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1RCW
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BU of 1rcw by Molmil
Crystal structure of CT610 from Chlamydia trachomatis
分子名称: CT610, FE (III) ION
著者Schwarzenbacher, R, Liddington, R.C.
登録日2003-11-04
公開日2004-05-04
最終更新日2011-07-13
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Structure of the Chlamydia protein CADD reveals a redox enzyme that modulates host cell apoptosis.
J.Biol.Chem., 279, 2004
7P44
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Structure of CgGBE in P21212 space group
分子名称: 1,2-ETHANEDIOL, 1,4-alpha-glucan-branching enzyme
著者Ballut, L, Conchou, L, Violot, S, Galisson, F, Aghajari, N.
登録日2021-07-09
公開日2022-07-27
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献The Candida glabrata glycogen branching enzyme structure reveals unique features of branching enzymes of the Saccharomycetaceae phylum.
Glycobiology, 32, 2022
7P45
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Structure of CgGBE in P212121 space group
分子名称: 1,2-ETHANEDIOL, 1,4-alpha-glucan-branching enzyme
著者Ballut, L, Conchou, L, Violot, S, Galisson, F, Aghajari, N.
登録日2021-07-09
公開日2022-07-27
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (2.09 Å)
主引用文献The Candida glabrata glycogen branching enzyme structure reveals unique features of branching enzymes of the Saccharomycetaceae phylum.
Glycobiology, 32, 2022
7P43
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Structure of CgGBE in complex with maltotriose
分子名称: 1,4-alpha-glucan-branching enzyme, alpha-D-glucopyranose-(1-4)-alpha-D-glucopyranose-(1-4)-alpha-D-glucopyranose
著者Ballut, L, Conchou, L, Violot, S, Galisson, F, Aghajari, N.
登録日2021-07-09
公開日2022-07-27
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (1.93 Å)
主引用文献The Candida glabrata glycogen branching enzyme structure reveals unique features of branching enzymes of the Saccharomycetaceae phylum.
Glycobiology, 32, 2022
2ICA
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BU of 2ica by Molmil
CD11a (LFA1) I-domain complexed with BMS-587101 aka 5-[(5S, 9R)-9-(4-cyanophenyl)-3-(3,5-dichlorophenyl)-1-methyl-2,4-dioxo-1,3,7-triazaspiro [4.4]non-7-yl]methyl]-3-thiophenecarboxylicacid
分子名称: 5-[(5S,9R)-9-(4-CYANOPHENYL)-3-(3,5-DICHLOROPHENYL)-1-METHYL-2,4-DIOXO-1,3,7-TRIAZASPIRO [4.4]NON-7-YL]METHYL]-3-THIOPHENECARBOXYLICACID, Integrin alpha-L
著者Sheriff, S, Einspahr, H.
登録日2006-09-12
公開日2006-12-19
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (1.56 Å)
主引用文献Discovery and Development of 5-[(5S,9R)-9- (4-Cyanophenyl)-3-(3,5-dichlorophenyl)-1- methyl-2,4-dioxo-1,3,7-triazaspiro[4.4]non- 7-yl-methyl]-3-thiophenecarboxylic acid (BMS-587101)-A Small Molecule Antagonist Leukocyte Function Associated Antigen-1.
J.Med.Chem., 49, 2006
3HAE
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BU of 3hae by Molmil
Rational development of high-affinity T-cell receptor-like antibodies
分子名称: Antibody heavy chain, Antibody light chain, Beta-2-microglobulin, ...
著者Stewart-Jones, G, Wadle, A, Hombach, A, Shenderov, E, Held, G, Fischer, E.
登録日2009-05-01
公開日2009-05-19
最終更新日2011-07-13
実験手法X-RAY DIFFRACTION (2.9 Å)
主引用文献Rational development of high-affinity T-cell receptor-like antibodies
Proc.Natl.Acad.Sci.USA, 106, 2009
3O1G
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BU of 3o1g by Molmil
Cathepsin K covalently bound to a 2-cyano pyrimidine inhibitor with a benzyl P3 group.
分子名称: Cathepsin K, N-benzyl-3-(2-cyano-6-propylpyrimidin-4-yl)-N-[2-(dimethylamino)ethyl]-5-(trifluoromethyl)benzamide, SULFATE ION
著者Fradera, X, van Zeeland, M, Uitdehaag, J.C.M.
登録日2010-07-21
公開日2010-10-06
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (1.65 Å)
主引用文献Optimisation of 2-cyano-pyrimidine inhibitors of cathepsin K: improving selectivity over hERG.
Bioorg.Med.Chem.Lett., 20, 2010
3O0U
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BU of 3o0u by Molmil
Cathepsin K covalently bound to a cyano-pyrimidine inhibitor with improved selectivity over hERG
分子名称: 3-{2-[(E)-iminomethyl]-6-propylpyrimidin-4-yl}-N,N-dimethyl-5-(trifluoromethyl)benzamide, Cathepsin K
著者Fradera, X, van Zeeland, M, Uitdehaag, J.C.M.
登録日2010-07-20
公開日2011-03-30
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Optimisation of 2-cyano-pyrimidine inhibitors of cathepsin K: improving selectivity over hERG.
Bioorg.Med.Chem.Lett., 20, 2010
8BUX
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BU of 8bux by Molmil
Rab-binding domain of human MiniBAR
分子名称: 1,2-ETHANEDIOL, Granule associated Rac and RHOG effector protein 1, MAGNESIUM ION, ...
著者Pylypenko, O, Hammich, H, Houdusse, A.
登録日2022-12-01
公開日2023-12-13
実験手法X-RAY DIFFRACTION (1.86 Å)
主引用文献MiniBAR/KIAA0355 is a dual Rac and Rab effector that controls actin contractility and trafficking for successful ciliogenesis
To Be Published
8BUY
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BU of 8buy by Molmil
Rac-binding domain of human MiniBAR
分子名称: 1,2-ETHANEDIOL, Granule associated Rac and RHOG effector protein 1, SULFATE ION
著者Pylypenko, O, Hammich, H, Houdusse, A.
登録日2022-12-01
公開日2023-12-13
実験手法X-RAY DIFFRACTION (1.6 Å)
主引用文献MiniBAR/KIAA0355 is a dual Rac and Rab effector that controls actin contractility and trafficking for successful ciliogenesis
To Be Published
2O7N
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BU of 2o7n by Molmil
CD11A (LFA1) I-domain complexed with 7A-[(4-cyanophenyl)methyl]-6-(3,5-dichlorophenyl)-5-oxo-2,3,5,7A-tetrahydro-1H-pyrrolo[1,2-A]pyrrole-7-carbonitrile
分子名称: 7A-[(4-cyanophenyl)methyl]-6-(3,5-dichlorophenyl)-5-oxo-2,3,5,7A-tetrahydro-1H-pyrrolo[1,2-A]pyrrole-7-carbonitrile, Integrin alpha-L
著者Sheriff, S.
登録日2006-12-11
公開日2007-03-20
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (1.75 Å)
主引用文献Design of LFA-1 antagonists based on a 2,3-dihydro-1H-pyrrolizin-5(7aH)-one scaffold.
Bioorg.Med.Chem.Lett., 17, 2007
8D2J
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BU of 8d2j by Molmil
A novel insecticidal protein from ferns IPD113_Cow.
分子名称: GLYCEROL, IPD113_Cow
著者Maher, M.J.
登録日2022-05-30
公開日2023-11-08
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Novel insecticidal proteins from ferns resemble insecticidal proteins from Bacillus thuringiensis.
Proc.Natl.Acad.Sci.USA, 120, 2023
1MRE
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BU of 1mre by Molmil
PREPARATION, CHARACTERIZATION AND CRYSTALLIZATION OF AN ANTIBODY FAB FRAGMENT THAT RECOGNIZES RNA. CRYSTAL STRUCTURES OF NATIVE FAB AND THREE FAB-MONONUCLEOTIDE COMPLEXES
分子名称: GUANOSINE-5'-DIPHOSPHATE, IGG2B-KAPPA JEL103 FAB (HEAVY CHAIN), IGG2B-KAPPA JEL103 FAB (LIGHT CHAIN), ...
著者Pokkuluri, P.R, Cygler, M.
登録日1994-06-13
公開日1995-02-14
最終更新日2024-06-05
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Preparation, characterization and crystallization of an antibody Fab fragment that recognizes RNA. Crystal structures of native Fab and three Fab-mononucleotide complexes.
J.Mol.Biol., 243, 1994
1MRF
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BU of 1mrf by Molmil
PREPARATION, CHARACTERIZATION AND CRYSTALLIZATION OF AN ANTIBODY FAB FRAGMENT THAT RECOGNIZES RNA. CRYSTAL STRUCTURES OF NATIVE FAB AND THREE FAB-MONONUCLEOTIDE COMPLEXES
分子名称: 2'-DEOXYINOSINE-5'-MONOPHOSPHATE, IGG2B-KAPPA JEL103 FAB (HEAVY CHAIN), IGG2B-KAPPA JEL103 FAB (LIGHT CHAIN), ...
著者Pokkuluri, P.R, Cygler, M.
登録日1994-06-13
公開日1995-02-14
最終更新日2024-06-05
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Preparation, characterization and crystallization of an antibody Fab fragment that recognizes RNA. Crystal structures of native Fab and three Fab-mononucleotide complexes.
J.Mol.Biol., 243, 1994
1MRD
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BU of 1mrd by Molmil
PREPARATION, CHARACTERIZATION AND CRYSTALLIZATION OF AN ANTIBODY FAB FRAGMENT THAT RECOGNIZES RNA. CRYSTAL STRUCTURES OF NATIVE FAB AND THREE FAB-MONONUCLEOTIDE COMPLEXES
分子名称: IGG2B-KAPPA JEL103 FAB (HEAVY CHAIN), IGG2B-KAPPA JEL103 FAB (LIGHT CHAIN), IMIDAZOLE, ...
著者Pokkuluri, P.R, Cygler, M.
登録日1994-06-13
公開日1995-02-14
最終更新日2024-06-05
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Preparation, characterization and crystallization of an antibody Fab fragment that recognizes RNA. Crystal structures of native Fab and three Fab-mononucleotide complexes.
J.Mol.Biol., 243, 1994
1MRC
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BU of 1mrc by Molmil
PREPARATION, CHARACTERIZATION AND CRYSTALLIZATION OF AN ANTIBODY FAB FRAGMENT THAT RECOGNIZES RNA. CRYSTAL STRUCTURES OF NATIVE FAB AND THREE FAB-MONONUCLEOTIDE COMPLEXES
分子名称: IGG2B-KAPPA JEL103 FAB (HEAVY CHAIN), IGG2B-KAPPA JEL103 FAB (LIGHT CHAIN), IMIDAZOLE, ...
著者Pokkuluri, P.R, Cygler, M.
登録日1994-06-13
公開日1995-02-14
最終更新日2024-06-05
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Preparation, characterization and crystallization of an antibody Fab fragment that recognizes RNA. Crystal structures of native Fab and three Fab-mononucleotide complexes.
J.Mol.Biol., 243, 1994
5IXF
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BU of 5ixf by Molmil
Solution structure of the STAM2 SH3 with AMSH derived peptide complex
分子名称: STAM-binding protein, Signal transducing adapter molecule 2
著者Hologne, M, Cantrelle, F.X, Trivelli, X, Walker, O.
登録日2016-03-23
公開日2016-12-07
最終更新日2024-06-19
実験手法SOLUTION NMR
主引用文献NMR Reveals the Interplay among the AMSH SH3 Binding Motif, STAM2, and Lys63-Linked Diubiquitin.
J.Mol.Biol., 428, 2016
6ENQ
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BU of 6enq by Molmil
Structure of human PPAR gamma LBD in complex with Lanifibranor (IVA337)
分子名称: 4-[1-(1,3-benzothiazol-6-ylsulfonyl)-5-chloro-indol-2-yl]butanoic acid, Peroxisome proliferator-activated receptor gamma
著者Boubia, B, Poupardin, O, Barth, M, Amaudrut, J, Broqua, P, Tallandier, M, Zeyer, D.
登録日2017-10-06
公開日2018-03-14
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Design, Synthesis, and Evaluation of a Novel Series of Indole Sulfonamide Peroxisome Proliferator Activated Receptor (PPAR) alpha / gamma / delta Triple Activators: Discovery of Lanifibranor, a New Antifibrotic Clinical Candidate.
J. Med. Chem., 61, 2018
3O31
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BU of 3o31 by Molmil
E81Q mutant of MtNAS in complex with a reaction intermediate
分子名称: BROMIDE ION, N-[(3S)-3-amino-3-carboxypropyl]-L-glutamic acid, ThermoNicotianamine Synthase
著者Dreyfus, C, Pignol, D, Arnoux, P.
登録日2010-07-23
公開日2011-06-08
最終更新日2014-11-12
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献The crystallographic structure of thermoNicotianamine synthase with a synthetic reaction intermediate highlights the sequential processing mechanism.
Chem.Commun.(Camb.), 47, 2011
8AIK
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BU of 8aik by Molmil
Crystal structure of DltE from L. plantarum, tartare bound form
分子名称: Beta-lactamase family protein, L(+)-TARTARIC ACID
著者Ravaud, S, Nikolopoulos, N, Grangeasse, C.
登録日2022-07-26
公開日2023-04-26
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (1.95 Å)
主引用文献Structure-function analysis of Lactiplantibacillus plantarum DltE& reveals D-alanylated lipoteichoic acids as direct cues supporting Drosophila juvenile growth.
Elife, 12, 2023
8AJI
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BU of 8aji by Molmil
Crystal structure of DltE from L. plantarum, TCEP form
分子名称: 3,3',3''-phosphanetriyltripropanoic acid, Beta-lactamase family protein, GLYCEROL, ...
著者Ravaud, S, Nikolopoulos, N, Grangeasse, C.
登録日2022-07-28
公開日2023-04-26
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (1.94 Å)
主引用文献Structure-function analysis of Lactiplantibacillus plantarum DltE& reveals D-alanylated lipoteichoic acids as direct cues supporting Drosophila juvenile growth.
Elife, 12, 2023
8AKH
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BU of 8akh by Molmil
Crystal structure of DltE from L. plantarum soaked with LTA
分子名称: Beta-lactamase family protein, GLYCEROL, L(+)-TARTARIC ACID, ...
著者Ravaud, S, Nikolopoulos, N, Grangeasse, C.
登録日2022-07-29
公開日2023-04-26
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (1.4 Å)
主引用文献Structure-function analysis of Lactiplantibacillus plantarum DltE& reveals D-alanylated lipoteichoic acids as direct cues supporting Drosophila juvenile growth.
Elife, 12, 2023
8AGR
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BU of 8agr by Molmil
Crystal structure of DltE from L. plantarum, apo form
分子名称: 1,2-ETHANEDIOL, Beta-lactamase family protein, SULFATE ION
著者Ravaud, S, Nikolopoulos, N, Grangeasse, C.
登録日2022-07-20
公開日2023-04-26
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (1.86 Å)
主引用文献Structure-function analysis of Lactiplantibacillus plantarum DltE& reveals D-alanylated lipoteichoic acids as direct cues supporting Drosophila juvenile growth.
Elife, 12, 2023
1CRL
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BU of 1crl by Molmil
INSIGHTS INTO INTERFACIAL ACTIVATION FROM AN 'OPEN' STRUCTURE OF CANDIDA RUGOSA LIPASE
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, LIPASE
著者Grochulski, P, Cygler, M.
登録日1993-03-02
公開日1994-01-31
最終更新日2020-07-29
実験手法X-RAY DIFFRACTION (2.06 Å)
主引用文献Insights into interfacial activation from an open structure of Candida rugosa lipase.
J.Biol.Chem., 268, 1993
1EWY
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BU of 1ewy by Molmil
ANABAENA PCC7119 FERREDOXIN:FERREDOXIN-NADP+-REDUCTASE COMPLEX
分子名称: FE2/S2 (INORGANIC) CLUSTER, FERREDOXIN I, FERREDOXIN-NADP REDUCTASE, ...
著者Morales, R, Charon, M.H, Frey, M.
登録日2000-04-28
公開日2001-02-07
最終更新日2023-08-09
実験手法X-RAY DIFFRACTION (2.38 Å)
主引用文献Crystallographic studies of the interaction between the ferredoxin-NADP+ reductase and ferredoxin from the cyanobacterium Anabaena: looking for the elusive ferredoxin molecule.
Acta Crystallogr.,Sect.D, 56, 2000

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