8D76
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![BU of 8d76 by Molmil](/molmil-images/mine/8d76) | Crystal Structure of EGFR LRTM with compound 24 | 分子名称: | (3S,4R)-3-fluoro-1-(4-{[8-{3-[(methanesulfonyl)methyl]azetidin-1-yl}-5-(propan-2-yl)-2,7-naphthyridin-3-yl]amino}pyrimidin-2-yl)-3-methylpiperidin-4-ol, Epidermal growth factor receptor, GLYCEROL | 著者 | Kim, J.L. | 登録日 | 2022-06-07 | 公開日 | 2022-07-27 | 最終更新日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (2.4 Å) | 主引用文献 | Discovery of BLU-945, a Reversible, Potent, and Wild-Type-Sparing Next-Generation EGFR Mutant Inhibitor for Treatment-Resistant Non-Small-Cell Lung Cancer. J.Med.Chem., 65, 2022
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8CAF
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![BU of 8caf by Molmil](/molmil-images/mine/8caf) | N8C_Fab3b in complex with NEDD8-CUL1(WHB) | 分子名称: | Cullin-1, Fab Heavy Chain, Fab Light Chain, ... | 著者 | Duda, D.M, Yanishevski, D, Henneberg, L.T, Schulman, B.A. | 登録日 | 2023-01-24 | 公開日 | 2023-09-13 | 最終更新日 | 2023-12-06 | 実験手法 | X-RAY DIFFRACTION (2.66 Å) | 主引用文献 | Activity-based profiling of cullin-RING E3 networks by conformation-specific probes. Nat.Chem.Biol., 19, 2023
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7WVL
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![BU of 7wvl by Molmil](/molmil-images/mine/7wvl) | |
7ROZ
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![BU of 7roz by Molmil](/molmil-images/mine/7roz) | |
7RQS
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![BU of 7rqs by Molmil](/molmil-images/mine/7rqs) | |
3KN7
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![BU of 3kn7 by Molmil](/molmil-images/mine/3kn7) | |
3KN8
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![BU of 3kn8 by Molmil](/molmil-images/mine/3kn8) | |
1BAK
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![BU of 1bak by Molmil](/molmil-images/mine/1bak) | |
3FH7
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![BU of 3fh7 by Molmil](/molmil-images/mine/3fh7) | |
3FH8
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![BU of 3fh8 by Molmil](/molmil-images/mine/3fh8) | |
3FUL
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![BU of 3ful by Molmil](/molmil-images/mine/3ful) | |
3FTZ
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![BU of 3ftz by Molmil](/molmil-images/mine/3ftz) | |
3FH5
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![BU of 3fh5 by Molmil](/molmil-images/mine/3fh5) | |
3FHE
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![BU of 3fhe by Molmil](/molmil-images/mine/3fhe) | |
3FTU
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![BU of 3ftu by Molmil](/molmil-images/mine/3ftu) | |
3FU6
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![BU of 3fu6 by Molmil](/molmil-images/mine/3fu6) | |
3FUN
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![BU of 3fun by Molmil](/molmil-images/mine/3fun) | |
3FTS
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![BU of 3fts by Molmil](/molmil-images/mine/3fts) | Leukotriene A4 hydrolase in complex with resveratrol | 分子名称: | ACETATE ION, IMIDAZOLE, Leukotriene A-4 hydrolase, ... | 著者 | Davies, D.R. | 登録日 | 2009-01-13 | 公開日 | 2009-07-28 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (2.33 Å) | 主引用文献 | Discovery of leukotriene A4 hydrolase inhibitors using metabolomics biased fragment crystallography. J.Med.Chem., 52, 2009
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3FTY
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![BU of 3fty by Molmil](/molmil-images/mine/3fty) | |
3FUF
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![BU of 3fuf by Molmil](/molmil-images/mine/3fuf) | |
3FU3
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![BU of 3fu3 by Molmil](/molmil-images/mine/3fu3) | |
3FTW
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![BU of 3ftw by Molmil](/molmil-images/mine/3ftw) | |
3FUD
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![BU of 3fud by Molmil](/molmil-images/mine/3fud) | |
3FUE
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![BU of 3fue by Molmil](/molmil-images/mine/3fue) | |
3FUK
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![BU of 3fuk by Molmil](/molmil-images/mine/3fuk) | |