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1V1M
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BU of 1v1m by Molmil
CROSSTALK BETWEEN COFACTOR BINDING AND THE PHOSPHORYLATION LOOP CONFORMATION IN THE BCKD MACHINE
分子名称: 2-OXOISOVALERATE DEHYDROGENASE ALPHA SUBUNIT, 2-OXOISOVALERATE DEHYDROGENASE BETA SUBUNIT, BENZAMIDINE, ...
著者Li, J, Wynn, R.M, Machius, M, Chuang, J.L, Karthikeyan, S, Tomchick, D.R, Chuang, D.T.
登録日2004-04-20
公開日2004-06-03
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Cross-Talk between Thiamin Diphosphate Binding and Phosphorylation Loop Conformation in Human Branched-Chain Alpha-Keto Acid Decarboxylase/Dehydrogenase.
J.Biol.Chem., 279, 2004
1V1R
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BU of 1v1r by Molmil
CROSSTALK BETWEEN COFACTOR BINDING AND THE PHOSPHORYLATION LOOP CONFORMATION IN THE BCKD MACHINE
分子名称: 2-OXOISOVALERATE DEHYDROGENASE ALPHA SUBUNIT, 2-OXOISOVALERATE DEHYDROGENASE BETA SUBUNIT, CHLORIDE ION, ...
著者Li, J, Wynn, R.M, Machius, M, Chuang, J.L, Karthikeyan, S, Tomchick, D.R, Chuang, D.T.
登録日2004-04-22
公開日2004-06-03
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Cross-Talk between Thiamin Diphosphate Binding and Phosphorylation Loop Conformation in Human Branched-Chain {Alpha}-Keto Acid Decarboxylase/Dehydrogenase
J.Biol.Chem., 279, 2004
1V16
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BU of 1v16 by Molmil
CROSSTALK BETWEEN COFACTOR BINDING AND THE PHOSPHORYLATION LOOP CONFORMATION IN THE BCKD MACHINE
分子名称: 2-OXOISOVALERATE DEHYDROGENASE ALPHA SUBUNIT, 2-OXOISOVALERATE DEHYDROGENASE BETA SUBUNIT, BENZAMIDINE, ...
著者Li, J, Wynn, R.M, Machius, M, Chuang, J.L, Karthikeyan, S, Tomchick, D.R, Chuang, D.T.
登録日2004-04-07
公開日2004-06-03
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Cross-Talk between Thiamin Diphosphate Binding and Phosphorylation Loop Conformation in Human Branched-Chain {Alpha}-Keto Acid Decarboxylase/Dehydrogenase
J.Biol.Chem., 279, 2004
1WCI
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BU of 1wci by Molmil
Reactivity modulation of human branched-chain alpha-ketoacid dehydrogenase by an internal molecular switch
分子名称: 2-OXOISOVALERATE DEHYDROGENASE ALPHA SUBUNIT, 2-OXOISOVALERATE DEHYDROGENASE BETA SUBUNIT, C2-1-HYDROXY-3-METHYL-BUTYL-THIAMIN, ...
著者Machius, M, Wynn, R.M, Chuang, J.L, Tomchick, D.R, Brautigam, C.A, Chuang, D.T.
登録日2004-11-16
公開日2006-02-16
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (1.84 Å)
主引用文献A Versatile Conformational Switch Regulates Reactivity in Human Branched-Chain Alpha-Ketoacid Dehydrogenase.
Structure, 14, 2006
8XHU
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BU of 8xhu by Molmil
Crystal structure of Helicobacter pylori IspDF
分子名称: 1,2-ETHANEDIOL, Bifunctional enzyme IspD/IspF, CHLORIDE ION, ...
著者Chen, X, Wu, D.
登録日2023-12-18
公開日2024-04-10
最終更新日2024-05-01
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Two natural compounds as potential inhibitors against the Helicobacter pylori and Acinetobacter baumannii IspD enzymes.
Int J Antimicrob Agents, 63, 2024
8XKG
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BU of 8xkg by Molmil
Crystal structure of Acinetobacter baumannii IspD
分子名称: 2-C-methyl-D-erythritol 4-phosphate cytidylyltransferase, GLYCEROL
著者Chen, X, Wu, D.
登録日2023-12-23
公開日2024-04-10
最終更新日2024-05-01
実験手法X-RAY DIFFRACTION (1.6 Å)
主引用文献Two natural compounds as potential inhibitors against the Helicobacter pylori and Acinetobacter baumannii IspD enzymes.
Int J Antimicrob Agents, 63, 2024
9BFL
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BU of 9bfl by Molmil
Solution structure of the scorpion toxin omega-Buthitoxin-Hf1a
分子名称: Buthitoxin-Hf1a
著者Rosengren, K.J, Payne, C.D.
登録日2024-04-18
公開日2024-06-05
実験手法SOLUTION NMR
主引用文献Novel Scorpion Toxin omega-Buthitoxin-Hf1a Selectively Inhibits Calcium Influx via Ca V 3.3 and Ca V 3.2 and Alleviates Allodynia in a Mouse Model of Acute Postsurgical Pain.
Int J Mol Sci, 25, 2024
7E4I
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BU of 7e4i by Molmil
Cryo-EM structure of the yeast mitochondrial SAM-Tom40/Tom5/Tom6 complex at 3.0 angstrom
分子名称: Mitochondrial import receptor subunit TOM40, Mitochondrial import receptor subunit TOM5, Mitochondrial import receptor subunit TOM6, ...
著者Wang, Q, Guan, Z.Y, Qi, L.B, Yan, C.Y, Yin, P.
登録日2021-02-13
公開日2021-09-01
最終更新日2024-06-05
実験手法ELECTRON MICROSCOPY (3.05 Å)
主引用文献Structural insight into the SAM-mediated assembly of the mitochondrial TOM core complex.
Science, 373, 2021
7E4H
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BU of 7e4h by Molmil
Cryo-EM structure of the yeast mitochondrial SAM-Tom40 complex at 3.0 angstrom
分子名称: Mitochondrial import receptor subunit TOM40, Sorting assembly machinery 35 kDa subunit, Sorting assembly machinery 37 kDa subunit, ...
著者Wang, Q, Guan, Z.Y, Qi, L.B, Yan, C.Y, Yin, P.
登録日2021-02-13
公開日2021-09-01
最終更新日2024-06-05
実験手法ELECTRON MICROSCOPY (3.01 Å)
主引用文献Structural insight into the SAM-mediated assembly of the mitochondrial TOM core complex.
Science, 373, 2021
4CLC
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BU of 4clc by Molmil
Crystal structure of Ybr137w protein
分子名称: UPF0303 PROTEIN YBR137W
著者Yeh, Y.-H, Lin, T.-W, Lin, C.-Y, Hsiao, C.-D.
登録日2014-01-14
公開日2014-11-19
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献Structural and Functional Characterization of Ybr137Wp Implicate its Involvement in the Targeting of Tail-Anchored Proteins to Membranes.
Mol.Cell.Biol., 34, 2014
8XKF
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BU of 8xkf by Molmil
Crystal structure of Helicobacter pylori IspDF with substrate CTP
分子名称: 1,2-ETHANEDIOL, Bifunctional enzyme IspD/IspF, CHLORIDE ION, ...
著者Chen, X, Wu, D.
登録日2023-12-23
公開日2024-04-10
最終更新日2024-05-01
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Two natural compounds as potential inhibitors against the Helicobacter pylori and Acinetobacter baumannii IspD enzymes.
Int J Antimicrob Agents, 63, 2024
7V7L
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BU of 7v7l by Molmil
Crystal Structure of the Heterodimeric HIF-3a:ARNT Complex
分子名称: Aryl hydrocarbon receptor nuclear translocator, Hypoxia-inducible factor 3-alpha
著者Diao, X, Ren, X, Li, F.W, Sun, X, Wu, D.
登録日2021-08-21
公開日2022-05-18
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Identification of oleoylethanolamide as an endogenous ligand for HIF-3 alpha.
Nat Commun, 13, 2022
7V7W
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BU of 7v7w by Molmil
Crystal Structure of the Heterodimeric HIF-3a:ARNT Complex with oleoylethanolamide (OEA)
分子名称: (Z)-N-(2-hydroxyethyl)octadec-9-enamide, Aryl hydrocarbon receptor nuclear translocator, Hypoxia-inducible factor 3-alpha
著者Diao, X, Ren, X, Li, F.W, Zhang, M, Sun, X, Wu, D.
登録日2021-08-21
公開日2022-05-18
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (2.507 Å)
主引用文献Identification of oleoylethanolamide as an endogenous ligand for HIF-3 alpha.
Nat Commun, 13, 2022
7W8O
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BU of 7w8o by Molmil
Solution structures of a disulfide-rich peptide that can bind mdm2
分子名称: drp2-a
著者Fan, S.H, Wu, Y.P, Wu, C.L.
登録日2021-12-08
公開日2022-06-08
最終更新日2023-06-14
実験手法SOLUTION NMR
主引用文献Structure-guided design of CPPC-paired disulfide-rich peptide libraries for ligand and drug discovery.
Chem Sci, 13, 2022
7W8K
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BU of 7w8k by Molmil
Solution structures of a disulfide-rich peptide that can bind mdm2
分子名称: drp1
著者Fan, S.H, Wu, Y.P, Wu, C.L.
登録日2021-12-08
公開日2022-06-08
最終更新日2023-06-14
実験手法SOLUTION NMR
主引用文献Structure-guided design of CPPC-paired disulfide-rich peptide libraries for ligand and drug discovery.
Chem Sci, 13, 2022
7W8R
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BU of 7w8r by Molmil
Solution structures of a disulfide-rich peptide that can bind mdm2
分子名称: drp2-b
著者Fan, S.H, Wu, Y.P, Wu, C.L.
登録日2021-12-08
公開日2022-06-08
最終更新日2023-06-14
実験手法SOLUTION NMR
主引用文献Structure-guided design of CPPC-paired disulfide-rich peptide libraries for ligand and drug discovery.
Chem Sci, 13, 2022
7W96
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BU of 7w96 by Molmil
Solution structures of a disulfide-rich peptide that can bind KEAP1
分子名称: drp6
著者Fan, S.H, Wu, Y.P, Wu, C.L.
登録日2021-12-09
公開日2022-11-09
実験手法SOLUTION NMR
主引用文献Structure-guided design of CPPC-paired disulfide-rich peptide libraries for ligand and drug discovery.
Chem Sci, 13, 2022
7WE3
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BU of 7we3 by Molmil
Solution structures of a disulfide-rich peptide that can bind CD28
分子名称: DRP8II
著者Fan, S.H, Wu, Y.P, Wu, C.L.
登録日2021-12-22
公開日2022-11-09
実験手法SOLUTION NMR
主引用文献Structure-guided design of CPPC-paired disulfide-rich peptide libraries for ligand and drug discovery.
Chem Sci, 13, 2022
7WEI
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BU of 7wei by Molmil
Solution structures of a disulfide-rich peptide that can bind CD28
分子名称: drp8I
著者Fan, S.H, Wu, Y.P, Wu, C.L.
登録日2021-12-23
公開日2022-11-09
実験手法SOLUTION NMR
主引用文献Structure-guided design of CPPC-paired disulfide-rich peptide libraries for ligand and drug discovery.
Chem Sci, 13, 2022
7W8T
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BU of 7w8t by Molmil
Solution structures of a disulfide-rich peptide that can bind KEAP1
分子名称: DRP3
著者Fan, S.H, Wu, Y.P, Wu, C.L.
登録日2021-12-08
公開日2022-06-08
最終更新日2023-06-14
実験手法SOLUTION NMR
主引用文献Structure-guided design of CPPC-paired disulfide-rich peptide libraries for ligand and drug discovery.
Chem Sci, 13, 2022
7W8Z
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BU of 7w8z by Molmil
Solution structures of a disulfide-rich peptide designed through sequence grafting
分子名称: drp4
著者Fan, S.H, Wu, Y.P, Wu, C.L.
登録日2021-12-09
公開日2022-06-08
最終更新日2023-06-14
実験手法SOLUTION NMR
主引用文献Structure-guided design of CPPC-paired disulfide-rich peptide libraries for ligand and drug discovery.
Chem Sci, 13, 2022
7XI3
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BU of 7xi3 by Molmil
Crystal Structure of the NPAS4-ARNT2 heterodimer in complex with DNA
分子名称: Aryl hydrocarbon receptor nuclear translocator 2, DNA (5'-D(P*CP*CP*AP*TP*CP*AP*CP*TP*CP*AP*CP*GP*AP*CP*CP*T)-3'), DNA (5'-D(P*GP*GP*AP*GP*GP*TP*CP*GP*TP*GP*AP*GP*TP*GP*AP*T)-3'), ...
著者Sun, X.N, Jing, L.Q, Li, F.W, Wu, D.L.
登録日2022-04-11
公開日2022-11-02
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (4.274 Å)
主引用文献Structures of NPAS4-ARNT and NPAS4-ARNT2 heterodimers reveal new dimerization modalities in the bHLH-PAS transcription factor family.
Proc.Natl.Acad.Sci.USA, 119, 2022
7XI4
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BU of 7xi4 by Molmil
Crystal Structure of the NPAS4-ARNT heterodimer in complex with DNA
分子名称: Aryl hydrocarbon receptor nuclear translocator, DNA (5'-D(*GP*GP*AP*GP*GP*TP*CP*GP*TP*GP*AP*GP*TP*GP*AP*T)-3'), DNA (5'-D(P*CP*CP*AP*TP*CP*AP*CP*TP*CP*AP*CP*GP*AP*CP*CP*T)-3'), ...
著者Sun, X.N, Jing, L.Q, Li, F.W, Wu, D.L.
登録日2022-04-12
公開日2022-11-02
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (4.707 Å)
主引用文献Structures of NPAS4-ARNT and NPAS4-ARNT2 heterodimers reveal new dimerization modalities in the bHLH-PAS transcription factor family.
Proc.Natl.Acad.Sci.USA, 119, 2022
7XHV
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BU of 7xhv by Molmil
Crystal Structure of the NPAS4-ARNT heterodimer in complex with DNA
分子名称: Aryl hydrocarbon receptor nuclear translocator, DNA (5'-D(P*CP*CP*AP*TP*CP*AP*CP*TP*CP*AP*CP*GP*AP*CP*CP*T)-3'), DNA (5'-D(P*GP*GP*AP*GP*GP*TP*CP*GP*TP*GP*AP*GP*TP*GP*AP*T)-3'), ...
著者Sun, X.N, Jing, L.Q, Li, F.W, Wu, D.L.
登録日2022-04-10
公開日2022-11-02
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (3.996 Å)
主引用文献Structures of NPAS4-ARNT and NPAS4-ARNT2 heterodimers reveal new dimerization modalities in the bHLH-PAS transcription factor family.
Proc.Natl.Acad.Sci.USA, 119, 2022

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