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7K48
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BU of 7k48 by Molmil
Structure of NavAb/Nav1.7-VS2A chimera trapped in the resting state by tarantula toxin m3-Huwentoxin-IV
分子名称: Maltose/maltodextrin-binding periplasmic protein,Ion transport protein,Sodium channel protein type 9 subunit alpha chimera, Mu-theraphotoxin-Hs2a
著者Wisedchaisri, G, Tonggu, L, Gamal El-Din, T.M, McCord, E, Zheng, N, Catterall, W.A.
登録日2020-09-15
公開日2020-12-02
最終更新日2021-01-20
実験手法ELECTRON MICROSCOPY (3.6 Å)
主引用文献Structural Basis for High-Affinity Trapping of the Na V 1.7 Channel in Its Resting State by Tarantula Toxin.
Mol.Cell, 81, 2021
7Y42
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BU of 7y42 by Molmil
Cryo-EM structure of the SARS-CoV-2 spike glycoprotein in complex with all-trans retinoic acid
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, RETINOIC ACID, Spike glycoprotein
著者Xiang, Y, Wang, L.
登録日2022-06-13
公開日2022-07-06
最終更新日2022-09-14
実験手法ELECTRON MICROSCOPY (3.45 Å)
主引用文献A Retinol Derivative Inhibits SARS-CoV-2 Infection by Interrupting Spike-Mediated Cellular Entry.
Mbio, 13, 2022
6Q21
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BU of 6q21 by Molmil
MOLECULAR SWITCH FOR SIGNAL TRANSDUCTION: STRUCTURAL DIFFERENCES BETWEEN ACTIVE AND INACTIVE FORMS OF PROTOONCOGENIC RAS PROTEINS
分子名称: C-H-RAS P21 PROTEIN CATALYTIC DOMAIN, MAGNESIUM ION, PHOSPHOMETHYLPHOSPHONIC ACID GUANYLATE ESTER
著者Kim, S.-H.
登録日1992-07-27
公開日1992-07-28
最終更新日2024-03-13
実験手法X-RAY DIFFRACTION (1.95 Å)
主引用文献Molecular switch for signal transduction: structural differences between active and inactive forms of protooncogenic ras proteins.
Science, 247, 1990
6OBY
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BU of 6oby by Molmil
The nucleotide-binding protein AF_226 in complex with ADP from Archaeoglobus fulgidus with Co found by PIXE. Based on 3KB1.
分子名称: ADENOSINE-5'-DIPHOSPHATE, COBALT (II) ION, Iron-sulfur cluster carrier protein
著者Snell, E.H, Garman, E.F, Lowe, E.D.
登録日2019-03-21
公開日2019-12-25
最終更新日2020-01-22
実験手法X-RAY DIFFRACTION (2.87 Å)
主引用文献High-Throughput PIXE as an Essential Quantitative Assay for Accurate Metalloprotein Structural Analysis: Development and Application.
J.Am.Chem.Soc., 142, 2020
1VCQ
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BU of 1vcq by Molmil
SEMLIKI FOREST VIRUS CAPSID PROTEIN (CRYSTAL FORM II)
分子名称: SEMLIKI FOREST VIRUS CAPSID PROTEIN
著者Lu, G, Choi, H.-K, Rossmann, M.G.
登録日1996-03-04
公開日1996-12-07
最終更新日2011-07-13
実験手法X-RAY DIFFRACTION (3.1 Å)
主引用文献Structure of Semliki Forest virus core protein.
Proteins, 27, 1997
9CSI
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BU of 9csi by Molmil
A. baumannii MsbA Bound to Cerastecin Compound 5
分子名称: 3,3'-[(1,4-dioxobutane-1,4-diyl)bis(azanediyl)]bis[(4-butylbenzene-1-sulfonamido)benzoic acid], Lipid A export ATP-binding/permease protein MsbA, MAGNESIUM ION, ...
著者Klein, D.J, Ishchenko, A, Soisson, S, Cheng, R, Hennig, M.
登録日2024-07-23
公開日2024-09-04
最終更新日2024-10-02
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献Cerastecin Inhibition of the Lipooligosaccharide Transporter MsbA to Combat Acinetobacter baumannii : From Screening Impurity to In Vivo Efficacy.
J.Med.Chem., 67, 2024
9CSG
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BU of 9csg by Molmil
Human Serum Albumin Bound to Cerastecin Compound 5e
分子名称: 2-(4-butylbenzene-1-sulfonamido)-5-(4-{3-carboxy-4-[4-(2-methoxyethyl)benzene-1-sulfonamido]anilino}-4-oxobutanamido)benzoic acid, Albumin, MYRISTIC ACID
著者Hruza, A, Klein, D.J, Ishchenko, A.
登録日2024-07-23
公開日2024-09-04
最終更新日2024-10-02
実験手法X-RAY DIFFRACTION (1.914 Å)
主引用文献Cerastecin Inhibition of the Lipooligosaccharide Transporter MsbA to Combat Acinetobacter baumannii : From Screening Impurity to In Vivo Efficacy.
J.Med.Chem., 67, 2024
3L0V
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BU of 3l0v by Molmil
Crystal structure of catalytic domain of TACE with the first hydantoin inhibitor occupying the S1' pocket
分子名称: (5R)-5-[(5-methoxy-3-oxo-1,3-dihydro-2H-indazol-2-yl)methyl]-5-methylimidazolidine-2,4-dione, Disintegrin and metalloproteinase domain-containing protein 17, ZINC ION
著者Orth, P.
登録日2009-12-10
公開日2010-03-02
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (1.75 Å)
主引用文献Discovery and SAR of hydantoin TACE inhibitors.
Bioorg.Med.Chem.Lett., 20, 2010
3L0T
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BU of 3l0t by Molmil
Crystal structure of catalytic domain of TACE with hydantoin inhibitor
分子名称: Disintegrin and metalloproteinase domain-containing protein 17, ISOPROPYL ALCOHOL, N-{(2R)-2-[2-(hydroxyamino)-2-oxoethyl]-4-methylpentanoyl}-3-methyl-L-valyl-N-(2-aminoethyl)-L-alaninamide, ...
著者Orth, P.
登録日2009-12-10
公開日2010-03-02
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (1.92 Å)
主引用文献Discovery and SAR of hydantoin TACE inhibitors.
Bioorg.Med.Chem.Lett., 20, 2010
7X2H
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BU of 7x2h by Molmil
Crystal structure of SARS-CoV-2 spike receptor-binding domain bound with 6-2C Fab
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 6-2C H chain, 6-2C L chain, ...
著者Wang, X, Wang, Z.
登録日2022-02-25
公開日2023-03-01
最終更新日2023-08-23
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Inactivated vaccine-elicited potent antibodies can broadly neutralize SARS-CoV-2 circulating variants.
Nat Commun, 14, 2023
1VYU
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BU of 1vyu by Molmil
Beta3 subunit of Voltage-gated Ca2+-channel
分子名称: CALCIUM CHANNEL BETA-3 SUBUNIT
著者Chen, Y.-H, Li, M.-H, Zhang, Y, He, L.-L, Yamada, Y, Fitzmaurice, A, Yang, S, Zhang, H, Liang, T, Yang, J.
登録日2004-05-07
公開日2004-06-15
最終更新日2011-07-13
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Structural Basis of the Alpha(1)-Beta Subunit Interaction of Voltage-Gated Ca(2+) Channels
Nature, 429, 2004
7XD2
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BU of 7xd2 by Molmil
SARS-CoV-2 S ectodomain trimer in complex with neutralizing antibody 10-5B
分子名称: H chain of antibody 10-5B, L chian of antibody 10-5B, Spike glycoprotein
著者Wang, X, Wang, Z.
登録日2022-03-26
公開日2023-07-12
最終更新日2024-10-09
実験手法ELECTRON MICROSCOPY (3.3 Å)
主引用文献Inactivated vaccine-elicited potent antibodies can broadly neutralize SARS-CoV-2 circulating variants.
Nat Commun, 14, 2023
4Q21
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BU of 4q21 by Molmil
MOLECULAR SWITCH FOR SIGNAL TRANSDUCTION: STRUCTURAL DIFFERENCES BETWEEN ACTIVE AND INACTIVE FORMS OF PROTOONCOGENIC RAS PROTEINS
分子名称: C-H-RAS P21 PROTEIN CATALYTIC DOMAIN, GUANOSINE-5'-DIPHOSPHATE, MAGNESIUM ION
著者Kim, S.-H.
登録日1991-09-25
公開日1992-07-15
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Molecular switch for signal transduction: structural differences between active and inactive forms of protooncogenic ras proteins.
Science, 247, 1990
3SPE
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BU of 3spe by Molmil
Crystal structure of the tail sheath protein protease resistant fragment from bacteriophage phiKZ
分子名称: GLYCEROL, PHIKZ029, PHOSPHATE ION
著者Aksyuk, A.A, Kurochkina, L.P, Fokine, A, Mesyanzhinov, V.V, Rossmann, M.G.
登録日2011-07-01
公開日2011-12-14
最終更新日2017-11-08
実験手法X-RAY DIFFRACTION (2.3996 Å)
主引用文献Structural conservation of the myoviridae phage tail sheath protein fold.
Structure, 19, 2011
6OE2
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BU of 6oe2 by Molmil
X-Ray Structure of the C-terminal domain (277-440) of Putative chitobiase from Bacteroides thetaiotaomicron. Northeast Structural Genomics Consortium Target BtR324A. Re-refinement of 3GGL with correct metal Mn replacing Zn. New metal confirmed with PIXE analysis of original sample.
分子名称: Chitobiase, DI(HYDROXYETHYL)ETHER, MANGANESE (II) ION
著者Snell, E.H, Garman, E.F, Lowe, E.D.
登録日2019-03-27
公開日2019-12-25
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (3 Å)
主引用文献High-Throughput PIXE as an Essential Quantitative Assay for Accurate Metalloprotein Structural Analysis: Development and Application.
J.Am.Chem.Soc., 142, 2020
2SNW
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BU of 2snw by Molmil
SINDBIS VIRUS CAPSID PROTEIN, TYPE3 CRYSTAL FORM
分子名称: COAT PROTEIN C
著者Choi, H.-K, Lee, S, Zhang, Y.-P, Mckinney, B.R, Wengler, G, Rossmann, M.G, Kuhn, R.J.
登録日1998-02-17
公開日1998-04-08
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (2.7 Å)
主引用文献Structural analysis of Sindbis virus capsid mutants involving assembly and catalysis.
J.Mol.Biol., 262, 1996
1KXA
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BU of 1kxa by Molmil
SINDBIS VIRUS CAPSID, (WILD-TYPE) RESIDUES 106-264, TETRAGONAL CRYSTAL FORM
分子名称: SINDBIS VIRUS CAPSID PROTEIN
著者Choi, H.-K, Rossmann, M.G.
登録日1996-05-05
公開日1996-11-08
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (3.1 Å)
主引用文献Structural analysis of Sindbis virus capsid mutants involving assembly and catalysis.
J.Mol.Biol., 262, 1996
1KXF
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BU of 1kxf by Molmil
SINDBIS VIRUS CAPSID, (WILD-TYPE) RESIDUES 1-264, TETRAGONAL CRYSTAL FORM (FORM II)
分子名称: SINDBIS VIRUS CAPSID PROTEIN
著者Choi, H.-K, Rossmann, M.G.
登録日1996-05-05
公開日1996-12-07
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2.38 Å)
主引用文献Structural analysis of Sindbis virus capsid mutants involving assembly and catalysis.
J.Mol.Biol., 262, 1996
1KXC
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BU of 1kxc by Molmil
SINDBIS VIRUS CAPSID (N190K MUTANT), TETRAGONAL CRYSTAL FORM
分子名称: SINDBIS VIRUS CAPSID PROTEIN
著者Choi, H.-K, Rossmann, M.G.
登録日1996-05-05
公開日1996-11-08
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (3.1 Å)
主引用文献Structural analysis of Sindbis virus capsid mutants involving assembly and catalysis.
J.Mol.Biol., 262, 1996
1KXD
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BU of 1kxd by Molmil
SINDBIS VIRUS CAPSID (N222L MUTANT), TETRAGONAL CRYSTAL FORM
分子名称: SINDBIS VIRUS CAPSID PROTEIN
著者Choi, H.-K, Rossmann, M.G.
登録日1996-05-05
公開日1996-11-08
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (3 Å)
主引用文献Structural analysis of Sindbis virus capsid mutants involving assembly and catalysis.
J.Mol.Biol., 262, 1996
1KXB
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BU of 1kxb by Molmil
SINDBIS VIRUS CAPSID (S215A MUTANT), TETRAGONAL CRYSTAL FORM
分子名称: SINDBIS VIRUS CAPSID PROTEIN
著者Choi, H.-K, Rossmann, M.G.
登録日1996-05-05
公開日1996-11-08
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2.9 Å)
主引用文献Structural analysis of Sindbis virus capsid mutants involving assembly and catalysis.
J.Mol.Biol., 262, 1996
1KXE
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BU of 1kxe by Molmil
SINDBIS VIRUS CAPSID (Y180S, E183G DOUBLE MUTANT), TETRAGONAL CRYSTAL FORM
分子名称: SINDBIS VIRUS CAPSID PROTEIN
著者Choi, H.-K, Rossmann, M.G.
登録日1996-05-05
公開日1996-11-08
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (3.2 Å)
主引用文献Structural analysis of Sindbis virus capsid mutants involving assembly and catalysis.
J.Mol.Biol., 262, 1996
1Q21
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CRYSTAL STRUCTURES AT 2.2 ANGSTROMS RESOLUTION OF THE CATALYTIC DOMAINS OF NORMAL RAS PROTEIN AND AN ONCOGENIC MUTANT COMPLEXED WITH GSP
分子名称: C-H-RAS P21 PROTEIN CATALYTIC DOMAIN, GUANOSINE-5'-DIPHOSPHATE, MAGNESIUM ION
著者Kim, S.-H.
登録日1991-09-25
公開日1992-07-15
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Crystal structures at 2.2 A resolution of the catalytic domains of normal ras protein and an oncogenic mutant complexed with GDP.
J.Mol.Biol., 217, 1991
4E2A
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BU of 4e2a by Molmil
Crystal Structure of the Putative acetyltransferase from Streptococcus mutans
分子名称: Putative acetyltransferase
著者Li, G.L, Nie, J.K, Li, L.F, Su, X.D.
登録日2012-03-08
公開日2013-03-13
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Crystal Structure of the Putative acetyltransferase from Streptococcus mutans
To be Published
1SVP
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BU of 1svp by Molmil
SINDBIS VIRUS CAPSID PROTEIN
分子名称: SINDBIS VIRUS CAPSID PROTEIN
著者Lee, S, Rossmann, M.G.
登録日1996-03-22
公開日1996-08-17
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Identification of a protein binding site on the surface of the alphavirus nucleocapsid and its implication in virus assembly.
Structure, 4, 1996

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