1X29
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1Y37
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7DCF
| Crystal structure of EHMT2 SET domain in complex with compound 10 | 分子名称: | 5'-methoxy-6'-(1-methyl-2,3,4,7-tetrahydroazepin-5-yl)spiro[cyclobutane-1,3'-indole]-2'-amine, Histone-lysine N-methyltransferase EHMT2, S-ADENOSYLMETHIONINE, ... | 著者 | Suzuki, M, Katayama, K. | 登録日 | 2020-10-26 | 公開日 | 2021-02-10 | 最終更新日 | 2024-03-27 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | Discovery of DS79932728: A Potent, Orally Available G9a/GLP Inhibitor for Treating beta-Thalassemia and Sickle Cell Disease. Acs Med.Chem.Lett., 12, 2021
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1G4X
| ASPARTATE AMINOTRANSFERASE ACTIVE SITE MUTANT N194A/R292L | 分子名称: | ASPARTATE AMINOTRANSFERASE, PYRIDOXAL-5'-PHOSPHATE | 著者 | Mizuguchi, H. | 登録日 | 2000-10-29 | 公開日 | 2000-11-22 | 最終更新日 | 2021-10-27 | 実験手法 | X-RAY DIFFRACTION (2.2 Å) | 主引用文献 | Strain is more important than electrostatic interaction in controlling the pKa of the catalytic group in aspartate aminotransferase. Biochemistry, 40, 2001
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1UIM
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1UIN
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1V2E
| |
1VB3
| |
1V7C
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1V2F
| |
1V72
| |
1VC3
| |
1VCO
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1VE4
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1VCM
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1VCN
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1V2D
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1X2A
| |
2COG
| |
2COI
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2DVX
| |
2DVT
| |
2COJ
| |
2EEO
| |
2DVU
| |