01-31 | 実験手法 | X-RAY DIFFRACTION (2.347 Å) | 主引用文献 | Structural convergence for tubulin binding of CPAP and vinca domain microtubule inhibitors. Proc.Natl.Acad.Sci.USA, 119, 2022
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7Z0G
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![BU of 7z0g by Molmil](/molmil-images/mine/7z0g) | CPAP:TUBULIN:IE5 ALPHAREP COMPLEX P1 SPACE GROUP | 分子名称: | 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, Centromere protein J, GUANOSINE-5'-DIPHOSPHATE, ... | 著者 | Gigant, B, Campanacci, V. | 登録日 | 2022-02-22 | 公開日 | 2022-04-13 | 最終更新日 | 2024-01-31 | 実験手法 | X-RAY DIFFRACTION (3.487 Å) | 主引用文献 | Structural convergence for tubulin binding of CPAP and vinca domain microtubule inhibitors. Proc.Natl.Acad.Sci.USA, 119, 2022
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7Z0F
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![BU of 7z0f by Molmil](/molmil-images/mine/7z0f) | CPAP:S-TUBULIN:IIH5 ALPHAREP COMPLEX | 分子名称: | Centromere protein J, GLYCEROL, GUANOSINE-5'-DIPHOSPHATE, ... | 著者 | Gigant, B, Campanacci, V. | 登録日 | 2022-02-22 | 公開日 | 2022-04-13 | 最終更新日 | 2024-01-31 | 実験手法 | X-RAY DIFFRACTION (2.396 Å) | 主引用文献 | Structural convergence for tubulin binding of CPAP and vinca domain microtubule inhibitors. Proc.Natl.Acad.Sci.USA, 119, 2022
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6XN6
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6XPA
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7F9F
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![BU of 7f9f by Molmil](/molmil-images/mine/7f9f) | Thrombocorticin | 分子名称: | MAGNESIUM ION, Thrombocorticin | 著者 | Kageyama, H, Onodera, K, Sakai, R, Tanaka, Y, Freymann, D.M. | 登録日 | 2021-07-04 | 公開日 | 2022-07-06 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (1.411 Å) | 主引用文献 | A marine sponge-derived lectin reveals hidden pathway for thrombopoietin receptor activation. Nat Commun, 13, 2022
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7F9G
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![BU of 7f9g by Molmil](/molmil-images/mine/7f9g) | Thrombocorticin in complex with Ca2+ and fucose | 分子名称: | CALCIUM ION, Thrombocorticin, alpha-L-fucopyranose | 著者 | Kageyama, H, Onodera, K, Sakai, R, Tanaka, Y. | 登録日 | 2021-07-04 | 公開日 | 2022-07-06 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (1.331 Å) | 主引用文献 | A marine sponge-derived lectin reveals hidden pathway for thrombopoietin receptor activation. Nat Commun, 13, 2022
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7F9J
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![BU of 7f9j by Molmil](/molmil-images/mine/7f9j) | Thrombocorticin Q25K in complex with Ca2+ | 分子名称: | CALCIUM ION, Thrombocorticin Q25K mutant | 著者 | Kageyama, H, Onodera, K, Sakai, R, Tanaka, Y. | 登録日 | 2021-07-04 | 公開日 | 2022-07-06 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (1.1 Å) | 主引用文献 | A marine sponge-derived lectin reveals hidden pathway for thrombopoietin receptor activation. Nat Commun, 13, 2022
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7F91
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7FBL
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![BU of 7fbl by Molmil](/molmil-images/mine/7fbl) | Thrombocorticin in complex with Ca2+ and mannose | 分子名称: | CALCIUM ION, Thrombocorticin, alpha-D-mannopyranose | 著者 | Kageyama, H, Onodera, K, Sakai, R, Tanaka, Y. | 登録日 | 2021-07-11 | 公開日 | 2022-07-13 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (1.419 Å) | 主引用文献 | A marine sponge-derived lectin reveals hidden pathway for thrombopoietin receptor activation. Nat Commun, 13, 2022
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7QDL
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![BU of 7qdl by Molmil](/molmil-images/mine/7qdl) | N-TERMINAL BROMODOMAIN OF HUMAN BRD4 with I-BET567 | 分子名称: | (2S,4R)-1-acetyl-4-((5-chloropyrimidin-2-yl)amino)-2-methyl-1,2,3,4-tetrahydroquinoline-6-carboxamide, 1,2-ETHANEDIOL, Bromodomain-containing protein 4 | 著者 | Chung, C. | 登録日 | 2021-11-27 | 公開日 | 2022-12-14 | 最終更新日 | 2024-05-01 | 実験手法 | X-RAY DIFFRACTION (1.67 Å) | 主引用文献 | Design, Synthesis, and Characterization of I-BET567, a Pan-Bromodomain and Extra Terminal (BET) Bromodomain Oral Candidate. J.Med.Chem., 65, 2022
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4YJP
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![BU of 4yjp by Molmil](/molmil-images/mine/4yjp) | THE KINASE DOMAIN OF HUMAN SPLEEN TYROSINE (SYK) IN COMPLEX WITH GTC000223 | 分子名称: | 2-[{2-[(1,1-dioxido-2,3-dihydro-1,2-benzothiazol-6-yl)amino]pyrimidin-4-yl}(1H-indazol-4-yl)amino]ethanol, DIMETHYL SULFOXIDE, Tyrosine-protein kinase SYK | 著者 | Somers, D.O, Neu, M. | 登録日 | 2015-03-03 | 公開日 | 2015-09-30 | 最終更新日 | 2024-05-01 | 実験手法 | X-RAY DIFFRACTION (1.83 Å) | 主引用文献 | Discovery of GSK143, a highly potent, selective and orally efficacious spleen tyrosine kinase inhibitor. Bioorg. Med. Chem. Lett., 21, 2011
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4YJU
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![BU of 4yju by Molmil](/molmil-images/mine/4yju) | THE KINASE DOMAIN OF HUMAN SPLEEN TYROSINE (SYK) IN COMPLEX WITH GTC000249 | 分子名称: | N~2~-(1,1-dioxido-2,3-dihydro-1,2-benzothiazol-6-yl)-5-fluoro-N~4~-(1H-indazol-4-yl)-N~4~-methylpyrimidine-2,4-diamine, Tyrosine-protein kinase SYK | 著者 | Somers, D.O, Neu, M, Stuckey, J. | 登録日 | 2015-03-03 | 公開日 | 2015-09-30 | 最終更新日 | 2024-05-01 | 実験手法 | X-RAY DIFFRACTION (1.67 Å) | 主引用文献 | Discovery of GSK143, a highly potent, selective and orally efficacious spleen tyrosine kinase inhibitor. Bioorg. Med. Chem. Lett., 21, 2011
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4YJT
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![BU of 4yjt by Molmil](/molmil-images/mine/4yjt) | THE KINASE DOMAIN OF HUMAN SPLEEN TYROSINE (SYK) IN COMPLEX WITH GTC000233 | 分子名称: | GLYCEROL, N~2~-(1,1-dioxido-2,3-dihydro-1,2-benzothiazol-6-yl)-N~4~-ethyl-5-fluoro-N~4~-(1H-indazol-4-yl)pyrimidine-2,4-diamine, Tyrosine-protein kinase SYK | 著者 | Somers, D.O, Neu, M, Stuckey, J. | 登録日 | 2015-03-03 | 公開日 | 2015-09-30 | 最終更新日 | 2024-05-01 | 実験手法 | X-RAY DIFFRACTION (1.52 Å) | 主引用文献 | Discovery of GSK143, a highly potent, selective and orally efficacious spleen tyrosine kinase inhibitor. Bioorg. Med. Chem. Lett., 21, 2011
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4YJR
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![BU of 4yjr by Molmil](/molmil-images/mine/4yjr) | SYK kinase domain in complex with inhibitor GTC000225 | 分子名称: | 3-(1H-indazol-4-yl{2-[(1-methyl-1H-indazol-5-yl)amino]pyrimidin-4-yl}amino)propan-1-ol, Tyrosine-protein kinase SYK | 著者 | Somers, D.O, Neu, M, Stuckey, J. | 登録日 | 2015-03-03 | 公開日 | 2015-09-30 | 最終更新日 | 2024-05-01 | 実験手法 | X-RAY DIFFRACTION (1.32 Å) | 主引用文献 | Discovery of GSK143, a highly potent, selective and orally efficacious spleen tyrosine kinase inhibitor. Bioorg. Med. Chem. Lett., 21, 2011
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4YJQ
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![BU of 4yjq by Molmil](/molmil-images/mine/4yjq) | SYK kinase domain in complex with inhibitor GTC000224 | 分子名称: | 3-[1H-indazol-4-yl(2-{[3-(4-methyl-1,3-oxazol-5-yl)phenyl]amino}pyrimidin-4-yl)amino]propan-1-ol, Tyrosine-protein kinase SYK | 著者 | Somers, D.O, Neu, M, Stuckey, J. | 登録日 | 2015-03-03 | 公開日 | 2015-09-30 | 最終更新日 | 2024-05-01 | 実験手法 | X-RAY DIFFRACTION (1.34 Å) | 主引用文献 | Discovery of GSK143, a highly potent, selective and orally efficacious spleen tyrosine kinase inhibitor. Bioorg. Med. Chem. Lett., 21, 2011
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5GU7
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![BU of 5gu7 by Molmil](/molmil-images/mine/5gu7) | Crystal Structure of human ERp44 form II | 分子名称: | Endoplasmic reticulum resident protein 44 | 著者 | Watanabe, S, Inaba, K. | 登録日 | 2016-08-26 | 公開日 | 2017-04-12 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (2.05 Å) | 主引用文献 | Structural basis of pH-dependent client binding by ERp44, a key regulator of protein secretion at the ER-Golgi interface Proc. Natl. Acad. Sci. U.S.A., 114, 2017
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5GU6
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![BU of 5gu6 by Molmil](/molmil-images/mine/5gu6) | Crystal structure of Human ERp44 form I | 分子名称: | CHLORIDE ION, Endoplasmic reticulum resident protein 44 | 著者 | Watanabe, S, Inaba, K. | 登録日 | 2016-08-26 | 公開日 | 2017-04-12 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Structural basis of pH-dependent client binding by ERp44, a key regulator of protein secretion at the ER-Golgi interface Proc. Natl. Acad. Sci. U.S.A., 114, 2017
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4YJO
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![BU of 4yjo by Molmil](/molmil-images/mine/4yjo) | THE KINASE DOMAIN OF HUMAN SPLEEN TYROSINE (SYK) IN COMPLEX WITH GTC000222 | 分子名称: | 5-chloro-N~2~-(1,1-dioxido-2,3-dihydro-1,2-benzothiazol-6-yl)-N~4~-ethyl-N~4~-(1H-indazol-4-yl)pyrimidine-2,4-diamine, GLYCEROL, Tyrosine-protein kinase SYK | 著者 | Somers, D.O, Neu, M. | 登録日 | 2015-03-03 | 公開日 | 2015-09-30 | 最終更新日 | 2024-05-01 | 実験手法 | X-RAY DIFFRACTION (1.6 Å) | 主引用文献 | Discovery of GSK143, a highly potent, selective and orally efficacious spleen tyrosine kinase inhibitor. Bioorg. Med. Chem. Lett., 21, 2011
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4YJV
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8PSD
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![BU of 8psd by Molmil](/molmil-images/mine/8psd) | SARS-CoV-2 XBB 1.0 closed conformation. | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, Spike glycoprotein | 著者 | Duhoo, Y, Lau, K. | 登録日 | 2023-07-13 | 公開日 | 2023-11-01 | 最終更新日 | 2023-12-06 | 実験手法 | ELECTRON MICROSCOPY (2.9 Å) | 主引用文献 | Broadly potent anti-SARS-CoV-2 antibody shares 93% of epitope with ACE2 and provides full protection in monkeys. J Infect, 87, 2023
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8PQ2
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![BU of 8pq2 by Molmil](/molmil-images/mine/8pq2) | XBB 1.0 RBD bound to P4J15 (Local) | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, P4J15 Fragment Antigen-Binding Heavy Chain, P4J15 Fragment Antigen-Binding Light Chain, ... | 著者 | Duhoo, Y, Lau, K. | 登録日 | 2023-07-10 | 公開日 | 2023-11-01 | 最終更新日 | 2023-12-06 | 実験手法 | ELECTRON MICROSCOPY (3.85 Å) | 主引用文献 | Broadly potent anti-SARS-CoV-2 antibody shares 93% of epitope with ACE2 and provides full protection in monkeys. J Infect, 87, 2023
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