7WJZ
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![BU of 7wjz by Molmil](/molmil-images/mine/7wjz) | Omicron Spike bitrimer with 6m6 antibody | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, 6m6 heavy chain, 6m6 light chain, ... | 著者 | Zhan, W.Q, Zhang, X, Chen, Z.G, Sun, L. | 登録日 | 2022-01-08 | 公開日 | 2022-07-13 | 最終更新日 | 2022-09-14 | 実験手法 | ELECTRON MICROSCOPY (3.34 Å) | 主引用文献 | A broadly neutralizing antibody against SARS-CoV-2 Omicron variant infection exhibiting a novel trimer dimer conformation in spike protein binding. Cell Res., 32, 2022
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8K6B
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8K6A
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![BU of 8k6a by Molmil](/molmil-images/mine/8k6a) | |
8K68
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8K67
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![BU of 8k67 by Molmil](/molmil-images/mine/8k67) | |
8K6C
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![BU of 8k6c by Molmil](/molmil-images/mine/8k6c) | |
8K6D
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7XUP
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![BU of 7xup by Molmil](/molmil-images/mine/7xup) | Crystal structure of TPe3.0 | 分子名称: | Transcriptional regulator, PadR-like family | 著者 | Chen, X, Qian, J.Y, Sun, N.N, Zhong, F.R, Wu, Y.Z. | 登録日 | 2022-05-19 | 公開日 | 2022-09-28 | 最終更新日 | 2024-05-08 | 実験手法 | X-RAY DIFFRACTION (2.602 Å) | 主引用文献 | Enantioselective [2+2]-cycloadditions with triplet photoenzymes. Nature, 611, 2022
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7XUQ
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![BU of 7xuq by Molmil](/molmil-images/mine/7xuq) | Crystal structure of Tpe3.0 complexed with N-Boc-3-alkenylindole | 分子名称: | Transcriptional regulator, PadR-like family, dimethyl 2-[[2-methyl-1-[(2-methylpropan-2-yl)oxycarbonyl]indol-3-yl]methyl]-2-prop-2-enyl-propanedioate | 著者 | Chen, X, Qian, J.Y, Sun, N.N, Zhong, F.R, Wu, Y.Z. | 登録日 | 2022-05-19 | 公開日 | 2022-09-28 | 最終更新日 | 2024-05-08 | 実験手法 | X-RAY DIFFRACTION (2.5 Å) | 主引用文献 | Enantioselective [2+2]-cycloadditions with triplet photoenzymes. Nature, 611, 2022
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7END
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7EN9
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![BU of 7en9 by Molmil](/molmil-images/mine/7en9) | Crystal structure of SARS-CoV-2 3CLpro in complex with the non-covalent inhibitor WU-02 | 分子名称: | 3C-like proteinase, 5-bromanyl-~{N}-methyl-3-nitro-2-[(4~{R},5~{S})-2-(7-oxidanylisoquinolin-4-yl)carbonyl-4-phenyl-2,7-diazaspiro[4.4]nonan-7-yl]benzamide | 著者 | Hou, N, Peng, C, Hu, Q. | 登録日 | 2021-04-16 | 公開日 | 2022-07-20 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Development of Highly Potent Noncovalent Inhibitors of SARS-CoV-2 3CLpro. Acs Cent.Sci., 9, 2023
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7EN8
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![BU of 7en8 by Molmil](/molmil-images/mine/7en8) | Crystal structure of SARS-CoV-2 3CLpro in complex with the non-covalent inhibitor WU-04 | 分子名称: | 3C-like proteinase, GLYCEROL, ~{N}-[(1~{S},2~{R})-2-[[4-bromanyl-2-(methylcarbamoyl)-6-nitro-phenyl]amino]cyclohexyl]isoquinoline-4-carboxamide | 著者 | Hou, N, Peng, C, Hu, Q. | 登録日 | 2021-04-16 | 公開日 | 2022-07-20 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (1.83 Å) | 主引用文献 | Development of Highly Potent Noncovalent Inhibitors of SARS-CoV-2 3CLpro. Acs Cent.Sci., 9, 2023
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7ENE
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7EPX
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![BU of 7epx by Molmil](/molmil-images/mine/7epx) | S protein of SARS-CoV-2 in complex with GW01 | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Spike glycoprotein, ... | 著者 | Shen, Y.P, Zhang, Y.Y, Yan, R.H, Li, Y.N, Zhou, Q. | 登録日 | 2021-04-28 | 公開日 | 2022-05-18 | 実験手法 | ELECTRON MICROSCOPY (3 Å) | 主引用文献 | Novel sarbecovirus bispecific neutralizing antibodies with exceptional breadth and potency against currently circulating SARS-CoV-2 variants and sarbecoviruses. Cell Discov, 8, 2022
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7VEG
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![BU of 7veg by Molmil](/molmil-images/mine/7veg) | Understanding NH-pi interaction between Gln and Phe | 分子名称: | (2~{S},4~{R})-4-oxidanylpyrrolidine-2-carboxamide, ACETYLAMINO-ACETIC ACID, peptide | 著者 | Fan, S, Xu, F. | 登録日 | 2021-09-08 | 公開日 | 2022-10-19 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (1.385 Å) | 主引用文献 | Structural Achievability of an NH-pi Interaction between Gln and Phe in a Crystal Structure of a Collagen-like Peptide. Biomolecules, 12, 2022
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7Y8F
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![BU of 7y8f by Molmil](/molmil-images/mine/7y8f) | Estrogen Receptor Alpha Ligand Binding Domain Y537S Mutant in Complex with an Inhibitor 30o and GRIP Peptide | 分子名称: | DI(HYDROXYETHYL)ETHER, Estrogen receptor, Grip peptide, ... | 著者 | Min, J, Hu, H.B, Yang, Y, Dong, C.E, Zhou, H.B, Chen, C.-C, Guo, R.-T. | 登録日 | 2022-06-23 | 公開日 | 2023-04-26 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (2.22 Å) | 主引用文献 | Structure-guided identification of novel dual-targeting estrogen receptor alpha degraders with aromatase inhibitory activity for the treatment of endocrine-resistant breast cancer. Eur.J.Med.Chem., 253, 2023
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7Y8G
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![BU of 7y8g by Molmil](/molmil-images/mine/7y8g) | Estrogen Receptor Alpha Ligand Binding Domain Y537S Mutant in Complex with an Inhibitor 30a and GRIP Peptide | 分子名称: | DI(HYDROXYETHYL)ETHER, Estrogen receptor, Grip peptide, ... | 著者 | Min, J, Hu, H.B, Yang, Y, Dong, C.E, Zhou, H.B, Chen, C.-C, Guo, R.-T. | 登録日 | 2022-06-23 | 公開日 | 2023-04-26 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (2.14 Å) | 主引用文献 | Structure-guided identification of novel dual-targeting estrogen receptor alpha degraders with aromatase inhibitory activity for the treatment of endocrine-resistant breast cancer. Eur.J.Med.Chem., 253, 2023
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7WOS
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![BU of 7wos by Molmil](/molmil-images/mine/7wos) | The state 3 of Omicron Spike with bispecific antibody FD01 | 分子名称: | 16L9 Fv, 2-acetamido-2-deoxy-beta-D-glucopyranose, GW01 Fv, ... | 著者 | Zhang, X, Zhan, W.Q, Chen, Z.G, Sun, L. | 登録日 | 2022-01-22 | 公開日 | 2022-11-30 | 実験手法 | ELECTRON MICROSCOPY (3.91 Å) | 主引用文献 | Combating the SARS-CoV-2 Omicron (BA.1) and BA.2 with potent bispecific antibodies engineered from non-Omicron neutralizing antibodies Cell Discov, 8, 2022
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7WOQ
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![BU of 7woq by Molmil](/molmil-images/mine/7woq) | The state 1 of Omicron Spike with bispecific antibody FD01 | 分子名称: | 16L9 Fv, 2-acetamido-2-deoxy-beta-D-glucopyranose, Spike glycoprotein | 著者 | Zhang, X, Zhan, W.Q, Chen, Z.G, Sun, L. | 登録日 | 2022-01-22 | 公開日 | 2022-11-30 | 実験手法 | ELECTRON MICROSCOPY (3.47 Å) | 主引用文献 | Combating the SARS-CoV-2 Omicron (BA.1) and BA.2 with potent bispecific antibodies engineered from non-Omicron neutralizing antibodies Cell Discov, 8, 2022
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7WOU
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![BU of 7wou by Molmil](/molmil-images/mine/7wou) | The state 4 of Omicron Spike with bispecific antibody FD01 | 分子名称: | 16L9 Fv, 2-acetamido-2-deoxy-beta-D-glucopyranose, GW01 Fv, ... | 著者 | Zhang, X, Zhan, W.Q, Chen, Z.G, Sun, L. | 登録日 | 2022-01-22 | 公開日 | 2022-11-30 | 実験手法 | ELECTRON MICROSCOPY (3.47 Å) | 主引用文献 | Combating the SARS-CoV-2 Omicron (BA.1) and BA.2 with potent bispecific antibodies engineered from non-Omicron neutralizing antibodies Cell Discov, 8, 2022
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7WOP
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![BU of 7wop by Molmil](/molmil-images/mine/7wop) | The local refined map of Omicron spike with bispecific antibody FD01 | 分子名称: | 16L9, GW01, Spike protein S1 | 著者 | Zhang, X, Zhan, W.Q, Chen, Z.G, Sun, L. | 登録日 | 2022-01-22 | 公開日 | 2022-11-30 | 実験手法 | ELECTRON MICROSCOPY (3.51 Å) | 主引用文献 | Combating the SARS-CoV-2 Omicron (BA.1) and BA.2 with potent bispecific antibodies engineered from non-Omicron neutralizing antibodies Cell Discov, 8, 2022
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7WOR
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![BU of 7wor by Molmil](/molmil-images/mine/7wor) | The state 2 of Omicron Spike with bispecific antibody FD01 | 分子名称: | 16L9 Fv, 2-acetamido-2-deoxy-beta-D-glucopyranose, GW01 Fv, ... | 著者 | Zhang, X, Zhan, W.Q, Chen, Z.G, Sun, L. | 登録日 | 2022-01-22 | 公開日 | 2022-11-30 | 実験手法 | ELECTRON MICROSCOPY (3.7 Å) | 主引用文献 | Combating the SARS-CoV-2 Omicron (BA.1) and BA.2 with potent bispecific antibodies engineered from non-Omicron neutralizing antibodies Cell Discov, 8, 2022
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7WOV
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![BU of 7wov by Molmil](/molmil-images/mine/7wov) | The state 5 of Omicron Spike with bispecific antibody FD01 | 分子名称: | 16L9 Fv, 2-acetamido-2-deoxy-beta-D-glucopyranose, GW01 Fv, ... | 著者 | Zhang, X, Zhan, W.Q, Sun, L, Chen, Z.G. | 登録日 | 2022-01-22 | 公開日 | 2022-11-30 | 実験手法 | ELECTRON MICROSCOPY (3.87 Å) | 主引用文献 | Combating the SARS-CoV-2 Omicron (BA.1) and BA.2 with potent bispecific antibodies engineered from non-Omicron neutralizing antibodies Cell Discov, 8, 2022
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7WOW
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![BU of 7wow by Molmil](/molmil-images/mine/7wow) | The state 6 of Omicron Spike with bispecific antibody FD01 | 分子名称: | 16L9 Fv, GW01 Fv, Spike glycoprotein | 著者 | Zhang, X, Zhan, W.Q, Chen, Z.G, Sun, L. | 登録日 | 2022-01-22 | 公開日 | 2022-11-30 | 実験手法 | ELECTRON MICROSCOPY (6.11 Å) | 主引用文献 | Combating the SARS-CoV-2 Omicron (BA.1) and BA.2 with potent bispecific antibodies engineered from non-Omicron neutralizing antibodies Cell Discov, 8, 2022
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7X1N
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![BU of 7x1n by Molmil](/molmil-images/mine/7x1n) | Crystal structure of MEF2D-MRE complex | 分子名称: | DNA (5'-D(P*AP*AP*CP*TP*AP*TP*TP*TP*AP*TP*AP*AP*G)-3'), DNA (5'-D(P*TP*CP*TP*TP*AP*TP*AP*AP*AP*TP*AP*GP*T)-3'), Myocyte enhancer factor 2D/deleted in azoospermia associated protein 1 fusion protein | 著者 | Zhang, H, Zhang, M, Wang, Q.Q, Chen, Z, Chen, S.J, Meng, G. | 登録日 | 2022-02-24 | 公開日 | 2022-05-25 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (3.315 Å) | 主引用文献 | Functional, structural, and molecular characterizations of the leukemogenic driver MEF2D-HNRNPUL1 fusion. Blood, 140, 2022
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