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1IY1
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Crystal structure of the FtsH ATPase domain with ADP from Thermus thermophilus
分子名称: ADENOSINE-5'-DIPHOSPHATE, ATP-dependent metalloprotease FtsH
著者Niwa, H, Tsuchiya, D, Makyio, H, Yoshida, M, Morikawa, K.
登録日2002-07-10
公開日2002-11-06
最終更新日2023-12-27
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献Hexameric ring structure of the ATPase domain of the membrane-integrated metalloprotease FtsH from Thermus thermophilus HB8
Structure, 10, 2002
1IY0
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Crystal structure of the FtsH ATPase domain with AMP-PNP from Thermus thermophilus
分子名称: ATP-dependent metalloprotease FtsH, PHOSPHOAMINOPHOSPHONIC ACID-ADENYLATE ESTER
著者Niwa, H, Tsuchiya, D, Makyio, H, Yoshida, M, Morikawa, K.
登録日2002-07-10
公開日2002-11-06
最終更新日2023-12-27
実験手法X-RAY DIFFRACTION (2.95 Å)
主引用文献Hexameric ring structure of the ATPase domain of the membrane-integrated metalloprotease FtsH from Thermus thermophilus HB8
Structure, 10, 2002
2E4W
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Crystal structure of the extracellular region of the group II metabotropic glutamate receptor complexed with 1S,3S-ACPD
分子名称: (1S,3S)-1-aminocyclopentane-1,3-dicarboxylic acid, 2-acetamido-2-deoxy-beta-D-glucopyranose, Metabotropic glutamate receptor 3
著者Muto, T, Tsuchiya, D, Morikawa, K, Jingami, H.
登録日2006-12-17
公開日2007-02-27
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Structures of the extracellular regions of the group II/III metabotropic glutamate receptors
Proc.Natl.Acad.Sci.Usa, 104, 2007
2E4V
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Crystal structure of the extracellular region of the group II metabotropic glutamate receptor complexed with DCG-IV
分子名称: (1R,2R)-3-[(S)-amino(carboxy)methyl]cyclopropane-1,2-dicarboxylic acid, 2-acetamido-2-deoxy-beta-D-glucopyranose, Metabotropic glutamate receptor 3
著者Muto, T, Tsuchiya, D, Morikawa, K, Jingami, H.
登録日2006-12-17
公開日2007-02-27
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Structures of the extracellular regions of the group II/III metabotropic glutamate receptors
Proc.Natl.Acad.Sci.Usa, 104, 2007
1GEF
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Crystal structure of the archaeal holliday junction resolvase HJC
分子名称: HOLLIDAY JUNCTION RESOLVASE, SULFATE ION
著者Nishino, T, Komori, K, Tsuchiya, D, Ishino, Y, Morikawa, K.
登録日2000-11-08
公開日2001-03-21
最終更新日2023-12-27
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Crystal structure of the archaeal holliday junction resolvase Hjc and implications for DNA recognition.
Structure, 9, 2001
4Y7S
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Crystal Structure of the CFEM protein Csa2
分子名称: 1,2-ETHANEDIOL, CHLORIDE ION, HEME B/C, ...
著者Dvir, H, Weissman, Z, Nasser, L, Hiya, D, Kornitzer, D.
登録日2015-02-16
公開日2016-08-03
最終更新日2016-10-12
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Structural basis of haem-iron acquisition by fungal pathogens.
Nat Microbiol, 1, 2016
8WIU
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Bromodomain and Extra-terminal Domain (BET) BRD4
分子名称: 7-[5-[1-(cyclopropylmethyl)-3,5-dimethyl-pyrazol-4-yl]pyridin-3-yl]-1~{H}-imidazo[4,5-b]pyridine, Isoform C of Bromodomain-containing protein 4
著者Cao, D, Zhiyan, D, Xiong, B.
登録日2023-09-25
公開日2024-01-03
実験手法X-RAY DIFFRACTION (1.4 Å)
主引用文献Discovery of a brain-permeable bromodomain and extra terminal domain (BET) inhibitor with selectivity for BD1 for the treatment of multiple sclerosis.
Eur.J.Med.Chem., 265, 2023
8IBQ
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Bromodomain and Extra-terminal Domain (BET) BRD4
分子名称: 7-[2-fluoranyl-3-(1,3,5-trimethylpyrazol-4-yl)phenyl]-1~{H}-imidazo[4,5-b]pyridine, Bromodomain-containing protein 4
著者Cao, D, Zhiyan, D, Xiong, B.
登録日2023-02-10
公開日2023-10-04
実験手法X-RAY DIFFRACTION (1.45 Å)
主引用文献Discovery of 1 H -Imidazo[4,5- b ]pyridine Derivatives as Potent and Selective BET Inhibitors for the Management of Neuropathic Pain.
J.Med.Chem., 66, 2023
8IDH
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Bromodomain and Extra-terminal Domain (BET) BRD4
分子名称: 7-[2-fluoranyl-3-(1,3,5-trimethylpyrazol-4-yl)phenyl]-1~{H}-imidazo[4,5-b]pyridine, Bromodomain-containing protein 4
著者Cao, D, Zhiyan, D, Xiong, B.
登録日2023-02-13
公開日2023-10-04
実験手法X-RAY DIFFRACTION (1.57 Å)
主引用文献Discovery of 1 H -Imidazo[4,5- b ]pyridine Derivatives as Potent and Selective BET Inhibitors for the Management of Neuropathic Pain.
J.Med.Chem., 66, 2023
1G7M
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CRYSTAL STRUCTURE OF HEN EGG WHITE LYSOZYME (HEL) COMPLEXED WITH THE MUTANT ANTI-HEL MONOCLONAL ANTIBODY D1.3 (VLW92V)
分子名称: ANTI-HEN EGG WHITE LYSOZYME MONOCLONAL ANTIBODY D1.3, LYSOZYME C
著者Sundberg, E.J, Urrutia, M, Braden, B.C, Isern, J, Mariuzza, R.A.
登録日2000-11-10
公開日2000-11-22
最終更新日2021-10-27
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Estimation of the hydrophobic effect in an antigen-antibody protein-protein interface.
Biochemistry, 39, 2000
1G7L
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CRYSTAL STRUCTURE OF HEN EGG WHITE LYSOZYME (HEL) COMPLEXED WITH THE MUTANT ANTI-HEL MONOCLONAL ANTIBODY D1.3 (VLW92S)
分子名称: ANTI-HEN EGG WHITE LYSOZYME MONOCLONAL ANTIBODY D1.3, LYSOZYME C
著者Sundberg, E.J, Urrutia, M, Braden, B.C, Isern, J, Mariuzza, R.A.
登録日2000-11-10
公開日2000-11-22
最終更新日2021-10-27
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Estimation of the hydrophobic effect in an antigen-antibody protein-protein interface.
Biochemistry, 39, 2000
1V5B
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The Structure Of The Mutant, S225A and E251L, Of 3-Isopropylmalate Dehydrogenase From Bacillus Coagulans
分子名称: 3-isopropylmalate dehydrogenase, SULFATE ION
著者Fujita, K, Minami, H, Suzuki, K, Tsunoda, M, Sekiguchi, T, Mizui, R, Tsuzaki, S, Nakamura, S, Takenaka, A.
登録日2003-11-22
公開日2005-02-15
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (2.95 Å)
主引用文献Crystal structure of a highly thermo-stabilized mutant of 3-isopropylmalate dehydrogenase from Bacillus coagulans: An evaluation of local packing density in the hydrophobic core
To be Published
1SBB
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BU of 1sbb by Molmil
T-CELL RECEPTOR BETA CHAIN COMPLEXED WITH SUPERANTIGEN SEB
分子名称: PROTEIN (14.3.D T CELL ANTIGEN RECEPTOR), PROTEIN (STAPHYLOCOCCAL ENTEROTOXIN B)
著者Li, H, Mariuzza, R.A.
登録日1999-02-22
公開日1999-03-01
最終更新日2023-08-23
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Three-dimensional structure of the complex between a T cell receptor beta chain and the superantigen staphylococcal enterotoxin B.
Immunity, 9, 1998
1G7H
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CRYSTAL STRUCTURE OF HEN EGG WHITE LYSOZYME (HEL) COMPLEXED WITH THE MUTANT ANTI-HEL MONOCLONAL ANTIBODY D1.3(VLW92A)
分子名称: ANTI-HEN EGG WHITE LYSOZYME MONOCLONAL ANTIBODY D1.3, LYSOZYME C
著者Sundberg, E.J, Urrutia, M, Braden, B.C, Isern, J, Mariuzza, R.A.
登録日2000-11-10
公開日2000-11-22
最終更新日2023-08-09
実験手法X-RAY DIFFRACTION (1.85 Å)
主引用文献Estimation of the hydrophobic effect in an antigen-antibody protein-protein interface.
Biochemistry, 39, 2000
1G7J
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CRYSTAL STRUCTURE OF HEN EGG WHITE LYSOZYME (HEL) COMPLEXED WITH THE MUTANT ANTI-HEL MONOCLONAL ANTIBODY D1.3 (VLW92H)
分子名称: ANTI-HEN EGG WHITE LYSOZYME MONOCLONAL ANTIBODY D1.3, LYSOZYME C
著者Sundberg, E.J, Urrutia, M, Braden, B.C, Isern, J, Mariuzza, R.A.
登録日2000-11-10
公開日2000-11-22
最終更新日2021-10-27
実験手法X-RAY DIFFRACTION (1.75 Å)
主引用文献Estimation of the hydrophobic effect in an antigen-antibody protein-protein interface.
Biochemistry, 39, 2000
1G7I
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CRYSTAL STRUCTURE OF HEN EGG WHITE LYSOZYME (HEL) COMPLEXED WITH THE MUTANT ANTI-HEL MONOCLONAL ANTIBODY D1.3 (VLW92F)
分子名称: ANTI-HEN EGG WHITE LYSOZYME MONOCLONAL ANTIBODY D1.3, LYSOZYME C, PHOSPHATE ION
著者Sundberg, E.J, Urrutia, M, Braden, B.C, Isern, J, Mariuzza, R.A.
登録日2000-11-10
公開日2000-11-22
最終更新日2021-10-27
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Estimation of the hydrophobic effect in an antigen-antibody protein-protein interface.
Biochemistry, 39, 2000
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