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8XSO
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BU of 8xso by Molmil
RNA polymerase II elongation complex transcribing genomic DNA extracted from human nuclei
分子名称: DNA, DNA-directed RNA polymerase II subunit RPB1, DNA-directed RNA polymerase II subunit RPB11-a, ...
著者Kujirai, T, Kato, J, Yamamoto, K, Hirai, S, Negishi, L, Ogasawara, M, Takizawa, Y, Kurumizaka, H.
登録日2024-01-09
公開日2025-05-07
最終更新日2025-06-11
実験手法ELECTRON MICROSCOPY (2.7 Å)
主引用文献Multiple structures of RNA polymerase II isolated from human nuclei by ChIP-CryoEM analysis.
Nat Commun, 16, 2025
5WR7
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BU of 5wr7 by Molmil
Crystal structure of Trk-A complexed with a selective inhibitor CH7057288
分子名称: High affinity nerve growth factor receptor, N-tert-butyl-2-[2-[6,6-dimethyl-8-(methylsulfonylamino)-11-oxidanylidene-naphtho[2,3-b][1]benzofuran-3-yl]ethynyl]-6-methyl-pyridine-4-carboxamide
著者Tanaka, H, Blaesse, M, Augustin, M, Goesser, C.
登録日2016-11-30
公開日2017-12-06
最終更新日2024-11-20
実験手法X-RAY DIFFRACTION (2.76 Å)
主引用文献Selective TRK Inhibitor CH7057288 against TRK Fusion-Driven Cancer.
Mol. Cancer Ther., 17, 2018
1ECS
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BU of 1ecs by Molmil
THE 1.7 A CRYSTAL STRUCTURE OF A BLEOMYCIN RESISTANCE DETERMINANT ENCODED ON THE TRANSPOSON TN5
分子名称: BLEOMYCIN RESISTANCE PROTEIN, CALCIUM ION, TETRAETHYLENE GLYCOL
著者Maruyama, M, Matoba, Y, Kumagai, T, Sugiyama, M.
登録日2000-01-25
公開日2001-05-02
最終更新日2023-08-09
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Crystal structures of the transposon Tn5-carried bleomycin resistance determinant uncomplexed and complexed with bleomycin.
J.Biol.Chem., 276, 2001
1EWJ
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BU of 1ewj by Molmil
CRYSTAL STRUCTURE OF BLEOMYCIN-BINDING PROTEIN COMPLEXED WITH BLEOMYCIN
分子名称: BLEOMYCIN A2, BLEOMYCIN RESISTANCE DETERMINANT
著者Maruyama, M, Kumagai, T, Matoba, Y, Hata, Y, Sugiyama, M.
登録日2000-04-26
公開日2001-04-26
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Crystal structures of the transposon Tn5-carried bleomycin resistance determinant uncomplexed and complexed with bleomycin.
J.Biol.Chem., 276, 2001
7VCP
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BU of 7vcp by Molmil
Frischella perrara beta-fructofuranosidase in complex with fructose
分子名称: DI(HYDROXYETHYL)ETHER, PENTAETHYLENE GLYCOL, Sucrose-6-phosphate hydrolase, ...
著者Tonozuka, T.
登録日2021-09-03
公開日2022-03-09
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Enzymatic and structural characterization of beta-fructofuranosidase from the honeybee gut bacterium Frischella perrara.
Appl.Microbiol.Biotechnol., 106, 2022
7VCO
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BU of 7vco by Molmil
Frischella perrara beta-fructofuranosidase
分子名称: DI(HYDROXYETHYL)ETHER, Sucrose-6-phosphate hydrolase, TRIETHYLENE GLYCOL
著者Tonozuka, T.
登録日2021-09-03
公開日2022-03-09
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (1.6 Å)
主引用文献Enzymatic and structural characterization of beta-fructofuranosidase from the honeybee gut bacterium Frischella perrara.
Appl.Microbiol.Biotechnol., 106, 2022
5B7V
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BU of 5b7v by Molmil
Human FGFR1 kinase in complex with CH5183284
分子名称: Fibroblast growth factor receptor 1, SULFATE ION, [5-amino-1-(2-methyl-1H-benzimidazol-6-yl)-1H-pyrazol-4-yl](1H-indol-2-yl)methanone
著者Fukami, T.A, Lukacs, C.M, Janson, C.
登録日2016-06-09
公開日2016-06-22
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (2.15 Å)
主引用文献The fibroblast growth factor receptor genetic status as a potential predictor of the sensitivity to CH5183284/Debio 1347, a novel selective FGFR inhibitor
Mol.Cancer Ther., 13, 2014
3WEA
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BU of 3wea by Molmil
Crystal structure of a Niemann-Pick type C2 protein from Japanese carpenter ant
分子名称: Niemann-Pick type C2 protein
著者Fujimoto, Z, Tsuchiya, W, Ishida, Y, Yamazaki, T.
登録日2013-07-02
公開日2014-02-05
最終更新日2024-11-06
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Niemann-Pick type C2 protein mediating chemical communication in the worker ant
Proc.Natl.Acad.Sci.USA, 111, 2014
5AZ0
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BU of 5az0 by Molmil
Crystal structure of aldo-keto reductase (AKR2E5) of the silkworm, Bombyx mori
分子名称: 1,2-ETHANEDIOL, ACETATE ION, CALCIUM ION, ...
著者Yamamoto, K, Higashiura, A, Suzuki, M, Nakagawa, A.
登録日2015-09-15
公開日2016-02-10
最終更新日2024-03-20
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Structural characterization of an aldo-keto reductase (AKR2E5) from the silkworm Bombyx mori
Biochem.Biophys.Res.Commun., 474, 2016
5AZ1
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BU of 5az1 by Molmil
Crystal structure of aldo-keto reductase (AKR2E5) complexed with NADPH
分子名称: 1,2-ETHANEDIOL, ACETATE ION, CALCIUM ION, ...
著者Yamamoto, K, Higashiura, A, Suzuki, M, Nakagawa, A.
登録日2015-09-15
公開日2016-02-10
最終更新日2024-03-20
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Structural characterization of an aldo-keto reductase (AKR2E5) from the silkworm Bombyx mori
Biochem.Biophys.Res.Commun., 474, 2016
1KRM
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BU of 1krm by Molmil
Crystal structure of bovine adenosine deaminase complexed with 6-hydroxyl-1,6-dihydropurine riboside
分子名称: 6-HYDROXY-1,6-DIHYDRO PURINE NUCLEOSIDE, ZINC ION, adenosine deaminase
著者Kinoshita, T.
登録日2002-01-10
公開日2003-01-14
最終更新日2024-03-13
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Structure of bovine adenosine deaminase complexed with 6-hydroxy-1,6-dihydropurine riboside.
Acta Crystallogr.,Sect.D, 59, 2003
2MME
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BU of 2mme by Molmil
Hybrid structure of the Shigella flexneri MxiH Type three secretion system needle
分子名称: MxiH
著者Demers, J.P, Habenstein, B, Loquet, A, Vasa, S.K, Becker, S, Baker, D, Lange, A, Sgourakis, N.G.
登録日2014-03-14
公開日2014-10-08
最終更新日2024-05-15
実験手法ELECTRON MICROSCOPY (7.7 Å), SOLID-STATE NMR
主引用文献High-resolution structure of the Shigella type-III secretion needle by solid-state NMR and cryo-electron microscopy.
Nat Commun, 5, 2014
4A61
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BU of 4a61 by Molmil
ParM from plasmid R1 in complex with AMPPNP
分子名称: MAGNESIUM ION, PHOSPHOAMINOPHOSPHONIC ACID-ADENYLATE ESTER, PLASMID SEGREGATION PROTEIN PARM
著者van den Ent, F, Moller-Jensen, J, Gayathri, P, Lowe, J.
登録日2011-10-31
公開日2012-11-07
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献A Bipolar Spindle of Antiparallel Parm Filaments Drives Bacterial Plasmid Segregation.
Science, 338, 2012
4A62
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BU of 4a62 by Molmil
ParM from R1 plasmid in complex with peptide from C-terminus of ParR
分子名称: MAGNESIUM ION, PHOSPHOAMINOPHOSPHONIC ACID-ADENYLATE ESTER, PLASMID SEGREGATION PROTEIN PARM, ...
著者Gayathri, P, Lowe, J.
登録日2011-10-31
公開日2012-11-07
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献A Bipolar Spindle of Antiparallel Parm Filaments Drives Bacterial Plasmid Segregation.
Science, 338, 2012
1WXY
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BU of 1wxy by Molmil
Crystal structure of adenosine deaminase ligated with a potent inhibitor
分子名称: Adenosine deaminase, N-[4,5-BIS(4-HYDROXYPHENYL)-1,3-THIAZOL-2-YL]HEXANAMIDE, ZINC ION
著者Kinoshita, T.
登録日2005-02-02
公開日2005-08-16
最終更新日2024-03-13
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Structural Basis of Compound Recognition by Adenosine Deaminase
Biochemistry, 44, 2005
1VFL
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BU of 1vfl by Molmil
Adenosine deaminase
分子名称: Adenosine deaminase, ZINC ION
著者Kinoshita, T.
登録日2004-04-16
公開日2005-08-16
最終更新日2023-12-27
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Structural Basis of Compound Recognition by Adenosine Deaminase
Biochemistry, 44, 2005
3WEB
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BU of 3web by Molmil
Crystal structure of a Niemann-Pick type C2 protein from Japanese carpenter ant in complex with oleic acid
分子名称: Niemann-Pick type C2 protein, OLEIC ACID
著者Fujimoto, Z, Tsuchiya, W, Ishida, Y, Yamazaki, T.
登録日2013-07-02
公開日2014-02-05
最終更新日2024-11-06
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Niemann-Pick type C2 protein mediating chemical communication in the worker ant
Proc.Natl.Acad.Sci.USA, 111, 2014
1ITX
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BU of 1itx by Molmil
Catalytic Domain of Chitinase A1 from Bacillus circulans WL-12
分子名称: GLYCEROL, Glycosyl Hydrolase
著者Iwahori, F, Matsumoto, T, Watanabe, T, Nonaka, T.
登録日2002-02-13
公開日2002-03-13
最終更新日2024-10-23
実験手法X-RAY DIFFRACTION (1.1 Å)
主引用文献Three-dimensional structure of the catalytic domain of chitinase A1 from Bacillus circulans WL-12 at a very high resolution
PROC.JPN.ACAD.,SER.B, 75, 1999
1UK0
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BU of 1uk0 by Molmil
Crystal structure of catalytic domain of human poly(ADP-ribose) polymerase with a novel inhibitor
分子名称: 2-{3-[4-(4-FLUOROPHENYL)-3,6-DIHYDRO-1(2H)-PYRIDINYL]PROPYL}-8-METHYL-4(3H)-QUINAZOLINONE, Poly [ADP-ribose] polymerase-1
著者Kinoshita, T.
登録日2003-08-13
公開日2004-01-27
最終更新日2023-12-27
実験手法X-RAY DIFFRACTION (3 Å)
主引用文献Inhibitor-induced structural change of the active site of human poly(ADP-ribose) polymerase.
Febs Lett., 556, 2004
1WZY
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BU of 1wzy by Molmil
Crystal structure of human ERK2 complexed with a pyrazolopyridazine derivative
分子名称: 1-ALLYL-5-(2-PHENYLPYRAZOLO[1,5-A]PYRIDIN-3-YL)-1H-PYRAZOLO[3,4-C]PYRIDAZIN-3-AMINE, Mitogen-activated protein kinase 1
著者Kinoshita, T.
登録日2005-03-10
公開日2005-12-20
最終更新日2024-03-13
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Crystal structure of human ERK2 complexed with a pyrazolo[3,4-c]pyridazine derivative
Bioorg.Med.Chem.Lett., 16, 2006
1JIE
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BU of 1jie by Molmil
Crystal structure of bleomycin-binding protein from bleomycin-producing Streptomyces verticillus complexed with metal-free bleomycin
分子名称: BLEOMYCIN A2, bleomycin-binding protein
著者Sugiyama, M, Kumagai, T, Hayashida, M, Maruyama, M, Matoba, Y.
登録日2001-07-02
公開日2002-02-06
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献The 1.6-A crystal structure of the copper(II)-bound bleomycin complexed with the bleomycin-binding protein from bleomycin-producing Streptomyces verticillus.
J.Biol.Chem., 277, 2002
1JIF
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BU of 1jif by Molmil
Crystal structure of bleomycin-binding protein from bleomycin-producing Streptomyces verticillus complexed with copper(II)-bleomycin
分子名称: BLEOMYCIN A2, CHLORIDE ION, COPPER (II) ION, ...
著者Sugiyama, M, Kumagai, T, Hayashida, M, Maruyama, M, Matoba, Y.
登録日2001-07-02
公開日2002-02-06
最終更新日2024-03-13
実験手法X-RAY DIFFRACTION (1.6 Å)
主引用文献The 1.6-A crystal structure of the copper(II)-bound bleomycin complexed with the bleomycin-binding protein from bleomycin-producing Streptomyces verticillus.
J.Biol.Chem., 277, 2002
7UTI
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BU of 7uti by Molmil
ALTERNATIVE MODELING OF TROPOMYOSIN IN HUMAN CARDIAC THIN FILAMENT IN THE CALCIUM BOUND STATE
分子名称: ADENOSINE-5'-DIPHOSPHATE, Actin, alpha skeletal muscle, ...
著者Rynkiewicz, M.J, Pavadai, E, Lehman, W.
登録日2022-04-27
公開日2022-09-21
実験手法ELECTRON MICROSCOPY (4.8 Å)
主引用文献Protein-Protein Docking Reveals Dynamic Interactions of Tropomyosin on Actin Filaments.
Biophys J, 119, 2020
7UTL
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BU of 7utl by Molmil
ALTERNATIVE MODELING OF TROPOMYOSIN IN HUMAN CARDIAC THIN FILAMENT IN THE CALCIUM FREE STATE
分子名称: ADENOSINE-5'-DIPHOSPHATE, Actin, alpha skeletal muscle, ...
著者Rynkiewicz, M.J, Pavadai, E, Lehman, W.
登録日2022-04-27
公開日2022-09-21
実験手法ELECTRON MICROSCOPY (6.6 Å)
主引用文献Protein-Protein Docking Reveals Dynamic Interactions of Tropomyosin on Actin Filaments.
Biophys J, 119, 2020
1YIQ
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BU of 1yiq by Molmil
Molecular cloning and structural analysis of quinohemoprotein alcohol dehydrogenase ADHIIG from Pseudomonas putida HK5. Compariison to the other quinohemoprotein alcohol dehydrogenase ADHIIB found in the same microorganism.
分子名称: CALCIUM ION, HEME C, PYRROLOQUINOLINE QUINONE, ...
著者Toyama, H, Chen, Z.W, Fukumoto, M, Adachi, O, Matsushita, K, Mathews, F.S.
登録日2005-01-12
公開日2005-08-16
最終更新日2024-11-20
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Molecular cloning and structural analysis of quinohemoprotein alcohol dehydrogenase ADH-IIG from Pseudomonas putida HK5
J.Mol.Biol., 352, 2005
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