5FCS
| Diabody | 分子名称: | Diabody, SULFATE ION | 著者 | Mosyak, L, Root, A. | 登録日 | 2015-12-15 | 公開日 | 2016-12-14 | 最終更新日 | 2019-11-13 | 実験手法 | X-RAY DIFFRACTION (2.01 Å) | 主引用文献 | Development of PF-06671008, a Highly Potent Anti-P-cadherin/Anti-CD3 Bispecific DART Molecule with Extended Half-Life for the Treatment of Cancer. Antibodies, 5, 2016
|
|
6XF6
| Cryo-EM structure of a biotinylated SARS-CoV-2 spike probe in the prefusion state (1 RBD up) | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Spike glycoprotein | 著者 | Cerutti, G, Gorman, J, Kwong, P.D, Shapiro, L. | 登録日 | 2020-06-15 | 公開日 | 2020-09-02 | 最終更新日 | 2020-12-02 | 実験手法 | ELECTRON MICROSCOPY (4 Å) | 主引用文献 | Structure-Based Design with Tag-Based Purification and In-Process Biotinylation Enable Streamlined Development of SARS-CoV-2 Spike Molecular Probes. SSRN, 2020
|
|
6XF5
| Cryo-EM structure of a biotinylated SARS-CoV-2 spike probe in the prefusion state (RBDs down) | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Spike glycoprotein | 著者 | Cerutti, G, Gorman, J, Kwong, P.D, Shapiro, L. | 登録日 | 2020-06-15 | 公開日 | 2020-09-02 | 最終更新日 | 2020-12-02 | 実験手法 | ELECTRON MICROSCOPY (3.45 Å) | 主引用文献 | Structure-Based Design with Tag-Based Purification and In-Process Biotinylation Enable Streamlined Development of SARS-CoV-2 Spike Molecular Probes. SSRN, 2020
|
|
7YR0
| |
7YQU
| SARS-CoV-2 BA.2.75 S Trimer (3 RBD Down) | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Spike glycoprotein | 著者 | Wang, L. | 登録日 | 2022-08-08 | 公開日 | 2022-10-19 | 最終更新日 | 2022-11-23 | 実験手法 | ELECTRON MICROSCOPY (3.19 Å) | 主引用文献 | Characterization of the enhanced infectivity and antibody evasion of Omicron BA.2.75. Cell Host Microbe, 30, 2022
|
|
7YQT
| SARS-CoV-2 BA.2.75 S Trimer (1 RBD Up) | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Spike glycoprotein | 著者 | Wang, L. | 登録日 | 2022-08-08 | 公開日 | 2022-10-19 | 最終更新日 | 2022-11-23 | 実験手法 | ELECTRON MICROSCOPY (3.45 Å) | 主引用文献 | Characterization of the enhanced infectivity and antibody evasion of Omicron BA.2.75. Cell Host Microbe, 30, 2022
|
|
7YQV
| pH 5.5 SARS-CoV-2 BA.2.75 S Trimer (1 RBD Up) | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Spike glycoprotein | 著者 | Wang, L. | 登録日 | 2022-08-08 | 公開日 | 2022-10-19 | 最終更新日 | 2022-11-23 | 実験手法 | ELECTRON MICROSCOPY (3.58 Å) | 主引用文献 | Characterization of the enhanced infectivity and antibody evasion of Omicron BA.2.75. Cell Host Microbe, 30, 2022
|
|
7YR1
| SARS-CoV-2 BA.2.75 S Trimer in complex with XG2v024 | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Spike glycoprotein, ... | 著者 | Wang, L. | 登録日 | 2022-08-08 | 公開日 | 2022-10-19 | 最終更新日 | 2022-11-23 | 実験手法 | ELECTRON MICROSCOPY (3.62 Å) | 主引用文献 | Characterization of the enhanced infectivity and antibody evasion of Omicron BA.2.75. Cell Host Microbe, 30, 2022
|
|
7YR2
| SARS-CoV-2 BA.2.75 S Trimer in complex with ACE2(state1) | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Angiotensin-converting enzyme 2, ... | 著者 | Wang, L. | 登録日 | 2022-08-08 | 公開日 | 2022-10-19 | 最終更新日 | 2022-11-23 | 実験手法 | ELECTRON MICROSCOPY (3.3 Å) | 主引用文献 | Characterization of the enhanced infectivity and antibody evasion of Omicron BA.2.75. Cell Host Microbe, 30, 2022
|
|
7YQX
| SARS-CoV-2 BA.2.75 S Trimer in complex with S309 (state1) | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, S309 heavy chain, ... | 著者 | Wang, L. | 登録日 | 2022-08-08 | 公開日 | 2022-10-19 | 最終更新日 | 2022-11-23 | 実験手法 | ELECTRON MICROSCOPY (3.72 Å) | 主引用文献 | Characterization of the enhanced infectivity and antibody evasion of Omicron BA.2.75. Cell Host Microbe, 30, 2022
|
|
7YR3
| SARS-CoV-2 BA.2.75 S Trimer in complex with ACE2(state2) | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Angiotensin-converting enzyme 2, ... | 著者 | Wang, L. | 登録日 | 2022-08-08 | 公開日 | 2022-10-19 | 最終更新日 | 2022-11-23 | 実験手法 | ELECTRON MICROSCOPY (3.52 Å) | 主引用文献 | Characterization of the enhanced infectivity and antibody evasion of Omicron BA.2.75. Cell Host Microbe, 30, 2022
|
|
7YQW
| SARS-CoV-2 BA.2.75 S Trimer (3 RBD Down) | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Spike glycoprotein, ... | 著者 | Wang, L. | 登録日 | 2022-08-08 | 公開日 | 2022-10-19 | 最終更新日 | 2022-11-23 | 実験手法 | ELECTRON MICROSCOPY (3.51 Å) | 主引用文献 | Characterization of the enhanced infectivity and antibody evasion of Omicron BA.2.75. Cell Host Microbe, 30, 2022
|
|
7YQY
| SARS-CoV-2 BA.2.75 S Trimer in complex with S309 (state2) | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, S309 heavy chain, ... | 著者 | Wang, L. | 登録日 | 2022-08-08 | 公開日 | 2022-10-19 | 最終更新日 | 2022-11-23 | 実験手法 | ELECTRON MICROSCOPY (3.74 Å) | 主引用文献 | Characterization of the enhanced infectivity and antibody evasion of Omicron BA.2.75. Cell Host Microbe, 30, 2022
|
|
7YQZ
| SARS-CoV-2 BA.2.75 S Trimer in complex with S309 (state3) | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, S309 heavy chain, S309 light chain, ... | 著者 | Wang, L. | 登録日 | 2022-08-08 | 公開日 | 2022-10-19 | 最終更新日 | 2022-11-23 | 実験手法 | ELECTRON MICROSCOPY (3.84 Å) | 主引用文献 | Characterization of the enhanced infectivity and antibody evasion of Omicron BA.2.75. Cell Host Microbe, 30, 2022
|
|
2FX4
| |
2FX6
| |
2FWW
| |
2FPZ
| |
2FS8
| Human beta-tryptase II with inhibitor CRA-29382 | 分子名称: | ALLYL {(1S)-1-[(5-{4-[(2,3-DIHYDRO-1H-INDEN-2-YLAMINO)CARBONYL]BENZYL}-1,2,4-OXADIAZOL-3-YL)CARBONYL]-3-PYRROLIDIN-3-YLPROPYL}CARBAMATE, Tryptase beta-2 | 著者 | Somoza, J.R. | 登録日 | 2006-01-21 | 公開日 | 2006-03-21 | 最終更新日 | 2017-10-18 | 実験手法 | X-RAY DIFFRACTION (2.5 Å) | 主引用文献 | Structure-guided design of Peptide-based tryptase inhibitors. Biochemistry, 45, 2006
|
|
2G8A
| |
2FS9
| Human beta tryptase II with inhibitor CRA-28427 | 分子名称: | ETHYL {(1S)-5-AMINO-1-[(5-{4-[(2,3-DIHYDRO-1H-INDEN-2-YLAMINO)CARBONYL]BENZYL}-1,2,4-OXADIAZOL-3-YL)CARBONYL]PENTYL}CARBAMATE, Tryptase beta-2 | 著者 | Somoza, J.R. | 登録日 | 2006-01-21 | 公開日 | 2006-03-07 | 最終更新日 | 2017-10-18 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Structure-guided design of Peptide-based tryptase inhibitors. Biochemistry, 45, 2006
|
|
2FXR
| |
7SUS
| Crystal structure of Apelin receptor in complex with small molecule | 分子名称: | (1R,2S)-N-[4-(2,6-dimethoxyphenyl)-5-(6-methylpyridin-2-yl)-1,2,4-triazol-3-yl]-1-(5-methylpyrimidin-2-yl)-1-oxidanyl-propane-2-sulfonamide, (2R)-2,3-dihydroxypropyl (9Z)-octadec-9-enoate, Apelin receptor, ... | 著者 | Xu, F, Yue, Y, Liu, L.E, Han, G.W, Hanson, M. | 登録日 | 2021-11-18 | 公開日 | 2022-07-27 | 最終更新日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (2.7 Å) | 主引用文献 | Structural insight into apelin receptor-G protein stoichiometry. Nat.Struct.Mol.Biol., 29, 2022
|
|
4FLH
| Crystal structure of human PI3K-gamma in complex with AMG511 | 分子名称: | 4-(2-[(5-fluoro-6-methoxypyridin-3-yl)amino]-5-{(1R)-1-[4-(methylsulfonyl)piperazin-1-yl]ethyl}pyridin-3-yl)-6-methyl-1,3,5-triazin-2-amine, Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform, SULFATE ION | 著者 | Whittington, D.A, Tang, J, Yakowec, P. | 登録日 | 2012-06-14 | 公開日 | 2012-08-29 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (2.6 Å) | 主引用文献 | Selective Class I Phosphoinositide 3-Kinase Inhibitors: Optimization of a Series of Pyridyltriazines Leading to the Identification of a Clinical Candidate, AMG 511. J.Med.Chem., 55, 2012
|
|
3L0I
| Complex structure of SidM/DrrA with the wild type Rab1 | 分子名称: | CHLORIDE ION, DrrA, Ras-related protein Rab-1A, ... | 著者 | Zhu, Y, Shao, F. | 登録日 | 2009-12-10 | 公開日 | 2009-12-22 | 最終更新日 | 2017-11-01 | 実験手法 | X-RAY DIFFRACTION (2.85 Å) | 主引用文献 | Structural mechanism of host Rab1 activation by the bifunctional Legionella type IV effector SidM/DrrA Proc.Natl.Acad.Sci.USA, 107, 2010
|
|