6TJP
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![BU of 6tjp by Molmil](/molmil-images/mine/6tjp) | Crystal structure of T7 bacteriophage portal protein, 13mer, closed valve - P212121 | 分子名称: | Portal protein | 著者 | Fabrega-Ferrer, M, Cuervo, A, Fernandez, F.J, Machon, C, Perez-Luque, R, Pous, J, Vega, M.C, Carrascosa, J.L, Coll, M. | 登録日 | 2019-11-26 | 公開日 | 2020-12-16 | 最終更新日 | 2024-05-01 | 実験手法 | X-RAY DIFFRACTION (3.74 Å) | 主引用文献 | Using a partial atomic model from medium-resolution cryo-EM to solve a large crystal structure. Acta Crystallogr D Struct Biol, 77, 2021
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7AVW
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![BU of 7avw by Molmil](/molmil-images/mine/7avw) | |
7BMK
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![BU of 7bmk by Molmil](/molmil-images/mine/7bmk) | ATP-Competitive Partial Antagonists-'PAIR's-Rheostatically Modulate IRE1alpha's Kinase Helix-alphaC to Segregate its RNase-Mediated Biological Outputs | 分子名称: | 1,2-ETHANEDIOL, 2,2,2-tris(fluoranyl)-~{N}-[4-[3-[2-[[(3~{S})-piperidin-3-yl]amino]pyrimidin-4-yl]pyridin-2-yl]oxynaphthalen-1-yl]ethanesulfonamide, DI(HYDROXYETHYL)ETHER, ... | 著者 | Feldman, H.C, Ghosh, R, Auyeung, V, Mueller, J.L, Vidadala, V.N, Olivier, A, Backes, B.J, Zikherman, J, Papa, F.R, Maly, D.J. | 登録日 | 2021-01-20 | 公開日 | 2021-09-29 | 最終更新日 | 2022-04-13 | 実験手法 | X-RAY DIFFRACTION (1.85 Å) | 主引用文献 | ATP-competitive partial antagonists of the IRE1 alpha RNase segregate outputs of the UPR. Nat.Chem.Biol., 17, 2021
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7F5X
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![BU of 7f5x by Molmil](/molmil-images/mine/7f5x) | GK domain of Drosophila P5CS filament with glutamate | 分子名称: | Delta-1-pyrroline-5-carboxylate synthase, GAMMA-L-GLUTAMIC ACID | 著者 | Liu, J.L, Zhong, J, Guo, C.J, Zhou, X. | 登録日 | 2021-06-23 | 公開日 | 2022-04-06 | 最終更新日 | 2024-06-12 | 実験手法 | ELECTRON MICROSCOPY (3.5 Å) | 主引用文献 | Structural basis of dynamic P5CS filaments. Elife, 11, 2022
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7F5U
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![BU of 7f5u by Molmil](/molmil-images/mine/7f5u) | |
7F5V
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![BU of 7f5v by Molmil](/molmil-images/mine/7f5v) | Drosophila P5CS filament with glutamate, ATP, and NADPH | 分子名称: | Delta-1-pyrroline-5-carboxylate synthase | 著者 | Liu, J.L, Zhong, J, Guo, C.J, Zhou, X. | 登録日 | 2021-06-22 | 公開日 | 2022-04-06 | 最終更新日 | 2024-06-12 | 実験手法 | ELECTRON MICROSCOPY (3.6 Å) | 主引用文献 | Structural basis of dynamic P5CS filaments. Elife, 11, 2022
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7DPW
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![BU of 7dpw by Molmil](/molmil-images/mine/7dpw) | Structural basis for ligand binding modes of CTP synthase | 分子名称: | CTP synthase, CYTIDINE-5'-TRIPHOSPHATE, MAGNESIUM ION | 著者 | Liu, J.L, Zhou, X, Guo, C.J, Chang, C.C. | 登録日 | 2020-12-21 | 公開日 | 2021-09-15 | 最終更新日 | 2024-06-05 | 実験手法 | ELECTRON MICROSCOPY (2.65 Å) | 主引用文献 | Structural basis for ligand binding modes of CTP synthase. Proc.Natl.Acad.Sci.USA, 118, 2021
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7DPT
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![BU of 7dpt by Molmil](/molmil-images/mine/7dpt) | Structural basis for ligand binding modes of CTP synthase | 分子名称: | 6-DIAZENYL-5-OXO-L-NORLEUCINE, ADENOSINE-5'-DIPHOSPHATE, CTP synthase, ... | 著者 | Liu, J.L, Zhou, X, Guo, C.J, Chang, C.C. | 登録日 | 2020-12-21 | 公開日 | 2021-09-15 | 実験手法 | ELECTRON MICROSCOPY (2.48 Å) | 主引用文献 | Structural basis for ligand binding modes of CTP synthase. Proc.Natl.Acad.Sci.USA, 118, 2021
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7F5T
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![BU of 7f5t by Molmil](/molmil-images/mine/7f5t) | Drosophila P5CS filament with glutamate | 分子名称: | Delta-1-pyrroline-5-carboxylate synthase, GLUTAMIC ACID | 著者 | Liu, J.L, Zhong, J, Guo, C.J, Zhou, X. | 登録日 | 2021-06-22 | 公開日 | 2022-05-18 | 最終更新日 | 2024-06-12 | 実験手法 | ELECTRON MICROSCOPY (4.1 Å) | 主引用文献 | Structural basis of dynamic P5CS filaments. Elife, 11, 2022
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7EKB
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![BU of 7ekb by Molmil](/molmil-images/mine/7ekb) | Crystal structure of 4E10 modified with pyrene acetamide | 分子名称: | ACETATE ION, Fab region of the heavy chain of broadly neutralizing antibody anti-HIV-1 4E10, Fab region of the light chain of the broadly neutralizing anti-HIV-1 antibody 4E10, ... | 著者 | Caaveiro, J.M.M, Rujas, E, Nieva, J.L. | 登録日 | 2021-04-05 | 公開日 | 2021-08-11 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (1.45 Å) | 主引用文献 | Focal accumulation of aromaticity at the CDRH3 loop mitigates 4E10 polyreactivity without altering its HIV neutralization profile. Iscience, 24, 2021
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7EKK
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![BU of 7ekk by Molmil](/molmil-images/mine/7ekk) | Anti-HIV-1 broadly neutralizing antibody delta-loop 4E10 modified with pyrene acetamide | 分子名称: | AMMONIUM ION, CHLORIDE ION, GLYCEROL, ... | 著者 | Caaveiro, J.M.M, Rujas, E, Nieva, J.L. | 登録日 | 2021-04-05 | 公開日 | 2021-08-11 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (1.7 Å) | 主引用文献 | Focal accumulation of aromaticity at the CDRH3 loop mitigates 4E10 polyreactivity without altering its HIV neutralization profile. Iscience, 24, 2021
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6XYY
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![BU of 6xyy by Molmil](/molmil-images/mine/6xyy) | Update of ACHE FROM DROSOPHILA MELANOGASTER COMPLEX WITH TACRINE DERIVATIVE 9-(3-PHENYLMETHYLAMINO)-1,2,3,4-TETRAHYDROACRIDINE | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, 9-(3-PHENYLMETHYLAMINO)-1,2,3,4-TETRAHYDROACRIDINE, Acetylcholinesterase, ... | 著者 | Nachon, F, Sussman, J.L. | 登録日 | 2020-01-31 | 公開日 | 2020-03-18 | 最終更新日 | 2024-01-24 | 実験手法 | X-RAY DIFFRACTION (2.7 Å) | 主引用文献 | A Second Look at the Crystal Structures ofDrosophila melanogasterAcetylcholinesterase in Complex with Tacrine Derivatives Provides Insights Concerning Catalytic Intermediates and the Design of Specific Insecticides. Molecules, 25, 2020
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6XSE
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![BU of 6xse by Molmil](/molmil-images/mine/6xse) | |
6XSH
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![BU of 6xsh by Molmil](/molmil-images/mine/6xsh) | |
6XH2
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![BU of 6xh2 by Molmil](/molmil-images/mine/6xh2) | |
6XLX
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![BU of 6xlx by Molmil](/molmil-images/mine/6xlx) | |
6XLV
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![BU of 6xlv by Molmil](/molmil-images/mine/6xlv) | |
6XSC
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![BU of 6xsc by Molmil](/molmil-images/mine/6xsc) | |
6XSI
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![BU of 6xsi by Molmil](/molmil-images/mine/6xsi) | |
6XRM
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![BU of 6xrm by Molmil](/molmil-images/mine/6xrm) | Crystal structure of human PI3K-gamma in complex with Compound 4 | 分子名称: | 5-[2-amino-3-(1-methyl-1H-pyrazol-4-yl)pyrazolo[1,5-a]pyrimidin-5-yl]-2-[(1S)-1-cyclopropylethyl]-7-(trifluoromethyl)-2,3-dihydro-1H-isoindol-1-one, Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform, SULFATE ION | 著者 | Walker, N.P, Jeffrey, J.L. | 登録日 | 2020-07-13 | 公開日 | 2020-09-16 | 最終更新日 | 2024-03-06 | 実験手法 | X-RAY DIFFRACTION (2.88 Å) | 主引用文献 | Discovery of Potent and Selective PI3K gamma Inhibitors. J.Med.Chem., 63, 2020
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1X7Z
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![BU of 1x7z by Molmil](/molmil-images/mine/1x7z) | Crystal structure of the human mitochondrial branched-chain alpha-ketoacid dehydrogenase | 分子名称: | 2-oxoisovalerate dehydrogenase alpha subunit, 2-oxoisovalerate dehydrogenase beta subunit, CHLORIDE ION, ... | 著者 | Wynn, R.M, Kato, M, Machius, M, Chuang, J.L, Li, J, Tomchick, D.R, Chuang, D.T. | 登録日 | 2004-08-16 | 公開日 | 2004-11-23 | 最終更新日 | 2023-08-23 | 実験手法 | X-RAY DIFFRACTION (1.72 Å) | 主引用文献 | Molecular mechanism for regulation of the human mitochondrial branched-chain alpha-ketoacid dehydrogenase complex by phosphorylation Structure, 12, 2004
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1X7Y
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![BU of 1x7y by Molmil](/molmil-images/mine/1x7y) | Crystal structure of the human mitochondrial branched-chain alpha-ketoacid dehydrogenase | 分子名称: | 2-oxoisovalerate dehydrogenase alpha subunit, 2-oxoisovalerate dehydrogenase beta subunit, CHLORIDE ION, ... | 著者 | Wynn, R.M, Kato, M, Machius, M, Chuang, J.L, Li, J, Tomchick, D.R, Chuang, D.T. | 登録日 | 2004-08-16 | 公開日 | 2004-11-23 | 最終更新日 | 2023-08-23 | 実験手法 | X-RAY DIFFRACTION (1.57 Å) | 主引用文献 | Molecular mechanism for regulation of the human mitochondrial branched-chain alpha-ketoacid dehydrogenase complex by phosphorylation Structure, 12, 2004
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6XN8
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![BU of 6xn8 by Molmil](/molmil-images/mine/6xn8) | Crystal Structure of 2-hydroxyacyl CoA lyase (HACL) from Rhodospirillales bacterium URHD0017 | 分子名称: | 2-hydroxyacyl-CoA lyase 1, 2-{3-[(4-AMINO-2-METHYLPYRIMIDIN-5-YL)METHYL]-4-METHYL-2-OXO-2,3-DIHYDRO-1,3-THIAZOL-5-YL}ETHYL TRIHYDROGEN DIPHOSPHATE, ADENOSINE-5'-DIPHOSPHATE, ... | 著者 | Miller, M.D, Xu, W, Olmos Jr, J.L, Chou, A, Clomburg, J.M, Gonzalez, R, Philips Jr, G.N. | 登録日 | 2020-07-02 | 公開日 | 2021-07-07 | 最終更新日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (1.95 Å) | 主引用文献 | Crystal Structure of 2-hydroxyacyl CoA lyase (HACL) from Rhodospirillales bacterium URHD0017 To Be Published
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6XU6
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![BU of 6xu6 by Molmil](/molmil-images/mine/6xu6) | Drosophila melanogaster Testis 80S ribosome | 分子名称: | 18S ribosomal RNA, 28S ribosomal RNA, 2S ribosomal RNA, ... | 著者 | Hopes, T, Agapiou, M, Norris, K, McCarthy, C.G.P, OConnell, M.J, Fontana, J, Aspden, J.L. | 登録日 | 2020-01-17 | 公開日 | 2021-07-28 | 最終更新日 | 2022-12-21 | 実験手法 | ELECTRON MICROSCOPY (3.5 Å) | 主引用文献 | Ribosome heterogeneity in Drosophila melanogaster gonads through paralog-switching. Nucleic Acids Res., 50, 2022
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6XU8
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![BU of 6xu8 by Molmil](/molmil-images/mine/6xu8) | Drosophila melanogaster Ovary 80S ribosome | 分子名称: | 18S ribosomal RNA, 28S ribosomal RNA, 2S ribosomal RNA, ... | 著者 | Hopes, T, Agapiou, M, Norris, K, McCarthy, C.G.P, OConnell, M.J, Fontana, J, Aspden, J.L. | 登録日 | 2020-01-17 | 公開日 | 2021-07-28 | 最終更新日 | 2022-12-21 | 実験手法 | ELECTRON MICROSCOPY (3 Å) | 主引用文献 | Ribosome heterogeneity in Drosophila melanogaster gonads through paralog-switching. Nucleic Acids Res., 50, 2022
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