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5XPR
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BU of 5xpr by Molmil
Human endothelin receptor type-B in complex with antagonist bosentan
分子名称: 4-tert-butyl-N-[6-(2-hydroxyethyloxy)-5-(2-methoxyphenoxy)-2-pyrimidin-2-yl-pyrimidin-4-yl]benzenesulfonamide, Endothelin B receptor,Endolysin,Endothelin B receptor, SULFATE ION
著者Shihoya, W, Nishizawa, T, Yamashita, K, Hirata, K, Okuta, A, Tani, K, Fujiyoshi, Y, Doi, T, Nureki, O.
登録日2017-06-04
公開日2017-08-16
最終更新日2024-10-16
実験手法X-RAY DIFFRACTION (3.6 Å)
主引用文献X-ray structures of endothelin ETB receptor bound to clinical antagonist bosentan and its analog
Nat. Struct. Mol. Biol., 24, 2017
1ISE
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BU of 1ise by Molmil
Crystal structure of a mutant of ribosome recycling factor from Escherichia coli, Arg132Gly
分子名称: Ribosome Recycling Factor
著者Nakano, H, Yoshida, T, Oka, S, Uchiyama, S, Nishina, K, Ohkubo, T, Kato, H, Yamagata, Y, Kobayashi, Y.
登録日2001-11-30
公開日2003-10-07
最終更新日2023-12-27
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Crystal structure of a mutant of ribosome recycling factor from Escherichia coli, Arg132Gly
To be Published
1IR7
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BU of 1ir7 by Molmil
IM mutant of lysozyme
分子名称: lysozyme
著者Ohmura, T, Ueda, T, Hashimoto, Y, Imoto, T.
登録日2001-09-19
公開日2001-10-03
最終更新日2024-10-16
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Tolerance of point substitution of methionine for isoleucine in hen egg white lysozyme.
Protein Eng., 14, 2001
1IR9
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BU of 1ir9 by Molmil
IM mutant of lysozyme
分子名称: lysozyme
著者Ohmura, T, Ueda, T, Hashimoto, Y, Imoto, T.
登録日2001-09-19
公開日2001-10-03
最終更新日2023-12-27
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Tolerance of point substitution of methionine for isoleucine in hen egg white lysozyme.
Protein Eng., 14, 2001
1EWT
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BU of 1ewt by Molmil
CRYSTAL STRUCTURE OF METABOTROPIC GLUTAMATE RECEPTOR SUBTYPE 1 LIGAND FREE FORM I
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, METABOTROPIC GLUTAMATE RECEPTOR SUBTYPE 1, SULFATE ION
著者Kunishima, N, Shimada, Y, Tsuji, Y, Jingami, H, Morikawa, K.
登録日2000-04-27
公開日2000-12-18
最終更新日2024-10-16
実験手法X-RAY DIFFRACTION (3.7 Å)
主引用文献Structural basis of glutamate recognition by a dimeric metabotropic glutamate receptor.
Nature, 407, 2000
1IYX
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BU of 1iyx by Molmil
Crystal structure of enolase from Enterococcus hirae
分子名称: ENOLASE, GLYCEROL, MAGNESIUM ION, ...
著者Hosaka, T, Meguro, T, Yamato, I, Shirakihara, Y.
登録日2002-09-12
公開日2003-07-29
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献Crystal Structure of Enterococcus hirae Enolase at 2.8 A Resolution
J.BIOCHEM.(TOKYO), 133, 2003
1IO7
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BU of 1io7 by Molmil
THERMOPHILIC CYTOCHROME P450 (CYP119) FROM SULFOLOBUS SOLFATARICUS: HIGH RESOLUTION STRUCTURAL ORIGIN OF ITS THERMOSTABILITY AND FUNCTIONAL PROPERTIES
分子名称: CYTOCHROME P450 CYP119, PROTOPORPHYRIN IX CONTAINING FE
著者Park, S.-Y, Yamane, K, Adachi, S, Shiro, Y, Sligar, S.G, RIKEN Structural Genomics/Proteomics Initiative (RSGI)
登録日2001-02-08
公開日2001-02-28
最終更新日2023-12-27
実験手法X-RAY DIFFRACTION (1.5 Å)
主引用文献Thermophilic cytochrome P450 (CYP119) from Sulfolobus solfataricus: high resolution structure and functional properties.
J.Inorg.Biochem., 91, 2002
8H8Q
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BU of 8h8q by Molmil
Fab-amyloid beta fragment complex at neutral pH
分子名称: CHLORIDE ION, Fab, GLN-LYS-CYS-VAL-PHE-PHE-ALA-GLU-ASP-VAL-GLY-SER-ASN-CYS-GLY, ...
著者Kita, A, Irie, K, Irie, Y, Matsushima, Y, Miki, K.
登録日2022-10-24
公開日2023-10-25
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Fab-amyloid beta fragment complex at neutral pH
To Be Published
8GCL
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BU of 8gcl by Molmil
Cryo-EM structure of hAQP2 in DDM
分子名称: Aquaporin-2
著者Kamegawa, A, Suzuki, S, Nishikawa, K, Numoto, N, Suzuki, H, Fujiyoshi, Y.
登録日2023-03-02
公開日2023-06-21
最終更新日2024-06-19
実験手法ELECTRON MICROSCOPY (2.89 Å)
主引用文献Structural analysis of the water channel AQP2 by single-particle cryo-EM.
J.Struct.Biol., 215, 2023
3UYW
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BU of 3uyw by Molmil
Crystal structures of globular head of 2009 pandemic H1N1 hemagglutinin
分子名称: 2-AMINOETHANESULFONIC ACID, Hemagglutinin
著者Xuan, C.L, Shi, Y, Qi, J.X, Xiao, H.X, Gao, G.F.
登録日2011-12-06
公開日2012-10-24
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (1.903 Å)
主引用文献Structural vaccinology: structure-based design of influenza A virus hemagglutinin subtype-specific subunit vaccines
Protein Cell, 2, 2011
4TQU
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BU of 4tqu by Molmil
Crystal structure of a bacterial ABC transporter involved in the import of the acidic polysaccharide alginate
分子名称: 4-deoxy-alpha-L-erythro-hex-4-enopyranuronic acid-(1-4)-beta-D-mannopyranuronic acid-(1-4)-beta-D-mannopyranuronic acid-(1-4)-beta-D-mannopyranuronic acid, AlgM1, AlgM2, ...
著者Maruyama, Y, Itoh, T, Kaneko, A, Nishitani, Y, Mikami, B, Hashimoto, W, Murata, K.
登録日2014-06-12
公開日2015-07-22
最終更新日2024-03-20
実験手法X-RAY DIFFRACTION (3.204 Å)
主引用文献Structure of a Bacterial ABC Transporter Involved in the Import of an Acidic Polysaccharide Alginate
Structure, 23, 2015
3UO8
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BU of 3uo8 by Molmil
Crystal structure of the MALT1 paracaspase (P1 form)
分子名称: Mucosa-associated lymphoid tissue lymphoma translocation protein 1, Z-Val-Arg-Pro-DL-Arg-fluoromethylketone
著者Jeffrey, P.D, Yu, J.W, Shi, Y.
登録日2011-11-16
公開日2011-12-21
最終更新日2024-03-20
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Crystal structure of the mucosa-associated lymphoid tissue lymphoma translocation 1 (MALT1) paracaspase region.
Proc.Natl.Acad.Sci.USA, 108, 2011
3UYX
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BU of 3uyx by Molmil
Crystal structures of globular head of 2009 pandemic H1N1 hemagglutinin
分子名称: Hemagglutinin, NITRATE ION
著者Xuan, C.L, Shi, Y, Qi, J.X, Xiao, H.X, Gao, G.F.
登録日2011-12-06
公開日2012-10-24
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Structural vaccinology: structure-based design of influenza A virus hemagglutinin subtype-specific subunit vaccines
Protein Cell, 2, 2011
5ZLG
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BU of 5zlg by Molmil
Human duodenal cytochrome b (Dcytb) in zinc ion and ascorbate bound form
分子名称: ASCORBIC ACID, Cytochrome b reductase 1, PROTOPORPHYRIN IX CONTAINING FE, ...
著者Ganasen, M, Togashi, H, Mauk, G.A, Shiro, Y, Sawai, H, Sugimoto, H.
登録日2018-03-27
公開日2018-10-31
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献Structural basis for promotion of duodenal iron absorption by enteric ferric reductase with ascorbate.
Commun Biol, 1, 2018
1EWV
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BU of 1ewv by Molmil
CRYSTAL STRUCTURE OF METABOTROPIC GLUTAMATE RECEPTOR SUBTYPE 1 LIGAND FREE FORM II
分子名称: METABOTROPIC GLUTAMATE RECEPTOR SUBTYPE 1
著者Kunishima, N, Shimada, Y, Tsuji, Y, Jingami, H, Morikawa, K.
登録日2000-04-27
公開日2000-12-18
最終更新日2023-08-09
実験手法X-RAY DIFFRACTION (4 Å)
主引用文献Structural basis of glutamate recognition by a dimeric metabotropic glutamate receptor.
Nature, 407, 2000
3YGS
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BU of 3ygs by Molmil
APAF-1 CARD IN COMPLEX WITH PRODOMAIN OF PROCASPASE-9
分子名称: APOPTOTIC PROTEASE ACTIVATING FACTOR 1, PROCASPASE 9
著者Qin, H, Srinivasula, S, Wu, G, Fernandes-Alnemri, T, Alnemri, E, Shi, Y.
登録日1999-05-08
公開日2000-04-19
最終更新日2023-12-27
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Structural basis of procaspase-9 recruitment by the apoptotic protease-activating factor 1.
Nature, 399, 1999
4TQV
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BU of 4tqv by Molmil
Crystal structure of a bacterial ABC transporter involved in the import of the acidic polysaccharide alginate
分子名称: AlgM1, AlgM2, AlgS
著者Maruyama, Y, Itoh, T, Kaneko, A, Nishitani, Y, Mikami, B, Hashimoto, W, Murata, K.
登録日2014-06-12
公開日2015-07-22
最終更新日2024-03-20
実験手法X-RAY DIFFRACTION (4.504 Å)
主引用文献Structure of a Bacterial ABC Transporter Involved in the Import of an Acidic Polysaccharide Alginate
Structure, 23, 2015
3UOA
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BU of 3uoa by Molmil
Crystal structure of the MALT1 paracaspase (P21 form)
分子名称: MAGNESIUM ION, Mucosa-associated lymphoid tissue lymphoma translocation protein 1, Z-Val-Arg-Pro-DL-Arg-fluoromethylketone
著者Jeffrey, P.D, Yu, J.W, Shi, Y.
登録日2011-11-16
公開日2011-12-21
最終更新日2024-10-09
実験手法X-RAY DIFFRACTION (1.75 Å)
主引用文献Crystal structure of the mucosa-associated lymphoid tissue lymphoma translocation 1 (MALT1) paracaspase region.
Proc.Natl.Acad.Sci.USA, 108, 2011
1IQP
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BU of 1iqp by Molmil
Crystal Structure of the Clamp Loader Small Subunit from Pyrococcus furiosus
分子名称: ADENOSINE-5'-DIPHOSPHATE, RFCS
著者Oyama, T, Ishino, Y, Cann, I.K.O, Ishino, S, Morikawa, K.
登録日2001-07-24
公開日2001-09-19
最終更新日2023-12-27
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献Atomic Structure of the Clamp Loader Small Subunit from Pyrococcus furiosus
Mol.Cell, 8, 2001
6JO1
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BU of 6jo1 by Molmil
Structure of the CYP102A1 Haem Domain with N-(S)-Ibuprofenoyl-L-Phenylalanine
分子名称: (2S)-2-[[(2S)-2-[4-(2-methylpropyl)phenyl]propanoyl]amino]-3-phenyl-propanoic acid, Bifunctional cytochrome P450/NADPH--P450 reductase, DIMETHYL SULFOXIDE, ...
著者Stanfield, J.K, Kasai, C, Sugimoto, H, Shiro, Y, Watanabe, Y, Shoji, O.
登録日2019-03-19
公開日2020-03-18
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Crystals in Minutes: Instant On-Site Microcrystallisation of Various Flavours of the CYP102A1 (P450BM3) Haem Domain.
Angew.Chem.Int.Ed.Engl., 59, 2020
6JS8
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Structure of the CYP102A1 Haem Domain with N-Dehydroabietoyl-L-Tryptophan
分子名称: (2S)-2-[[(1R,4aS,10aR)-1,4a-dimethyl-7-propan-2-yl-2,3,4,9,10,10a-hexahydrophenanthren-1-yl]carbonylamino]-3-(1H-indol-3-yl)propanoic acid, Bifunctional cytochrome P450/NADPH--P450 reductase, DIMETHYL SULFOXIDE, ...
著者Stanfield, J.K, Kasai, C, Sugimoto, H, Shiro, Y, Watanabe, Y, Shoji, O.
登録日2019-04-07
公開日2020-03-18
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (1.36 Å)
主引用文献Crystals in Minutes: Instant On-Site Microcrystallisation of Various Flavours of the CYP102A1 (P450BM3) Haem Domain.
Angew.Chem.Int.Ed.Engl., 59, 2020
6K58
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BU of 6k58 by Molmil
Structure of the CYP102A1 Haem Domain with N-Enanthyl-L-Prolyl-L-Phenylalanine
分子名称: (2S)-2-[[(2S)-1-heptylpyrrolidin-2-yl]carbonylamino]-3-phenyl-propanoic acid, Bifunctional cytochrome P450/NADPH--P450 reductase, DIMETHYL SULFOXIDE, ...
著者Stanfield, J.K, Kasai, C, Sugimoto, H, Shiro, Y, Watanabe, Y, Shoji, O.
登録日2019-05-28
公開日2020-03-18
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (1.41 Å)
主引用文献Crystals in Minutes: Instant On-Site Microcrystallisation of Various Flavours of the CYP102A1 (P450BM3) Haem Domain.
Angew.Chem.Int.Ed.Engl., 59, 2020
6JVC
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BU of 6jvc by Molmil
Structure of the Cobalt Protoporphyrin IX-Reconstituted CYP102A1 Haem Domain with N-Abietoyl-L-Tryptophan
分子名称: (2S)-2-[[(1R,4aR,4bR,10aR)-1,4a-dimethyl-7-propan-2-yl-2,3,4,4b,5,6,10,10a-octahydrophenanthren-1-yl]carbonylamino]-3-( 1H-indol-3-yl)propanoic acid, 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, Bifunctional cytochrome P450/NADPH--P450 reductase, ...
著者Stanfield, J.K, Matsumoto, A, Kasai, C, Sugimoto, H, Shiro, Y, Watanabe, Y, Shoji, O.
登録日2019-04-16
公開日2020-03-18
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (1.75 Å)
主引用文献Crystals in Minutes: Instant On-Site Microcrystallisation of Various Flavours of the CYP102A1 (P450BM3) Haem Domain.
Angew.Chem.Int.Ed.Engl., 59, 2020
6K9S
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Structure of the Carbonylruthenium Mesoporphyrin IX-Reconstituted CYP102A1 Haem Domain with N-Abietoyl-L-Tryptophan
分子名称: (2S)-2-[[(1R,4aR,4bR,10aR)-1,4a-dimethyl-7-propan-2-yl-2,3,4,4b,5,6,10,10a-octahydrophenanthren-1-yl]carbonylamino]-3-( 1H-indol-3-yl)propanoic acid, Bifunctional cytochrome P450/NADPH--P450 reductase, CARBON MONOXIDE, ...
著者Stanfield, J.K, Omura, K, Kasai, C, Sugimoto, H, Shiro, Y, Watanabe, Y, Shoji, O.
登録日2019-06-17
公開日2020-03-18
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (1.55 Å)
主引用文献Crystals in Minutes: Instant On-Site Microcrystallisation of Various Flavours of the CYP102A1 (P450BM3) Haem Domain.
Angew.Chem.Int.Ed.Engl., 59, 2020
6K24
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Structure of the Rhodium Mesoporphyrin IX-Reconstituted CYP102A1 Haem Domain with N-Abietoyl-L-Tryptophan
分子名称: (2S)-2-[[(1R,4aR,4bR,10aR)-1,4a-dimethyl-7-propan-2-yl-2,3,4,4b,5,6,10,10a-octahydrophenanthren-1-yl]carbonylamino]-3-( 1H-indol-3-yl)propanoic acid, Bifunctional cytochrome P450/NADPH--P450 reductase, DIMETHYL SULFOXIDE, ...
著者Stanfield, J.K, Matsumoto, A, Kasai, C, Sugimoto, H, Shiro, Y, Watanabe, Y, Shoji, O.
登録日2019-05-13
公開日2020-03-18
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Crystals in Minutes: Instant On-Site Microcrystallisation of Various Flavours of the CYP102A1 (P450BM3) Haem Domain.
Angew.Chem.Int.Ed.Engl., 59, 2020

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