6LUB
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![BU of 6lub by Molmil](/molmil-images/mine/6lub) | Crystal Structure of EGFR(L858R/T790M/C797S) in complex with CH7233163 | 分子名称: | Epidermal growth factor receptor, N-[2-(1-cyclopropylsulfonylpyrazol-4-yl)pyrimidin-4-yl]-7-(4-methylpiperazin-1-yl)-5-propan-2-yl-9-[2,2,2-tris(fluoranyl)ethoxy]pyrido[4,3-b]indol-3-amine | 著者 | Kawauchi, H, Fukami, T.A, Sato, S, Endo, M, Torizawa, T, Kashima, K, Chiba, T, Sakamoto, H. | 登録日 | 2020-01-27 | 公開日 | 2020-10-07 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (2.315 Å) | 主引用文献 | CH7233163 Overcomes Osimertinib-Resistant EGFR-Del19/T790M/C797S Mutation. Mol.Cancer Ther., 19, 2020
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7DC7
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![BU of 7dc7 by Molmil](/molmil-images/mine/7dc7) | Crystal structure of D12 Fab-ATP complex | 分子名称: | ADENOSINE-5'-TRIPHOSPHATE, D12 Fab heavy chain, D12 Fab light chain | 著者 | Kawauchi, H, Fukami, T.A, Tatsumi, K, Torizawa, T, Mimoto, F. | 登録日 | 2020-10-23 | 公開日 | 2021-01-13 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (1.77 Å) | 主引用文献 | Exploitation of Elevated Extracellular ATP to Specifically Direct Antibody to Tumor Microenvironment. Cell Rep, 33, 2020
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6LUD
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![BU of 6lud by Molmil](/molmil-images/mine/6lud) | Crystal Structure of EGFR(L858R/T790M/C797S) in complex with Osimertinib | 分子名称: | Epidermal growth factor receptor, N-(2-{[2-(dimethylamino)ethyl](methyl)amino}-4-methoxy-5-{[4-(1-methyl-1H-indol-3-yl)pyrimidin-2-yl]amino}phenyl)prop-2-enamide | 著者 | Kawauchi, H, Fukami, T.A, Sato, S, Endo, M, Torizawa, T, Kashima, K, Chiba, T, Sakamoto, H. | 登録日 | 2020-01-27 | 公開日 | 2020-10-07 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (2.05 Å) | 主引用文献 | CH7233163 Overcomes Osimertinib-Resistant EGFR-Del19/T790M/C797S Mutation. Mol.Cancer Ther., 19, 2020
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8QFW
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![BU of 8qfw by Molmil](/molmil-images/mine/8qfw) | Murine pyridoxal phosphatase in complex with 7,8-dihydroxyflavone | 分子名称: | 7,8-bis(oxidanyl)-2-phenyl-chromen-4-one, CITRIC ACID, Chronophin, ... | 著者 | Schindelin, H, Gohla, A. | 登録日 | 2023-09-05 | 公開日 | 2024-06-12 | 最終更新日 | 2024-06-26 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | 7,8-Dihydroxyflavone is a direct inhibitor of human and murine pyridoxal phosphatase. Elife, 13, 2024
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8T8A
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![BU of 8t8a by Molmil](/molmil-images/mine/8t8a) | |
7PKJ
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![BU of 7pkj by Molmil](/molmil-images/mine/7pkj) | Streptococcus pyogenes apo GapN | 分子名称: | BETA-MERCAPTOETHANOL, GLYCEROL, Putative NADP-dependent glyceraldehyde-3-phosphate dehydrogenase, ... | 著者 | Schindelin, H, Albert, L. | 登録日 | 2021-08-25 | 公開日 | 2022-03-16 | 最終更新日 | 2024-01-31 | 実験手法 | X-RAY DIFFRACTION (1.989 Å) | 主引用文献 | The Non-phosphorylating Glyceraldehyde-3-Phosphate Dehydrogenase GapN Is a Potential New Drug Target in Streptococcus pyogenes. Front Microbiol, 13, 2022
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7PKC
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![BU of 7pkc by Molmil](/molmil-images/mine/7pkc) | Streptococcus pyogenes Apo-GapN C284S variant | 分子名称: | GLYCEROL, Putative NADP-dependent glyceraldehyde-3-phosphate dehydrogenase, SULFATE ION | 著者 | Schindelin, H, Albert, L. | 登録日 | 2021-08-25 | 公開日 | 2022-03-16 | 最終更新日 | 2024-05-01 | 実験手法 | X-RAY DIFFRACTION (1.5 Å) | 主引用文献 | The Non-phosphorylating Glyceraldehyde-3-Phosphate Dehydrogenase GapN Is a Potential New Drug Target in Streptococcus pyogenes. Front Microbiol, 13, 2022
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6QSE
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![BU of 6qse by Molmil](/molmil-images/mine/6qse) | Crystal structure of Pizza6S in the presence of Anderson-Evans (TEW) | 分子名称: | 6-tungstotellurate(VI), Pizza6S | 著者 | Noguchi, H, Vandebroek, L, Kamata, K, Tame, J.R.H, Van Meervelt, L, Parac-Vogt, T.N, Voet, A.R.D. | 登録日 | 2019-02-20 | 公開日 | 2020-03-18 | 最終更新日 | 2024-01-24 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Hybrid assemblies of a symmetric designer protein and polyoxometalates with matching symmetry. Chem.Commun.(Camb.), 56, 2020
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6QSF
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![BU of 6qsf by Molmil](/molmil-images/mine/6qsf) | Crystal structure of Pizza6S in the presence of Keggin (STA) | 分子名称: | Keggin (STA), Pizza6S | 著者 | Noguchi, H, Vandebroek, L, Kamata, K, Tame, J.R.H, Van Meervelt, L, Parac-Vogt, T.N, Voet, A.R.D. | 登録日 | 2019-02-20 | 公開日 | 2020-03-18 | 最終更新日 | 2024-01-24 | 実験手法 | X-RAY DIFFRACTION (1.5 Å) | 主引用文献 | Hybrid assemblies of a symmetric designer protein and polyoxometalates with matching symmetry. Chem.Commun.(Camb.), 56, 2020
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6QSD
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![BU of 6qsd by Molmil](/molmil-images/mine/6qsd) | Crystal structure of Pizza6S | 分子名称: | Pizza6S, SULFATE ION | 著者 | Noguchi, H, Vandebroek, L, Kamata, K, Tame, J.R.H, Van Meervelt, L, Parac-Vogt, T.N, Voet, A.R.D. | 登録日 | 2019-02-20 | 公開日 | 2020-03-18 | 最終更新日 | 2024-01-24 | 実験手法 | X-RAY DIFFRACTION (1.45 Å) | 主引用文献 | Hybrid assemblies of a symmetric designer protein and polyoxometalates with matching symmetry. Chem.Commun.(Camb.), 56, 2020
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6QSH
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![BU of 6qsh by Molmil](/molmil-images/mine/6qsh) | Crystal structure of the hybrid bioinorganic complex of Pizza6S linked by the 1:2 Ce-substituted Keggin | 分子名称: | 1:2 Ce-substituted Keggin, Pizza6S | 著者 | Noguchi, H, Vandebroek, L, Kamata, K, Tame, J.R.H, Van Meervelt, L, Parac-Vogt, T.N, Voet, A.R.D. | 登録日 | 2019-02-20 | 公開日 | 2020-03-18 | 最終更新日 | 2024-01-24 | 実験手法 | X-RAY DIFFRACTION (2.5 Å) | 主引用文献 | Hybrid assemblies of a symmetric designer protein and polyoxometalates with matching symmetry. Chem.Commun.(Camb.), 56, 2020
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6QSG
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![BU of 6qsg by Molmil](/molmil-images/mine/6qsg) | Crystal structure of the hybrid bioinorganic complex of Pizza6S and Keggin (STA) | 分子名称: | Keggin (STA), Pizza6S | 著者 | Noguchi, H, Vandebroek, L, Kamata, K, Tame, J.R.H, Van Meervelt, L, Parac-Vogt, T.N, Voet, A.R.D. | 登録日 | 2019-02-20 | 公開日 | 2020-03-18 | 最終更新日 | 2024-01-24 | 実験手法 | X-RAY DIFFRACTION (1.15 Å) | 主引用文献 | Hybrid assemblies of a symmetric designer protein and polyoxometalates with matching symmetry. Chem.Commun.(Camb.), 56, 2020
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1X1D
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![BU of 1x1d by Molmil](/molmil-images/mine/1x1d) | Crystal structure of BchU complexed with S-adenosyl-L-homocysteine and Zn-bacteriopheophorbide d | 分子名称: | CrtF-related protein, GLYCEROL, S-ADENOSYL-L-HOMOCYSTEINE, ... | 著者 | Yamaguchi, H, Wada, K, Fukuyama, K. | 登録日 | 2005-04-04 | 公開日 | 2006-07-18 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (2.7 Å) | 主引用文献 | Crystal Structures of BchU, a Methyltransferase Involved in Bacteriochlorophyll c Biosynthesis, and its Complex with S-adenosylhomocysteine: Implications for Reaction Mechanism. J.Mol.Biol., 360, 2006
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1X1B
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![BU of 1x1b by Molmil](/molmil-images/mine/1x1b) | Crystal structure of BchU complexed with S-adenosyl-L-homocysteine | 分子名称: | CrtF-related protein, GLYCEROL, S-ADENOSYL-L-HOMOCYSTEINE, ... | 著者 | Yamaguchi, H, Wada, K, Fukuyama, K. | 登録日 | 2005-04-03 | 公開日 | 2006-07-18 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (2.6 Å) | 主引用文献 | Crystal Structures of BchU, a Methyltransferase Involved in Bacteriochlorophyll c Biosynthesis, and its Complex with S-adenosylhomocysteine: Implications for Reaction Mechanism. J.Mol.Biol., 360, 2006
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1X19
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![BU of 1x19 by Molmil](/molmil-images/mine/1x19) | Crystal structure of BchU involved in bacteriochlorophyll c biosynthesis | 分子名称: | CrtF-related protein, SULFATE ION | 著者 | Yamaguchi, H, Wada, K, Fukuyama, K. | 登録日 | 2005-04-02 | 公開日 | 2006-07-18 | 最終更新日 | 2024-03-13 | 実験手法 | X-RAY DIFFRACTION (2.27 Å) | 主引用文献 | Crystal Structures of BchU, a Methyltransferase Involved in Bacteriochlorophyll c Biosynthesis, and its Complex with S-adenosylhomocysteine: Implications for Reaction Mechanism. J.Mol.Biol., 360, 2006
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1X1A
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![BU of 1x1a by Molmil](/molmil-images/mine/1x1a) | Crystal structure of BchU complexed with S-adenosyl-L-methionine | 分子名称: | CrtF-related protein, GLYCEROL, S-ADENOSYLMETHIONINE, ... | 著者 | Yamaguchi, H, Wada, K, Fukuyama, K. | 登録日 | 2005-04-03 | 公開日 | 2006-07-18 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (2.6 Å) | 主引用文献 | Crystal Structures of BchU, a Methyltransferase Involved in Bacteriochlorophyll c Biosynthesis, and its Complex with S-adenosylhomocysteine: Implications for Reaction Mechanism. J.Mol.Biol., 360, 2006
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1X1C
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![BU of 1x1c by Molmil](/molmil-images/mine/1x1c) | Crystal structure of BchU complexed with S-adenosyl-L-homocysteine and Zn2+ | 分子名称: | CrtF-related protein, GLYCEROL, S-ADENOSYL-L-HOMOCYSTEINE, ... | 著者 | Yamaguchi, H, Wada, K, Fukuyama, K. | 登録日 | 2005-04-03 | 公開日 | 2006-07-18 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (2.85 Å) | 主引用文献 | Crystal Structures of BchU, a Methyltransferase Involved in Bacteriochlorophyll c Biosynthesis, and its Complex with S-adenosylhomocysteine: Implications for Reaction Mechanism. J.Mol.Biol., 360, 2006
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5Z5E
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![BU of 5z5e by Molmil](/molmil-images/mine/5z5e) | |
5X7X
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![BU of 5x7x by Molmil](/molmil-images/mine/5x7x) | The crystal structure of the nucleosome containing H3.3 at 2.18 angstrom resolution | 分子名称: | CHLORIDE ION, DNA (146-MER), Histone H2A type 1-B/E, ... | 著者 | Arimura, Y, Taguchi, H, Kurumizaka, H. | 登録日 | 2017-02-27 | 公開日 | 2017-04-19 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (2.184 Å) | 主引用文献 | Crystal Structure and Characterization of Novel Human Histone H3 Variants, H3.6, H3.7, and H3.8 Biochemistry, 56, 2017
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5XM1
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![BU of 5xm1 by Molmil](/molmil-images/mine/5xm1) | The mouse nucleosome structure containing H2A, H2B type3-A, H3mm7, and H4 | 分子名称: | DNA (146-MER), Histone H2A type 1-B, Histone H2B type 3-A, ... | 著者 | Taguchi, H, Horikoshi, N, Kurumizaka, H. | 登録日 | 2017-05-12 | 公開日 | 2018-03-07 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (3.45 Å) | 主引用文献 | Histone H3.3 sub-variant H3mm7 is required for normal skeletal muscle regeneration. Nat Commun, 9, 2018
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5XM0
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![BU of 5xm0 by Molmil](/molmil-images/mine/5xm0) | The mouse nucleosome structure containing H2A, H2B type3-A, H3.3, and H4 | 分子名称: | DNA (146-MER), Histone H2A type 1-B, Histone H2B type 3-A, ... | 著者 | Taguchi, H, Horikoshi, N, Kurumizaka, H. | 登録日 | 2017-05-12 | 公開日 | 2018-03-07 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (2.874 Å) | 主引用文献 | Histone H3.3 sub-variant H3mm7 is required for normal skeletal muscle regeneration. Nat Commun, 9, 2018
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1YSE
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![BU of 1yse by Molmil](/molmil-images/mine/1yse) | |
3WFL
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![BU of 3wfl by Molmil](/molmil-images/mine/3wfl) | Crtstal structure of glycoside hydrolase family 5 beta-mannanase from Talaromyces trachyspermus | 分子名称: | 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, 2-acetamido-2-deoxy-beta-D-glucopyranose, GLYCEROL, ... | 著者 | Suzuki, K, Ichinose, H, Kamino, K, Ogasawara, W, Kaneko, S, Fushinobu, S. | 登録日 | 2013-07-19 | 公開日 | 2014-07-23 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (1.6 Å) | 主引用文献 | Purification, cloning, functional expression, structure, and characterization of a thermostable beta-mannanase from Talaromyces trachyspermus and its efficiency in production of mannooligosaccharides from coffee wastes To be Published
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5Y6Q
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3A22
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![BU of 3a22 by Molmil](/molmil-images/mine/3a22) | Crystal Structure of beta-L-Arabinopyranosidase complexed with L-arabinose | 分子名称: | 2-(2-{2-[2-(2-METHOXY-ETHOXY)-ETHOXY]-ETHOXY}-ETHOXY)-ETHANOL, 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, GLYCEROL, ... | 著者 | Fujimoto, Z, Ichinose, H, Kaneko, S. | 登録日 | 2009-04-27 | 公開日 | 2009-07-14 | 最終更新日 | 2023-11-01 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | A beta-l-Arabinopyranosidase from Streptomyces avermitilis is a novel member of glycoside hydrolase family 27. J.Biol.Chem., 284, 2009
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