8GOL
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![BU of 8gol by Molmil](/molmil-images/mine/8gol) | crystal structure of SulE | 分子名称: | 2-[(4-chloranyl-6-methoxy-pyrimidin-2-yl)carbamoylsulfamoyl]benzoic acid, Alpha/beta fold hydrolase, GLYCEROL | 著者 | Liu, B, Ran, T, Wang, W, He, J. | 登録日 | 2022-08-25 | 公開日 | 2023-08-02 | 最終更新日 | 2024-05-29 | 実験手法 | X-RAY DIFFRACTION (1.6 Å) | 主引用文献 | Crystal structures of herbicide-detoxifying esterase reveal a lid loop affecting substrate binding and activity. Nat Commun, 14, 2023
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8GP0
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![BU of 8gp0 by Molmil](/molmil-images/mine/8gp0) | crystal structure of SulE | 分子名称: | Alpha/beta fold hydrolase, CITRIC ACID, GLYCEROL | 著者 | Liu, B, Ran, T, wang, W, He, J. | 登録日 | 2022-08-25 | 公開日 | 2023-08-02 | 最終更新日 | 2024-05-29 | 実験手法 | X-RAY DIFFRACTION (1.46 Å) | 主引用文献 | Crystal structures of herbicide-detoxifying esterase reveal a lid loop affecting substrate binding and activity. Nat Commun, 14, 2023
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7UFZ
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![BU of 7ufz by Molmil](/molmil-images/mine/7ufz) | Crystal structure of TDP1 complexed with compound XZ768 | 分子名称: | (4-{[(4S)-2-phenylimidazo[1,2-a]pyridin-3-yl]amino}phenyl)phosphonic acid, 1,2-ETHANEDIOL, DIMETHYL SULFOXIDE, ... | 著者 | Lountos, G.T, Zhao, X.Z, Wang, W, Tropea, J.E, Needle, D, Pommier, Y, Burke, T.R. | 登録日 | 2022-03-23 | 公開日 | 2023-04-12 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (1.559 Å) | 主引用文献 | Phosphonic acid-containing inhibitors of tyrosyl-DNA phosphodiesterase 1. Front Chem, 10, 2022
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7UFY
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![BU of 7ufy by Molmil](/molmil-images/mine/7ufy) | Crystal structure of TDP1 complexed with compound XZ766 | 分子名称: | 1,2-ETHANEDIOL, Tyrosyl-DNA phosphodiesterase 1, [(4-{[(4S)-2,7-diphenylimidazo[1,2-a]pyridin-3-yl]amino}phenyl)methyl]phosphonic acid | 著者 | Lountos, G.T, Zhao, X.Z, Wang, W, Tropea, J.E, Needle, D, Pommier, Y, Burke, T.R. | 登録日 | 2022-03-23 | 公開日 | 2023-04-12 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (1.584 Å) | 主引用文献 | Phosphonic acid-containing inhibitors of tyrosyl-DNA phosphodiesterase 1. Front Chem, 10, 2022
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8HEH
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![BU of 8heh by Molmil](/molmil-images/mine/8heh) | Crystal structure of GCN5-related N-acetyltransferase 05790 | 分子名称: | COENZYME A, GLYCEROL, GNAT family N-acetyltransferase | 著者 | Xu, M.X, Ran, T.T, Wang, W. | 登録日 | 2022-11-08 | 公開日 | 2022-12-21 | 最終更新日 | 2024-05-29 | 実験手法 | X-RAY DIFFRACTION (1.4 Å) | 主引用文献 | Crystal structure of prodigiosin binding protein PgbP, a GNAT family protein, in Serratia marcescens FS14. Biochem.Biophys.Res.Commun., 640, 2022
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8H4E
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![BU of 8h4e by Molmil](/molmil-images/mine/8h4e) | Blasnase-T13A/P55N with D-asn | 分子名称: | D-ASPARAGINE, FORMIC ACID, L-asparaginase, ... | 著者 | Lu, F, Wang, W, Chi, H, Ran, T. | 登録日 | 2022-10-10 | 公開日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (2.06 Å) | 主引用文献 | Structure-based rational design of Bacillus licheniformis L-asparaginase with low/no D-asparaginase activity for a safer enzyme To Be Published
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8H46
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![BU of 8h46 by Molmil](/molmil-images/mine/8h46) | Blasnase-T13A/P55N with L-asn | 分子名称: | ASPARAGINE, FORMIC ACID, GLYCEROL, ... | 著者 | Lu, F, Wang, W, Chi, H, Ran, T. | 登録日 | 2022-10-10 | 公開日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | Structure-based rational design of Bacillus licheniformis L-asparaginase with low/no D-asparaginase activity for a safer enzyme To Be Published
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8H47
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![BU of 8h47 by Molmil](/molmil-images/mine/8h47) | Blasnase-T13A/P55F | 分子名称: | FORMIC ACID, GLYCEROL, L-asparaginase, ... | 著者 | Lu, F, Wang, W, Chi, H, Ran, T. | 登録日 | 2022-10-10 | 公開日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Structure-based rational design of Bacillus licheniformis L-asparaginase with low/no D-asparaginase activity for a safer enzyme To Be Published
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8H4B
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![BU of 8h4b by Molmil](/molmil-images/mine/8h4b) | Blasnase-T13A/M57P with L-asn | 分子名称: | ASPARAGINE, FORMIC ACID, L-asparaginase, ... | 著者 | Lu, F, Wang, W, Chi, H, Ran, T. | 登録日 | 2022-10-10 | 公開日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Structure-based rational design of Bacillus licheniformis L-asparaginase with low/no D-asparaginase activity for a safer enzyme To Be Published
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8H4D
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![BU of 8h4d by Molmil](/molmil-images/mine/8h4d) | Blasnase-T13A/M57N | 分子名称: | FORMIC ACID, GLYCEROL, L-asparaginase, ... | 著者 | Lu, F, Wang, W, Chi, H, Ran, T. | 登録日 | 2022-10-10 | 公開日 | 2023-10-18 | 最終更新日 | 2024-05-01 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Structure-based rational design of Bacillus licheniformis L-asparaginase with low/no D-asparaginase activity for a safer enzyme To Be Published
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8H44
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![BU of 8h44 by Molmil](/molmil-images/mine/8h44) | Blasnase-P55N | 分子名称: | FORMIC ACID, L-asparaginase, MAGNESIUM ION | 著者 | Lu, F, Wang, W, Chi, H, Ran, T. | 登録日 | 2022-10-10 | 公開日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | Structure-based rational design of Bacillus licheniformis L-asparaginase with low/no D-asparaginase activity for a safer enzyme To Be Published
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8H45
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![BU of 8h45 by Molmil](/molmil-images/mine/8h45) | Blasnase-T13A/P55N | 分子名称: | FORMIC ACID, L-asparaginase, MAGNESIUM ION | 著者 | Lu, F, Wang, W, Chi, H, Ran, T. | 登録日 | 2022-10-10 | 公開日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (1.97 Å) | 主引用文献 | Structure-based rational design of Bacillus licheniformis L-asparaginase with low/no D-asparaginase activity for a safer enzyme To Be Published
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8H48
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![BU of 8h48 by Molmil](/molmil-images/mine/8h48) | Blasnase-T13A/P55F with L-asn | 分子名称: | ASPARAGINE, FORMIC ACID, L-asparaginase, ... | 著者 | Lu, F, Wang, W, Chi, H, Ran, T. | 登録日 | 2022-10-10 | 公開日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | Structure-based rational design of Bacillus licheniformis L-asparaginase with low/no D-asparaginase activity for a safer enzyme To Be Published
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8H49
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![BU of 8h49 by Molmil](/molmil-images/mine/8h49) | Blasnase-M57P | 分子名称: | FORMIC ACID, L-asparaginase, MAGNESIUM ION | 著者 | Lu, F, Wang, W, Chi, H, Ran, T. | 登録日 | 2022-10-10 | 公開日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Structure-based rational design of Bacillus licheniformis L-asparaginase with low/no D-asparaginase activity for a safer enzyme To Be Published
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8H4A
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![BU of 8h4a by Molmil](/molmil-images/mine/8h4a) | Blasnase-T13A/M57P | 分子名称: | FORMIC ACID, L-asparaginase, MAGNESIUM ION | 著者 | Lu, F, Wang, W, Chi, H, Ran, T. | 登録日 | 2022-10-10 | 公開日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Structure-based rational design of Bacillus licheniformis L-asparaginase with low/no D-asparaginase activity for a safer enzyme To Be Published
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8H4C
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![BU of 8h4c by Molmil](/molmil-images/mine/8h4c) | Blasnase-T13A/M57P | 分子名称: | FORMIC ACID, L-asparaginase, MAGNESIUM ION | 著者 | Lu, F, Wang, W, Chi, H, Ran, T. | 登録日 | 2022-10-10 | 公開日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (1.6 Å) | 主引用文献 | Structure-based rational design of Bacillus licheniformis L-asparaginase with low/no D-asparaginase activity for a safer enzyme To Be Published
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8H4G
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![BU of 8h4g by Molmil](/molmil-images/mine/8h4g) | Blasnase-T13A/M57N | 分子名称: | FORMIC ACID, L-asparaginase, MAGNESIUM ION | 著者 | Lu, F, Wang, W, Chi, H, Ran, T. | 登録日 | 2022-10-10 | 公開日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (1.81 Å) | 主引用文献 | Structure-based rational design of Bacillus licheniformis L-asparaginase with low/no D-asparaginase activity for a safer enzyme To Be Published
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8H4F
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![BU of 8h4f by Molmil](/molmil-images/mine/8h4f) | Blasnase-T13A/P55F with D-asn | 分子名称: | D-ASPARAGINE, FORMIC ACID, L-asparaginase, ... | 著者 | Lu, F, Wang, W, Chi, H, Ran, T. | 登録日 | 2022-10-10 | 公開日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Structure-based rational design of Bacillus licheniformis L-asparaginase with low/no D-asparaginase activity for a safer enzyme To Be Published
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3VPI
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![BU of 3vpi by Molmil](/molmil-images/mine/3vpi) | |
6N9T
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![BU of 6n9t by Molmil](/molmil-images/mine/6n9t) | Structure of a peptide-based photo-affinity cross-linker with Herceptin Fc | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-2)-alpha-D-mannopyranose-(1-6)-[alpha-D-mannopyranose-(1-3)]beta-D-mannopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-[alpha-L-fucopyranose-(1-6)]2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-2)-alpha-D-mannopyranose-(1-6)-[alpha-D-mannopyranose-(1-3)]beta-D-mannopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-[beta-L-fucopyranose-(1-6)]2-acetamido-2-deoxy-beta-D-glucopyranose, Immunoglobulin G1 FC, ... | 著者 | Sadowsky, J, Ultsch, M, Vance, N, Wang, W. | 登録日 | 2018-12-04 | 公開日 | 2019-01-16 | 最終更新日 | 2020-07-29 | 実験手法 | X-RAY DIFFRACTION (2.576 Å) | 主引用文献 | Development, Optimization, and Structural Characterization of an Efficient Peptide-Based Photoaffinity Cross-Linking Reaction for Generation of Homogeneous Conjugates from Wild-Type Antibodies. Bioconjug. Chem., 30, 2019
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3VPJ
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![BU of 3vpj by Molmil](/molmil-images/mine/3vpj) | |
5URY
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![BU of 5ury by Molmil](/molmil-images/mine/5ury) | Crystal structure of Frizzled 5 CRD in complex with PAM | 分子名称: | Frizzled-5, PALMITOLEIC ACID, alpha-L-fucopyranose-(1-3)-[alpha-L-fucopyranose-(1-4)][alpha-L-fucopyranose-(1-6)]2-acetamido-2-deoxy-beta-D-glucopyranose | 著者 | Mukund, S, Nile, A.H, Stanger, K, Hannoush, R.N, Wang, W. | 登録日 | 2017-02-13 | 公開日 | 2017-05-10 | 最終更新日 | 2020-07-29 | 実験手法 | X-RAY DIFFRACTION (2.098 Å) | 主引用文献 | Unsaturated fatty acyl recognition by Frizzled receptors mediates dimerization upon Wnt ligand binding. Proc. Natl. Acad. Sci. U.S.A., 114, 2017
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5VZX
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![BU of 5vzx by Molmil](/molmil-images/mine/5vzx) | Crystal structure of crenezumab Fab | 分子名称: | 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, Crenezumab Fab heavy chain, ... | 著者 | Ultsch, M, Wang, W. | 登録日 | 2017-05-29 | 公開日 | 2017-08-09 | 実験手法 | X-RAY DIFFRACTION (2.501 Å) | 主引用文献 | Structure of Crenezumab Complex with Abeta Shows Loss of beta-Hairpin. Sci Rep, 6, 2016
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5W96
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![BU of 5w96 by Molmil](/molmil-images/mine/5w96) | Solution structure of phage derived peptide inhibitor of frizzled 7 receptor | 分子名称: | Fz7 binding peptide | 著者 | Nile, A.H, de Sousa e Melo, F, Mukund, S, Piskol, R, Hansen, S, Zhou, L, Zhang, Y, Fu, Y, Gogol, E.B, Komuves, L.G, Modrusan, Z, Angers, S, Franke, Y, Koth, C, Fairbrother, W.J, Wang, W, de Sauvage, F.J, Hannoush, R.N. | 登録日 | 2017-06-22 | 公開日 | 2018-04-18 | 最終更新日 | 2023-06-14 | 実験手法 | SOLUTION NMR | 主引用文献 | A selective peptide inhibitor of Frizzled 7 receptors disrupts intestinal stem cells. Nat. Chem. Biol., 14, 2018
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5VRQ
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![BU of 5vrq by Molmil](/molmil-images/mine/5vrq) | Crystal structure of Legionella pneumophila effector AnkC | 分子名称: | Ankyrin repeat-containing protein | 著者 | Kozlov, G, Wong, K, Wang, W, Skubak, P, Munoz-Escobar, J, Liu, Y, Pannu, N.S, Gehring, K, Montreal-Kingston Bacterial Structural Genomics Initiative (BSGI) | 登録日 | 2017-05-11 | 公開日 | 2017-11-29 | 最終更新日 | 2024-03-13 | 実験手法 | X-RAY DIFFRACTION (3.205 Å) | 主引用文献 | Ankyrin repeats as a dimerization module. Biochem. Biophys. Res. Commun., 495, 2018
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