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4IE6
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BU of 4ie6 by Molmil
Crystal structure of the human fat mass and obesity associated protein (FTO) in complex with N-[(1-chloro-4-hydroxyisoquinolin-3-yl)carbonyl]glycine (IOX3/UN9)
分子名称: Alpha-ketoglutarate-dependent dioxygenase FTO, N-[(1-CHLORO-4-HYDROXYISOQUINOLIN-3-YL)CARBONYL]GLYCINE, ZINC ION
著者Aik, W.S, McDonough, M.A, Schofield, C.J.
登録日2012-12-13
公開日2013-04-03
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (2.5036 Å)
主引用文献Structural basis for inhibition of the fat mass and obesity associated protein (FTO)
J.Med.Chem., 56, 2013
4IDZ
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BU of 4idz by Molmil
Crystal structure of the human fat mass and obesity associated protein (FTO) in complex with N-oxalylglycine (NOG)
分子名称: Alpha-ketoglutarate-dependent dioxygenase FTO, GLYCEROL, N-OXALYLGLYCINE, ...
著者Aik, W.S, McDonough, M.A, Schofield, C.J.
登録日2012-12-13
公開日2013-04-03
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (2.46 Å)
主引用文献Structural basis for inhibition of the fat mass and obesity associated protein (FTO)
J.Med.Chem., 56, 2013
4IE4
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BU of 4ie4 by Molmil
Crystal structure of the human fat mass and obesity associated protein (FTO) in complex with 5-carboxy-8-hydroxyquinoline (IOX1)
分子名称: 8-hydroxyquinoline-5-carboxylic acid, Alpha-ketoglutarate-dependent dioxygenase FTO, GLYCEROL, ...
著者Aik, W.S, McDonough, M.A, Schofield, C.J.
登録日2012-12-13
公開日2013-04-03
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (2.5048 Å)
主引用文献Structural basis for inhibition of the fat mass and obesity associated protein (FTO)
J.Med.Chem., 56, 2013
4J8S
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BU of 4j8s by Molmil
Crystal structure of human CNOT1 MIF4G domain in complex with a TTP peptide
分子名称: CCR4-NOT transcription complex subunit 1, Tristetraprolin
著者Frank, F, Fabian, M.R, Rouya, C, Siddiqui, N, Lai, W.S, Karetnikov, A, Blackshear, P.J, Sonenberg, N, Nagar, B.
登録日2013-02-14
公開日2013-05-08
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (1.55 Å)
主引用文献Structural basis for the recruitment of the human CCR4-NOT deadenylase complex by tristetraprolin.
Nat.Struct.Mol.Biol., 20, 2013
4JIT
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BU of 4jit by Molmil
Crystal Structure of E. coli XGPRT in complex with (S)-3-(Guanin-9-yl)pyrrolidin-N-ylacetylphosphonic acid
分子名称: Xanthine phosphoribosyltransferase, {2-[(3S)-3-(2-amino-6-oxo-1,6-dihydro-9H-purin-9-yl)pyrrolidin-1-yl]-2-oxoethyl}phosphonic acid
著者Keough, D.T, Hockova, D, Rejman, D, Spacek, P, Vrbkova, S, Krecmerova, M, Eng, W.S, Jans, H, West, N.P, Naesens, L.M.J, de Jersey, J, Guddat, L.W.
登録日2013-03-07
公開日2014-12-24
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献Inhibition of the Escherichia coli 6-oxopurine phosphoribosyltransferases by nucleoside phosphonates: potential for new antibacterial agents.
J.Med.Chem., 56, 2013
4JLS
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BU of 4jls by Molmil
Crystal Structure of E. coli XGPRT in complex with (3R,4S)-4-(Guanin-9-yl)-3-hydroxypyrrolidin-1-N-ylacetylphosphonic acid
分子名称: Xanthine phosphoribosyltransferase, {2-[(3S,4R)-3-(2-amino-6-oxo-1,6-dihydro-9H-purin-9-yl)-4-hydroxypyrrolidin-1-yl]-2-oxoethyl}phosphonic acid
著者Keough, D.T, Hockova, D, Rejman, D, Spacek, P, Vrbkova, S, Krecmerova, M, Eng, W.S, Jans, H, West, N.P, Naesens, L.M.J, de Jersey, J, Guddat, L.W.
登録日2013-03-12
公開日2014-12-24
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Inhibition of the Escherichia coli 6-oxopurine phosphoribosyltransferases by nucleoside phosphonates: potential for new antibacterial agents.
J.Med.Chem., 56, 2013
4KGS
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BU of 4kgs by Molmil
Backbone Modifications in the Protein GB1 Loops: beta-3-Val21, beta-3-Asp40
分子名称: GLYCEROL, Streptococcal Protein GB1 Backbone Modified Variant: beta-3-Val21, beta-3-Asp40
著者Reinert, Z.E, Lengyel, G.A, Horne, W.S.
登録日2013-04-29
公開日2013-09-04
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (1.95 Å)
主引用文献Protein-like Tertiary Folding Behavior from Heterogeneous Backbones.
J.Am.Chem.Soc., 135, 2013
4KGR
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BU of 4kgr by Molmil
Backbone Modifications in the Protein GB1 Helix: beta-3-Ala24, beta-3-Lys28, beta-3-Lys31, beta-3-Asn35
分子名称: GLYCEROL, Streptococcal Protein GB1 Backbone Modified Variant: beta-3-Ala24, beta-3-Lys28, ...
著者Reinert, Z.E, Lengyel, G.A, Horne, W.S.
登録日2013-04-29
公開日2013-09-04
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Protein-like Tertiary Folding Behavior from Heterogeneous Backbones.
J.Am.Chem.Soc., 135, 2013
4KGT
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BU of 4kgt by Molmil
Backbone Modifications in the Protein GB1 Turns: Aib10, D-Pro47
分子名称: Streptococcal Protein GB1 Backbone Modified Variant: Aib10, D-Pro47
著者Reinert, Z.E, Lengyel, G.A, Horne, W.S.
登録日2013-04-29
公開日2013-09-04
最終更新日2023-12-06
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Protein-like Tertiary Folding Behavior from Heterogeneous Backbones.
J.Am.Chem.Soc., 135, 2013
4LFM
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BU of 4lfm by Molmil
Crystal Structure of D-galactose-6-phosphate isomerase in complex with D-psicose
分子名称: D-psicose, Galactose-6-phosphate isomerase subunit A, Galactose-6-phosphate isomerase subunit B
著者Jung, W.S, Pan, C.H.
登録日2013-06-27
公開日2013-11-27
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (1.65 Å)
主引用文献Crystal structure and substrate specificity of D-galactose-6-phosphate isomerase complexed with substrates.
Plos One, 8, 2013
4LFN
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BU of 4lfn by Molmil
Crystal Structure of D-galactose-6-phosphate isomerase in complex with D-ribulose
分子名称: D-ribulose, Galactose-6-phosphate isomerase subunit A, Galactose-6-phosphate isomerase subunit B
著者Jung, W.S, Pan, C.H.
登録日2013-06-27
公開日2013-11-27
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (1.65 Å)
主引用文献Crystal structure and substrate specificity of D-galactose-6-phosphate isomerase complexed with substrates.
Plos One, 8, 2013
4LFK
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BU of 4lfk by Molmil
Crystal Structure of D-galactose-6-phosphate isomerase in a substrate-free form
分子名称: Galactose-6-phosphate isomerase subunit A, Galactose-6-phosphate isomerase subunit B
著者Jung, W.S, Pan, C.H.
登録日2013-06-27
公開日2013-11-27
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (1.96 Å)
主引用文献Crystal structure and substrate specificity of D-galactose-6-phosphate isomerase complexed with substrates.
Plos One, 8, 2013
4LFL
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BU of 4lfl by Molmil
Crystal Structure of D-galactose-6-phosphate isomerase in complex with D-tagatose-6-phosphate
分子名称: 6-O-phosphono-D-tagatose, Galactose-6-phosphate isomerase subunit A, Galactose-6-phosphate isomerase subunit B
著者Jung, W.S, Pan, C.H.
登録日2013-06-27
公開日2013-11-27
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (1.65 Å)
主引用文献Crystal structure and substrate specificity of D-galactose-6-phosphate isomerase complexed with substrates.
Plos One, 8, 2013
5U5B
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BU of 5u5b by Molmil
Coiled Coil Peptide Metal Coordination Framework: Trimer Fold
分子名称: COPPER (II) ION, Designed trimeric coiled coil peptide with two terpyridine side chains, GLYCEROL
著者Tavenor, N.A, Murnin, M.J, Horne, W.S.
登録日2016-12-06
公開日2017-02-22
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Supramolecular Metal-Coordination Polymers, Nets, and Frameworks from Synthetic Coiled-Coil Peptides.
J. Am. Chem. Soc., 139, 2017
5U59
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BU of 5u59 by Molmil
Coiled Coil Peptide Metal Coordination Framework: Dimer Fold Grown with Citrate
分子名称: CITRIC ACID, COPPER (II) ION, Designed dimeric coiled coil peptide with two terpyridine side chains
著者Tavenor, N.A, Murnin, M.J, Horne, W.S.
登録日2016-12-06
公開日2017-02-22
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Supramolecular Metal-Coordination Polymers, Nets, and Frameworks from Synthetic Coiled-Coil Peptides.
J. Am. Chem. Soc., 139, 2017
5U5C
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BU of 5u5c by Molmil
Coiled Coil Peptide Metal Coordination Framework: Tetramer Fold
分子名称: COPPER (II) ION, Designed tetrameric coiled coil peptide with one terpyridine side chain, HEXANE-1,6-DIOL
著者Tavenor, N.A, Murnin, M.J, Horne, W.S.
登録日2016-12-06
公開日2017-02-22
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Supramolecular Metal-Coordination Polymers, Nets, and Frameworks from Synthetic Coiled-Coil Peptides.
J. Am. Chem. Soc., 139, 2017
5U5A
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BU of 5u5a by Molmil
Coiled Coil Peptide Metal Coordination Framework: Dimer Fold
分子名称: COPPER (II) ION, Designed dimeric coiled coil peptide with two terpyridine side chains
著者Tavenor, N.A, Murnin, M.J, Horne, W.S.
登録日2016-12-06
公開日2017-02-22
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (3.23 Å)
主引用文献Supramolecular Metal-Coordination Polymers, Nets, and Frameworks from Synthetic Coiled-Coil Peptides.
J. Am. Chem. Soc., 139, 2017
5UX1
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BU of 5ux1 by Molmil
Protein 43 with aldehyde deformylating oxygenase activity from Synechococcus
分子名称: FE (III) ION, tRNA-(MS(2)IO(6)A)-hydroxylase-like
著者Wilson, D.K, Mak, W.S, Siegel, J.B.
登録日2017-02-21
公開日2018-02-28
最終更新日2024-03-06
実験手法X-RAY DIFFRACTION (1.5 Å)
主引用文献Protein 43 with aldehyde deformylating oxygenase activity from Synechococcus
To Be Published
5UUN
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BU of 5uun by Molmil
Crystal structure of SARO_2595 from Novosphingobium aromaticivorans
分子名称: ACETATE ION, GLUTATHIONE, Glutathione S-transferase-like protein
著者Bingman, C.A, Kontur, W.S, Olmsted, C.N, Fox, B.G, Donohue, T.J.
登録日2017-02-17
公開日2018-02-28
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (1.45 Å)
主引用文献Novosphingobium aromaticivoransuses a Nu-class glutathioneS-transferase as a glutathione lyase in breaking the beta-aryl ether bond of lignin.
J. Biol. Chem., 293, 2018
5UXI
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BU of 5uxi by Molmil
Protein 4 with aldehyde deformylating oxygenase activity from Nostoc puntiforme
分子名称: Aldehyde decarbonylase, DECYLAMINE-N,N-DIMETHYL-N-OXIDE
著者Wilson, D.K, Mak, W.S, Siegel, J.B.
登録日2017-02-22
公開日2018-02-28
最終更新日2024-03-06
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Protein 4 with aldehyde deformylating oxygenase activity from Nostoc puntiforme
To Be Published
5UX2
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BU of 5ux2 by Molmil
Protein 19 with aldehyde deformylating oxidase activity from Synechococcus
分子名称: Aldehyde decarbonylase, FE (III) ION, PROPANOIC ACID
著者Wilson, D.K, Mak, W.S, Siegel, J.B.
登録日2017-02-21
公開日2018-02-28
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (1.99 Å)
主引用文献Protein 19 with aldehyde deformylating oxidase activity from Synechococcus
To Be Published
5UUO
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BU of 5uuo by Molmil
Crystal structure of SARO_2595 from Novosphingobium aromaticivorans
分子名称: 1,2-ETHANEDIOL, GLUTATHIONE, Glutathione S-transferase-like protein, ...
著者Bingman, C.A, Kontur, W.S, Olmsted, C.N, Fox, B.G, Donohue, T.J.
登録日2017-02-17
公開日2018-02-28
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (1.25 Å)
主引用文献Novosphingobium aromaticivoransuses a Nu-class glutathioneS-transferase as a glutathione lyase in breaking the beta-aryl ether bond of lignin.
J. Biol. Chem., 293, 2018
5UXG
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BU of 5uxg by Molmil
Protein 84 with aldehyde deformylating oxygenase activity from Sulfolobus tokodaii (monoclinic)
分子名称: PHOSPHATE ION, aldehyde deformylating oxygenase
著者Wilson, D.K, Mak, W.S, Siegel, J.B.
登録日2017-02-22
公開日2018-02-28
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (1.72 Å)
主引用文献Protein 84 with aldehyde deformylating oxygenase activity from Sulfolobus tokodaii (monoclinic)
To Be Published
5V4T
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BU of 5v4t by Molmil
Protein 84 with aldehyde deformylating oxygenase activity from Sulfolobus tokodaii (orthorhombic form)
分子名称: 1,2-ETHANEDIOL, FE (III) ION, hypothetic aldehyde deformylating oxygenase
著者Wilson, D.K, Mak, W.S, Siegel, J.B.
登録日2017-03-10
公開日2018-03-14
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Protein 84 with aldehyde deformylating oxygenase activity from Sulfolobus tokodaii (orthorhombic form)
To Be Published
5US3
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BU of 5us3 by Molmil
Heterogeneous-backbone Foldamer Mimic of the Sp1-3 Zinc Finger
分子名称: Heterogeneous-Backbone Variant of the Sp1-3 Zinc Finger: N-Me-Ala3, N-Me-Arg10, beta-3-Asp15, ...
著者George, K.L, Horne, W.S.
登録日2017-02-13
公開日2017-05-31
最終更新日2023-11-15
実験手法SOLUTION NMR
主引用文献Heterogeneous-Backbone Foldamer Mimics of Zinc Finger Tertiary Structure.
J. Am. Chem. Soc., 139, 2017

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件を2024-05-29に公開中

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